Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Productos de "Receptor GABA"
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Kavain
CAS:Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation ofFórmula:C14H14O3Pureza:99.35% - ≥95%Forma y color:SolidPeso molecular:230.26Radequinil
CAS:Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).Fórmula:C18H14N4O3Pureza:98%Forma y color:SolidPeso molecular:334.33Riluzole
CAS:Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.Fórmula:C8H5F3N2OSPureza:99.71% - 99.88%Forma y color:PowderPeso molecular:234.2Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Fórmula:C10H14ClNO2Pureza:99.93%Forma y color:White Crystalline PowderPeso molecular:215.68Chlormezanone
CAS:Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.Fórmula:C11H12ClNO3SPureza:99.89% - 99.97%Forma y color:Crystals SolidPeso molecular:273.74Chlorothymol
CAS:Chlorothymol (AI3-00120) is a disinfectant used in oral.Fórmula:C10H13ClOPureza:99.50%Forma y color:White Crystals Or PowderPeso molecular:184.66Ref: TM-T20242
5mg48,00€10mg66,00€25mg97,00€50mg154,00€100mg216,00€200mg324,00€500mg543,00€1mL*10mM (DMSO)48,00€Saclofen
CAS:Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.Fórmula:C9H12ClNO3SPureza:99.17%Forma y color:White Crystalline SolidPeso molecular:249.71(-)-Bicuculline methochloride
CAS:(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.Fórmula:C21H20ClNO6Pureza:98%Forma y color:SolidPeso molecular:417.84Tuclazepam
CAS:Tuclazepam (KC 1956) is a derivative of the benzodiazepine class of drugs, exhibiting anti-anxiety and sedative properties.Fórmula:C17H16Cl2N2OForma y color:SolidPeso molecular:335.23Brexanolone caprilcerbate
CAS:Brexanolone caprilcerbate is an effective positive allosteric modulator of the GABAA receptor.Fórmula:C48H78O12Forma y color:SolidPeso molecular:847.13Temgicoluril
CAS:Temgicoluril (mebikar) acts on GABA Receptor.Fórmula:C8H14N4O2Pureza:99.80%Forma y color:SolidPeso molecular:198.22Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Fórmula:C22H21FN4O3SPureza:98.42% - 99.29%Forma y color:SolidPeso molecular:440.49ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Fórmula:C14H16ClN3OPureza:100%Forma y color:SolidPeso molecular:277.75Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Fórmula:C18H17N3O2Pureza:98.74%Forma y color:SolidPeso molecular:307.35TPA 023
CAS:TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).Fórmula:C20H22FN7OPureza:99.06%Forma y color:SolidPeso molecular:395.43Ref: TM-T17144
1mg227,00€5mg550,00€10mg825,00€25mg1.216,00€50mg1.644,00€100mg2.213,00€1mL*10mM (DMSO)605,00€2'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Fórmula:C16H14O4Pureza:98.75%Forma y color:SolidPeso molecular:270.28GABAB receptor antagonist 1
CAS:(E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM.GABAB receptor antagonist 1 is a selectiveFórmula:C18H24O4Pureza:98%Forma y color:SolidPeso molecular:304.38rac-BHFF
CAS:rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.Fórmula:C17H21F3O3Pureza:100% - 98.43%Forma y color:SolidPeso molecular:330.34Ref: TM-T4176
2mg43,00€5mg60,00€10mg96,00€25mg187,00€50mg311,00€100mg472,00€200mg657,00€1mL*10mM (DMSO)71,00€COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Fórmula:C16H16ClNO3SPureza:99.56%Forma y color:SolidPeso molecular:337.82Ref: TM-T36520
1mg52,00€2mg75,00€5mg116,00€10mg178,00€25mg324,00€50mg452,00€100mg620,00€200mg843,00€1mL*10mM (DMSO)128,00€Furosemide sodium
CAS:Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.Fórmula:C12H10ClN2NaO5SPureza:100%Forma y color:SolidPeso molecular:352.73
