Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Products of "Opioid Receptor"
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Loperamide hydrochloride
CAS:Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.Formula:C29H34Cl2N2O2Purity:100% - 99.94%Color and Shape:Crystals Practically Insoluble In WaterMolecular weight:513.498AH 8532
CAS:AH 8532 is an opioid compound with analgesic effects and is effective in inhibiting the quinone-induced writhing response in mice, with an oral ED50 of 16 mg/kg.Formula:C16H23ClN2OColor and Shape:SolidMolecular weight:294.82[D-Ala2]leucine-enkephalin
CAS:[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.Formula:C29H39N5O7Purity:98.06%Color and Shape:SolidMolecular weight:569.65Sinomenine hydrochloride
CAS:Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.Formula:C19H24ClNO4Purity:99.43%Color and Shape:SolidMolecular weight:365.851Deltorphin I
CAS:Deltorphin I is an agonist of δ-opioid receptor.Formula:C37H52N8O10Purity:100%Color and Shape:SolidMolecular weight:768.86Gluten Exorphin C
CAS:Gluten exorphin C is an opioid peptide derived from wheat gluten.Formula:C29H45N5O8Purity:100%Color and Shape:SolidMolecular weight:591.7Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).Formula:C50H72N15O15SPurity:100%Color and Shape:SolidMolecular weight:1326.26Ref: TM-T7567L
1mg48.00€5mg125.00€10mg180.00€25mg325.00€50mg467.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)187.00€DAMGO TFA (78123-71-4(Free base))
DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.Formula:C28H36F3N5O8Purity:98.67% - 99.76%Color and Shape:SolidMolecular weight:627.6ML-335
CAS:ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.Formula:C25H32N2O3Purity:98.52%Color and Shape:SolidMolecular weight:408.53Ref: TM-T23002
2mg40.00€5mg62.00€10mg87.00€25mg170.00€50mg264.00€100mg380.00€200mg540.00€1mL*10mM (DMSO)35.00€Trimebutine maleate
CAS:Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.Formula:C26H33NO9Purity:99.76% - 99.88%Color and Shape:White SolidMolecular weight:503.55DPI-3290
CAS:DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potentFormula:C30H34FN3O2Purity:98%Color and Shape:SolidMolecular weight:487.61[Leu5]-Enkephalin
CAS:[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nMFormula:C28H37N5O7Purity:99.87%Color and Shape:SolidMolecular weight:555.62ZT 52656A hydrochloride
CAS:ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.Formula:C19H26ClF3N2OPurity:98.78%Color and Shape:SolidMolecular weight:390.87Salvinorin A
CAS:Salvinorin A is a non-nitrogenous κ-opioid selective agonist.Formula:C23H28O8Purity:99.06%Color and Shape:SolidMolecular weight:432.46Ref: TM-T23306
1mg274.00€5mg663.00€10mg947.00€25mg1,415.00€50mg1,890.00€100mg2,547.00€1mL*10mM (DMSO)735.00€AP-238
CAS:AP-238 is a novel synthetic opioid (NSO) that acts as an agonist for the μ-opioid receptor (MOR), with an EC50 of 248 nM. Additionally, AP-238 exhibits analgesic properties.Formula:C18H26N2OColor and Shape:SolidMolecular weight:286.41AR-M 1000390 hydrochloride
CAS:ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.Formula:C23H29ClN2OPurity:99.68%Color and Shape:SolidMolecular weight:384.94BPR1M97
CAS:BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.Formula:C18H18Cl2N2OPurity:98.13% - 99.15%Color and Shape:SolidMolecular weight:349.25Ref: TM-T10593
1mg96.00€5mg227.00€10mg359.00€25mg660.00€50mg1,035.00€100mg1,454.00€500mg2,822.00€1mL*10mM (DMSO)215.00€DPDPE TFA (88373-73-3 free base)
CAS:DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and is antinociceptive in vivo.Formula:C32H40F3N5O9S2Purity:99.39%Color and Shape:SolidMolecular weight:759.81Nalmefene
CAS:Nalmefene (ORF 11676) is a μ-opioid antagonist and partial κ agonist used in the study of opioid overdose and alcohol dependence.Formula:C21H25NO3Purity:99.86%Color and Shape:SolidMolecular weight:339.43Spinorphin
CAS:Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.Formula:C45H64N8O10Purity:99.68%Color and Shape:SolidMolecular weight:877μ opioid receptor agonist 3
