GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor
- Adenosine Receptor
- Adrenergic Receptor
- Bombesin Receptor
- Bradykinin Receptor
- Cannabinoid Receptor
- CaSR
- Cholecystokinin
- CXCR
- Dopamine Receptor
- Endothelin Receptor
- Glucagon Receptor
- GNRH Receptor
- GPCR19
- GRK
- GTPase
- Hedgehog/Smoothened
- Histamine Receptor
- LPA Receptor
- Melatonin Receptor
- Opioid Receptor
- OX Receptor
- PAFR
- PKA
- S1P Receptor
- SGLT
- Sigma receptor
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Products of "GPCR/G-Protein"
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(Rac)-Norcisapride
CAS:Norcisapride, a 5-HT3 and 5-HT4 agonist, treats GI, orofacial, and ENT disorders.Formula:C14H20ClN3O3Purity:99.13%Color and Shape:SoildMolecular weight:313.78PSB-603
CAS:PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.Formula:C24H25ClN6O4SPurity:97.13%Color and Shape:SolidMolecular weight:529.01Ref: TM-T23203
1mg37.00€5mg97.00€10mg160.00€25mg344.00€50mg562.00€100mg938.00€200mg1,264.00€1mL*10mM (DMSO)111.00€CGP71683 hydrochloride
CAS:CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).Formula:C26H30ClN5O2SPurity:99.92%Color and Shape:SolidMolecular weight:512.07LUF6096
CAS:LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFormula:C22H21Cl2N3OPurity:100%Color and Shape:SolidMolecular weight:414.33PD128907 HCl
CAS:PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.Formula:C14H20ClNO3Purity:98%Color and Shape:SolidMolecular weight:285.77Eloralintide
CAS:Eloralintide (LY 3841136) is an AMYR agonist, anticipated for research in type 2 diabetes and obesity.Formula:C201H319N49O65S2Color and Shape:SolidMolecular weight:4526.1TCS 1102
CAS:TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).Formula:C27H26N4O2SPurity:99.35% - 99.52%Color and Shape:SolidMolecular weight:470.59Empagliflozin
CAS:Empagliflozin (BI 10773) is an SGLT-2 inhibitor (IC50=3.1 nM) that is potent and selective, with more than 300-fold selectivity for SGLT-1/4/5/6.Formula:C23H27ClO7Purity:98% - 99.89%Color and Shape:SolidMolecular weight:450.91Ref: TM-T1766
1g278.00€5mg47.00€10mg60.00€50mg79.00€100mg96.00€200mg144.00€500mg188.00€1mL*10mM (DMSO)50.00€BMS 182874
CAS:BMS 182874: Oral ETA antagonist, IC50=0.150 μM, Ki=0.055 μM, lowers hypertension in rats.Formula:C17H19N3O3SPurity:98.38%Color and Shape:SolidMolecular weight:345.42S 14506 hydrochloride
CAS:S 14506 hydrochloride is a 5-HT1A receptor full agonist.Formula:C24H27ClFN3O2Purity:99.5%Color and Shape:SolidMolecular weight:443.94Capromorelin Tartrate
CAS:Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).Formula:C32H41N5O10Purity:97.69%Color and Shape:SolidMolecular weight:655.7Ref: TM-TQ0022
5mg39.00€10mg64.00€25mg126.00€50mg215.00€100mg319.00€200mg455.00€1mL*10mM (DMSO)52.00€Amezinium methylsulfate
CAS:Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.Formula:C12H15N3O5SPurity:99.64%Color and Shape:SolidMolecular weight:313.335-HT3 antagonist 2
CAS:5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.Formula:C18H21N3OPurity:98%Color and Shape:SolidMolecular weight:295.38SNAP 94847 hydrochloride
CAS:SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)Formula:C29H33ClF2N2O2Purity:100% - 99.85%Color and Shape:SolidMolecular weight:515.03Ref: TM-T8004
2mg42.00€5mg64.00€10mg97.00€25mg187.00€50mg316.00€100mg455.00€200mg635.00€1mL*10mM (DMSO)71.00€AAZ-A 154 hydrobromide
CAS:AAZ-A 154 hydrobromide is a selective, competitive, non-hallucinogenic 5-HT2AR antagonist. It promotes neuronal growth in rodents and yields enduring beneficial behavioral effects.Formula:C14H21BrN2OColor and Shape:SolidMolecular weight:313.23GnRH antagonist 2
CAS:GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.Formula:C28H27F2N9O5Purity:98.08%Color and Shape:SolidMolecular weight:607.57Latozinemab
Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.Purity:> 95%Color and Shape:LiquidMolecular weight:146.28 kDaUridine 5'-diphosphate
CAS:Uridine 5'-diphosphate acts as a P2Y6 receptor agonist, exhibiting an EC50 value of 0.013 μM for the human P2Y6 receptor [1].Formula:C9H14N2O12P2Purity:98%Color and Shape:SolidMolecular weight:404.16Ondansetron hydrochloride dihydrate
CAS:Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.Formula:C18H19N3O·HCl·2H2OPurity:99.92%Color and Shape:White Crystal PowderMolecular weight:365.86Tienoxolol FA
Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.Formula:C22H30N2O7SPurity:97.05% - 99.47%Color and Shape:SoildMolecular weight:466.55
