Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Productos de "Receptor de histamina"
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H4R antagonist 3
CAS:H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study ofFórmula:C19H21ClN4SPureza:98%Forma y color:SolidPeso molecular:372.92Perphenazine
CAS:Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.Fórmula:C21H26ClN3OSPureza:99.3% - 99.72%Forma y color:SolidPeso molecular:403.97S 38093
CAS:S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).Fórmula:C17H24N2O2Pureza:99.95%Forma y color:SolidPeso molecular:288.38Ref: TM-T4099
2mg38,00€5mg52,00€10mg80,00€25mg131,00€50mg210,00€100mg334,00€200mg467,00€1mL*10mM (DMSO)52,00€Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Fórmula:C18H18ClNOSPureza:99.78%Forma y color:SolidPeso molecular:331.86Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Fórmula:C18H21ClN2Pureza:98% - 98.75%Forma y color:SolidPeso molecular:300.83Meclizine dihydrochloride
CAS:Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiationFórmula:C25H27ClN2·2HClPureza:98.05% - 99.79%Forma y color:White Slightly Yellowish Crystalline PowderPeso molecular:463.87Dothiepin
CAS:Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancingFórmula:C19H21NSPureza:98%Forma y color:SolidPeso molecular:295.44Pimethixene
CAS:Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Fórmula:C19H19NSPureza:97.50%Forma y color:SolidPeso molecular:293.43Ref: TM-T12489
2mg34,00€5mg50,00€10mg65,00€25mg106,00€50mg158,00€100mg226,00€200mg339,00€1mL*10mM (DMSO)52,00€Tecastemizole
CAS:Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.Fórmula:C19H21FN4Pureza:99.66%Forma y color:SolidPeso molecular:324.4Ref: TM-T26253
1mg57,00€5mg125,00€10mg177,00€25mg304,00€50mg437,00€100mg615,00€500mg1.225,00€1mL*10mM (DMSO)138,00€Bamirastine
CAS:Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect onFórmula:C31H37N5O3Pureza:96.68%Forma y color:SolidPeso molecular:527.66Dimenhydrinate
CAS:Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.Fórmula:C24H28ClN5O3Pureza:99.57% - 99.77%Forma y color:Crystals Physical Description Crystalline White Powder (Ntp 1992)Peso molecular:469.96Mianserin hydrochloride
CAS:Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.Fórmula:C18H21ClN2Pureza:99.63% - 99.82%Forma y color:White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedPeso molecular:300.83Betahistine mesylate
CAS:Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks with asthma/ulcers.Fórmula:C8H12N2·2(CH4O3S)Pureza:98%Forma y color:CoaPeso molecular:328.4Impromidine hydrochloride
CAS:Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.Fórmula:C14H26Cl3N7SPureza:99.50%Forma y color:SolidPeso molecular:430.83Triprolidine hydrochloride monohydrate
CAS:Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.Fórmula:C19H25ClN2OPureza:99.68% - 99.81%Forma y color:White Crystalline PowderPeso molecular:332.87Ketotifen fumarate
CAS:Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.Fórmula:C23H23NO5SPureza:99.25% - 99.73%Forma y color:SolidPeso molecular:425.5Niaprazine
CAS:Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.Fórmula:C20H25FN4OPureza:99.5%Forma y color:SolidPeso molecular:356.44Ref: TM-T36949
2mg40,00€5mg58,00€10mg96,00€25mg144,00€50mg210,00€100mg309,00€200mg444,00€1mL*10mM (DMSO)64,00€Histamine Phosphate
CAS:Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.Fórmula:C5H9N·2H3O4PPureza:100%Forma y color:White Crystal PowderPeso molecular:307.14Nizatidine
CAS:Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.Fórmula:C12H21N5O2S2Pureza:99.43% - 99.87%Forma y color:White To Off-White Crystalline PowderPeso molecular:331.46Mequitazine
CAS:Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Fórmula:C20H22N2SPureza:99.98%Forma y color:SolidPeso molecular:322.47