CAS:Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.Formula:C22H28N2O2Purity:98%Color and Shape:SolidMolecular weight:352.47Sinomenine
CAS:Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.Formula:C19H23NO4Purity:99.02% - 99.89%Color and Shape:White PowderMolecular weight:329.39Trimebutine CTB salt
CAS:Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.Formula:C29H36N2O8S2Purity:100% - 99.53%Color and Shape:SolidMolecular weight:604.74Nociceptin
CAS:Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.Formula:C79H129N27O22Purity:99.35%Color and Shape:SolidMolecular weight:1809.04SR17018
CAS:SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.Formula:C19H18Cl3N3OPurity:99.89%Color and Shape:SolidMolecular weight:410.72Meptazinol hydrochloride
CAS:Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.Formula:C15H23NO·HClPurity:99.75%Color and Shape:White SolidMolecular weight:269.81Bisacodyl
CAS:Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.Formula:C22H19NO4Purity:99.45% - 99.78%Color and Shape:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderMolecular weight:361.39Orphine
CAS:Orphine is an opioid compound that can amplify the antinociceptive effects reduced by naloxone in mice.Formula:C20H23N3OColor and Shape:SolidMolecular weight:321.42Adrenorphin
CAS:Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).Formula:C44H69N15O9SPurity:98%Color and Shape:SolidMolecular weight:984.18LY2795050
CAS:LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).Formula:C23H22ClN3O2Purity:97.77%Color and Shape:SolidMolecular weight:407.89Ref: TM-TQ0091
1mg52.00€2mg74.00€5mg116.00€10mg180.00€25mg298.00€50mgTo inquire1mL*10mM (DMSO)127.00€AH 7563
CAS:AH 7563 is structurally classified as an opioid compound with analgesic properties. In mice, its ED50 for pain relief was 15.3 mg/kg when administered orally in the Phenylquinone test, and 15.5 mg/kg when injected subcutaneously in the Hot plate test.Formula:C16H24N2OColor and Shape:SolidMolecular weight:260.38Deltorphin 2
CAS:Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.Formula:C38H54N8O10Purity:100%Color and Shape:SolidMolecular weight:782.88PZM21
CAS:PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).Formula:C19H27N3O2SPurity:99.59%Color and Shape:SolidMolecular weight:361.5Ref: TM-T4386
1mg47.00€2mg60.00€5mg87.00€10mg127.00€25mg205.00€50mg298.00€100mg472.00€1mL*10mM (DMSO)97.00€(-)-Menthol
CAS:(-)-Menthol (Levomenthol) is a levo isomer of menthol, an organic compound obtained from peppermint or mint oils with flavoring and local anesthetic properties.Formula:C10H20OPurity:99.01%Color and Shape:Whitish To White Solid Solid CrystallineMolecular weight:156.2722-Thiocyanatosalvinorin A
CAS:22-Thiocyanatosalvinorin A (RB-64) is a potent selective agonist for the kappa-opioid receptor, exhibiting an EC50 value of 0.077 nM.Formula:C24H27NO8SColor and Shape:SolidMolecular weight:489.54SNC 162
CAS:SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.Formula:C27H37N3OPurity:98%Color and Shape:SolidMolecular weight:419.6MOR agonist-1
CAS:MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associatedFormula:C22H26ClFN2O2Purity:98%Color and Shape:SolidMolecular weight:404.91U-48520
CAS:U-48520 is an agonist of the μ-opioid receptor (μ-opioid receptor) with an EC50 of 1561 nM.Formula:C16H23ClN2OColor and Shape:SolidMolecular weight:294.82Matrine
CAS:Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.Formula:C15H24N2OPurity:100% - 97.16%Color and Shape:SolidMolecular weight:248.36Piperidylthiambutene hydrochloride
CAS:Piperidylthiambutene hydrochloride is an opioid compound that exhibits analgesic effects in animal models.Formula:C17H22ClNS2Color and Shape:SolidMolecular weight:339.95GSK1521498 free base (hydrochloride)
CAS:GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).Formula:C24H21ClF2N4Purity:98%Color and Shape:SolidMolecular weight:438.9GR 89696 fumarate
CAS:GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.Formula:C23H29Cl2N3O7Purity:99.19%Color and Shape:SolidMolecular weight:530.4JTC-801
