Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Productos de "Receptor 5-HT"
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Pizotifen Malate
CAS:Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based on benzocycloheptane.Fórmula:C19H21NS·C4H6O5Pureza:100%Forma y color:SolidPeso molecular:429.53Repinotan
CAS:Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.Fórmula:C21H24N2O4SPureza:99%Forma y color:SolidPeso molecular:400.49Gentisein
CAS:Gentisein (NSC-329491), a primary metabolite of Mangiferin, exhibits significant inhibition of serotonin uptake, demonstrating potency with an IC50 value of 4.7Fórmula:C13H8O5Pureza:96.74%Forma y color:SolidPeso molecular:244.2(Rac)-Norcisapride
CAS:Norcisapride, a 5-HT3 and 5-HT4 agonist, treats GI, orofacial, and ENT disorders.Fórmula:C14H20ClN3O3Pureza:99.13%Forma y color:SoildPeso molecular:313.78(S)-Amisulpride
CAS:(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.Fórmula:C17H27N3O4SPureza:98.38%Forma y color:SolidPeso molecular:369.48Ref: TM-T26375
1mg50,00€2mg71,00€5mg114,00€10mg178,00€25mg340,00€50mg538,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)126,00€AAZ-A 154 hydrobromide
CAS:AAZ-A 154 hydrobromide is a selective, competitive, non-hallucinogenic 5-HT2AR antagonist. It promotes neuronal growth in rodents and yields enduring beneficial behavioral effects.Fórmula:C14H21BrN2OForma y color:SolidPeso molecular:313.23Ondansetron hydrochloride dihydrate
CAS:Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.Fórmula:C18H19N3O·HCl·2H2OPureza:99.92%Forma y color:White Crystal PowderPeso molecular:365.86SB 243213 hydrochloride
CAS:SB 243213 hydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8).ItFórmula:C22H20ClF3N4O2Pureza:98%Forma y color:SolidPeso molecular:464.87Ipsapirone
CAS:Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.Fórmula:C19H23N5O3SPureza:99.01%Forma y color:SolidPeso molecular:401.485-HT1A modulator 4
CAS:5-HT1A modulator 4 (Compound 1) is a ligand for the 5-HT receptor, with Ki values of 2.18 μM for 5-HT1A and 19.7 μM for 5-HT2A.Fórmula:C9H14N4Forma y color:SolidPeso molecular:178.234SB-200646A
CAS:SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.Fórmula:C15H15ClN4OPureza:98%Forma y color:SolidPeso molecular:302.76Adatanserin
CAS:Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.Fórmula:C21H31N5OPureza:99.17%Forma y color:SolidPeso molecular:369.5ST1936
CAS:ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.Fórmula:C13H17ClN2Pureza:98.00%Forma y color:SolidPeso molecular:236.74Ref: TM-T23396
1mg47,00€5mg117,00€10mg188,00€25mg334,00€50mg497,00€100mg720,00€200mg1.008,00€1mL*10mM (DMSO)130,00€Cyproheptadine hydrochloride
CAS:Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.Fórmula:C21H21N·HClPureza:99.88% - 99.97%Forma y color:SolidPeso molecular:323.86Tropanserin
CAS:Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.Fórmula:C17H23NO2Pureza:99.74%Forma y color:SolidPeso molecular:273.37Sarizotan 2HCl
CAS:Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.Fórmula:C22H23Cl2FN2OPureza:98.83%Forma y color:SoildPeso molecular:421.345-HT2C agonist-3 free base
CAS:5-HT2C agonist-3 ((+)-19) free base, a selective 5-HT2C agonist (EC50: 24 nM, Ki: 78 nM), exhibits antipsychotic drug-like activity and inhibits Amphetamine-Fórmula:C19H22FNO2Pureza:98%Forma y color:SolidPeso molecular:315.38Sulamserod hydrochloride
CAS:Sulamserod hydrochloride is a 5-HT4 receptor antagonist. It is utilized in research related to gastrointestinal disorders.Fórmula:C19H29Cl2N3O5SForma y color:SolidPeso molecular:482.42LY 344864
CAS:LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.Fórmula:C21H22FN3OPureza:98%Forma y color:SolidPeso molecular:351.42γ-Mangostin
CAS:Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.Fórmula:C23H24O6Pureza:98.55% - 99.08%Forma y color:SolidPeso molecular:396.43WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Fórmula:C14H18N2Pureza:98%Forma y color:SolidPeso molecular:214.315-HT7 agonist 1
CAS:5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).Fórmula:C19H20ClN3Pureza:98.61%Forma y color:SolidPeso molecular:325.84Ref: TM-T10170
1mg115,00€2mg172,00€5mg255,00€10mg375,00€25mg562,00€50mg787,00€100mg1.074,00€1mL*10mM (DMSO)255,00€YM-31636 free base
CAS:YM-31636 (free base) is an orally active, potent, and selective agonist of the 5-HT3 receptor with a pKi value of 9.67. This compound induces contraction in isolated guinea pig distal colon and provokes tachycardia in isolated guinea pig right atrium, demonstrating a relative intrinsic activity of about 0.23. YM-31636 (free base) holds potential for research in constipation management.Fórmula:C14H11N3SForma y color:SolidPeso molecular:253.325-HT2 agonist-1 free base
CAS:Compound 24 (5-HT2 agonist-1 free base) is a potent agonist for 5-HT2A, 5-HT2B, and 5-HT2C receptors, exhibiting IC50 values of 10 nM, 8.3 nM, and 1.6 nM,Fórmula:C19H22N2O2Pureza:98%Forma y color:SolidPeso molecular:310.39Thioridazine hydrochloride
CAS:Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4Fórmula:C21H27ClN2S2Pureza:99.55% - 99.55%Forma y color:White To Off-White SolidPeso molecular:407.0425N-NBOMe hydrochloride
