Transferasa
Las transferasas son una gran clase de enzimas que catalizan la transferencia de grupos funcionales, como grupos metilo, glicosilo y fosfato, de una molécula a otra. Los inhibidores de transferasas se utilizan para estudiar una amplia gama de procesos biológicos, incluyendo la transducción de señales, el metabolismo y la expresión génica. Estos inhibidores son herramientas esenciales en áreas de investigación como el cáncer, las enfermedades metabólicas y la epigenética, donde está implicada la disfunción de la actividad de las transferasas. En CymitQuimica, ofrecemos una selección integral de inhibidores de transferasas para apoyar su investigación en enzimología, señalización celular y mecanismos de enfermedad.
Productos de "Transferasa"
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Ibiglustat (L-Malic acid)
CAS:Ibiglustat (L-Malic acid) (Ibiglustat L-Malic acid) is a selective, brain-penetrant, and allosteric inhibitor of glucosylceramide synthase.Fórmula:C24H30FN3O7SPureza:99.79%Forma y color:SolidPeso molecular:523.57Ref: TM-T11599
1mg60,00€2mg88,00€5mg153,00€10mg217,00€25mg368,00€50mg547,00€100mg782,00€1mL*10mM (DMSO)170,00€GGTI-2133
CAS:GGTI-2133: potent GGTase I inhibitor, IC50=38 nM; blocks inflammatory cell invasion in mice asthma.Fórmula:C27H28N4O3Pureza:99.80%Forma y color:SolidPeso molecular:456.54GPAT-IN-1
CAS:GPAT-IN-1 is a glycerol 3-phosphate acyltransferase (GPAT) inhibitor, which can be used to study obesity and diabetes.Fórmula:C21H26ClNO4SPureza:99.61% - 99.61%Forma y color:SolidPeso molecular:423.95P-3FAX-Neu5Ac
CAS:P-3FAX-Neu5Ac is a sialic acid analog and a sialyltransferase inhibitor.Fórmula:C22H30FNO14Pureza:97.08%Forma y color:SolidPeso molecular:551.47Nitecapone
CAS:Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)Fórmula:C12H11NO6Pureza:98.39%Forma y color:SolidPeso molecular:265.22CP-609754
CAS:CP-609754 shows selective inhibition of farnesyltransferase.Fórmula:C29H22ClN3O2Pureza:98.8% - 99.04%Forma y color:SolidPeso molecular:479.96Ref: TM-T38050
1mg55,00€5mg116,00€10mg187,00€25mg319,00€50mg449,00€100mg638,00€200mg840,00€1mL*10mM (DMSO)134,00€GSK2973980A
CAS:GSK2973980A is a selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor (IC50: 3 nM).Fórmula:C25H19F5N4O4Pureza:98%Forma y color:SolidPeso molecular:534.43LB42708
CAS:LB42708 is an orally active farnesyltransferase (FTase) inhibitor (IC50: 0.8/1.2/2.0 nM toward H/N/K-ras).Fórmula:C30H27BrN4O2Pureza:97.83%Forma y color:SolidPeso molecular:555.47Ref: TM-T2678
1mg49,00€2mg64,00€5mg96,00€10mg145,00€25mg278,00€50mg414,00€100mg580,00€1mL*10mM (DMSO)133,00€Lucerastat
CAS:Lucerastat(NBDGJ) is an orally available inhibitor of GCS for Fabry disease by reducing harmful substrates.. GCS is a key enzyme in sphingolipid synthesiss.Fórmula:C10H21NO4Pureza:98%Forma y color:SolidPeso molecular:219.28Risedronic Acid
CAS:Risedronic Acid (Risedronate), a pyridinyl biphosphonate, can inhibit osteoclast-mediated bone resorption.Fórmula:C7H11NO7P2Pureza:99.77% - 99.85%Forma y color:White Crystalline PowderPeso molecular:283.11Lapaquistat acetate
CAS:Lapaquistat acetate (TAK-475) is a squalene synthase inhibitor that reduces the cytotoxicity induced by statins in human skeletal muscle cells.Fórmula:C33H41ClN2O9Pureza:100% - 99.74%Forma y color:SolidPeso molecular:645.14Entacapone acid
CAS:Entacapone acid (AG 1290) is a selective and reversible inhibitor of catechol-O-methyltransferase(COMT).Fórmula:C10H6N2O6Pureza:99.76%Forma y color:SolidPeso molecular:250.16GGsTop
CAS:GGsTop (Nahlsgen) is a GGT inhibitor with anti-aging activity.Fórmula:C13H18NO7PPureza:98.96%Forma y color:SolidPeso molecular:331.26OU749
CAS:OU749 is a γ-glutamyl transferase (GGT) inhibitor with an intrinsic Ki of 17.6 μM.Fórmula:C16H15N3O3S2Pureza:99.7%Forma y color:SolidPeso molecular:361.44Ref: TM-T22128
2mg49,00€5mg88,00€10mg127,00€25mg208,00€50mg309,00€100mg460,00€500mg1.008,00€1mL*10mM (DMSO)70,00€JNJ-DGAT2-A
CAS:JNJ-DGAT2-A, a specific inhibitor of DGAT2(IC50 = 0.14 μM), can be used in studies about the synthesis of triglycerides.Fórmula:C24H16BrFN4O2SPureza:98.2%Forma y color:SolidPeso molecular:523.38Tipifarnib
CAS:Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.Fórmula:C27H22Cl2N4OPureza:97.1% - 99.22%Forma y color:Off-White To Pale Beige SolidPeso molecular:489.4FGTI-2734
CAS:FGTI-2734, a dual FT/GGT-1 inhibitor (IC50: 250/520 nM), blocks KRAS membrane binding and curbs KRAS-driven pancreatic cancer.Fórmula:C26H31FN6O2SPureza:99.36%Forma y color:SolidPeso molecular:510.63Ref: TM-T11282
1mg51,00€5mg119,00€10mg188,00€25mg393,00€50mg587,00€100mg835,00€1mL*10mM (DMSO)136,00€Minodronic acid monohydrate
CAS:Minodronic acid monohydrate 是一种法尼基二磷酸合成酶抑制剂,可作为骨吸收抑制剂。Fórmula:C9H14N2O8P2Pureza:≥95%Forma y color:SolidPeso molecular:340.16Entacapone
CAS:Entacapone (OR-611) is a selective and reversible inhibitor of catechol-O-methyltransferase (COMT).Fórmula:C14H15N3O5Pureza:100% - 99.79%Forma y color:Yellow Crystalline SolidPeso molecular:305.29Ref: TM-T2216
5mg35,00€10mg51,00€25mg80,00€50mg96,00€100mg144,00€200mg207,00€500mg350,00€1mL*10mM (DMSO)49,00€Ibiglustat
CAS:Ibiglustat (GZ402671) inhibits Glucosylceramide synthase, may treat Fabry disease by preventing GL-3 synthesis.Fórmula:C20H24FN3O2SPureza:97.97% - 99.14%Forma y color:SolidPeso molecular:389.49Ref: TM-T4473
1mg39,00€5mg97,00€10mg168,00€25mg298,00€50mg430,00€100mg605,00€200mg815,00€1mL*10mM (DMSO)90,00€