CAS:JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.Formula:C26H25N3O2·HClPurity:98.91% - 99.27%Color and Shape:SolidMolecular weight:447.96Methylnaltrexone bromide
CAS:Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.Formula:C21H26BrNO4Purity:99.02%Color and Shape:SolidMolecular weight:436.35Dermorphin
CAS:Dermorphin is agonist of μ-opioid receptor (MOR) agonist.Formula:C40H50N8O10Purity:98.82%Color and Shape:SolidMolecular weight:802.87DAMGO
CAS:DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.Formula:C26H35N5O6Purity:98.83% - 99.92%Color and Shape:SolidMolecular weight:513.59Ref: TM-T4351
1mg50.00€2mg60.00€5mg87.00€10mg140.00€25mg283.00€50mg423.00€100mg623.00€1mL*10mM (DMSO)88.00€Aticaprant
CAS:Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.Formula:C26H27FN2O2Purity:99.53% - 99.93%Color and Shape:SolidMolecular weight:418.5Ref: TM-TQ0082
1mg40.00€2mg52.00€5mg88.00€10mg126.00€25mg259.00€50mg406.00€100mg607.00€1mL*10mM (DMSO)87.00€N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formula:C17H17ClN4Purity:97.25%Color and Shape:Yellow Crystalline SolidMolecular weight:312.8Ref: TM-T5158
2mg35.00€5mg50.00€10mg84.00€25mg160.00€50mg248.00€100mg364.00€200mg517.00€1mL*10mM (DMSO)62.00€Valorphin
CAS:Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.Formula:C44H61N9O11Purity:98%Color and Shape:SolidMolecular weight:892.01GR103545
CAS:GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.Formula:C23H29Cl2N3O7Purity:99.75%Color and Shape:SolidMolecular weight:530.4Ref: TM-T9459
1mg87.00€2mg143.00€5mg188.00€10mg283.00€25mg509.00€50mg727.00€100mg1,017.00€1mL*10mM (DMSO)250.00€DPDPE
CAS:DPDPE is selective δ-opioid receptor agonist peptide.Formula:C30H39N5O7S2Purity:98%Color and Shape:SolidMolecular weight:645.79Corynantheidine
CAS:Corynantheidine ((-)-Corynantheidine) is a partial agonist of the mu opioid receptor (MOR) and demonstrates MOR-dependent analgesic effects in mice.Formula:C22H28N2O3Color and Shape:SolidMolecular weight:368.47N-Phenethylnoroxymorphone
CAS:N-Phenethylnoroxymorphone is an opioid compound that can enhance morphine-induced analgesia in rats. It is used in the research of neurological disorders.Formula:C24H25NO4Color and Shape:SolidMolecular weight:391.46MCOPPB triHydrochloride
CAS:MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.Formula:C26H43Cl3N4Purity:99.89% - 99.91%Color and Shape:SolidMolecular weight:518.01Ref: TM-T2071
2mg34.00€5mg50.00€10mg87.00€25mg163.00€50mg255.00€100mg375.00€200mg535.00€1mL*10mM (DMSO)58.00€Naltrexone hydrochloride
CAS:Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.Formula:C20H24ClNO4Purity:100% - 99%Color and Shape:White Crystalline PowderMolecular weight:377.862ADL-5747
CAS:ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletalFormula:C24H28N2O3Purity:100% - 99.44%Color and Shape:SolidMolecular weight:392.49Trimebutine
CAS:Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioidFormula:C22H29NO5Purity:98.13% - 99.49%Color and Shape:SolidMolecular weight:387.47BTRX-335140
CAS:BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.Formula:C25H32FN5O2Purity:98% - 99.89%Color and Shape:SolidMolecular weight:453.55Ref: TM-T14835
1mg105.00€2mg155.00€5mg250.00€10mg406.00€25mg840.00€50mg1,378.00€100mg1,882.00€200mg2,632.00€1mL*10mM (DMSO)283.00€Nociceptin (1-13), amide
CAS:Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrainFormula:C61H100N22O15Purity:98%Color and Shape:SolidMolecular weight:1381.59BW-180C
CAS:BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.Formula:C29H39N5O7Purity:100%Color and Shape:SolidMolecular weight:569.65Ref: TM-TP1905
1mg47.00€2mg62.00€5mg89.00€10mg139.00€25mg254.00€50mg400.00€100mg595.00€1mL*10mM (DMSO)111.00€BMS-986122
CAS:BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1Formula:C16H15BrClNO3S2Purity:98.42%Color and Shape:SolidMolecular weight:448.78Ref: TM-T26869
1mg48.00€5mg96.00€10mg160.00€25mg344.00€50mg550.00€100mg787.00€500mg1,568.00€1mL*10mM (DMSO)96.00€Endomorphin 2