CAS:25N-NBOMe hydrochloride is a derivative of 2C-N and acts as an agonist for the 5-HT2A and 5-HT2C receptors, with Ki values of 0.144 nM and 1.06 nM, respectively. It has minimal effect on the release of preloaded neurotransmitters from recombinant dopamine, serotonin, and norepinephrine transporters.Fórmula:C18H23ClN2O5Forma y color:SolidPeso molecular:382.84Landipirdine
CAS:Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.Fórmula:C18H19FN2O3SPureza:97.50% - 99.33%Forma y color:SolidPeso molecular:362.42Venlafaxine hydrochloride
CAS:Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Fórmula:C17H28ClNO2Pureza:99.86%Forma y color:White Crystalline PowderPeso molecular:313.863Adatanserin hydrochloride
CAS:Adatanserin hydrochloride (WY50324 hydrochloride) is a 5-HT(1A)/5-HT(2) receptor ligand that is neuroprotective and may be used in the study of depression.Fórmula:C21H32ClN5OPureza:99.64%Forma y color:SolidPeso molecular:405.96Olopatadine hydrochloride
CAS:Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.Fórmula:C21H23NO3·HClPureza:99.62% - 99.64%Forma y color:White SolidPeso molecular:373.87Latrepirdine dihydrochloride
CAS:Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Fórmula:C21H25N3·2HClPureza:98.45%Forma y color:SolidPeso molecular:392.37SR 57227 hydrochloride
CAS:SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.Fórmula:C10H14ClN3·HClPureza:99.89%Forma y color:SolidPeso molecular:248.15Ref: TM-T23394
5mg50,00€10mg74,00€25mg126,00€50mg210,00€100mg313,00€200mg445,00€1mL*10mM (DMSO)49,00€RS 56812 hydrochloride
CAS:5-HT3 partial agonistFórmula:C18H22ClN3O2Pureza:97.69%Forma y color:SolidPeso molecular:347.84N-Desmethyl Pimavanserin
CAS:N-Desmethyl Pimavanserin (AC-279) is the active metabolite of Pimavanserin and is used in the treatment of insomnia and other sleep disorders.Fórmula:C24H32FN3O2Pureza:98.02%Forma y color:SolidPeso molecular:413.53Urapidil
CAS:Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Fórmula:C20H29N5O3Pureza:100% - 99.85%Forma y color:SolidPeso molecular:387.48Gepirone
CAS:Gepirone is a 5-HT1A receptor agonist belonging to the buspirone family. Gepirone HCl possesses greater selectivity for the 5-HT1A receptor than SSRIs.Fórmula:C19H29N5O2Pureza:99.35% - 99.77%Forma y color:SolidPeso molecular:359.47Pizotifen
CAS:Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.Fórmula:C19H21NSPureza:99.93%Forma y color:SolidPeso molecular:295.44Ondansetron
CAS:Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.Fórmula:C18H19N3OPureza:99.92%Forma y color:White To Yellow CrystalsPeso molecular:293.364-Hydroxy MPT
CAS:4-Hydroxy MPT (4-OH-MPT) is a serotonin-active compound that acts as an agonist for 5-HT2A and 5-HT2B receptors, with EC50 values of 3.82 nM and 3.4 nM, respectively.Fórmula:C14H20N2OForma y color:SolidPeso molecular:232.32Olanzapine
CAS:Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Fórmula:C17H20N4SPureza:100% - ≥95%Forma y color:Yellowish Crystalline PowderPeso molecular:312.43Desvenlafaxine succinate hydrate
CAS:Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).Fórmula:C20H33NO7Pureza:99.26%Forma y color:White Crystalline PowdePeso molecular:399.48Dolasetron Mesylate hydrate
CAS:Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.Fórmula:C20H26N2O7SPureza:99.86% - 99.9%Forma y color:SolidPeso molecular:438.49cis-(Z)-Flupentixol dihydrochloride
CAS:cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.Fórmula:C23H27Cl2F3N2OSPureza:98.07%Forma y color:SolidPeso molecular:507.44Ebalzotan
CAS:NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.Fórmula:C19H30N2O2Pureza:99.08% - 99.41%Forma y color:SolidPeso molecular:318.45Relenopride
CAS:YKP 10811 (Relenopride) is a novel 5-HT4 receptor partial agonist, which can be used to study irritable bowel syndrome with constipation.Fórmula:C24H30ClFN4O4Pureza:98.91% - 99.20%Forma y color:SoildPeso molecular:492.97MM 77 dihydrochloride
CAS:MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.Fórmula:C19H29Cl2N3O3Pureza:100.00%Forma y color:SolidPeso molecular:418.36Ref: TM-T23007
1mg86,00€5mg157,00€10mg215,00€25mg472,00€50mg687,00€100mg938,00€500mg1.882,00€1mL*10mM (DMSO)281,00€AL 34662
CAS:AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also aFórmula:C10H13N3OPureza:99.77%Forma y color:SolidPeso molecular:191.23Naluzotan hydrochloride
CAS:Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.Fórmula:C23H39ClN4O3SPureza:98.61%Forma y color:SolidPeso molecular:487.1PNU 22394 hydrochloride
CAS:PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonistFórmula:C13H17ClN2Pureza:97.83%Forma y color:SolidPeso molecular:236.74RS-67333
CAS:RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.Fórmula:C19H29ClN2O2Pureza:99.24%Forma y color:SolidPeso molecular:352.9(E)-3,4,5-Trimethoxycinnamic acid
CAS:(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Fórmula:C12H14O5Pureza:99.83%Forma y color:SolidPeso molecular:238.24Clovoxamine
CAS:Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant and anticonvulsant activity.Fórmula:C14H21ClN2O2Pureza:98.88% - 99.16%Forma y color:SolidPeso molecular:284.78Mosapride
