Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Productos de "Receptor de histamina"
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ROS 234 dioxalate
CAS:ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)Fórmula:C17H19N5O8Pureza:98%Forma y color:SolidPeso molecular:421.37Bavisant
CAS:Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.Fórmula:C19H27N3O2Pureza:96.06% - 98%Forma y color:SolidPeso molecular:329.44Ref: TM-TQ0046
1mg43,00€5mg96,00€10mg134,00€25mg221,00€50mg325,00€100mg465,00€500mgA consultar1mL*10mM (DMSO)94,00€(±)-Tazifylline
CAS:(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Fórmula:C23H32N6O3SPureza:98.97%Forma y color:SolidPeso molecular:472.6Ref: TM-T10000
1mg148,00€5mg284,00€10mg411,00€25mg645,00€50mg867,00€100mg1.121,00€1mL*10mM (DMSO)369,00€BMY 25368 HCl
CAS:BMY 25368 HCl is a competitive histamine H2 receptor antagonist that antagonizes gastric secretion stimulated by pentagastrin, ethacrynic choline, and food.Fórmula:C19H26ClN3O3Pureza:98.73% - 99.81%Forma y color:SoildPeso molecular:379.88Lodoxamide tromethamine
CAS:Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergicFórmula:C19H28ClN5O12Pureza:99.58%Forma y color:SolidPeso molecular:553.91Mifentidine
CAS:Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.Fórmula:C13H16N4Pureza:100% - 99.20%Forma y color:SolidPeso molecular:228.29Clemastine fumarate
CAS:Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.Fórmula:C25H30ClNO5Pureza:99.52% - 99.8%Forma y color:Colorless To Faintly Yellow Crystalline Powder Appearance White Or Almost White Crystalline PowderPeso molecular:459.97Fexofenadine
CAS:Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Fórmula:C32H39NO4Pureza:99.87%Forma y color:White To Off-White SolidPeso molecular:501.66Ref: TM-T21390
10mg50,00€25mg71,00€50mg97,00€100mg145,00€200mg212,00€500mg373,00€1mL*10mM (DMSO)58,00€NP10679
CAS:NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, hERG channels, and CYPase.Fórmula:C23H26F3N3O3Pureza:99.43%Forma y color:SolidPeso molecular:449.47Carebastine
CAS:Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.Fórmula:C32H37NO4Pureza:99.16%Forma y color:Off-White SolidPeso molecular:499.64Lavoltidine
CAS:Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.Fórmula:C19H29N5O2Pureza:100% - 100%Forma y color:SolidPeso molecular:359.47Azelastine
CAS:Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.Fórmula:C22H24ClN3OPureza:99.35%Forma y color:White Crystal PowderPeso molecular:381.9Benztropine mesylate
CAS:Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSONFórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Forma y color:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53Levodropropizine
CAS:Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.Fórmula:C13H20N2O2Pureza:100% - 99.93%Forma y color:White Or Off White Crystalline PowderPeso molecular:236.31Diphenhydramine
CAS:Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.Fórmula:C17H21NOPureza:99.49%Forma y color:SolidPeso molecular:255.35Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Fórmula:C18H18ClNS·HClPureza:99.16%Forma y color:White PowderPeso molecular:352.322-Pyridylethylamine dihydrochloride
CAS:2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Fórmula:C7H12Cl2N2Pureza:99.42%Forma y color:SolidPeso molecular:195.09Thioperamide maleate
CAS:Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Fórmula:C19H28N4O4SPureza:99.88%Forma y color:SolidPeso molecular:408.52ReN-1869
CAS:ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseasesFórmula:C24H27NO2Pureza:99.87% - 99.89%Forma y color:SolidPeso molecular:361.48Pheniramine maleate
CAS:Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.Fórmula:C16H20N2·C4H4O4Pureza:99.85%Forma y color:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CPeso molecular:356.42
