Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Products of "Adenosine Receptor"
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KI-7
CAS:KI-7 is an adenosine A2B receptor positive allosteric modulator.Formula:C23H18N2O2Purity:98.03%Color and Shape:SolidMolecular weight:354.4Ref: TM-T9238
2mg38.00€5mg58.00€10mg90.00€25mg182.00€50mg279.00€100mg420.00€200mg592.00€1mL*10mM (DMSO)65.00€Acefylline
CAS:Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.Formula:C9H10N4O4Purity:99.57%Color and Shape:White Crystalline SolidMolecular weight:238.2YGZ-331
CAS:YGZ-331, a sedative hypnotic, acts by elevating GABA levels as a derivative of the adenosine nucleoside NGBA. It functions through activating A1R and A2aR, and inhibiting the phosphorylation of CaMKII (pCaMKII), thereby exerting its calming effects. Additionally, YGZ-331 reduces spontaneous motor activity in mice.Formula:C19H23N5O4Color and Shape:SolidMolecular weight:385.42MRS1220
CAS:MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeuticFormula:C21H14ClN5O2Purity:96.59%Color and Shape:SolidMolecular weight:403.82LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Formula:C18H14FN5OPurity:100% - 99.03%Color and Shape:SolidMolecular weight:335.34Swertisin
CAS:Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.Formula:C22H22O10Purity:99.74% - 99.79%Color and Shape:SolidMolecular weight:446.4SCH 58261
CAS:SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Formula:C18H15N7OPurity:99.07% - 99.75%Color and Shape:SolidMolecular weight:345.36Ref: TM-T6979
1mg40.00€2mg51.00€5mg85.00€10mg125.00€25mg225.00€50mg364.00€100mg582.00€1mL*10mM (DMSO)86.00€Diphylline
CAS:Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.Formula:C10H14N4O4Purity:98.54%Color and Shape:Crystals From Alcohol SolidMolecular weight:254.24MRS 1754
CAS:MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.Formula:C26H26N6O4Purity:96.12% - 97.48%Color and Shape:SolidMolecular weight:486.52A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effectiveFormula:C28H34N6O6Purity:98%Color and Shape:SolidMolecular weight:550.61Taminadenant
CAS:Taminadenant is an adenosine receptor antagonist.Formula:C10H8BrN7Purity:99.11%Color and Shape:SolidMolecular weight:306.12Ref: TM-T16980
5mg51.00€10mg88.00€25mg127.00€50mg170.00€100mg250.00€200mg374.00€1mL*10mM (DMSO)57.00€BAY 60-6583
CAS:BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3Formula:C19H17N5O2SPurity:100% - 98.87%Color and Shape:SolidMolecular weight:379.44Ref: TM-T14506
1mg44.00€5mg92.00€10mg123.00€25mg245.00€50mg418.00€100mg627.00€200mg877.00€1mL*10mM (DMSO)106.00€Rolofylline
CAS:Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Formula:C20H28N4O2Purity:99.53%Color and Shape:SolidMolecular weight:356.46VPC171
CAS:VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Formula:C18H12F3NOSPurity:99.52%Color and Shape:SolidMolecular weight:347.35Ref: TM-T29112
1mg73.00€2mg96.00€5mg131.00€10mg182.00€25mg335.00€50mg467.00€100mg662.00€200mg892.00€1mL*10mM (DMSO)134.00€
