Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Productos de "Proteasa del VIH"
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Dolutegravir
CAS:Dolutegravir (GSK1349572), HIV integrase inhibitor with IC50 of 2.7 nM, partly effective against some raltegravir-resistant HIV strains.Fórmula:C20H19F2N3O5Pureza:98.97% - 99.08%Forma y color:White To Pale Yellow SolidPeso molecular:419.38Ref: TM-T6198
1g1.111,00€1mg35,00€2mg50,00€5mg74,00€10mg115,00€25mg172,00€50mg274,00€100mg427,00€200mg607,00€500mg850,00€1mL*10mM (DMSO)69,00€INCB-9471
CAS:INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.Fórmula:C30H40F3N5O2Pureza:98%Forma y color:SolidPeso molecular:559.666TAK-220
CAS:TAK-220: Oral CCR5 antagonist. IC50: 3.5 nM (RANTES), 1.4 nM (MIP-1α).Fórmula:C31H41ClN4O3Pureza:98%Forma y color:SolidPeso molecular:553.14Bis-T-23
CAS:Bis-T-23 is a promoter of actin-dependent dynamin oligomerization, an HIV-I integrase inhibitor, and a Telstar derivative.Fórmula:C23H20N4O8Pureza:96.81% - 98.77%Forma y color:SolidPeso molecular:480.43Indinavir sulfate
CAS:Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM.Fórmula:C36H49N5O8SPureza:100% - 99.75%Forma y color:White PowderPeso molecular:711.87Ganoderic acid B
CAS:Ganoderic acid B: quality marker for G. lucidum products, inhibits telomerase & EBV activation, moderates HIV-1 protease.Fórmula:C30H44O7Pureza:99.09% - 99.95%Forma y color:SolidPeso molecular:516.67Cyclotriazadisulfonamide hydrochloride
CAS:Cyclotriazadisulfonamide HCl blocks HIV entry by hindering CD4 translocation into the ER.Fórmula:C31H40ClN3O4S2Pureza:98%Forma y color:SolidPeso molecular:618.25Ref: TM-T39264L
1mg185,00€5mg415,00€10mg622,00€25mg1.119,00€50mg1.679,00€100mg2.520,00€200mg3.780,00€Islatravir
CAS:Islatravir (MK-8591) is an effective anti-HIV-1 agent.Fórmula:C12H12FN5O3Pureza:98.77%Forma y color:SolidPeso molecular:293.25Ref: TM-T16098
1mg80,00€5mg170,00€10mg259,00€25mg454,00€50mg615,00€100mg827,00€200mg1.111,00€1mL*10mM (DMSO)182,00€Vesnarinone
CAS:Vesnarinone (Arkin) (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, positive inotropic activity, butFórmula:C22H25N3O4Pureza:96.69% - 98.13%Forma y color:SolidPeso molecular:395.45PKF050-638
CAS:PKF050-638 disrupts CRM1-NES, inhibits HIV-1 Rev export; selective with IC50=0.04 μM.Fórmula:C13H13ClN4O2Pureza:98%Forma y color:SolidPeso molecular:292.72LDC4297 hydrochloride
CAS:LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.Fórmula:C23H29ClN8OForma y color:SolidPeso molecular:468.98Ancriviroc
CAS:Ancriviroc (SCH-351125) is an orally bioavailable small molecule chemokine receptor CCR5 antagonist.Cost-effective and quality-assured.Fórmula:C28H37BrN4O3Pureza:97.31% - 99.74%Forma y color:SolidPeso molecular:557.52Apricitabine
CAS:Apricitabine (SPD754) is a highly selective and orally active HIV-1 reverse transcriptase inhibitor (Ki=0.08 μM), the (-) enantiomer of 2′-deoxy-3′-oxy-4′-Fórmula:C8H11N3O3SPureza:100%Forma y color:SolidPeso molecular:229.26Ref: TM-T14313
1mg299,00€5mg535,00€10mg663,00€25mg1.014,00€50mg1.690,00€100mg2.832,00€1mL*10mM (DMSO)625,00€SB 206553 hydrochloride
CAS:SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disordersFórmula:C17H17ClN4OPureza:99.56%Forma y color:SolidPeso molecular:328.84-Chloro-2-(trifluoroacetyl)aniline hydrochloride
CAS:4-Chloro-2-(trifluoroacetyl)aniline hydrochloride is an inhibitor of HIV-1 RT (HIV reverse transcriptase) .Fórmula:C8H6Cl2F3NOPureza:97.15%Forma y color:SolidPeso molecular:260.04GSK-364735
CAS:GSK-364735 is an HIV-1 IN inhibitor.Fórmula:C19H18FN3O4Pureza:97.89%Forma y color:SolidPeso molecular:371.36Tenofovir alafenamide fumarate
CAS:Tenofovir alafenamide fumarate (GS-7340) is an oral anti-HIV drug that prevents infection.Fórmula:C25H33N6O9PPureza:99.95%Forma y color:SolidPeso molecular:592.54Amprenavir
CAS:Amprenavir (KVX-478) is a synthetic derivative of hydroxyethylamine sulfonamide that selectively binds to and inhibits human immunodeficiency virus (HIV)Fórmula:C25H35N3O6SPureza:99.60% - 99.79%Forma y color:Off-White To Pale YellowPeso molecular:505.63Saquinavir mesylate
CAS:Saquinavir mesylate (Ro 31-8959/003) is an Inhibitor of HIV Proteaseused in antiretroviral therapyFórmula:C39H54N6O8SPureza:99.19%Forma y color:White Or Pale Yellow PowderPeso molecular:766.9NBD-556
CAS:NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.Fórmula:C17H24ClN3O2Pureza:99.79%Forma y color:SolidPeso molecular:337.84
