Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Productos de "Receptor GABA"
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GS 39783
CAS:GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement andFórmula:C15H23N5O2SPureza:99.94%Forma y color:SolidPeso molecular:337.44Isonipecotic acid
CAS:Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.Fórmula:C6H11NO2Pureza:99.82%Forma y color:White To Faint Pink-Beige PowderPeso molecular:129.16Piperazine citrate
CAS:Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.Fórmula:C24H46N6O14Pureza:≥98%Forma y color:Crystals IndicationPeso molecular:642.65Lorediplon
CAS:Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.Fórmula:C20H15FN4O2SPureza:99.12% - 99.19%Forma y color:SolidPeso molecular:394.42L-655708
CAS:L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.Fórmula:C18H19N3O4Pureza:98.41%Forma y color:PowderPeso molecular:341.36U 89843A
CAS:U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.Fórmula:C16H23N5Pureza:99.53%Forma y color:SolidPeso molecular:285.39Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Fórmula:C7H12ClNO2Pureza:≥95% - ≥98%Forma y color:SolidPeso molecular:177.63Ref: TM-T5799
2mg35,00€5mg50,00€10mg71,00€25mg105,00€50mg158,00€100mg225,00€200mg334,00€1mL*10mM (DMSO)51,00€Nerisopam
CAS:Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.Fórmula:C18H19N3O2Pureza:97.27%Forma y color:SolidPeso molecular:309.36Ref: TM-T28159
1mg93,00€5mg200,00€10mg303,00€25mg490,00€50mg710,00€100mg998,00€200mg1.349,00€1mL*10mM (DMSO)270,00€ONO-8590580
CAS:ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.Fórmula:C21H21FN6Pureza:99.43%Forma y color:SolidPeso molecular:376.43Ref: TM-TQ0040
1mg66,00€2mg93,00€5mg126,00€10mg170,00€25mg376,00€50mg562,00€100mg802,00€1mL*10mM (DMSO)140,00€SKF89976A hydrochloride
CAS:SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFórmula:C22H26ClNO2Pureza:98.72%Forma y color:SolidPeso molecular:371.9Ref: TM-T12930
1mg35,00€5mg69,00€10mg95,00€25mg178,00€50mg283,00€100mg454,00€200mg650,00€1mL*10mM (DMSO)74,00€4-Acetamidobutanoic acid
CAS:4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Fórmula:C6H11NO3Pureza:99.79%Forma y color:SolidPeso molecular:145.16U-89843A
CAS:U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].Fórmula:C16H24ClN5Pureza:98%Forma y color:SolidPeso molecular:321.85Broflanilide
CAS:Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.Fórmula:C25H14BrF11N2O2Pureza:98.95%Forma y color:SolidPeso molecular:663.29Ref: TM-T10618
1mg52,00€2mg74,00€5mg111,00€10mg180,00€25mg358,00€50mg588,00€100mg835,00€1mL*10mM (DMSO)131,00€Tracazolate hydrochloride
CAS:Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.Fórmula:C16H25ClN4O2Pureza:99.07%Forma y color:SolidPeso molecular:340.85GABA receptor Antagonist 1
GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 of 7.08 nmol/L and demonstrates insecticidal efficacy against P.Pureza:98%Forma y color:Odour Solid6-(4-Methoxyphenyl)-3-pyridazinamine
CAS:6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFórmula:C11H11N3OPureza:99.03%Forma y color:SolidPeso molecular:201.22TET-13
TET-13 is a positive allosteric modulator of the GABAA receptor with an EC50 of 5.65 μM, which is more potent than Etomidate (EC50: 9.29 μM). It exhibits strong anesthetic effects in both mice and rats, with an ED50 of 0.48 mg/kg in mice and 0.69 mg/kg in rats.Fórmula:C15H16N2O3SForma y color:SolidPeso molecular:304.36PZ-II-029
CAS:PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.Fórmula:C18H15N3O3Pureza:99.72%Forma y color:SolidPeso molecular:321.33Ref: TM-T28479
1mg52,00€5mg111,00€10mg170,00€25mg305,00€50mg472,00€100mg723,00€500mg1.454,00€1mL*10mM (DMSO)202,00€(R)-baclofen
CAS:(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.Fórmula:C10H12ClNO2Pureza:98.94%Forma y color:SolidPeso molecular:213.66NS-2710
CAS:NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.Fórmula:C22H20N4OPureza:98.10% - 99.82%Forma y color:SolidPeso molecular:356.42