CAS:EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.Formula:C32H37N5O5Purity:99.64%Color and Shape:SolidMolecular weight:571.67MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Formula:C37H47Cl2N5O3Purity:98%Color and Shape:SolidMolecular weight:680.71Asimadoline
CAS:Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.Formula:C27H30N2O2Color and Shape:SolidMolecular weight:414.54Urotensin-II receptor antagonist-1
CAS:Urotensin-II receptor antagonist-1 (compound 1) is a human Urotensin II receptor antagonist with low oral bioavailability (F=0-3% in rats) and a Ki of 16 nM in HEK293 cells expressing human recombinant UT receptors. It inhibits cytochrome P450 enzymes (IC50=0.75 μM for CYP2D6; 1.4 μM for CYP3A4), suppresses κ opioid receptors (EC50=3.2 μM), and targets cardiac sodium channels (Ki=2.5 μM).Formula:C25H31Cl2N3OColor and Shape:SolidMolecular weight:460.439ICI 204,448
CAS:ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.Formula:C23H27Cl3N2O4Purity:100%Color and Shape:SolidMolecular weight:501.83Opioid receptor agonist 1
Opioid receptor agonist1 (Compound 2638-28) is an orally active opioid receptor agonist that shows strong affinity for MOR, DOR, and KOR, with Ki values of 5, 24, and 212 nM, respectively. It exhibits analgesic activity in both the mouse warm water tail-flick model and the acetic acid writhing model.Formula:C32H45N5OMolecular weight:515.73LY255582
CAS:LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM,Formula:C22H35NO2Purity:98%Color and Shape:SolidMolecular weight:345.526'-GNTI dihydrochloride
CAS:6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over recruitment of β-aspirin 2.Formula:C27H29N5O3·2ClHPurity:99.08%Color and Shape:SolidMolecular weight:544.47IPAG
CAS:IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.Formula:C17H22IN3Purity:98.8%Color and Shape:SolidMolecular weight:395.28SNC 80
CAS:SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.Formula:C28H39N3O2Purity:98.67%Color and Shape:SolidMolecular weight:449.63Anilopam
CAS:Anilopam is an opioid analgesic belonging to the benzazepine class and acts as an agonist at opioid receptors.Formula:C20H26N2OColor and Shape:SolidMolecular weight:310.43Cebranopadol
CAS:Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP)Formula:C24H27FN2OPurity:99.61% - 99.78%Color and Shape:SolidMolecular weight:378.48Ref: TM-T5167
2mg40.00€5mg60.00€10mg87.00€25mg170.00€50mg274.00€100mg406.00€200mg592.00€1mL*10mM (DMSO)66.00€KOR agonist 3
KOR agonist 3 (Compound 5) is an agonist of the κ opioid receptor (κOR) with an EC50 of 0.88 nM. It also exhibits some activation of μOR, with an EC50 of 720 nM. However, KOR agonist 3 does not activate δOR at concentrations below 1 μM. Its ability to recruit β-Arrestin-2 is lower than that of U50488.Formula:C24H24N2O3Color and Shape:SolidMolecular weight:388.46LY2444296
CAS:LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).Formula:C24H22F2N2O2Purity:98.03%Color and Shape:SolidMolecular weight:408.44AH 8529
CAS:AH 8529 is an orally active opioid compound with analgesic properties.Formula:C16H23ClN2OColor and Shape:SolidMolecular weight:294.82Samidorphan HCl
CAS:Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ-opioid, κ-opioid, and delta-opioid receptors.Formula:C21H27ClN2O4Purity:98.25% - 99.60%Color and Shape:SoildMolecular weight:406.9DuP 747 HCl
CAS:DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two conformations.Formula:C24H29Cl3N2O2Purity:99.81%Color and Shape:SoildMolecular weight:483.86NNC 63-0532
CAS:NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.Formula:C27H29N3O3Purity:98.75%Color and Shape:SolidMolecular weight:443.54Apitegromab
CAS:Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases includingPurity:95%Color and Shape:Liquid(-)-9-Hydroxycorynantheidine
CAS:(-)-9-Hydroxycorynantheidine (9-O-Desmethyl mitragynine) is a demethylated analog of Mitragynine, functioning as a selective and partial agonist for the μ-opioid receptor (μ-opioid receptor). This compound inhibits electrically stimulated twitch contractions in the guinea pig ileum.Formula:C22H28N2O4Color and Shape:SolidMolecular weight:384.47EST73502 HCl
