
Receptor de glucagón
Los receptores de glucagón son GPCR que median los efectos del glucagón, una hormona involucrada en la regulación de la homeostasis de la glucosa al promover la descomposición del glucógeno y la liberación de glucosa desde el hígado. Estos receptores son cruciales en la gestión de los niveles de azúcar en sangre y son de particular interés en el estudio de la diabetes y los trastornos metabólicos. Los antagonistas de los receptores de glucagón se están explorando como posibles tratamientos para la hiperglucemia en la diabetes tipo 2. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de glucagón de alta calidad para apoyar su investigación en endocrinología, diabetes y regulación metabólica.
Productos de "Receptor de glucagón"
Ordenar por
(S, R)-LSN 3318839
CAS:(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.Fórmula:C26H23Cl2N3O2Pureza:99.57%Forma y color:SoildPeso molecular:480.39NNC 92-1687
CAS:NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.Fórmula:C15H12N2O3SPureza:100% - 99.72%Forma y color:SolidPeso molecular:300.33Avexitide
CAS:Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.Fórmula:C149H234N40O47SPureza:98% - 99.65%Forma y color:SolidPeso molecular:3369.76Exendin-4 acetate
CAS:Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).Fórmula:C186H286N50O62SPureza:98.65%Forma y color:SolidPeso molecular:4247Lotiglipron
CAS:Lotiglipron (PF-07081532) is a GLP-1R agonist that lowers blood glucose and may be used in the study of type 2 diabetes mellitus (T2DM) and excess obesity.Fórmula:C31H31ClN4O5Pureza:98.3%Forma y color:SolidPeso molecular:575.05V-0219
CAS:V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.Fórmula:C20H25F3N4O2Pureza:100%Forma y color:SoildPeso molecular:410.43Orforglipron
CAS:Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1Fórmula:C48H48F2N10O5Pureza:99.15% - 99.61%Forma y color:SolidPeso molecular:882.96Ref: TM-T11408
1mg244,00€5mg597,00€10mg938,00€25mg1.882,00€50mg2.593,00€100mg3.505,00€1mL*10mM (DMSO)47,00€V-0219 hydrochloride
V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.Fórmula:C20H26ClF3N4O2Pureza:100%Forma y color:SoildPeso molecular:446.89Ref: TM-T60047L
1mg59,00€5mg125,00€10mg205,00€25mg393,00€50mg585,00€100mg832,00€200mg1.121,00€1mL*10mM (DMSO)136,00€Semaglutide
CAS:Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).Fórmula:C187H291N45O59Pureza:96.92% - 99.78%Forma y color:SolidPeso molecular:4114Ref: TM-T19850
1mg126,00€5mg264,00€10mg378,00€25mg562,00€50mg780,00€100mg1.054,00€200mg1.419,00€500µg85,00€GLP-1 (9-36) amide
CAS:GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.Fórmula:C140H214N36O43Pureza:97%Forma y color:SolidPeso molecular:3089.41LGD-6972
CAS:LGD-6972 is an antagonist of glucagon receptor.Fórmula:C43H46N2O5SPureza:98.8% - 99.33%Forma y color:SolidPeso molecular:702.9Ref: TM-T11845
1mg88,00€5mg187,00€10mg274,00€25mg472,00€50mg692,00€100mg938,00€1mL*10mM (DMSO)283,00€Shanzhiside methyl ester
CAS:Shanzhiside methylester soothes neuropathic pain by triggering spinal GLP-1 receptors, boosting microglial β-endorphin through p38 MAPK.Fórmula:C17H26O11Pureza:99.32%Forma y color:SolidPeso molecular:406.38GLP-1 receptor agonist 9
CAS:1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.Fórmula:C32H31ClFN3O5Pureza:98%Forma y color:SolidPeso molecular:592.06Tirzepatide
CAS:Tirzepatide (LY-3298176) is a dual agonist of GIP and GLP-1 receptors with neuroprotective activity and can be used to study diabetes and obesity.Fórmula:C225H348N48O68Pureza:99.52% - 99.99%Forma y color:SolidPeso molecular:4813.45Exendin-4
CAS:Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.Fórmula:C184H282N50O60SPureza:97.71% - 99.72%Forma y color:SolidPeso molecular:4186.57PF-06882961 Tris
CAS:PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Fórmula:C35H41FN6O7Pureza:98.11% - 99.79%Forma y color:SolidPeso molecular:676.7GLP-1(7-37) acetate(106612-94-6 free base)
CAS:Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.Fórmula:C151H228N40O47Pureza:98.89%Forma y color:SolidPeso molecular:3355.67PF-06291874
CAS:PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.Fórmula:C26H28F3N3O4Pureza:99.12%Forma y color:SolidPeso molecular:503.51GLP-1(7-36), amide
CAS:GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.Fórmula:C149H226N40O45Pureza:99.85%Forma y color:White PowderPeso molecular:3297.63Adomeglivant
CAS:Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.Fórmula:C32H36F3NO4Pureza:99.97%Forma y color:SolidPeso molecular:555.63Ref: TM-T14130
5mg116,00€10mg188,00€25mg323,00€50mg568,00€100mg949,00€200mg1.424,00€1mL*10mM (DMSO)137,00€