Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Productos de "Receptor GABA"
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NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Fórmula:C21H23ClN2O3Pureza:99.92%Forma y color:SolidPeso molecular:386.87FG 7142
CAS:FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.Fórmula:C13H11N3OPureza:98.75%Forma y color:SolidPeso molecular:225.25Ref: TM-T11277
2mg34,00€5mg64,00€10mg97,00€25mg158,00€50mg225,00€100mg335,00€200mg465,00€1mL*10mM (DMSO)42,00€AZD7325
CAS:AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.Fórmula:C19H19FN4O2Pureza:99.83%Forma y color:SolidPeso molecular:354.38BGT1-IN-1
CAS:BGT1-IN-1 (compound 9) is an effective inhibitor of BGT1, demonstrating IC50 values of 13.9 µM for hBGT1 and 58.3 µM for GAT3. It exhibits no cytotoxic effects and possesses neuroprotective activity.Fórmula:C6H9NO2Forma y color:SolidPeso molecular:127.14RO 4938581
CAS:RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).Fórmula:C13H8BrF2N5Pureza:98%Forma y color:SolidPeso molecular:352.143,4,5-Trimethoxycinnamic acid
CAS:3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at theFórmula:C12H14O5Pureza:98.91%Forma y color:SolidPeso molecular:238.24Riluzole-13C,15N2
CAS:Riluzole-13C,15N2 (PK 26124-13C,15N2) is a 13C and 15N labeled form of Riluzole, a glutamate antagonist with anticonvulsant activity, inhibiting GABA uptake.Fórmula:CC7H5F3OS15N2Forma y color:SolidPeso molecular:237.18L-Cycloserine
CAS:L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.Fórmula:C3H6N2O2Pureza:99.45% - 99.92%Forma y color:Crystals White PowderPeso molecular:102.09SCH 50911 hydrochloride
CAS:SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).Fórmula:C8H16ClNO3Pureza:98%Forma y color:SolidPeso molecular:209.67Phaclofen
CAS:GABAB antagonistFórmula:C9H13ClNO3PPureza:99.32%Forma y color:White SolidPeso molecular:249.63
