GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor
- Adenosine Receptor
- Adrenergic Receptor
- Bombesin Receptor
- Bradykinin Receptor
- Cannabinoid Receptor
- CaSR
- Cholecystokinin
- CXCR
- Dopamine Receptor
- Endothelin Receptor
- Glucagon Receptor
- GNRH Receptor
- GPCR19
- GRK
- GTPase
- Hedgehog/Smoothened
- Histamine Receptor
- LPA Receptor
- Melatonin Receptor
- Opioid Receptor
- OX Receptor
- PAFR
- PKA
- S1P Receptor
- SGLT
- Sigma receptor
Show 19 more subcategories
Products of "GPCR/G-Protein"
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LY255582
CAS:LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM,Formula:C22H35NO2Purity:98%Color and Shape:SolidMolecular weight:345.52Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formula:C19H25NOSPurity:98.08% - 99.59%Color and Shape:SolidMolecular weight:315.47Ref: TM-T6647
5mg52.00€10mg78.00€25mg145.00€50mg255.00€100mg378.00€200mg552.00€500mg868.00€1mL*10mM (DMSO)55.00€Fasiglifam
CAS:Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.Formula:C29H32O7SPurity:99.61% - 99.82%Color and Shape:SolidMolecular weight:524.63Ref: TM-T2351
1mg49.00€5mg96.00€10mg161.00€25mg284.00€50mg470.00€100mg567.00€200mg820.00€1mL*10mM (DMSO)124.00€PF-4363467
CAS:PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.Formula:C22H30N2O3SColor and Shape:SolidMolecular weight:402.55Uridine-5'-diphosphate disodium salt
CAS:UDP disodium salt is a P2Y6 agonist (EC50 = 13 nM), enhances inflammation, phagocytosis, vasoconstriction, and inhibits P2Y14.Formula:C9H12N2Na2O12P2Purity:100% - 98.86%Color and Shape:White Fine CrystalsMolecular weight:448.12Terazosin hydrochloride
CAS:Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.Formula:C19H26ClN5O4Purity:99.69% - 99.91%Color and Shape:SolidMolecular weight:423.89CAY10526
CAS:CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.Formula:C12H7BrO3SPurity:98.75%Color and Shape:SolidMolecular weight:311.15SB-423562
CAS:SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.Formula:C26H32N2O4Purity:98.64%Color and Shape:SolidMolecular weight:436.54Ref: TM-T12846
1mg39.00€5mg85.00€10mg126.00€25mg221.00€50mg338.00€100mg467.00€200mg640.00€1mL*10mM (DMSO)94.00€CB2R/FAAH modulator-3
CAS:CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.Formula:C22H31NO2Purity:99.02%Color and Shape:SoildMolecular weight:341.49Ref: TM-T67747
2mg38.00€5mg58.00€10mg90.00€25mg164.00€50mg259.00€100mg383.00€200mg545.00€1mL*10mM (DMSO)64.00€Strontium chloride
CAS:Strontium chloride is an agonist of Calcium sensing receptor (CaSR) and directly affects C-type nerve fibers.Formula:Cl2SrPurity:98%Color and Shape:White Solid CrystallineMolecular weight:158.52TD-5471 hydrochloride
CAS:TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (Formula:C32H32ClN3O4Purity:99.57%Color and Shape:SolidMolecular weight:558.07Tiopinac
CAS:Tiopinac: tricyclic with anti-inflammatory, analgesic, antipyretic properties; inhibits prostaglandin synthesis; mild anti-platelet effects in humans.Formula:C16H12O3SPurity:100%Color and Shape:SolidMolecular weight:284.33Gentisein
CAS:Gentisein (NSC-329491), a primary metabolite of Mangiferin, exhibits significant inhibition of serotonin uptake, demonstrating potency with an IC50 value of 4.7Formula:C13H8O5Purity:96.74%Color and Shape:SolidMolecular weight:244.2AR 231453
CAS:Azenosertib (ZN-c3) is an orally active, specific GPR119 agonist. Cost-effective and quality-assured.Formula:C21H24FN7O5SPurity:99.31% - 99.45%Color and Shape:SolidMolecular weight:505.52Cicloprolol hydrochloride
CAS:Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.Formula:C18H30ClNO4Purity:97.26%Color and Shape:SolidMolecular weight:359.89BAR501
CAS:BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。Formula:C26H46O3Purity:99.29% - 99.34%Color and Shape:SolidMolecular weight:406.64Balixafortide
CAS:Balixafortide (POL6326), a potent CXCR4 blocker with IC50 < 10 nM, mobilizes HSPCs and is anti-cancer, 1000x more selective than CXCR7.Formula:C84H118N24O21S2Purity:98%Color and Shape:SolidMolecular weight:1864.14Pro8-Oxytocin TFA
Pro8-Oxytocin TFA, a modified oxytocin (OXT) ligand, exhibits greater potency and efficacy than the standard mammalian OXT ligand, Leu8-Oxytocin, at primateFormula:C42H62N12O12S2·xC2HF3O2Purity:98%Color and Shape:SolidFlupentixol dihydrochloride
CAS:Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.Formula:C23H27Cl2F3N2OSPurity:100% - 99.35%Color and Shape:White Or Off-White SolidMolecular weight:507.43Betaxolol
CAS:Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.Formula:C18H29NO3Purity:99.01%Color and Shape:White Crystalline SolidMolecular weight:307.43
