Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Productos de "Receptor de histamina"
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GSK189254A
CAS:GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).Fórmula:C21H25N3O2Pureza:98.04% - 98.71%Forma y color:SolidPeso molecular:351.44Dioxopromethazine hydrochloride
CAS:Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.Fórmula:C17H20N2O2S·HClPureza:99.58%Forma y color:SolidPeso molecular:352.88Decloxizine dihydrochloride
CAS:Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.Fórmula:C21H28N2O2·2ClHPureza:99.73%Forma y color:SolidPeso molecular:413.39Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Fórmula:C19H29ClN2O4Pureza:99.49%Forma y color:SolidPeso molecular:384.9Rupatadine Fumarate
CAS:Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM.Fórmula:C26H26ClN3·C4H4O4Pureza:99.86%Forma y color:White Or Almost-White PowderPeso molecular:532.03Mebhydrolin napadisylate
CAS:Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergicFórmula:C19H20N2C10H8O6S2Pureza:99.35% - 99.77%Forma y color:White Or Almost White CrystallinePeso molecular:420.52Tesmilifene fumarate
CAS:Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。Fórmula:C23H29NO5Pureza:99.86%Forma y color:SolidPeso molecular:399.48Ref: TM-T22746
5mg47,00€10mg64,00€25mg116,00€50mg167,00€100mg249,00€200mg369,00€1mL*10mM (DMSO)52,00€Desloratadine
CAS:Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties.Fórmula:C19H19ClN2Pureza:100% - 99.79%Forma y color:SolidPeso molecular:310.82Oxmetidine FA
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.Fórmula:C20H23N5O5SPureza:97.34%Forma y color:SoildPeso molecular:445.49S 38093 HCl
CAS:S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.Fórmula:C17H25ClN2O2Pureza:97.91%Forma y color:SolidPeso molecular:324.85Ref: TM-T4087
1mg51,00€2mg71,00€5mg97,00€10mg138,00€25mg239,00€50mg341,00€100mg487,00€200mg658,00€1mL*10mM (DMSO)97,00€Osthole
CAS:Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.Fórmula:C15H16O3Pureza:99.93% - 99.96%Forma y color:Fine White PowderPeso molecular:244.29Toreforant
CAS:Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).Fórmula:C23H32N6Pureza:98%Forma y color:SolidPeso molecular:392.54Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Fórmula:C27H25F2N3OSPureza:99.45% - 99.89%Forma y color:SolidPeso molecular:477.574-Methylhistamine
CAS:4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer andFórmula:C6H11N3Pureza:98%Forma y color:SolidPeso molecular:125.17Fenclozine Maleate
CAS:Fenclozine Maleate (S 1429) is a potential histamine H1 receptor antagonist , which can be used to study fever, inflammation and pain.Fórmula:C45H47ClN2O12Pureza:98.47%Forma y color:SoildPeso molecular:843.314Astemizole
CAS:Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.Fórmula:C28H31FN4OPureza:98.24% - 99.67%Forma y color:White Crystals SolidPeso molecular:458.57Alcaftadine
CAS:Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.Fórmula:C19H21N3OPureza:98% - 99.99%Forma y color:SolidPeso molecular:307.39Betazole dihydrochloride
CAS:Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.Fórmula:C5H11Cl2N3Pureza:99.12%Forma y color:SolidPeso molecular:184.067Ref: TM-T8599
1mg35,00€5mg60,00€10mg96,00€25mg170,00€50mg306,00€100mg399,00€200mg568,00€1mL*10mM (DMSO)60,00€PF-03654764
CAS:PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.Fórmula:C20H28F2N2OPureza:100%Forma y color:SolidPeso molecular:350.45Immethridine dihydrobromide
CAS:Immethridine dihydrobromide is a histamine H3 receptor agonist.Fórmula:C9H11Br2N3Pureza:97.49% - 98.16%Forma y color:SolidPeso molecular:321.01
