Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Products of "Opioid Receptor"
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Loperamide hydrochloride
CAS:Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.Formula:C29H34Cl2N2O2Purity:100% - 99.94%Color and Shape:Crystals Practically Insoluble In WaterMolecular weight:513.498AH 8532
CAS:AH 8532 is an opioid compound with analgesic effects and is effective in inhibiting the quinone-induced writhing response in mice, with an oral ED50 of 16 mg/kg.Formula:C16H23ClN2OColor and Shape:SolidMolecular weight:294.82[D-Ala2]leucine-enkephalin
CAS:[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.Formula:C29H39N5O7Purity:98.06%Color and Shape:SolidMolecular weight:569.65Sinomenine hydrochloride
CAS:Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.Formula:C19H24ClNO4Purity:99.43%Color and Shape:SolidMolecular weight:365.851Deltorphin I
CAS:Deltorphin I is an agonist of δ-opioid receptor.Formula:C37H52N8O10Purity:100%Color and Shape:SolidMolecular weight:768.86Gluten Exorphin C
CAS:Gluten exorphin C is an opioid peptide derived from wheat gluten.Formula:C29H45N5O8Purity:100%Color and Shape:SolidMolecular weight:591.7Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).Formula:C50H72N15O15SPurity:100%Color and Shape:SolidMolecular weight:1326.26Ref: TM-T7567L
1mg48.00€5mg125.00€10mg180.00€25mg325.00€50mg467.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)187.00€DAMGO TFA (78123-71-4(Free base))
DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.Formula:C28H36F3N5O8Purity:98.67% - 99.76%Color and Shape:SolidMolecular weight:627.6ML-335
CAS:ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.Formula:C25H32N2O3Purity:98.52%Color and Shape:SolidMolecular weight:408.53Ref: TM-T23002
2mg40.00€5mg62.00€10mg87.00€25mg170.00€50mg264.00€100mg380.00€200mg540.00€1mL*10mM (DMSO)35.00€Trimebutine maleate
CAS:Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.Formula:C26H33NO9Purity:99.76% - 99.88%Color and Shape:White SolidMolecular weight:503.55DPI-3290
CAS:DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potentFormula:C30H34FN3O2Purity:98%Color and Shape:SolidMolecular weight:487.61[Leu5]-Enkephalin
CAS:[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nMFormula:C28H37N5O7Purity:99.87%Color and Shape:SolidMolecular weight:555.62ZT 52656A hydrochloride
CAS:ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.Formula:C19H26ClF3N2OPurity:98.78%Color and Shape:SolidMolecular weight:390.87Salvinorin A
CAS:Salvinorin A is a non-nitrogenous κ-opioid selective agonist.Formula:C23H28O8Purity:99.06%Color and Shape:SolidMolecular weight:432.46Ref: TM-T23306
1mg274.00€5mg663.00€10mg947.00€25mg1,415.00€50mg1,890.00€100mg2,547.00€1mL*10mM (DMSO)735.00€AP-238
CAS:AP-238 is a novel synthetic opioid (NSO) that acts as an agonist for the μ-opioid receptor (MOR), with an EC50 of 248 nM. Additionally, AP-238 exhibits analgesic properties.Formula:C18H26N2OColor and Shape:SolidMolecular weight:286.41AR-M 1000390 hydrochloride
CAS:ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.Formula:C23H29ClN2OPurity:99.68%Color and Shape:SolidMolecular weight:384.94BPR1M97
CAS:BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.Formula:C18H18Cl2N2OPurity:98.13% - 99.15%Color and Shape:SolidMolecular weight:349.25Ref: TM-T10593
1mg96.00€5mg227.00€10mg359.00€25mg660.00€50mg1,035.00€100mg1,454.00€500mg2,822.00€1mL*10mM (DMSO)215.00€DPDPE TFA (88373-73-3 free base)
CAS:DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and is antinociceptive in vivo.Formula:C32H40F3N5O9S2Purity:99.39%Color and Shape:SolidMolecular weight:759.81Nalmefene
CAS:Nalmefene (ORF 11676) is a μ-opioid antagonist and partial κ agonist used in the study of opioid overdose and alcohol dependence.Formula:C21H25NO3Purity:99.86%Color and Shape:SolidMolecular weight:339.43Spinorphin
CAS:Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.Formula:C45H64N8O10Purity:99.68%Color and Shape:SolidMolecular weight:877μ opioid receptor agonist 3
CAS:Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.Formula:C22H28N2O2Purity:98%Color and Shape:SolidMolecular weight:352.47Sinomenine
CAS:Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.Formula:C19H23NO4Purity:99.02% - 99.89%Color and Shape:White PowderMolecular weight:329.39Trimebutine CTB salt
CAS:Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.Formula:C29H36N2O8S2Purity:100% - 99.53%Color and Shape:SolidMolecular weight:604.74Nociceptin
CAS:Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.Formula:C79H129N27O22Purity:99.35%Color and Shape:SolidMolecular weight:1809.04SR17018
CAS:SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.Formula:C19H18Cl3N3OPurity:99.89%Color and Shape:SolidMolecular weight:410.72Meptazinol hydrochloride
