GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor
- Adenosine Receptor
- Adrenergic Receptor
- Bombesin Receptor
- Bradykinin Receptor
- Cannabinoid Receptor
- CaSR
- Cholecystokinin
- CXCR
- Dopamine Receptor
- Endothelin Receptor
- Glucagon Receptor
- GNRH Receptor
- GPCR19
- GRK
- GTPase
- Hedgehog/Smoothened
- Histamine Receptor
- LPA Receptor
- Melatonin Receptor
- Opioid Receptor
- OX Receptor
- PAFR
- PKA
- S1P Receptor
- SGLT
- Sigma receptor
Show 19 more subcategories
Products of "GPCR/G-Protein"
Sort by
Cyamemazine
CAS:Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Formula:C19H21N3SPurity:97.01%Color and Shape:SolidMolecular weight:323.46Fenoterol
CAS:Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.Formula:C17H21NO4Purity:99.56%Color and Shape:SolidMolecular weight:303.35SARS-CoV-2-IN-57
CAS:SARS-CoV-2-IN-57 (compound (+)-R-26) is a potent inhibitor of SARS-CoV-2 with an IC50 of 80 nM and demonstrates high affinity for the Sigma Receptor, exhibitingFormula:C23H37N3OPurity:98%Color and Shape:SolidMolecular weight:371.564-Deoxypyridoxine hydrochloride
CAS:4-Deoxypyridoxine HCl halts S1P breakdown by blocking SPL, reducing apoptosis in insulinoma cells like S1P.Formula:C8H12ClNO2Purity:99.86%Color and Shape:White To Off White Crystalline PowderMolecular weight:189.64Diquafosol tetrasodium
CAS:Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear filmFormula:C18H22N4Na4O23P4Purity:98.7% - 99.97%Color and Shape:SolidMolecular weight:878.23Isoetharine mesylate salt
CAS:Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.Formula:C14H25NO6SPurity:99.35% - 99.75%Color and Shape:SolidMolecular weight:335.42Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formula:C26H28FN3O9Purity:99.68%Color and Shape:SolidMolecular weight:545.51JHU 75528
CAS:JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can be used to study the cannabinoid system in schizophrenic patients.Formula:C23H21Cl2N5O2Purity:99.97%Color and Shape:SolidMolecular weight:470.35Paynantheine
CAS:Paynantheine is an alkaloid with antinociceptive properties, found in Mitragyna speciosa. It also acts as an agonist at 5-HT1AR and 5-HT2BR receptors, inducing lower lip contraction and providing antinociception in rats.Formula:C23H28N2O4Color and Shape:SolidMolecular weight:396.48R 396 acetate
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.Formula:C41H55N9O12Purity:99.52%Color and Shape:SolidMolecular weight:865.93Ref: TM-T24697L
1mg115.00€2mg162.00€5mg249.00€10mg369.00€25mg562.00€50mg787.00€100mg1,054.00€200mg1,406.00€[D-Phe12]-Bombesin acetate
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.Formula:C76H116N22O20SPurity:99.81%Color and Shape:SolidMolecular weight:1689.94Ref: TM-TP2239L
1mg159.00€5mg349.00€10mg522.00€25mg938.00€50mg1,404.00€100mg2,108.00€200mg3,162.00€500mg4,745.00€Butopamine hydrochloride
CAS:Butopamine hydrochloride is an orally active inotropic compound that is more effective at increasing heart rate compared to Dobutamine.Formula:C18H24ClNO3Color and Shape:SolidMolecular weight:337.84Spantide acetate
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.Formula:C77H112N20O15Purity:98.92%Color and Shape:SolidMolecular weight:1557.84Maprotiline hydrochloride
CAS:Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.Formula:C20H24ClNPurity:99.68% - 99.84%Color and Shape:White PowderMolecular weight:313.864CRF (6-33) acetate(120066-38-8 free base)
CRFBP inhibitor peptide; reduces weight gain, boosts activity in obese rats.Formula:C143H235N41O45SPurity:97.12%Color and Shape:SolidMolecular weight:3280.76Duloxetine hydrochloride
CAS:Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.Formula:C18H20ClNOSPurity:100% - 99.93%Color and Shape:White Or White Crystalline PowderMolecular weight:333.88Ticalopride
CAS:Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formula:C14H20ClN3O3Purity:100%Color and Shape:SolidMolecular weight:313.78Proxyfan
CAS:Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.Formula:C13H16N2OPurity:99.68%Color and Shape:SolidMolecular weight:216.28Solabegron
CAS:Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-ARFormula:C23H23ClN2O3Purity:97.89%Color and Shape:SolidMolecular weight:410.89Ref: TM-T12970
1mg58.00€5mg164.00€10mg259.00€25mg472.00€50mg638.00€100mg848.00€200mg1,121.00€1mL*10mM (DMSO)170.00€Amiselimod hydrochloride
CAS:Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.Formula:C19H31ClF3NO3Purity:99.55%Color and Shape:SolidMolecular weight:413.9Ref: TM-T10305
1mg38.00€2mg49.00€5mg80.00€10mg120.00€25mg215.00€50mg354.00€100mg512.00€200mg738.00€1mL*10mM (DMSO)88.00€
![[D-Phe12]-Bombesin acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP2239L.webp&w=3840&q=75)
