Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Productos de "Receptor de histamina"
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PF-03654746
CAS:PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.Fórmula:C18H24F2N2OPureza:98.83% - 99.1%Forma y color:SolidPeso molecular:322.39HTMT dimaleate
CAS:HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Fórmula:C27H33F3N4O9Pureza:98.51%Forma y color:SolidPeso molecular:614.57VUF10460
CAS:VUF10460 is a non-imidazole histamine H4 receptor agonist.Fórmula:C15H19N5Pureza:99.44% - 99.57%Forma y color:SolidPeso molecular:269.34Antazoline hydrochloride
CAS:Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenousFórmula:C17H19N3·HClPureza:98% - 99.53%Forma y color:White Or Almost White Crystalline PowderPeso molecular:301.82Imetit dihydrobromide
CAS:Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in triggering a shape change in eosinophils (EC50: 25 nM).Fórmula:C6H12Br2N4SPureza:98%Forma y color:SolidPeso molecular:332.06Betahistine dihydrochloride
CAS:Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.Fórmula:C8H14Cl2N2Pureza:99.34% - 99.88%Forma y color:White To Light Yellow Crystalline PowderPeso molecular:209.12Diphenhydramine hydrochloride
CAS:DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.Fórmula:C17H22ClNOPureza:99.84%Forma y color:Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)Peso molecular:291.82H4 Receptor antagonist 1
CAS:H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Fórmula:C16H17ClN4OPureza:98.81%Forma y color:SolidPeso molecular:316.79Ref: TM-T5829
2mg46,00€5mg66,00€10mg92,00€25mg177,00€50mg305,00€100mg439,00€500mg938,00€1mL*10mM (DMSO)73,00€Ciproxifan
CAS:Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).Fórmula:C16H18N2O2Pureza:98.00%Forma y color:SolidPeso molecular:270.33KSK94
CAS:KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.Fórmula:C25H26N4OPureza:99.56%Forma y color:SolidPeso molecular:398.5Famotidine
CAS:Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.Fórmula:C8H15N7O2S3Pureza:98.93% - 99.75%Forma y color:White To Off-White Crystalline PowderPeso molecular:337.45Enerisant
CAS:Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.Fórmula:C22H30N4O3Pureza:99.7%Forma y color:SoildPeso molecular:398.50Ref: TM-T67828
1mg86,00€5mg180,00€10mg296,00€25mg627,00€50mg810,00€100mg1.140,00€200mg1.510,00€1mL*10mM (DMSO)188,00€Clemizole
CAS:Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.Fórmula:C19H20ClN3Pureza:98% - 99.15%Forma y color:SolidPeso molecular:325.84Ref: TM-T1822
1mg44,00€5mg87,00€10mg106,00€25mg160,00€50mg270,00€100mg487,00€500mg1.026,00€1mL*10mM (DMSO)87,00€Betahistine EP Impurity C
CAS:Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Fórmula:C15H19N3Pureza:≥95%Forma y color:SolidPeso molecular:241.33H3R-IN-1 Hydrochloride
CAS:H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .Fórmula:C19H24ClN3O3Pureza:98%Forma y color:SolidPeso molecular:377.86Nedocromil
CAS:Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).Fórmula:C19H17NO7Pureza:95.00%Forma y color:SolidPeso molecular:371.34Meclizine
CAS:Meclizine, also known as Meclozine, is a piperazine class H1 antagonist with antihistamine properties that inhibits the interaction of histamine at H1 receptorsFórmula:C25H27ClN2Pureza:95.16%Forma y color:SolidPeso molecular:390.95Brompheniramine maleate
CAS:Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.Fórmula:C16H19BrN2·C4H4O4Pureza:99.80%Forma y color:Crystal PowderPeso molecular:435.31Chlorpheniramine maleate
CAS:Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.Fórmula:C20H23ClN2O4Pureza:99.64% - 99.98%Forma y color:Odorless White Crystalline Solid Or White Powder With A Bitter TastePeso molecular:390.87Cinnarizine
CAS:Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.Fórmula:C26H28N2Pureza:99.94%Forma y color:SolidPeso molecular:368.51
