Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Productos de "Receptor de histamina"
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Adriforant
CAS:Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.Fórmula:C13H22N6Pureza:99.84%Forma y color:SolidPeso molecular:262.35KP136
CAS:KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).Fórmula:C16H18N4O3Pureza:98.16% - 99.86%Forma y color:SolidPeso molecular:314.34Oxmetidine
CAS:Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.Fórmula:C19H21N5O3SPureza:99.67%Forma y color:SolidPeso molecular:399.47Ref: TM-T68122
1mg378,00€5mg895,00€10mg1.216,00€25mg1.786,00€50mg2.442,00€100mg3.287,00€500mg6.603,00€Histamine
CAS:Histamine (Ergamine) is an amine derived by enzymatic decarboxylation of HISTIDINE.Fórmula:C5H9N3Pureza:100% - 96.63%Forma y color:Needles From Chloroform SolidPeso molecular:111.15Terfenadine
CAS:Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Fórmula:C32H41NO2Pureza:98.76% - 99.75%Forma y color:SolidPeso molecular:471.67WZ4141
CAS:WZ4141 is an intermediate in compound synthesis.Fórmula:C16H13N3O2Pureza:98%Forma y color:SolidPeso molecular:279.29MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.Fórmula:C24H26F3N3O4Pureza:100%Forma y color:SolidPeso molecular:477.48Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Fórmula:C17H20N4OPureza:100% - 100%Forma y color:SoildPeso molecular:296.37Hydroxyzine
CAS:Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.Fórmula:C21H27ClN2O2Pureza:99.54% - ≥95%Forma y color:Oil SolidPeso molecular:374.9JNJ 10191584 maleate
CAS:JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM).Fórmula:C17H19ClN4O5Pureza:99.82%Forma y color:SolidPeso molecular:394.81Nα-Methylhistamine FA
Nα-Methylhistamine FA is a histamine H3 receptor agonistFórmula:C7H13N3O2Pureza:100%Forma y color:SolidPeso molecular:171.2Amitriptyline hydrochloride
CAS:Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptiveFórmula:C20H24ClNPureza:97% - 99.94%Forma y color:Crystals White To Off-White PowderPeso molecular:313.86Donetidine
CAS:Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Fórmula:C20H25N5O3SPureza:99.12%Forma y color:SolidPeso molecular:415.51Mepyramine maleate
CAS:Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.Fórmula:C21H27N3O5Pureza:99.51% - 99.7%Forma y color:White Crystalline PowderPeso molecular:401.47Abt-288
CAS:ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.Fórmula:C23H24N4OPureza:98% - 98.84%Forma y color:SolidPeso molecular:372.46Levocetirizine
CAS:Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.Fórmula:C21H25ClN2O3Pureza:98% - 99.9%Forma y color:White PowderPeso molecular:388.89Cetirizine Impurity B dihydrochloride
CAS:Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.Fórmula:C19H23Cl3N2O2Pureza:99.24%Forma y color:SolidPeso molecular:417.76BMY-25271
CAS:BMY-25271 is an antagonist of histamine H2 receptor.Fórmula:C12H19N5O2S2Pureza:98%Forma y color:SolidPeso molecular:329.44Iodophenpropit dihydrobromide
CAS:Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).Fórmula:C15H20BrIN4SPureza:98%Forma y color:SolidPeso molecular:495.22Pitolisant hydrochloride
CAS:Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).Fórmula:C17H27Cl2NOPureza:99.26% - 99.72%Forma y color:SolidPeso molecular:332.31Ref: TM-T7176
5mg50,00€10mg74,00€25mg124,00€50mg197,00€100mg311,00€200mg467,00€500mg747,00€1mL*10mM (DMSO)52,00€