CAS:Mosapride (AS-4370) is a selective 5HT4 agonistFórmula:C21H25ClFN3O3Pureza:99.56%Forma y color:White To Off-White Crystalline SolidPeso molecular:421.89SB 216641 hydrochloride
CAS:SB 216641 hydrochloride (SB-216641A) is a 5-HT1B/D receptor antagonist with anxiolytic properties.Fórmula:C28H31ClN4O4Pureza:98.40% - 99.23%Forma y color:SolidPeso molecular:523.02Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Fórmula:C22H29N3O4SPureza:99.94%Forma y color:Yellowish White Crystalline PowderPeso molecular:431.55Vilazodone
CAS:Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.Fórmula:C26H27N5O2Pureza:99.61%Forma y color:Light Yellow SolidPeso molecular:441.52Agomelatine (L(+)-Tartaric acid)
CAS:Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, andFórmula:C19H23NO8Forma y color:SolidPeso molecular:393.39LP-211
CAS:LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.Fórmula:C30H34N4OPureza:98.65%Forma y color:SolidPeso molecular:466.62Ref: TM-T5387
2mg47,00€5mg70,00€10mg96,00€25mg180,00€50mg305,00€100mg487,00€200mg695,00€1mL*10mM (DMSO)77,00€Usmarapride free base
CAS:Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.Fórmula:C21H29N5O2Pureza:99.91% - 99.91%Forma y color:SolidPeso molecular:383.49Glemanserin
CAS:Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.Fórmula:C20H25NOPureza:99.52%Forma y color:SolidPeso molecular:295.42Ref: TM-T22964
1mg40,00€5mg88,00€10mg126,00€25mg273,00€50mg432,00€100mg638,00€500mg1.359,00€1mL*10mM (DMSO)88,00€DA-6886
CAS:DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Fórmula:C19H28Cl2N6O2Pureza:99% - 99.89%Forma y color:SolidPeso molecular:443.37Litoxetine
CAS:Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.Fórmula:C16H19NOPureza:99.12%Forma y color:SolidPeso molecular:241.33Ref: TM-T67956
1mg97,00€5mg217,00€10mg325,00€25mg557,00€50mg797,00€100mg1.103,00€500mg2.205,00€1mL*10mM (DMSO)188,00€RG-12915
CAS:RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).Fórmula:C20H25ClN2O2Pureza:98%Forma y color:SolidPeso molecular:360.88VUF 10166
CAS:VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.Fórmula:C13H15ClN4Pureza:99.66%Forma y color:SolidPeso molecular:262.74Trazodone hydrochloride
CAS:Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.Fórmula:C19H23Cl2N5OPureza:99.50% - 99.52%Forma y color:SolidPeso molecular:408.335-HT6R antagonist 1
Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stabilityFórmula:C17H22F2N6OPureza:98%Forma y color:SolidPeso molecular:364.39Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderateFórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Forma y color:SolidPeso molecular:427.41Ref: TM-T4577
1mg51,00€5mg108,00€10mg180,00€25mg316,00€50mg472,00€100mg658,00€200mg938,00€1mL*10mM (DMSO)108,00€Faxeladol
CAS:Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.Fórmula:C15H23NOPureza:99.11% - 99.13%Forma y color:SolidPeso molecular:233.35Cyamemazine
CAS:Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Fórmula:C19H21N3SPureza:97.01%Forma y color:SolidPeso molecular:323.46Ziprasidone hydrochloride
CAS:Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFórmula:C21H22CL2N4OSPureza:97.97% - 99.82%Forma y color:SolidPeso molecular:449.4p-MPPF dihydrochloride
CAS:p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.Fórmula:C25H29Cl2FN4O2Pureza:99.78%Forma y color:SolidPeso molecular:507.43Citalopram
CAS:Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.Fórmula:C20H21FN2OPureza:99.89%Forma y color:SolidPeso molecular:324.39AGH-107
CAS:AGH-107 is a highly selective 5-HT7 receptor agonist that can cross the blood-brain barrier, featuring a Ki value of 6 nM and an EC50 value of 19 nM. Demonstrating high selectivity for central nervous system targets, AGH-107 also exhibits high metabolic stability and low toxicity in HEK-293 and HepG2 cell cultures.Fórmula:C13H12IN3Forma y color:SolidPeso molecular:337.162-Methyl-5-HT
CAS:2-Methyl-5-HT (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.Fórmula:C11H14N2OPureza:95.64%Forma y color:SolidPeso molecular:190.24Ref: TM-T10075
5mg50,00€10mg88,00€25mg187,00€50mg354,00€100mg528,00€500mg1.159,00€1mL*10mM (DMSO)52,00€Pumosetrag Hydrochloride
CAS:Pumosetrag Hydrochloride is an orally available 5-HT3 partial agonist. It is developed for the treatment of irritable bowel syndrome and gastroesophageal reflux disease.Fórmula:C15H18ClN3O2SPureza:98%Forma y color:SolidPeso molecular:339.845HT6-ligand-1
CAS:5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).Fórmula:C20H22BrN3O2SPureza:98.48% - 98.95%Forma y color:SolidPeso molecular:448.38Remlifanserin
CAS:Remlifanserin is a potent inverse agonist of the serotonin receptor (5-HT2A).Fórmula:C24H29F2N3O2Forma y color:SolidPeso molecular:429.50S 14506 hydrochloride
CAS:S 14506 hydrochloride is a 5-HT1A receptor full agonist.Fórmula:C24H27ClFN3O2Pureza:99.5%Forma y color:SolidPeso molecular:443.945-HT3 antagonist 2
CAS:5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.Fórmula:C18H21N3OPureza:98%Forma y color:SolidPeso molecular:295.38Ocaperidone
