Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Productos de "Receptor de histamina"
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Samelisant
CAS:Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.Fórmula:C21H31N3O3Pureza:99.09%Forma y color:SolidPeso molecular:373.49Ref: TM-T9770
1mg111,00€2mg166,00€5mg274,00€10mg439,00€25mg725,00€50mg1.017,00€100mg1.359,00€500mg2.745,00€1mL*10mM (DMSO)283,00€Fexofenadine-d6
CAS:Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.Fórmula:C32H39NO4Pureza:98%Forma y color:SolidPeso molecular:507.69Dimaprit dihydrochloride
CAS:Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Fórmula:C6H15N3S·2HClPureza:99.79%Forma y color:SolidPeso molecular:234.19Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Fórmula:C18H18ClNSPureza:98.77% - 99.69%Forma y color:Pale Yellow Crystals SolidPeso molecular:315.86Bepotastine
CAS:Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.Fórmula:C21H25ClN2O3Pureza:99.96%Forma y color:SolidPeso molecular:388.89Ref: TM-T7893
2mg39,00€5mg57,00€10mg87,00€25mg156,00€50mg230,00€100mg344,00€200mg512,00€1mL*10mM (DMSO)63,00€Conessine
CAS:Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.Fórmula:C24H40N2Pureza:99.65%Forma y color:SolidPeso molecular:356.59Mizolastine
CAS:Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.Fórmula:C24H25FN6OPureza:98% - 99.75%Forma y color:SolidPeso molecular:432.49Antazoline
CAS:Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Fórmula:C17H19N3Pureza:≥95%Forma y color:White Crystalline Powder SolidPeso molecular:265.35Mebhydrolin
CAS:Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.Fórmula:C19H20N2Pureza:99.73% - ≥98%Forma y color:SolidPeso molecular:276.38JNJ-39220675
CAS:JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.Fórmula:C21H24FN3O2Pureza:97.95% - 99.78%Forma y color:SolidPeso molecular:369.43OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Fórmula:C18H22N2O2SPureza:99.49%Forma y color:SolidPeso molecular:330.44Hydroxyzine dihydrochloride
CAS:Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.Fórmula:C21H27ClN2O2·2HClPureza:99.46% - 99.79%Forma y color:Oil PowderPeso molecular:447.83Lodoxamide
CAS:Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.Fórmula:C11H6ClN3O6Pureza:99.13% - 99.81%Forma y color:SolidPeso molecular:311.63FR-145715
CAS:FR-145715 is a histamine H2 receptor antagonist characterized by its specific anti-Helicobacter pylori activity. This compound is utilized in the study of gastric lesions.Fórmula:C16H21N5O2SForma y color:SolidPeso molecular:347.44Niperotidine
CAS:Niperotidine is an antagonist of histamine H2-receptor.Fórmula:C20H26N4O5SPureza:98%Forma y color:SolidPeso molecular:434.51Thonzylamine
CAS:Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.Fórmula:C16H22N4OPureza:99.45%Forma y color:SolidPeso molecular:286.37Levocarnitine propionate hydrochloride
CAS:Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Fórmula:C10H20ClNO4Pureza:90% - 98%Forma y color:SolidPeso molecular:253.72Pemirolast potassium
CAS:Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.Fórmula:C10H7KN6OPureza:98.91% - 99.63%Forma y color:Crystals From Dimethylformamide Crystalline SolidPeso molecular:266.31Epinastine hydrochloride
CAS:Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Fórmula:C16H15N3·HClPureza:99.26% - 99.62%Forma y color:White SolidPeso molecular:285.77Levocetirizine Dihydrochloride
CAS:Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.Fórmula:C21H27Cl3N2O3Pureza:99.75%Forma y color:White Or Off-White Crystalline PowderPeso molecular:461.81Ref: TM-T22354
1g692,00€10mg50,00€25mg86,00€50mg131,00€100mg188,00€200mg283,00€500mg487,00€1mL*10mM (DMSO)52,00€
