Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Productos de "Receptor GABA"
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CP-409092
CAS:CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.Fórmula:C17H19N3O2Pureza:98%Forma y color:SolidPeso molecular:297.35(E)-GABAB receptor antagonist 1
CAS:(E)-GABAB antagonist 1 inhibits GABA IP3 production, with an IC50 of 37.9 μM and acts as a selective negative modulator.Fórmula:C18H24O4Pureza:95.26%Forma y color:SolidPeso molecular:304.38Ref: TM-T11137
1mg115,00€5mg255,00€10mg375,00€25mg562,00€50mg787,00€100mg1.074,00€200mg1.454,00€1mL*10mM (DMSO)246,00€Cyproflanilide
CAS:Cyproflanilide is a GABAR antagonist that exhibits high activity against a variety of pests, including those from the Lepidoptera, Coleoptera, and Thysanoptera orders.Fórmula:C28H17BrF12N2O2Forma y color:SolidPeso molecular:721.33Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Fórmula:C22H17Cl2F6N3O3Pureza:99.72% - 99.90%Forma y color:Solid PowderPeso molecular:556.29(-)-Bicuculline methobromide
CAS:(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .Fórmula:C21H20BrNO6Forma y color:WhitePeso molecular:462.29Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Fórmula:C58H94O26Pureza:100% - 99.05%Forma y color:SolidPeso molecular:1207.35Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Fórmula:C20H29N3O5SPureza:99.39% - ≥95%Forma y color:SolidPeso molecular:423.53NS11394
CAS:NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Fórmula:C23H19N3OPureza:99.44% - 99.86%Forma y color:SolidPeso molecular:353.42Ref: TM-T2067
2mg34,00€5mg50,00€10mg80,00€25mg131,00€50mg212,00€100mg321,00€200mg460,00€1mL*10mM (DMSO)58,00€Cannabidivarin
CAS:Cannabidivarin (GWP42006) inhibits GABAA receptors, potentially controlling childhood absence epilepsy.Fórmula:C19H26O2Pureza:98.06% - 98.51%Forma y color:SolidPeso molecular:286.41Ref: TM-T8162
1mg52,00€2mg74,00€5mg87,00€10mg140,00€25mg264,00€50mg416,00€100mg615,00€1mL*10mM (DMSO)111,00€SSD114 HCl
CAS:SSD114 is a novel GABAB receptor positive allosteric modulator.Fórmula:C18H21ClF3N3OPureza:99.03% - 99.95%Forma y color:SolidPeso molecular:387.83Ref: TM-T4522
1mg38,00€2mg50,00€5mg88,00€10mg119,00€25mg188,00€50mg300,00€100mg512,00€1mL*10mM (DMSO)74,00€Fipronil
CAS:Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Fórmula:C12H4Cl2F6N4OSPureza:97.48%Forma y color:Solid PowderPeso molecular:437.15Ocinaplon
CAS:Ocinaplon (DOV 273547) is a GABAA receptors modulator.Fórmula:C17H11N5OPureza:98.78%Forma y color:SolidPeso molecular:301.3Padsevonil
CAS:Padsevonil (UCB-0942) is a potential GABA A receptor orthosteric modulator with antiepileptic activity for the treatment of epilepsy.Fórmula:C14H14ClF5N4O2SPureza:99.63%Forma y color:SolidPeso molecular:432.80Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Fórmula:C10H12N2O3Pureza:99.38%Forma y color:White Crystalline PowderPeso molecular:208.21Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Fórmula:C15H18BrN3O3Pureza:98.51%Forma y color:SolidPeso molecular:368.23DMCM hydrochloride
CAS:DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Fórmula:C17H19ClN2O4Pureza:98.95%Forma y color:SolidPeso molecular:350.8Ref: TM-T11061
1mg37,00€2mg49,00€5mg85,00€10mg111,00€25mg250,00€50mg464,00€100mg655,00€1mL*10mM (DMSO)93,00€(S)-SNAP5114
CAS:(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.Fórmula:C30H35NO6Pureza:97%Forma y color:SolidPeso molecular:505.6Ref: TM-T16831
1mg35,00€5mg80,00€10mg116,00€25mg259,00€50mg375,00€100mg545,00€500mg1.093,00€1mL*10mM (DMSO)87,00€Tiagabine hydrochloride
CAS:Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.Fórmula:C20H25NO2S2·HClPureza:99.09% - 99.77%Forma y color:White To Off-White SolidPeso molecular:412.01MRK-016
CAS:MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.Fórmula:C17H20N8O2Pureza:99.76%Forma y color:SolidPeso molecular:368.39Guvacine hydrobromide
CAS:Guvacine hydrobromide, an alkaloid derived from the Areca catechu nut, serves as a potent inhibitor of GABA (GABA uptakp) uptake.Fórmula:C6H10BrNO2Pureza:98%Forma y color:SolidPeso molecular:208.05
