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GluR

GluR

Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.

Productos de "GluR"

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productos por página.Hay 147 productos en esta categoría.
  • 3-MATIDA

    CAS:
    3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).
    Fórmula:C8H9NO4S
    Pureza:98.41% - 99.05%
    Forma y color:Solid
    Peso molecular:215.23

    Ref: TM-T3486

    2mg
    35,00€
    5mg
    51,00€
    10mg
    84,00€
    25mg
    154,00€
    50mg
    240,00€
    100mg
    359,00€
    200mg
    510,00€
  • KRP-199 sodium


    KRP-199 sodium sodium is highly potent and selective for AMPA-R in vitro and exhibits good neuroprotection in vivo.
    Fórmula:C22H12F3N5Na2O7
    Pureza:96.85%
    Forma y color:Soild
    Peso molecular:561.33

    Ref: TM-T27748L

    1mg
    185,00€
    5mg
    459,00€
    10mg
    657,00€
    25mg
    1.026,00€
    50mg
    1.415,00€
    100mg
    1.872,00€
    500mg
    3.734,00€
  • LY3020371 hydrochloride

    CAS:
    LY3020371 HCl: potent mGlu2/3 antagonist, antidepressant-like; Ki: 5.3/2.5 nM, IC50: 16.2 nM for cAMP inhibition.
    Fórmula:C15H16ClF2NO5S
    Forma y color:Solid
    Peso molecular:395.81

    Ref: TM-T11911

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • JNJ-46778212

    CAS:
    JNJ-46778212 (VU 0409551) is a selective and potent mGlu5 allosteric modulator (EC50: 260 nM) for the study of neurodissection.
    Fórmula:C20H17FN2O3
    Pureza:99.24%
    Forma y color:Solid
    Peso molecular:352.36

    Ref: TM-T15619

    5mg
    62,00€
    10mg
    97,00€
    25mg
    202,00€
    50mg
    344,00€
    100mg
    552,00€
    1mL*10mM (DMSO)
    67,00€
  • A-794282

    CAS:
    A-794282 is a selective antagonist of mGluR1.
    Fórmula:C19H18N4OS
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:350.44

    Ref: TM-T26486

    1mg
    279,00€
    2mg
    414,00€
    5mg
    685,00€
    10mg
    938,00€
    25mg
    1.444,00€
    50mg
    1.882,00€
  • GET73

    CAS:
    GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.
    Fórmula:C13H16F3NO2
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:275.27

    Ref: TM-T11393

    1mg
    65,00€
    5mg
    131,00€
    10mg
    202,00€
    25mg
    340,00€
    50mg
    452,00€
    100mg
    638,00€
    200mg
    842,00€
    1mL*10mM (DMSO)
    177,00€
  • γ-DGG

    CAS:
    gamma-DGG is a competitive blocker of AMPA receptor.
    Fórmula:C7H12N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:204.18

    Ref: TM-T15369

    5mg
    47,00€
    10mg
    60,00€
  • VU0483605

    CAS:
    VU0483605 is an effective and selective positive allosteric modulator of mGluR1 with EC50s of 390 and 356 nM for human and rat, respectively.
    Fórmula:C20H10Cl3N3O3
    Pureza:97.03%
    Forma y color:Solid
    Peso molecular:446.67

    Ref: TM-T21747

    2mg
    42,00€
    5mg
    64,00€
    10mg
    97,00€
    25mg
    183,00€
    50mg
    284,00€
    100mg
    425,00€
    200mg
    562,00€
    1mL*10mM (DMSO)
    78,00€
  • E4CPG

    CAS:
    E4CPG is a novel group I/II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG.
    Fórmula:C11H13NO4
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:223.23

    Ref: TM-T3477

    2mg
    35,00€
    5mg
    52,00€
    10mg
    70,00€
    25mg
    144,00€
    50mg
    250,00€
    100mg
    376,00€
  • L-AP4

    CAS:
    L-APB is an effective and specific agonist for the group III mGluRs (EC50s: 0.13, 0.29, 1.0, 249 μM for mGlu4, mGlu8, mGlu6, and mGlu7 receptors, respectively).
    Fórmula:C4H10NO5P
    Pureza:98%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:183.1

    Ref: TM-T15692

    1mg
    A consultar
    5mg
    A consultar
    10mg
    A consultar
    50mg
    A consultar
  • LY-2300559

    CAS:
    LY-2300559 is an agonist of metabotropic glutamate receptor 2 (mGluR2) and can be used in studies about the treatment of migraine.
    Fórmula:C26H26O6
    Pureza:100%
    Forma y color:Solid
    Peso molecular:434.48