CAS:Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.Fórmula:C24H25FN4O2Pureza:99.33%Forma y color:SolidPeso molecular:420.484-hydroxy DiPT hydrochloride
CAS:4-hydroxy DiPT (hydrochloride) is a 5-HT2A agonist that can induce head twitch response (HTR) in mice, indicating its hallucinogenic potential. This compound holds promise for research into hallucinogens.Fórmula:C16H25ClN2OForma y color:SolidPeso molecular:296.84Renzapride
CAS:Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.Fórmula:C16H22ClN3O2Pureza:98.97% - 99.09%Forma y color:SolidPeso molecular:323.82GR 125743
CAS:GR 125743 is a novel antagonist of 5-HT1B/1D receptor.Fórmula:C25H28N4O2Pureza:99.76%Forma y color:SolidPeso molecular:416.52Ref: TM-T8737
1mg43,00€2mg56,00€5mg88,00€10mg119,00€25mg235,00€50mg350,00€100mg522,00€1mL*10mM (DMSO)87,00€Pardoprunox hydrochloride
CAS:Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)Fórmula:C12H16ClN3O2Pureza:98.73% - 99.13%Forma y color:SolidPeso molecular:269.73LY266097 hydrochloride
CAS:LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.Fórmula:C21H24Cl2N2O2Pureza:99.63%Forma y color:SolidPeso molecular:407.33Alosetron hydrochloride
CAS:Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.Fórmula:C17H19ClN4OPureza:99.90%Forma y color:Off-White PowderPeso molecular:330.81(Rac)-WAY-161503
CAS:(Rac)-WAY-161503 is a selective and high-affinity agonist of the 5-HT2C receptor (Ki: 4 nM; EC50: 12 nM), with anti-obesity and antidepressant effects.Fórmula:C11H11Cl2N3OPureza:98.08%Forma y color:SolidPeso molecular:272.13Org-13011 fumarate
CAS:Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.Fórmula:C22H29F3N4O5Pureza:98.61%Forma y color:SolidPeso molecular:486.48Azaphen dihydrochloride monohydrate
CAS:Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.Fórmula:C16H23Cl2N5O2Pureza:99.85%Forma y color:SolidPeso molecular:388.29Metadoxine
CAS:Metadoxine (Metadoxil) is a neurotransmitter stimulant.Fórmula:C8H11NO3·C5H7NO3Pureza:99.19%Forma y color:Off-White PowderPeso molecular:298.29Geissoschizine methyl ether
CAS:Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.Fórmula:C22H26N2O3Pureza:99.68% - 99.86%Forma y color:SolidPeso molecular:366.45Ref: TM-TN1032
1mg137,00€5mg404,00€10mg587,00€25mg914,00€50mg1.225,00€100mg1.663,00€1mL*10mM (DMSO)375,00€Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Fórmula:C22H28FNO3Pureza:98.94% - 99.95%Forma y color:SolidPeso molecular:373.46Methiothepin maleate
CAS:Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.Fórmula:C24H28N2O4S2Pureza:98%Forma y color:SolidPeso molecular:472.62Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。Fórmula:C21H25ClN2O4SPureza:99.04%Forma y color:SolidPeso molecular:436.95SB 271046 hydrochloride
CAS:SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.Fórmula:C20H22ClN3O3S2·HClPureza:99.57%Forma y color:SolidPeso molecular:488.455-Methyltryptamine hydrochloride
CAS:5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.Fórmula:C11H15ClN2Pureza:99.45%Forma y color:SolidPeso molecular:210.703Dolasetron
CAS:Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.Fórmula:C19H20N2O3Pureza:99.84% - 99.86%Forma y color:White PowderPeso molecular:324.37Harmine hydrochloride
CAS:Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.Fórmula:C13H13ClN2OPureza:100% - 99.45%Forma y color:Yellow To Slightly Green Crystalline PowderPeso molecular:248.71Almotriptan Malate
CAS:Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.Fórmula:C17H25N3O2S·C4H6O5Pureza:99.95%Forma y color:Pale Yellow SolidPeso molecular:469.55A-582941 dihydrochloride
CAS:A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partialFórmula:C17H22Cl2N4Pureza:99.55%Forma y color:SolidPeso molecular:353.29Ref: TM-T22016
1mg42,00€5mg88,00€10mg120,00€25mg235,00€50mg354,00€100mg533,00€200mg743,00€1mL*10mM (DMSO)87,00€ECPLA
CAS:ECPLA is an LSD analog and a potent 5-HT2A agonist (EC50 of 14.6 nM), capable of stimulating Gq-mediated calcium flux. It exhibits high affinity for most serotonin receptors, α2-adrenergic receptors, and D2-like dopamine receptors.Fórmula:C21H25N3OForma y color:SolidPeso molecular:335.44AC-90179 HCl
CAS:AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Fórmula:C23H31ClN2O2Pureza:99.14%Forma y color:SolidPeso molecular:402.96Ref: TM-T26543
1mg52,00€2mg74,00€5mg96,00€10mg137,00€25mg215,00€50mg391,00€100mg582,00€1mL*10mM (DMSO)127,00€Litoxetine HCl
Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles without antimuscarinic effects.Fórmula:C16H20ClNOPureza:98.98% - 99.19%Forma y color:SoildPeso molecular:277.79Ref: TM-T67956L
1mg97,00€5mg217,00€10mg325,00€25mg557,00€50mg797,00€100mg1.103,00€1mL*10mM (DMSO)208,00€Asenapine Maleate
CAS:Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.Fórmula:C21H20ClNO5Pureza:99.28%Forma y color:SolidPeso molecular:401.84Ref: TM-T1951
5mg35,00€10mg51,00€25mg80,00€50mg96,00€100mg135,00€200mg225,00€500mg373,00€1mL*10mM (DMSO)55,00€RS-127445
CAS:RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.Fórmula:C17H16FN3Pureza:99.32%Forma y color:SolidPeso molecular:281.33AVN-492