CAS:EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.Formula:C19H27ClF2N2O2Purity:97.66%Color and Shape:SolidMolecular weight:388.88Ref: TM-T39284
1mg92.00€5mg180.00€10mg258.00€25mg424.00€50mg598.00€100mg792.00€200mg1,074.00€1mL*10mM (DMSO)197.00€DBPR116
CAS:DBPR116 is a prodrug of BPRMU191 that can penetrate the blood-brain barrier. It significantly enhances the delivery efficiency of drugs targeting the central nervous system. When combined with the antagonist Naltrexone, DBPR116 demonstrates superior safety and analgesic effects compared to morphine in various in vivo pharmacological studies, including thermal pain models, cancer pain models, constipation, sedation, psychological dependence, heart rate, and respiratory frequency. As a strategy for peripheral administration, DBPR116 effectively alleviates pain while reducing adverse effects, showing promise as a safer opioid analgesic.Formula:C19H18FNO3SColor and Shape:SolidMolecular weight:359.42CP-866087
CAS:CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.Formula:C24H28N2O2Purity:100% - 99.44%Color and Shape:SoildMolecular weight:376.49(R,S)-Ivosidenib
CAS:(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .Formula:C28H22ClF3N6O3Color and Shape:SolidMolecular weight:582.96Propiram fumarate HCl
CAS:Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.Formula:C16H25N3O·xClHPurity:99.25%Color and Shape:SoildBMS986187
CAS:BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.Formula:C31H34O4Purity:99.09%Color and Shape:SolidMolecular weight:470.6KOR agonist 5
KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).Formula:C38H38N2O5Color and Shape:SolidMolecular weight:602.72Tyr-Gly-Gly-Phe-Met-OH
CAS:Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.Formula:C27H35N5O7SPurity:≥95%Color and Shape:White Lyophilised SolidMolecular weight:573.66SCH 221510
CAS:SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.Formula:C28H31NOPurity:99.10%Color and Shape:SolidMolecular weight:397.55GSK1521498
CAS:GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).Formula:C24H23F2N4O4PPurity:98%Color and Shape:SolidMolecular weight:500.43Opioid receptor modulator 1
CAS:Opioid receptor modulator 1 is a modulator of opioid receptor.Formula:C18H23NO2Purity:98%Color and Shape:SolidMolecular weight:285.38BAN ORL 24 dihydrochloride
CAS:BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that can be used to study neurological diseases.Formula:C27H37Cl2N3O2Purity:95.03%Color and Shape:SolidMolecular weight:506.51R-6890
CAS:R-6890 is an opioid compound with analgesic properties.Formula:C21H24ClN3OColor and Shape:SolidMolecular weight:369.89ADL-5859
CAS:ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for theFormula:C24H28N2O3·HClPurity:98.78% - 99.11%Color and Shape:SolidMolecular weight:428.95Ref: TM-T6175
1mg52.00€2mg70.00€5mg96.00€10mg170.00€25mg338.00€50mg520.00€100mg748.00€500mg1,549.00€1mL*10mM (DMSO)114.00€Dermorphin TFA
CAS:Dermorphin TFA is a new class of opioids-like peptidesFormula:C42H51F3N8O12Purity:100% - 98%Color and Shape:SolidMolecular weight:916.89Mu opioid receptor antagonist 7
CAS:Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (Formula:C22H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:386.914-Hydroxy-1-(2-phenylethyl)piperidine
CAS:4-Hydroxy-1-(2-phenylethyl)piperidine is a synthetic ligand for muscarinic acetylcholine receptors (mAChR) or non-opioid intracellular sigma-1 receptors (σ1 receptors). It serves as a metabolite of the opioid compounds furanylfentanyl and 4-fluoroisobutyryl fentanyl (FIBF).Formula:C13H19NOColor and Shape:SolidMolecular weight:205.3ICI 199,441 hydrochloride
CAS:ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.Formula:C21H25Cl3N2OPurity:99.46%Color and Shape:SolidMolecular weight:427.8Ref: TM-T22849
2mg34.00€5mg50.00€10mg80.00€25mg145.00€50mg226.00€100mg331.00€200mg465.00€1mL*10mM (DMSO)62.00€
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