    Ref: TM-T27932

    1mg
    333,00€
    5mg
    787,00€
    10mg
    1.074,00€
    25mg
    1.510,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
    500mg
    4.655,00€
  • (S)-MCPG

    CAS:
    (S)-MCPG is the active isomer of (RS)-MCPG, non-selective group I/group II metabotropic glutamate receptor antagonist.
    Fórmula:C10H11NO4
    Pureza:98.72%
    Forma y color:Solid
    Peso molecular:209.20

    Ref: TM-T13452

    1mg
    35,00€
    5mg
    A consultar
  • VU 0357121

    CAS:
    VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly antagonizing at other mGlu receptor subtypes.
    Fórmula:C17H17F2NO2
    Pureza:99% - 99.99%
    Forma y color:Solid
    Peso molecular:305.32

    Ref: TM-T6725

    2mg
    42,00€
    5mg
    59,00€
    10mg
    95,00€
    25mg
    175,00€
    50mg
    281,00€
    100mg
    439,00€
    1mL*10mM (DMSO)
    59,00€
  • Fenobam

    CAS:
    Fenobam shows inverse agonist activity which blocks the mGlu5 receptor basal activity(IC50: 84 nM).
    Fórmula:C11H11ClN4O2
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:266.68

    Ref: TM-T15275

    1mg
    35,00€
    5mg
    64,00€
    10mg
    101,00€
    25mg
    170,00€
    50mg
    248,00€
    100mg
    359,00€
    200mg
    497,00€
    1mL*10mM (DMSO)
    96,00€
  • DNQX

    CAS:
    DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)
    Fórmula:C8H4N4O6
    Pureza:97.15% - 99.10%
    Forma y color:Off-White Powder With A Yellow Tinge
    Peso molecular:252.14

    Ref: TM-T7304

    25mg
    56,00€
    50mg
    89,00€
    100mg
    115,00€
    1mL*10mM (DMSO)
    55,00€
  • JNJ-40411813

    CAS:
    JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).
    Fórmula:C20H25ClN2O
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:344.88

    Ref: TM-TQ0094

    1mg
    55,00€
    5mg
    117,00€
    10mg
    183,00€
    25mg
    306,00€
    50mg
    437,00€
    100mg
    562,00€
    200mg
    743,00€
    1mL*10mM (DMSO)
    131,00€
  • S 18986

    CAS:
    S 18986 is a selective, orally active, brain penetrant positive allosteric modulator of AMPA-type receptors, showcasing cognitive-enhancing properties in
    Fórmula:C10H12N2O2S
    Pureza:99.25%
    Forma y color:Solid
    Peso molecular:224.28

    Ref: TM-T16816

    1mg
    35,00€
    5mg
    64,00€
    10mg
    97,00€
    25mg
    A consultar
    50mg
    A consultar
  • 1H-Pyrrolo[2,1-c][1,2,4]benzothiadiazine, 2,3,3a,4-tetrahydro-, 5,5-dioxide, (3aR)-

    CAS:
    1H-Pyrrolo[2,1-c][1,2,4]benzothiadiazine, 2,3,3a,4-tetrahydro-, 5,5-dioxide, (3aR)- is a low activity isomer of S 18986.
    Fórmula:C10H12N2O2S
    Pureza:99.69%
    Forma y color:Soild
    Peso molecular:224.28

    Ref: TM-T60224

    1mg
    77,00€
    5mg
    158,00€
    10mg
    225,00€
    25mg
    338,00€
    50mg
    475,00€
    1mL*10mM (DMSO)
    137,00€
  • VU0155041

    CAS:
    VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).
    Fórmula:C14H15Cl2NO3
    Pureza:99.52% - 99.56%
    Forma y color:Solid
    Peso molecular:316.18

    Ref: TM-T3565

    2mg
    40,00€
    5mg
    58,00€
    10mg
    85,00€
    25mg
    145,00€
    50mg
    188,00€
    100mg
    301,00€
    200mg
    435,00€
    1mL*10mM (DMSO)
    64,00€
  • (S)-ATPO

    CAS:
    (S)-ATPO is Competitive antagonist at GluR1-4 (AMPA-preferring) receptors.
    Fórmula:C11H19N2O7P
    Pureza:98.37% - 99.41%
    Forma y color:Solid
    Peso molecular:322.25

    Ref: TM-T3473

    1mg
    52,00€
    2mg
    74,00€
    5mg
    97,00€
    10mg
    157,00€
    25mg
    285,00€
    50mg
    447,00€
    100mg
    653,00€