Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Productos de "Receptor de dopamina"
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Desmethyl cariprazine
CAS:Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (Ki: 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM).Fórmula:C20H30Cl2N4OPureza:98%Forma y color:SolidPeso molecular:413.38Triflupromazine hydrochloride
CAS:Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.Fórmula:C18H20ClF3N2SPureza:99.73% - 99.76%Forma y color:CrystalsPeso molecular:388.88LP-211
CAS:LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.Fórmula:C30H34N4OPureza:98.65%Forma y color:SolidPeso molecular:466.62Ref: TM-T5387
2mg47,00€5mg70,00€10mg96,00€25mg180,00€50mg305,00€100mg487,00€200mg695,00€1mL*10mM (DMSO)77,00€CY 208-243
CAS:CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity.Fórmula:C19H18N2Pureza:98%Forma y color:SolidPeso molecular:274.36ACEPROMAZINE MALEATE
CAS:ACEPROMAZINE MALEATE is a dopamine receptor antagonistFórmula:C23H26N2O5SPureza:98.87% - 99.30%Forma y color:Off White Or Yellow Crystalline PowderPeso molecular:442.53PF-184298
CAS:PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.Fórmula:C15H20Cl2N2OPureza:98.30%Forma y color:SolidPeso molecular:315.24Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderateFórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Forma y color:SolidPeso molecular:427.41Ref: TM-T4577
1mg51,00€5mg108,00€10mg180,00€25mg316,00€50mg472,00€100mg658,00€200mg938,00€1mL*10mM (DMSO)108,00€ML417
CAS:ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).Fórmula:C22H25N3O3Pureza:98.81% - 99.42%Forma y color:SolidPeso molecular:379.45Escitalopram
CAS:Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.Fórmula:C20H21FN2OPureza:99.82%Forma y color:White Or White Crystalline PowderPeso molecular:324.39SKF 81297
CAS:SKF 81297 is a selective and potent agonist for the dopamine D1 receptor [1].Fórmula:C16H16ClNO2Pureza:98%Forma y color:SolidPeso molecular:289.76Trazpiroben
CAS:Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Fórmula:C31H39N3O4Pureza:98.85% - 99.41%Forma y color:SolidPeso molecular:517.66Fluoroclebopride
CAS:Fluoroclebopride is a dopamine (DA) D2 receptor ligand.Fórmula:C20H23ClFN3O2Pureza:99.68% - 99.91%Forma y color:SolidPeso molecular:391.87Ref: TM-T3187
1mg35,00€5mg74,00€10mg96,00€25mg159,00€50mg235,00€100mg376,00€500mg867,00€1mL*10mM (DMSO)96,00€Duloxetine hydrochloride
CAS:Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.Fórmula:C18H20ClNOSPureza:100% - 99.93%Forma y color:White Or White Crystalline PowderPeso molecular:333.88Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Fórmula:C19H25NOSPureza:98.08% - 99.59%Forma y color:SolidPeso molecular:315.47Ref: TM-T6647
5mg52,00€10mg78,00€25mg145,00€50mg255,00€100mg378,00€200mg552,00€500mg868,00€1mL*10mM (DMSO)55,00€D4R agonist-1
CAS:D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.Fórmula:C19H22N4SPureza:98.16%Forma y color:SolidPeso molecular:338.47Ref: TM-T78825
1mg333,00€5mg922,00€10mg1.140,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.664,00€PF-4363467
CAS:PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.Fórmula:C22H30N2O3SForma y color:SolidPeso molecular:402.55Flupentixol dihydrochloride
CAS:Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.Fórmula:C23H27Cl2F3N2OSPureza:100% - 99.35%Forma y color:White Or Off-White SolidPeso molecular:507.43PD128907 HCl
CAS:PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.Fórmula:C14H20ClNO3Pureza:98%Forma y color:SolidPeso molecular:285.77Zatebradine
CAS:Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).Fórmula:C26H36N2O5Pureza:98%Forma y color:SolidPeso molecular:456.57Remoxipride hydrochloride
CAS:Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-Fórmula:C16H24BrClN2O3Pureza:99.32%Forma y color:SolidPeso molecular:407.73
