GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor
- Adenosine Receptor
- Adrenergic Receptor
- Bombesin Receptor
- Bradykinin Receptor
- Cannabinoid Receptor
- CaSR
- Cholecystokinin
- CXCR
- Dopamine Receptor
- Endothelin Receptor
- Glucagon Receptor
- GNRH Receptor
- GPCR19
- GRK
- GTPase
- Hedgehog/Smoothened
- Histamine Receptor
- LPA Receptor
- Melatonin Receptor
- Opioid Receptor
- OX Receptor
- PAFR
- PKA
- S1P Receptor
- SGLT
- Sigma receptor
Show 19 more subcategories
Products of "GPCR/G-Protein"
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Mibenratide TFA
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].Purity:98%Color and Shape:Odour SolidAS19
CAS:AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).Formula:C18H25N3Purity:98%Color and Shape:SolidMolecular weight:283.41Spns2-IN-1
Spns2-IN-1 is a potent Spns2 inhibitor, effectively impeding Spns2-dependent S1P transport with an IC50 value of 1.4±0.3 μM, crucial for modulating the immunePurity:98%Color and Shape:Odour SolidCP 96021
CAS:"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."Formula:C29H21FN4OSPurity:97.81% - 99.11%Color and Shape:SoildMolecular weight:492.57MK-571 sodium
CAS:MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.Formula:C26H27ClN2O3S2·NaPurity:97% - 98.69%Color and Shape:SolidMolecular weight:537.07SKF 81297
CAS:SKF 81297 is a selective and potent agonist for the dopamine D1 receptor [1].Formula:C16H16ClNO2Purity:98%Color and Shape:SolidMolecular weight:289.76LP-471756
CAS:LP-471756 is a specific antagonist of GPR139 and inhibits LP-360924-stimulated cAMP production (IC50 = 640 nM).Formula:C19H23NO2SPurity:99.59%Color and Shape:SolidMolecular weight:329.46Ref: TM-T27850
5mg48.00€10mg71.00€25mg135.00€50mg212.00€100mg340.00€200mg480.00€1mL*10mM (DMSO)49.00€Almorexant
CAS:Almorexant (ACT 078573), a strong dual orexin receptor antagonist, has Ki of 1.3 nM for OX1 and 0.17 nM for OX2.Formula:C29H31F3N2O3Purity:97.75% - 98.02%Color and Shape:SolidMolecular weight:512.56Felypressin acetate
CAS:Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.Formula:C48H69N13O13S2Purity:97.06%Color and Shape:SolidMolecular weight:1100.27Trazpiroben
CAS:Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Formula:C31H39N3O4Purity:98.85% - 99.41%Color and Shape:SolidMolecular weight:517.66AM-1638
CAS:AM-1638 is an orally active GPR40/FFA1 agonist, useful for studying type II diabetes.Formula:C33H35FO4Color and Shape:SolidMolecular weight:514.63Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formula:C22H31N3O2Purity:97.21% - 99.49%Color and Shape:SolidMolecular weight:369.5Ref: TM-T2278
1mg40.00€2mg52.00€5mg88.00€10mg125.00€25mg233.00€50mg424.00€100mg613.00€500mg1,264.00€1mL*10mM (DMSO)127.00€Men 10376 TFA(135306-85-3,free)
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4Formula:C59H69F3N12O12Purity:99.22%Color and Shape:SolidMolecular weight:1195.25Dazmegrel HCl
Dazmegrel HCl is a platelet thromboxane inhibitor used in the study of myocardial infarction and arrhythmias.Formula:C16H18ClN3O2Purity:98.63%Color and Shape:SolidMolecular weight:319.79OPC-51803
CAS:OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.Formula:C26H32ClN3O2Purity:100% - 100%Color and Shape:SolidMolecular weight:454Ref: TM-T28257
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€Talibegron hydrochloride
CAS:Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.Formula:C18H22ClNO4Purity:99.82%Color and Shape:SolidMolecular weight:351.83Amitriptyline
CAS:Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.Formula:C20H23NPurity:98.24% - 99.64%Color and Shape:Crystals SolidMolecular weight:277.4A2B receptor antagonist 2
CAS:A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).Formula:C12H15N5Purity:100%Color and Shape:SolidMolecular weight:229.28GLP-1R agonist 3
CAS:GLP-1R agonist 3 is a GLP-1R agonist, an imidazole derivative.GLP-1R agonist 3 can be used to study diabetes and obesity.Formula:C31H28FN5O4Purity:97.19%Color and Shape:SolidMolecular weight:553.582,6-DMA hydrochloride
CAS:2,6-DMA hydrochloride is a phenethylamine and acts as an agonist of the serotonin 5-HT2 receptor, with a pA2 value of 5.09.Formula:C11H18ClNO2Color and Shape:SolidMolecular weight:231.72
