Receptor de andrógenos
El receptor de andrógenos (AR) es un receptor hormonal nuclear que se activa al unirse a andrógenos, como la testosterona y la dihidrotestosterona. Este receptor juega un papel crucial en el desarrollo y mantenimiento de las características masculinas, así como en la regulación de varios procesos fisiológicos, incluyendo el crecimiento muscular, la libido y la densidad ósea. Los inhibidores del receptor de andrógenos son ampliamente estudiados en el contexto del cáncer de próstata, donde la señalización del AR a menudo está sobreexpresada. En CymitQuimica, ofrecemos una gama de moduladores del receptor de andrógenos de alta calidad para apoyar su investigación en endocrinología, biología del cáncer y regulación hormonal.
Productos de "Receptor de andrógenos"
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Darolutamide
CAS:Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).Fórmula:C19H19ClN6O2Pureza:97.36% - 99.62%Forma y color:SolidPeso molecular:398.85Ref: TM-T6915
1mg49,00€2mg70,00€5mg105,00€10mg166,00€25mg265,00€50mg378,00€100mg560,00€500mg1.216,00€1mL*10mM (DMSO)106,00€UT-155
CAS:UT-155 is a selective and potent antagonist of the androgen receptor (AR) (Ki: 267 nM for UT-155 binding to AR-LBD).Fórmula:C20H15F4N3O2Pureza:98.94%Forma y color:SolidPeso molecular:405.35Ref: TM-T13272
1mg62,00€5mg135,00€10mg207,00€25mg333,00€50mg452,00€100mg645,00€200mg872,00€1mL*10mM (DMSO)149,00€MK-0773 FA
MK-0773 FA (MK-0773 FA (606101-58-0 Free base)) is an androgen receptor modulator used for the prevention and treatment of cancer-related muscle wasting.Fórmula:C28H36FN5O4Pureza:99.17%Forma y color:SoildPeso molecular:525.61Nandrolone decanoate
CAS:Nandrolone decanoate is an anabolic steroid similar to testosterone, stimulating muscle, bone growth, and red blood cell production.Fórmula:C28H44O3Pureza:98.43% - 99.03%Forma y color:SolidPeso molecular:428.65Luxdegalutamide
CAS:Luxdegalutamide (ARV-766) is an orally available and effective protein degrader of protein hydrolysis-targeted chimeras (PROTAC).Luxdegalutamide degrades theFórmula:C45H54FN7O6Pureza:100%Forma y color:SolidPeso molecular:807.95Androgen receptor degrader-3
CAS:Androgen Receptor Degrader-3 (ARD-3) is a compound that inhibits androgen receptor signaling and promotes the degradation of the receptor, with potentialFórmula:C45H51ClN8O5Pureza:98%Forma y color:SolidPeso molecular:819.39Celiprolol hydrochloride
CAS:Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.Fórmula:C20H33N3O4·HClForma y color:White Crystalline SolidPeso molecular:415.96Anticancer agent 135
Anticancer agent 135 (compound 26h) acts as a potent androgen receptor (AR) antagonist, effectively blocking AR nuclear translocation and inhibiting AR/AR-V7Fórmula:C23H21F3N4OSPureza:98%Forma y color:SolidPeso molecular:458.5AS-601811
CAS:AS-601811 is a bio-active chemical.Fórmula:C15H17NOPureza:98.05% - 99.49%Forma y color:SolidPeso molecular:227.3Androgen receptor degrader-1
CAS:Androgen Receptor Degrader-1 (Compound 18) is a potent agent for androgen receptor degradation, applicable in cancer research [1].Fórmula:C15H14ClN3O4Pureza:98%Forma y color:SolidPeso molecular:335.74AZD3514
CAS:AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.Phase 1.Fórmula:C25H32F3N7O2Pureza:96.6%Forma y color:SolidPeso molecular:519.56Ralaniten triacetate
CAS:Ralaniten triacetate (EPI-506) is a precursor of Ralaniten, an AR-NTD inhibitor, which can be used in the study of prostate and breast cancer.Fórmula:C27H33ClO8Pureza:99.37%Forma y color:SolidPeso molecular:521.00Ref: TM-T36375
1mg162,00€5mg393,00€10mg655,00€25mg1.415,00€50mg1.882,00€100mg2.375,00€1mL*10mM (DMSO)449,00€Anti-Androgen receptor Antibody (8H883)
Anti-Androgen receptor Antibody (8H883) is an antibody targeting Androgen receptor. Anti-Androgen receptor Antibody (8H883) can be used in ELISA, IHC.Forma y color:Odour LiquidVPC-14449
CAS:VPC-14449 is a selective androgen receptor DNA-binding domain (AR-DBD) inhibitor, useful in prostate cancer research.Fórmula:C10H10Br2N4OSPureza:99.56%Forma y color:SolidPeso molecular:394.09S-23
CAS:S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (Fórmula:C18H13ClF4N2O3Pureza:98.55%Forma y color:SolidPeso molecular:416.75CLP-3094
CAS:CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor.Fórmula:C15H13ClN2OSPureza:99.84%Forma y color:SolidPeso molecular:304.79Ref: TM-T9179
1mg52,00€5mg114,00€10mg188,00€25mg331,00€50mg495,00€100mg705,00€500mg1.415,00€1mL*10mM (DMSO)125,00€ORM-15341
CAS:ORM-15341 is a potent and full antagonist for human AR (hAR)( with IC50 values of 38 nM as shown by transactivation assays in AR-HEK293 cells)Fórmula:C19H17ClN6O2Pureza:98.01%Forma y color:SolidPeso molecular:396.83Clascoterone
CAS:Clascoterone (CB-03-01) is a new topical and peripherally selective androgen antagonist.Fórmula:C24H34O5Pureza:99.26% - 99.32%Forma y color:SolidPeso molecular:402.52RU 59063
CAS:RU 59063 is a prototype of a new class of high-affinity nonsteroidal androgen receptor (AR) ligands.Fórmula:C17H18F3N3O2SPureza:98.21%Forma y color:SolidPeso molecular:385.4Ref: TM-T20761
1mg87,00€5mg192,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€200mg1.130,00€1mL*10mM (DMSO)208,00€VPC-14228
CAS:VPC-14228 is a specific AR-DBD inhibitor that acts by inhibiting both Y594A and Q592A mutants.Fórmula:C13H14N2OSPureza:99.88%Forma y color:SolidPeso molecular:246.33
