Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Productos de "Receptor de histamina"
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Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Fórmula:C19H21N3OPureza:99.30% - 99.37%Forma y color:SolidPeso molecular:307.39Doxepin hydrochloride
CAS:Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.Fórmula:C19H22ClNOPureza:99.57% - 99.91%Forma y color:White To Off-White PowderPeso molecular:315.837Psoralenoside
CAS:Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.Fórmula:C17H18O9Pureza:99.03% - 99.49%Forma y color:SolidPeso molecular:366.32Ref: TM-TN1008
1mg119,00€5mg283,00€10mg418,00€25mg687,00€50mg938,00€100mg1.264,00€1mL*10mM (DMSO)319,00€Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFórmula:C28H33ClN2·2HClPureza:98.05%Forma y color:Off-White PowderPeso molecular:505.95JNJ-5207852 dihydrochloride
CAS:JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptorFórmula:C20H34Cl2N2OPureza:99.51%Forma y color:SolidPeso molecular:389.4JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Fórmula:C20H32N2OPureza:97.19%Forma y color:SolidPeso molecular:316.48FRG8701
CAS:FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.Fórmula:C22H30N2O4SPureza:98%Forma y color:SolidPeso molecular:418.55H3R antagonist 1
CAS:H3R-IN-1 is an effective inverse agonist of the histamine receptor 3 (H3R).Fórmula:C19H23N3O3Forma y color:SolidPeso molecular:341.4Clemastine
CAS:Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.Fórmula:C21H26ClNOPureza:99.83%Forma y color:SolidPeso molecular:343.89Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Fórmula:C21H27Cl3N2O3Pureza:99.4% - 99.97%Forma y color:SolidPeso molecular:461.81Ranitidine Hydrochloride
CAS:Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.Fórmula:C13H23ClN4O3SPureza:99.30% - 99.49%Forma y color:SolidPeso molecular:350.86Ebastine
CAS:Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.Fórmula:C32H39NO2Pureza:100% - 99.93%Forma y color:White To Off-White PowderPeso molecular:469.66Azacyclonol
CAS:Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.Fórmula:C18H21NOPureza:99.46%Forma y color:Solid PowderPeso molecular:267.37Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Fórmula:C21H24ClNOPureza:100% - 99.77%Forma y color:White To Slightly Yellowish Crystalline SolidPeso molecular:341.88Alginic acid
CAS:Alginic acid, a polysaccharide from brown seaweed, has anti-anaphylactic and anti-inflammatory properties and is used in food industry.Fórmula:C14H22O13Pureza:≥98%Forma y color:SolidPeso molecular:398.317Fexofenadine hydrochloride
CAS:Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, withFórmula:C32H40ClNO4Pureza:100%Forma y color:White Crystalline PowderPeso molecular:538.12ReN-1869 hydrochloride
CAS:ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.Fórmula:C24H28ClNO2Pureza:98%Forma y color:SolidPeso molecular:397.94Azatadine dimaleate
CAS:Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).Fórmula:C28H30N2O8Pureza:100% - 99.70%Forma y color:PowderPeso molecular:522.55LML134
CAS:LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).Fórmula:C19H29N5O3Pureza:99.36%Forma y color:SolidPeso molecular:375.47Ref: TM-T8514
1mg52,00€5mg105,00€10mg170,00€25mg306,00€50mg452,00€100mg672,00€200mg905,00€1mL*10mM (DMSO)117,00€SUN 1334H
CAS:SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).Fórmula:C23H28Cl2F2N2O3Pureza:98%Forma y color:SolidPeso molecular:489.38