CAS:AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Fórmula:C17H21N5O2SPureza:99.81%Forma y color:SolidPeso molecular:359.45Ref: TM-T5179
1mg39,00€2mg49,00€5mg81,00€10mg120,00€25mg236,00€50mg354,00€100mg510,00€1mL*10mM (DMSO)89,00€Befiradol hydrochloride
CAS:Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 aggregation.Fórmula:C20H23Cl2F2N3OPureza:99.1%Forma y color:SolidPeso molecular:430.32Levodropropizine
CAS:Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.Fórmula:C13H20N2O2Pureza:100% - 99.93%Forma y color:White Or Off White Crystalline PowderPeso molecular:236.31R 59-022
CAS:R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.Fórmula:C27H26FN3OSPureza:98.55%Forma y color:SolidPeso molecular:459.58AVN-322
CAS:AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.Fórmula:C17H20ClN5O2SPureza:98.83%Forma y color:SolidPeso molecular:393.89BW 723C86
CAS:BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.Fórmula:C16H19ClN2OSPureza:99.35%Forma y color:SolidPeso molecular:322.85Pardoprunox
CAS:Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Fórmula:C12H15N3O2Pureza:98%Forma y color:SolidPeso molecular:233.27CI 169369
CAS:CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and depression.Fórmula:C19H21ClN2SPureza:100%Forma y color:SoildPeso molecular:344.9Paroxetine hydrochloride
CAS:Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.Fórmula:C19H21ClFNO3Pureza:98% - 99.99%Forma y color:White Crystalline PowderPeso molecular:365.8265-HT2A receptor agonist-5
CAS:5-HT2A receptor agonist-5 (compound I-3) is a potent 5-HT2A agonist with a Ki value of 0.017 µM and exhibits antidepressant activity.Fórmula:C23H29N3OForma y color:SolidPeso molecular:363.5Cannabidiolic acid methyl ester
CAS:Cannabidiolic acid methyl ester (HU-580) is an orally active analogue of cannabidiolic acid. It enhances the activation of 5-HT1A receptors and increases the expression of c-Fos and NeuN in specific hypothalamic nuclei in rats. Cannabidiolic acid methyl ester exhibits anti-nausea, anxiolytic, and anti-nociceptive effects.Fórmula:C23H32O4Forma y color:SolidPeso molecular:372.5Nefazodone hydrochloride
CAS:Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Forma y color:White SolidPeso molecular:506.47Ref: TM-T3275
5mg47,00€10mg70,00€25mg120,00€50mg216,00€100mg325,00€200mg472,00€500mg775,00€1mL*10mM (DMSO)77,00€LY334370
CAS:LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFórmula:C21H22FN3OPureza:99.32%Forma y color:SolidPeso molecular:351.42CJ 033466
CAS:CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.Fórmula:C19H28ClN5OPureza:98.41%Forma y color:SolidPeso molecular:377.91Ref: TM-T22671
1mg48,00€5mg101,00€10mg170,00€25mg270,00€50mg386,00€100mg520,00€1mL*10mM (DMSO)158,00€4-fluoro MBZP
CAS:4-fluoro MBZP is a novel psychoactive substance in the phenylpiperazine class, utilized for studies on the 5-HT2 receptors in the central nervous system.Fórmula:C12H17FN2Forma y color:SolidPeso molecular:208.28Intepirdine
CAS:Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.Fórmula:C19H19N3O2SPureza:98% - 98.63%Forma y color:SolidPeso molecular:353.44Lesopitron HCl
CAS:Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.Fórmula:C15H22Cl2N6Pureza:97.05% - 98.18%Forma y color:SoildPeso molecular:357.28Minesapride
CAS:Minesapride: novel 5-HT4 partial agonist, may treat constipation-predominant IBS.Fórmula:C21H31ClN4O5Pureza:99% - 99.35%Forma y color:SolidPeso molecular:454.95Ref: TM-T28043L
1mg115,00€5mg245,00€10mg363,00€25mg562,00€50mg802,00€100mg1.111,00€200mg1.491,00€1mL*10mM (DMSO)284,00€LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Fórmula:C27H38ClN3OSPureza:98.06%Forma y color:SolidPeso molecular:488.13Methiothepin mesylate
CAS:Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.Fórmula:C21H28N2O3S3Pureza:98% - 99.92%Forma y color:SolidPeso molecular:452.65Pheniramine maleate
CAS:Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.Fórmula:C16H20N2·C4H4O4Pureza:99.85%Forma y color:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CPeso molecular:356.42Tipindole
CAS:Tipindole is a serotonin antagonist utilized in research related to depression.Fórmula:C16H20N2O2SForma y color:SolidPeso molecular:304.41Cerlapirdine
CAS:Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.Fórmula:C22H23N3O3SPureza:98.60%Forma y color:SolidPeso molecular:409.5Ref: TM-T30798
1mg81,00€5mg170,00€10mg274,00€25mg543,00€50mg780,00€100mg1.074,00€1mL*10mM (DMSO)198,00€SEP-363856 hydrochloride
CAS:SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.Fórmula:C9H14ClNOSPureza:99.86% - 99.99%Forma y color:SolidPeso molecular:219.73Ref: TM-T12899L
1mg70,00€2mg92,00€5mg154,00€10mg243,00€25mg425,00€50mg628,00€100mg938,00€500mg1.882,00€1mL*10mM (DMSO)169,00€AAZ-A 154 hydrochloride
CAS:AAZ-A 154 hydrochloride is a selective, competitive, non-hallucinogenic antagonist of 5-HT2AR. It promotes neuronal growth in rodents and results in enduring beneficial behavioral effects.Fórmula:C14H21ClN2OForma y color:SolidPeso molecular:268.78Triazolomethylindole-3-acetic acid