CAS:Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.Formula:C15H23NO·HClPurity:99.75%Color and Shape:White SolidMolecular weight:269.81Bisacodyl
CAS:Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.Formula:C22H19NO4Purity:99.45% - 99.78%Color and Shape:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderMolecular weight:361.39Orphine
CAS:Orphine is an opioid compound that can amplify the antinociceptive effects reduced by naloxone in mice.Formula:C20H23N3OColor and Shape:SolidMolecular weight:321.42Adrenorphin
CAS:Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).Formula:C44H69N15O9SPurity:98%Color and Shape:SolidMolecular weight:984.18LY2795050
CAS:LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).Formula:C23H22ClN3O2Purity:97.77%Color and Shape:SolidMolecular weight:407.89Ref: TM-TQ0091
1mg52.00€2mg74.00€5mg116.00€10mg180.00€25mg298.00€50mgTo inquire1mL*10mM (DMSO)127.00€AH 7563
CAS:AH 7563 is structurally classified as an opioid compound with analgesic properties. In mice, its ED50 for pain relief was 15.3 mg/kg when administered orally in the Phenylquinone test, and 15.5 mg/kg when injected subcutaneously in the Hot plate test.Formula:C16H24N2OColor and Shape:SolidMolecular weight:260.38Deltorphin 2
CAS:Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.Formula:C38H54N8O10Purity:100%Color and Shape:SolidMolecular weight:782.88PZM21
CAS:PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).Formula:C19H27N3O2SPurity:99.59%Color and Shape:SolidMolecular weight:361.5Ref: TM-T4386
1mg47.00€2mg60.00€5mg87.00€10mg127.00€25mg205.00€50mg298.00€100mg472.00€1mL*10mM (DMSO)97.00€(-)-Menthol
CAS:(-)-Menthol (Levomenthol) is a levo isomer of menthol, an organic compound obtained from peppermint or mint oils with flavoring and local anesthetic properties.Formula:C10H20OPurity:99.01%Color and Shape:Whitish To White Solid Solid CrystallineMolecular weight:156.2722-Thiocyanatosalvinorin A
CAS:22-Thiocyanatosalvinorin A (RB-64) is a potent selective agonist for the kappa-opioid receptor, exhibiting an EC50 value of 0.077 nM.Formula:C24H27NO8SColor and Shape:SolidMolecular weight:489.54SNC 162
CAS:SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.Formula:C27H37N3OPurity:98%Color and Shape:SolidMolecular weight:419.6MOR agonist-1
CAS:MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associatedFormula:C22H26ClFN2O2Purity:98%Color and Shape:SolidMolecular weight:404.91U-48520
CAS:U-48520 is an agonist of the μ-opioid receptor (μ-opioid receptor) with an EC50 of 1561 nM.Formula:C16H23ClN2OColor and Shape:SolidMolecular weight:294.82Matrine
CAS:Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.Formula:C15H24N2OPurity:100% - 97.16%Color and Shape:SolidMolecular weight:248.36Piperidylthiambutene hydrochloride
CAS:Piperidylthiambutene hydrochloride is an opioid compound that exhibits analgesic effects in animal models.Formula:C17H22ClNS2Color and Shape:SolidMolecular weight:339.95GSK1521498 free base (hydrochloride)
CAS:GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).Formula:C24H21ClF2N4Purity:98%Color and Shape:SolidMolecular weight:438.9GR 89696 fumarate
CAS:GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.Formula:C23H29Cl2N3O7Purity:99.19%Color and Shape:SolidMolecular weight:530.4JTC-801
CAS:JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.Formula:C26H25N3O2·HClPurity:98.91% - 99.27%Color and Shape:SolidMolecular weight:447.96Methylnaltrexone bromide
CAS:Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.Formula:C21H26BrNO4Purity:99.02%Color and Shape:SolidMolecular weight:436.35Dermorphin
CAS:Dermorphin is agonist of μ-opioid receptor (MOR) agonist.Formula:C40H50N8O10Purity:98.82%Color and Shape:SolidMolecular weight:802.87DAMGO
CAS:DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.Formula:C26H35N5O6Purity:98.83% - 99.92%Color and Shape:SolidMolecular weight:513.59Ref: TM-T4351
1mg50.00€2mg60.00€5mg87.00€10mg140.00€25mg283.00€50mg423.00€100mg623.00€1mL*10mM (DMSO)88.00€Aticaprant
CAS:Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.Formula:C26H27FN2O2Purity:99.53% - 99.93%Color and Shape:SolidMolecular weight:418.5Ref: TM-TQ0082
1mg40.00€2mg52.00€5mg88.00€10mg126.00€25mg259.00€50mg406.00€100mg607.00€1mL*10mM (DMSO)87.00€N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formula:C17H17ClN4Purity:97.25%Color and Shape:Yellow Crystalline SolidMolecular weight:312.8Ref: TM-T5158
2mg35.00€5mg50.00€10mg84.00€25mg160.00€50mg248.00€100mg364.00€200mg517.00€1mL*10mM (DMSO)62.00€Valorphin
CAS:Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.Formula:C44H61N9O11Purity:98%Color and Shape:SolidMolecular weight:892.01
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