GPR
Los receptores acoplados a proteínas G (GPRs) son una gran familia de receptores de superficie celular que desempeñan un papel crucial en la transmisión de señales de hormonas, neurotransmisores y otros ligandos extracelulares hacia el interior de la célula. Los GPRs están involucrados en una amplia gama de procesos fisiológicos, incluyendo la regulación hormonal, la respuesta inmune y la percepción sensorial. Modificar la actividad de los GPR es una estrategia clave en el desarrollo de terapias para diversas enfermedades, incluyendo trastornos endocrinos, enfermedades cardiovasculares y condiciones neurológicas. En CymitQuimica, ofrecemos una selección de moduladores de GPR de alta calidad para apoyar su investigación en señalización celular, endocrinología y descubrimiento de fármacos.
Productos de "GPR"
Ordenar por
TUG-469
CAS:TUG-469 is an agonist of free fatty acid 1(FFA) receptor.Fórmula:C23H23NO2Pureza:100%Forma y color:SolidPeso molecular:345.43CRTh2 antagonist 2
CAS:CRTh2 antagonist 2 is a selective and potent CRTH2 antagonist, IC50≤10 nM. CRTh2 antagonist 2 can be used to study the direction of androgenic alopecia.Fórmula:C26H23ClN4O3Pureza:99.53%Forma y color:SolidPeso molecular:474.94Ref: TM-T10889
1mg71,00€5mg128,00€10mg200,00€25mg320,00€50mg437,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)170,00€JNJ-63533054
CAS:JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.Fórmula:C17H17ClN2O2Pureza:98.38% - 99.87%Forma y color:SolidPeso molecular:316.78Ref: TM-T3119
1mg35,00€5mg66,00€10mg89,00€25mg185,00€50mg329,00€100mg487,00€500mg1.026,00€1mL*10mM (DMSO)74,00€4-CMTB
CAS:4-CMTB is a selective agonist of FFA2 and GPR43.It also is a positive allosteric modulator (pEC50=6.38).Fórmula:C14H15ClN2OSPureza:99.59%Forma y color:SolidPeso molecular:294.8Ref: TM-T8642
1mg48,00€2mg65,00€5mg96,00€10mg138,00€25mg230,00€50mg341,00€100mg507,00€1mL*10mM (DMSO)92,00€GPR120 Agonist 3
CAS:GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62).Fórmula:C19H23ClF3NO3Pureza:99.29%Forma y color:SolidPeso molecular:405.84Ref: TM-T15413
1mg37,00€5mg88,00€10mg144,00€25mg274,00€50mg393,00€100mg588,00€200mg833,00€1mL*10mM (DMSO)87,00€ML 145
CAS:ML 145 is a selective antagonist of GPR35/CXCR8 (IC50/EC50 of 20.1 nM)Fórmula:C24H22N2O5S2Pureza:97.74%Forma y color:SolidPeso molecular:482.57Ref: TM-T12074
1mg52,00€5mg111,00€10mg178,00€25mg350,00€50mg522,00€100mg750,00€200mg1.075,00€1mL*10mM (DMSO)120,00€PW0787
CAS:PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).Fórmula:C23H20F4N4O2Pureza:98.42%Forma y color:SolidPeso molecular:460.42Ref: TM-T9452
1mg37,00€5mg80,00€10mg117,00€25mg235,00€50mg353,00€100mg500,00€200mg690,00€1mL*10mM (DMSO)96,00€LP-471756
CAS:LP-471756 is a specific antagonist of GPR139 and inhibits LP-360924-stimulated cAMP production (IC50 = 640 nM).Fórmula:C19H23NO2SPureza:99.59%Forma y color:SolidPeso molecular:329.46Ref: TM-T27850
5mg48,00€10mg71,00€25mg135,00€50mg212,00€100mg340,00€200mg480,00€1mL*10mM (DMSO)49,00€Fasiglifam
CAS:Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.Fórmula:C29H32O7SPureza:99.61% - 99.82%Forma y color:SolidPeso molecular:524.63Ref: TM-T2351
1mg49,00€5mg96,00€10mg161,00€25mg284,00€50mg470,00€100mg567,00€200mg820,00€1mL*10mM (DMSO)124,00€AR 231453
CAS:Azenosertib (ZN-c3) is an orally active, specific GPR119 agonist. Cost-effective and quality-assured.Fórmula:C21H24FN7O5SPureza:99.31% - 99.45%Forma y color:SolidPeso molecular:505.52RTI-13951-33
CAS:RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional assay).Fórmula:C28H33N3O3Pureza:98%Forma y color:SolidPeso molecular:459.58AMG 837 calcium hydrate
CAS:AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM.Fórmula:C52H44CaF6O8Pureza:98.07%Forma y color:SolidPeso molecular:950.97Ref: TM-TQ0020
2mg37,00€5mg52,00€10mg80,00€25mg150,00€50mg284,00€100mg415,00€200mg665,00€1mL*10mM (DMSO)58,00€GPR35 agonist 3
CAS:GPR35 agonist 3 is a synthetic GPR35 agonist used in the study of cancer, type 2 diabetes and cardiovascular disease.Fórmula:C12H9NO5SPureza:98.79%Forma y color:SolidPeso molecular:279.27CID 2745687
CAS:CID 2745687 blocks human GPR35, countering cromolyn disodium & zaprinast effects.Fórmula:C17H19F2N5O2SPureza:99.11%Forma y color:SolidPeso molecular:395.43Ref: TM-T21874
1mg40,00€2mg52,00€5mg88,00€10mg126,00€25mg274,00€50mg432,00€100mg638,00€1mL*10mM (DMSO)87,00€AMG 837
CAS:Prinaberel (ERB 041) is an ERβ agonist with anticancer activity and anti-inflammatory activity that inhibits the NFκB pro-inflammatory signaling pathway.Fórmula:C26H21F3O3Pureza:98%Forma y color:SolidPeso molecular:438.44YE 120
CAS:YE 120 is a GPR35 agonist.Fórmula:C16H9Cl2N3OPureza:99.67%Forma y color:SolidPeso molecular:330.17GPR120 Agonist 2
CAS:GPR120 Agonist 2 is a potent and selective GPR120 receptor agonist.Fórmula:C22H25ClO4Pureza:98.64% - 99.52%Forma y color:SolidPeso molecular:388.88Ref: TM-T4312
1mg38,00€5mg101,00€10mg145,00€25mg235,00€50mg338,00€100mg455,00€200mg625,00€1mL*10mM (DMSO)101,00€CID1231538
CAS:CID1231538 is a potent GPR35 antagonist.Fórmula:C26H22ClN3O3S2Pureza:98.79%Forma y color:SolidPeso molecular:524.052-(pentylsulfanyl)pyrimidine-4,6-diol
CAS:2-(pentylsulfanyl)pyrimidine-4,6-diol 是一种新型 GRP84 激动剂。Fórmula:C9H14N2O2SPureza:97.58%Forma y color:SolidPeso molecular:214.28Palosuran
CAS:Palosuran (ACT-058362) (ACT-058362) is a new potent and specific antagonist of the human UT receptor.Fórmula:C25H30N4O2Pureza:98.46%Forma y color:SolidPeso molecular:418.53Ref: TM-T2058
2mg47,00€5mg74,00€10mg107,00€25mg235,00€50mg393,00€100mg645,00€200mg898,00€1mL*10mM (DMSO)202,00€