CAS:Triazolomethylindole-3-acetic acid is a metabolite of Rizatriptan, which acts as an agonist for the serotonin (5-HT) receptor subtypes 5-HT1B and 5-HT1D.Fórmula:C13H12N4O2Forma y color:SolidPeso molecular:256.26Cannabigerol
CAS:Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFórmula:C21H32O2Pureza:99.23% - 99.92%Forma y color:SolidPeso molecular:316.48Ref: TM-TN1465
1mg145,00€2mg215,00€5mg314,00€10mg474,00€25mg808,00€50mg1.111,00€100mg1.501,00€1mL*10mM (DMSO)324,00€Serotonin
CAS:Serotonin (5-hydroxytryptamine) is a natural product from animalsFórmula:C10H12N2OPureza:95.94% - 99.92%Forma y color:SolidPeso molecular:176.22Ref: TM-TN2437
1mg78,00€5mg139,00€10mg202,00€25mg360,00€50mg540,00€100mg810,00€500mg1.596,00€1mL*10mM (DMSO)117,00€m-Chlorophenylbiguanide hydrochloride
CAS:m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.Fórmula:C8H11Cl2N5Pureza:99.43% - 99.87%Forma y color:SolidPeso molecular:248.11Viloxazine
CAS:Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activityFórmula:C13H19NO3Pureza:99.8%Forma y color:SolidPeso molecular:237.29Fluoxetine
CAS:Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.Fórmula:C17H18F3NOPureza:99.07% - 99.28%Forma y color:SolidPeso molecular:309.332-Methyl-N,N-dimethyltryptamine
CAS:2-Methyl-N,N-dimethyltryptamine (2,N,N-TMT, compound 15) exhibits binding affinity for the serotonin (5-HT) receptor, with a pA2 value of 6.04. It plays a significant role in neurological disease research.Fórmula:C13H18N2Forma y color:SolidPeso molecular:202.3Bromperidol
CAS:Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.Fórmula:C21H23BrFNO2Pureza:99.89%Forma y color:Tan SolidPeso molecular:420.32Cinitapride
CAS:Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.Fórmula:C21H30N4O4Pureza:98.99%Forma y color:SolidPeso molecular:402.49Ref: TM-T21385
1mg78,00€5mg163,00€10mg253,00€25mg505,00€50mg730,00€100mg1.026,00€1mL*10mM (DMSO)187,00€p-MPPF
CAS:p-MPPF is a 5-HT antagonist that can be used to study neurological diseases.Fórmula:C25H27FN4O2Pureza:99.79%Forma y color:SolidPeso molecular:434.51Mirtazapine
CAS:Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.Fórmula:C17H19N3Pureza:99.98%Forma y color:SolidPeso molecular:265.35PRX933 hydrochloride
CAS:PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.Fórmula:C16H22ClN5O2Pureza:97.99% - 99.72%Forma y color:SolidPeso molecular:351.84Ref: TM-T12565
1mg356,00€5mg568,00€10mg907,00€25mg1.339,00€50mg1.815,00€100mg2.432,00€1mL*10mM (DMSO)652,00€Iprindole
CAS:Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].Fórmula:C19H28N2Pureza:99.06%Forma y color:SolidPeso molecular:284.44Ref: TM-T37015
2mg37,00€5mg52,00€10mg80,00€25mg154,00€50mg266,00€100mg455,00€200mg652,00€1mL*10mM (DMSO)84,00€MDL 100009
CAS:MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.Fórmula:C22H28FNO3Pureza:98.96%Forma y color:SolidPeso molecular:373.46Ref: TM-T22359
1mg148,00€2mg188,00€5mg283,00€10mg424,00€25mg655,00€50mg883,00€100mg1.169,00€200mg1.596,00€1mL*10mM (DMSO)335,00€Tropisetron
CAS:Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.Fórmula:C17H20N2O2Pureza:99.95%Forma y color:White SolidPeso molecular:284.35Flucopride
CAS:Flucopride (Compound 4a) acts as an acetylcholinesterase inhibitor (AChE) with an IC50 value of 24 nM and serves as a partial agonist for the human 5-HT4 receptor (5-HT4R) with a Ki of 9.6 nM for (h)5-HT4R. It promotes non-amyloidogenic processing of APP in COS-7 cells transiently expressing (h)5-HT4R with an EC50 of 23.0 nM. Flucopride is also likely to exhibit significant gastrointestinal tract (GIT) penetration and blood-brain barrier (BBB) permeability, as determined in PAMPA experiments.Fórmula:C22H33FN2O2Forma y color:SolidPeso molecular:376.51GR 46611
CAS:GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.Fórmula:C23H27N3O2Pureza:99.9%Forma y color:SolidPeso molecular:377.48Sertindole
CAS:Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).Fórmula:C24H26ClFN4OPureza:99.74%Forma y color:Off-White To Pale Yellow SolidPeso molecular:440.94Xanthotoxol
CAS:Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.Fórmula:C11H6O4Pureza:99.97%Forma y color:SolidPeso molecular:202.16SKF-83566
CAS:SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.Fórmula:C17H18BrNOPureza:95.00% - 99.82%Forma y color:SolidPeso molecular:332.23Arotinolol
CAS:Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency for inhibiting the binding of the radioligand [125I-ICYP] to [5HT1B-serotonergic] receptor sites. It is an antihypertensive agent.Fórmula:C15H21N3O2S3Forma y color:White SolidPeso molecular:371.54Wf-516
CAS:Wf-516 is a 5-HT reuptake inhibitor (Kis: 5 nM and 40 nM for 5-HT1A receptor and 5-HT2A receptor in humans, respectively), and with potent antidepressantFórmula:C25H25Cl2N3O4Pureza:98%Forma y color:SolidPeso molecular:502.395-HT2C agonist-3
CAS:5-HT2C agonist-3 ((+)-19), a selective 5-HT2C agonist (EC 50: 24 nM, Ki: 78 nM), exhibits antipsychotic-like activity by blocking amphetamine-inducedFórmula:C19H23ClFNO2Pureza:98%Forma y color:SolidPeso molecular:351.84Puerarin
CAS:Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.Fórmula:C21H20O9Pureza:98.90% - 99.21%Forma y color:Yellow Brown Fine PowderPeso molecular:416.38Cilansetron
