Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Productos de "Receptor GABA"
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Vigabatrin
CAS:Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-Fórmula:C6H11NO2Pureza:98.2% - 99.76%Forma y color:SolidPeso molecular:129.16Anticonvulsant agent 9
Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.Fórmula:C22H24N4O2Forma y color:SolidPeso molecular:376.45Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFórmula:C2H5NO3·5HClPureza:98.03%Forma y color:Light Beige Crystalline PowderPeso molecular:109.3Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFórmula:C15H14FN3O3Pureza:100% - 99.98%Forma y color:Less Crystals Colourless CrystalsPeso molecular:303.29U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Fórmula:C17H21N3O2Pureza:99.65% - 99.76%Forma y color:SolidPeso molecular:299.37CGP 36742
CAS:CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).Fórmula:C7H18NO2PForma y color:SolidPeso molecular:179.2Lotilaner
CAS:Lotilaner is a parasiticide.Fórmula:C20H14Cl3F6N3O3SPureza:99.56%Forma y color:SolidPeso molecular:596.76Ref: TM-T15775
1mg92,00€5mg188,00€10mg311,00€25mg563,00€50mg753,00€100mg1.103,00€500mg2.205,00€1mL*10mM (DMSO)255,00€Guvacine hydrochloride
CAS:Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)Fórmula:C6H10ClNO2Pureza:98.42%Forma y color:SolidPeso molecular:163.602Afloqualone
CAS:Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.Fórmula:C16H14FN3OPureza:99.72%Forma y color:SolidPeso molecular:283.3Losigamone
CAS:Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.Fórmula:C12H11ClO4Pureza:100%Forma y color:SolidPeso molecular:254.67Oxiracetam
CAS:Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.Fórmula:C6H10N2O3Pureza:99.67%Forma y color:White Crystalline PowderPeso molecular:158.16Primidone
CAS:Primidone (NCI-C56360) is a potent anticonvulsant agent.Fórmula:C12H14N2O2Pureza:99.91%Forma y color:Crystals (Ntp 1992)Peso molecular:218.25L-822179
CAS:L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.Fórmula:C17H14N8O2Pureza:98.34% - 98.74%Forma y color:SolidPeso molecular:362.35α5-GABAA receptor modulator 1
α5-GABAA receptor modulator 1 (Compound A-4) is a selective silent allosteric modulator (SAM) targeting the α5 subunit of GABAA receptors, useful for research into central nervous system (CNS) disorders.Fórmula:C21H20FN3O4Forma y color:SolidPeso molecular:397.4CGP 35348
CAS:CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。Fórmula:C8H20NO4PPureza:≥98%Forma y color:SolidPeso molecular:225.22Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Fórmula:C10H12ClNO2Pureza:98% - 99.85%Forma y color:1992)Peso molecular:213.66CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Fórmula:C15H24Cl2NO4PPureza:98.75%Forma y color:SolidPeso molecular:384.24Muscimol HBr
CAS:Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.Fórmula:C4H7BrN2O2Pureza:100%Forma y color:Off-White PowderPeso molecular:195.01Ref: TM-T20657
1mg119,00€2mg172,00€5mg253,00€10mg406,00€25mg657,00€50mg948,00€100mg1.264,00€500mg2.555,00€1mL*10mM (DMSO)215,00€(-)-Securinine
CAS:(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Fórmula:C13H15NO2Pureza:99.58% - 99.87%Forma y color:SolidPeso molecular:217.266,2'-Dihydroxyflavone
CAS:6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.Fórmula:C15H10O4Pureza:99.03%Forma y color:SolidPeso molecular:254.24
