GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor
- Adenosine Receptor
- Adrenergic Receptor
- Bombesin Receptor
- Bradykinin Receptor
- Cannabinoid Receptor
- CaSR
- Cholecystokinin
- CXCR
- Dopamine Receptor
- Endothelin Receptor
- Glucagon Receptor
- GNRH Receptor
- GPCR19
- GRK
- GTPase
- Hedgehog/Smoothened
- Histamine Receptor
- LPA Receptor
- Melatonin Receptor
- Opioid Receptor
- OX Receptor
- PAFR
- PKA
- S1P Receptor
- SGLT
- Sigma receptor
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Products of "GPCR/G-Protein"
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SR59230A
CAS:SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).Formula:C23H29NO6Purity:98.84%Color and Shape:SolidMolecular weight:415.48Ref: TM-T13016
1mg52.00€2mg77.00€5mg107.00€10mg172.00€25mg343.00€50mg510.00€100mg737.00€1mL*10mM (DMSO)125.00€PF-184298
CAS:PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.Formula:C15H20Cl2N2OPurity:98.30%Color and Shape:SolidMolecular weight:315.24Trazodone hydrochloride
CAS:Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.Formula:C19H23Cl2N5OPurity:99.50% - 99.52%Color and Shape:SolidMolecular weight:408.33Fenoterol hydrobromide
CAS:Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.Formula:C17H22BrNO4Purity:99.88%Color and Shape:SolidMolecular weight:384.27AP1189 acetate
CAS:AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.Formula:C16H18N6O4Purity:98.73%Color and Shape:SolidMolecular weight:358.35Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderateFormula:C21H32Cl2N4OPurity:99.68% - 99.87%Color and Shape:SolidMolecular weight:427.41Ref: TM-T4577
1mg51.00€5mg108.00€10mg180.00€25mg316.00€50mg472.00€100mg658.00€200mg938.00€1mL*10mM (DMSO)108.00€ML417
CAS:ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).Formula:C22H25N3O3Purity:98.81% - 99.42%Color and Shape:SolidMolecular weight:379.45[Ala17]-MCH acetate
[Ala17]-MCH acetate is a selective ligand for MCHR1 with a Ki of 0.16 nM and Kd of 0.37 nM(Eu3+ chelate-labeled).Formula:C99H159N29O28S4Purity:98.92%Color and Shape:SolidMolecular weight:2331.76CB2R/FAAH modulator-1
CAS:CB2R/FAAH modulator-1: agonizes CB2R, inhibits FAAH (IC50=4 μM), alters cytokine production; used in inflammation research. Ki: CB2R=14.8 nM, CB1R=241.3 nM.Formula:C24H27NO2Purity:100%Color and Shape:SoildMolecular weight:361.48Ref: TM-T67896
1mg77.00€5mg158.00€10mg225.00€25mg338.00€50mg472.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)163.00€CB2 modulator 1
CAS:CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.Formula:C18H19F3N4O2Purity:99.02%Color and Shape:SolidMolecular weight:380.36Ref: TM-T10696
1mg35.00€5mg56.00€10mg79.00€25mg114.00€50mg167.00€100mgTo inquire1mL*10mM (DMSO)64.00€Etelcalcetide hydrochloride
CAS:Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.Formula:C38H73N21O10S2HClPurity:100%Color and Shape:SolidMolecular weight:1353.332-Oleoylglycerol
CAS:2-Oleoylglycerol is a lipid found in palm kernels that acts as a GPR119 agonist with neuroprotective properties and can be used in steatohepatitis modeling.Formula:C21H40O4Purity:98%Color and Shape:SolidMolecular weight:356.54Rocastine
CAS:Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.Formula:C13H19N3OSPurity:98.26%Color and Shape:SolidMolecular weight:265.37CXCR2-IN-1
CAS:CXCR2-IN-1 has a pIC50 of 9.3 and is a CXCR2 antagonist of the central nervous system penetration agent.Formula:C19H20Cl2FN3O4SPurity:99.53%Color and Shape:SolidMolecular weight:476.35NIBR189
CAS:NIBR189 is a potent and selective antagonist of EBI2 (GPR183) receptor (IC50 of 11 and 15 nM for human and mouse EBI2 receptors, respectively)Formula:C21H21BrN2O3Purity:97%Color and Shape:ColourlessMolecular weight:429.31Escitalopram
CAS:Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.Formula:C20H21FN2OPurity:99.82%Color and Shape:White Or White Crystalline PowderMolecular weight:324.39Calcitonin(salmon) Acetate(47931-85-1(free base))
Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5Formula:C145H240N44O48S2Purity:99.29%Color and Shape:SolidMolecular weight:3431.85Efaroxan hydrochloride
CAS:Efaroxan hydrochloride a selective, oral α2-adrenoceptor antagonist significantly potentiates adrenaline-induced increases in insulin levels.Formula:C13H17ClN2OPurity:98%Color and Shape:SolidMolecular weight:252.74PW0787
CAS:PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).Formula:C23H20F4N4O2Purity:98.42%Color and Shape:SolidMolecular weight:460.42Ref: TM-T9452
1mg37.00€5mg80.00€10mg117.00€25mg235.00€50mg353.00€100mg500.00€200mg690.00€1mL*10mM (DMSO)96.00€Evofolin B
CAS:Evofolin B is a natural compound isolated from the stem bark of Zanthoxylum ailanthoides.Formula:C17H18O6Purity:98%Color and Shape:SolidMolecular weight:318.32
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