CAS:Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.Fórmula:C20H21N3OPureza:99.77% - 99.85%Forma y color:SolidPeso molecular:319.4Clothiapine
CAS:Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Fórmula:C18H18ClN3SPureza:99.93%Forma y color:SolidPeso molecular:343.87GSK163090
CAS:GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).Fórmula:C25H29N5OPureza:99.20%Forma y color:SolidPeso molecular:415.53Ref: TM-TQ0311
1mg37,00€2mg52,00€5mg80,00€10mg125,00€25mgA consultar50mgA consultar1mL*10mM (DMSO)87,00€JPC0323
JPC0323 is a dual positive allosteric modulator of the 5-HT2C and 5-HT2A receptors, featuring on-target properties, acceptable plasma exposure, and adequateFórmula:C22H43NO4Pureza:98%Forma y color:SolidPeso molecular:385.585-HT2C agonist-4
CAS:Compound 3i, a 5-HT2C agonist-4, acts as an agonist for the 5-HT2C receptor with an EC50 of 5.7 nM. It is capable of reducing locomotor activity in zebrafish larvae.Fórmula:C24H25N5OForma y color:SolidPeso molecular:399.49Risperidone
CAS:Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.Fórmula:C23H27FN4O2Pureza:99.73%Forma y color:Crystalline SolidPeso molecular:410.48MRS7925
MRS7925 (Compound 43) serves as a potent antagonist of the 5-HT2B receptor, with an inhibition constant (Ki) of 17 nM, and is utilized in the study of fibrosisFórmula:C20H26IN5O3Pureza:98%Forma y color:SolidPeso molecular:511.36Escin IB
CAS:Escin Ib inhibits gastric emptying, at least in part, mediated by capsaicin-sensitive sensory nerves, to stimulate the synthesis and/or release of dopamine, toFórmula:C55H86O24Pureza:99.09% - 99.81%Forma y color:SolidPeso molecular:1131.26Indophagolin
CAS:Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Fórmula:C19H15BrClF3N2O3SPureza:99.76%Forma y color:SolidPeso molecular:523.75Ref: TM-T8946
1mg58,00€5mg111,00€10mg170,00€25mg284,00€50mg393,00€100mg552,00€200mg748,00€1mL*10mM (DMSO)129,00€Pipamperone
CAS:Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.Fórmula:C21H30FN3O2Pureza:99.94%Forma y color:White PowderPeso molecular:375.48Ref: TM-T12480
1mg62,00€2mg85,00€5mg119,00€10mg170,00€25mg283,00€50mg430,00€100mg622,00€1mL*10mM (DMSO)131,00€WAY208466 dihydrochloride
CAS:WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.Fórmula:C17H20Cl2FN3O2SPureza:98.43%Forma y color:SolidPeso molecular:420.33WAY-100635 maleate
CAS:WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Fórmula:C25H34N4O2·xC4H4O4Pureza:100%Forma y color:White SolidPeso molecular:538.645Ref: TM-T3453
2mg46,00€5mg66,00€10mg95,00€25mg159,00€50mg226,00€100mg334,00€500mg807,00€1mL*10mM (DMSO)79,00€5-HT2A receptor agonist-6
CAS:5-HT2A receptor agonist-6 (compound 47) is a selective agonist of the 5-HT2A receptor with a pEC50 value of 6.58.Fórmula:C18H19N3O3Forma y color:SolidPeso molecular:325.36Niaprazine
CAS:Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.Fórmula:C20H25FN4OPureza:99.5%Forma y color:SolidPeso molecular:356.44Ref: TM-T36949
2mg40,00€5mg58,00€10mg96,00€25mg144,00€50mg210,00€100mg309,00€200mg444,00€1mL*10mM (DMSO)64,00€Brexpiprazole
CAS:Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Fórmula:C25H27N3O2SPureza:99.06% - 99.96%Forma y color:SolidPeso molecular:433.57SB 243213
CAS:SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.Fórmula:C22H19F3N4O2Pureza:100% - 100%Forma y color:SolidPeso molecular:428.41Bemesetron
CAS:Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.Fórmula:C15H17Cl2NO2Pureza:97.37%Forma y color:SolidPeso molecular:314.21Prucalopride
CAS:Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.Fórmula:C18H26ClN3O3Pureza:100%Forma y color:SolidPeso molecular:367.87Ro4368554
CAS:Ro4368554 is a selective 5-HT6 antagonist capable of crossing the blood-brain barrier. It can reverse memory deficits caused by scopolamine and tryptophan depletion. Ro4368554 is applicable for research related to memory impairments.Fórmula:C19H21N3O2SForma y color:SolidPeso molecular:355.454lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Fórmula:C31H36FN3O4SPureza:95.83% - 98.57%Forma y color:SolidPeso molecular:565.7F 14679
CAS:F 14679 is a potent 5-HT1A agonist (pKi=10.23) with a maximum Ca2t response similar to 5-HT.Fórmula:C21H25ClF2N4OPureza:99.09%Forma y color:SolidPeso molecular:422.9FFN246
CAS:FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation andFórmula:C15H13FN2OPureza:98%Forma y color:SolidPeso molecular:256.27SB 242084
CAS:SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.Fórmula:C21H19ClN4O2Pureza:99.77% - ≥98%Forma y color:SolidPeso molecular:394.85Ref: TM-T7277
1mg42,00€2mg55,00€5mg90,00€10mg115,00€25mg246,00€50mg472,00€100mg720,00€1mL*10mM (DMSO)89,00€Cisapride
CAS:Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.Fórmula:C23H29ClFN3O4Pureza:99.77%Forma y color:White To Slightly Biege Powder SolidPeso molecular:465.95Ref: TM-T1291
5mg47,00€10mg59,00€25mg77,00€50mg99,00€100mg135,00€200mg235,00€500mg394,00€1mL*10mM (DMSO)55,00€(S)-Bexicaserin
CAS:(S)-Bexcaserin (compound 2) serves as a 5-HT2C receptor agonist, presenting research possibilities in obesity and psychiatric disorders [1].Fórmula:C15H19F2N3OPureza:98%Forma y color:SolidPeso molecular:295.33Frovatriptan succinate hydrate
CAS:Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.Fórmula:C18H25N3O6Pureza:99.95%Forma y color:SolidPeso molecular:379.41Hypidone hydrochloride
CAS:Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitorFórmula:C18H23ClN2O2Pureza:99.82% - 99.93%Forma y color:SolidPeso molecular:334.84Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Fórmula:C23H27Cl2N3O2Pureza:99.43% - 99.62%Forma y color:Colourless Flake Crystalline SolidPeso molecular:448.39Naratriptan
CAS:Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.Fórmula:C17H25N3O2SPureza:99.08%Forma y color:SolidPeso molecular:335.47Metoclopramide hydrochloride
CAS:Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.Fórmula:C14H22ClN3O2·HClPureza:99.99%Forma y color:White To Off-White PowderPeso molecular:336.26Tiflucarbine
CAS:Tiflucarbine is a potential non-selective 5-HT agonist with antidepressant activity.Tiflucarbine dose-dependently increased the specific activity of solubleFórmula:C16H17FN2SPureza:100%Forma y color:SolidPeso molecular:288.38pCPA methyl ester hydrochloride
CAS:pCPA methyl ester HCl inhibits tryptophan hydroxylase, 5-HT synthesis, crosses blood-brain barrier, lowers central 5-HT.Fórmula:C10H13Cl2NO2Pureza:99.08% - 99.88%Forma y color:SolidPeso molecular:250.12Loxapine
CAS:Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.Fórmula:C18H18ClN3OPureza:99.88%Forma y color:Pale Yellowish Crystals From Petroleum Ether SolidPeso molecular:327.815-HT2 agonist-1
CAS:Compound 24, a 5-HT2 agonist-1, selectively activates 5-HT2A, 5-HT2B, and 5-HT2C receptors with IC50 values of 10 nM, 8.3 nM, and 1.6 nM, respectively.Fórmula:C19H23ClN2O2Pureza:98%Forma y color:SolidPeso molecular:346.85Gevotroline
CAS:Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.Fórmula:C19H20FN3Pureza:98.79%Forma y color:SolidPeso molecular:309.385-HT1AR/5-HT6R ligand-1
5-HT1AR/5-HT6R ligand-1 (Compound PP13) functions as a ligand for the 5-HT receptor, demonstrating high affinity for 5-HT1AR, 5-HT6R, and 5-HT7R with Ki values of 19, 69, and 198 nM, respectively. In HEK293 cells, it inhibits cAMP production with EC50 values of 1535, 488, and 53 nM for these receptors. Additionally, 5-HT1AR/5-HT6R ligand-1 exhibits antiproliferative effects on several cancer cell lines, including 1321N1, U87MG, MCF7, and AsPC-1, with IC50 values of 9.6, 13.6, 19.3, and 14.6 μM, respectively. The compound also shows antagonistic activity towards the dopamine receptor D2R, with a Ki of 1903 nM.Fórmula:C25H29ClN4O2SForma y color:SolidPeso molecular:485.04GTS-21 dihydrochloride
CAS:GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by the binding of the neurotransmitter ACh.Fórmula:C19H20N2O2·2HClPureza:100% - 99.62%Forma y color:SolidPeso molecular:381.3Ref: TM-T2663
5mg51,00€10mg85,00€25mg115,00€50mg144,00€100mg216,00€200mg325,00€500mg545,00€1mL*10mM (DMSO)57,00€4-Iodoamphetamine hydrochloride
CAS:4-Iodoamphetamine (p-Iodoamphetamine) hydrochloride is a halogenated phenethylamine characterized by the presence of an iodine atom at the para position of the phenyl group. It selectively induces serotonin release and inhibits reuptake in rat brain synaptosomes.Fórmula:C9H13ClINForma y color:SolidPeso molecular:297.56Citalopram hydrobromide
CAS:Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, therebyFórmula:C20H22BrFN2OPureza:99.81%Forma y color:White Crystalline PowderPeso molecular:405.304SB 204741
CAS:SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.Fórmula:C14H14N4OSPureza:99.83%Forma y color:SolidPeso molecular:286.35Eletriptan hydrobromide
CAS:Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D receptor.Fórmula:C22H27BrN2O2SPureza:100% - 99.69%Forma y color:Tan SolidPeso molecular:463.43Ref: TM-T0216
2mg39,00€5mg57,00€10mg70,00€25mg134,00€50mg230,00€100mg373,00€200mg555,00€1mL*10mM (DMSO)63,00€Cinitapride Hydrogen Tartrate
CAS:Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptorsFórmula:C25H36N4O10Pureza:98%Forma y color:SolidPeso molecular:552.5812-Methyl-5-HT maleate
CAS:2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.Fórmula:C15H18N2O5Pureza:98%Forma y color:SolidPeso molecular:306.31WAY-607695
CAS:WAY-607695 is a potential 5-HT1A receptor agonist.Fórmula:C13H12FNO2Pureza:99.82%Forma y color:SolidPeso molecular:233.24Rotigotine Hydrochloride
CAS:Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.Fórmula:C19H26ClNOSPureza:99.53% - 99.56%Forma y color:Almost White To White Crystalline PowderPeso molecular:351.93D3/5-HT receptor modulator-1
CAS:D3/5-HT receptor modulator-1 (compound 5i) is a selective antagonist of the dopamine D3 and 5-HT2A receptors, and a partial agonist at the 5-HT1A receptor. It exhibits Ki values of 4.5 nM, 11.9 nM, and 15.3 nM for the dopamine D3, 5-HT2A, and 5-HT1A receptors respectively. The compound shows lower affinity for the dopamine D2 receptor, 5-HT2C receptor, and hERG channel. D3/5-HT receptor modulator-1 possesses atypical antipsychotic properties.Fórmula:C24H29N3O2Forma y color:SolidPeso molecular:391.506
