Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Productos de "Proteasa del VIH"
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BRD-6929
CAS:BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.Fórmula:C19H17N3O2SPureza:99.05%Forma y color:SolidPeso molecular:351.42Ref: TM-T10603
5mg50,00€10mg90,00€25mg170,00€50mg305,00€100mg442,00€200mg620,00€1mL*10mM (DMSO)51,00€Hck-IN-1
CAS:Hck-IN-1 selectively inhibits Nef:Hck, IC50: 2.8 μM; >20 μM for Hck alone. Potent HIV-1 Nef antagonist, IC50: 100-300 nM for HIV-1 replication.Fórmula:C16H11ClN6O3SPureza:99.07%Forma y color:SolidPeso molecular:402.81Ref: TM-T11538
1mg97,00€5mg216,00€10mg344,00€25mg567,00€50mg825,00€100mg1.121,00€200mg1.510,00€1mL*10mM (DMSO)240,00€AMD 3465 hexahydrobromide
CAS:AMD 3465 hexahydrobromide (GENZ-644494 (hexahydrobromide)) is a CXCR4 receptor antagonist with potential anticancer and anti-HIV activity.Fórmula:C24H44Br6N6Pureza:99.39%Forma y color:SolidPeso molecular:896.07Dolutegravir sodium
CAS:Dolutegravir sodium (GSK-1349572A) salt(DTG; GSK1349572) is an HIV integrase inhibitor(IC50: 2.7 nM), modest activity against raltegravir-resistant signatureFórmula:C20H18F2N3NaO5Pureza:98% - 99.74%Forma y color:SolidPeso molecular:441.36CK-666
CAS:CK-666 inhibits Arp2/3 complex, blocking Arp2/3 activation and actin filament formation.Fórmula:C18H17FN2OPureza:99.93%Forma y color:SolidPeso molecular:296.34Ref: TM-T10826
1mg40,00€5mg87,00€10mg140,00€25mg281,00€50mg545,00€100mg755,00€200mg945,00€1mL*10mM (DMSO)95,00€Acetyl-binankadsurin A
CAS:Acetyl-binankadsurin A (compound 5), a lignan obtained from Kadsura longipedunculata, exhibits weak inhibitory effects on HIV-1 protease, demonstrating an IC50Fórmula:C24H28O8Pureza:98%Forma y color:SolidPeso molecular:444.47HIV-1 Inhibitor 18A
CAS:HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) specifically inhibits the entry of multiple HIV-1 isolates.Fórmula:C14H11N5O2SPureza:91.64%Forma y color:SolidPeso molecular:313.33Ref: TM-T24141
1mg115,00€5mg227,00€10mg313,00€25mg535,00€50mg752,00€100mg1.064,00€1mL*10mM (DMSO)217,00€Benzalphthalide
CAS:Benzalphthalide (NSC-2824) is a chemical compound with anti-HIV activity.Fórmula:C15H10O2Pureza:98.41%Forma y color:Pale Yellow To Yellow Crystalline PowderPeso molecular:222.24PDDC inhibitor
CAS:PDDC inhibitor (Phenyl (R)-(1-(3-(3,4-dimethoxyphenyl)-2,6-dimethylimidazo[1,2-b]pyridazin-8-yl)pyrrolidin-3-yl)carbamate) is an nSMase2 inhibitor.Fórmula:C27H29N5O4Pureza:96.09% - 99.39%Forma y color:SolidPeso molecular:487.55Emtricitabine S-oxide
CAS:Emtricitabine treats HIV; its degradation byproduct is Emtricitabine S-oxide.Fórmula:C8H10FN3O4SPureza:98%Forma y color:SolidPeso molecular:263.25Salicylanilide
CAS:Salicylanilide (2-Hydroxybenzanilide)s are a group of compounds with antiviral potency, antibacterial and antifungal activities.Fórmula:C13H11NO2Pureza:99.55%Forma y color:White To Off-White Crystalline PowderPeso molecular:213.23Thiamine disulfide
CAS:Thiamine disulfide (Algoneurina) , also known as thiamin or vitamin B1, is a vitamin found in food and manufactured as a dietary supplement and medication.Fórmula:C24H34N8O4S2Pureza:99.18%Forma y color:CoaPeso molecular:562.71DRB
CAS:DRB is a nucleoside analog that inhibits several carboxyl-terminal domain (CTD) kinases including casein kinase II (IC50 range of 4-10 μM)Fórmula:C12H12Cl2N2O4Pureza:99.46%Forma y color:White To Off-White Crystalline SolidPeso molecular:319.14Efavirenz
CAS:Efavirenz (DMP 266) is an HIV-1 inhibitor, affecting reverse transcriptase and various cytochrome P450 enzymes.Fórmula:C14H9ClF3NO2Pureza:99.2% - 99.83%Forma y color:White To Slightly Pink Crystalline PowderPeso molecular:315.67Ref: TM-T2393
1g404,00€5mg42,00€10mg52,00€25mg71,00€50mg89,00€100mg116,00€500mg273,00€1mL*10mM (DMSO)49,00€Mk-6186 HCl
MK-6186 HCl, a novel non-nucleoside reverse transcriptase inhibitor with antiviral activity, can be used to study HIV.Fórmula:C21H13Cl3N6OPureza:98.19%Forma y color:SoildPeso molecular:471.732-Amino-6-bromopyridine
CAS:2-Amino-6-bromopyridine has inhibitory effect on HIV-68 protease.Fórmula:C5H5BrN2Pureza:99.87%Forma y color:SolidPeso molecular:173.01NNRTIs-IN-3
NNRTIs-IN-3 (compound 8) is an HIV-1 non-nucleoside reverse transcriptase inhibitor, displaying potent efficacy with an EC50 value of 0.01 µM [1].Fórmula:C17H20ClN5OPureza:98%Forma y color:SolidPeso molecular:345.83Fostemsavir
CAS:Fostemsavir (BMS-663068) is an HIV-1 attachment inhibitor in development for the treatment of HIV-1 infection.Fórmula:C25H26N7O8PPureza:98.95%Forma y color:SolidPeso molecular:583.49Ref: TM-T3523
1mg59,00€5mg120,00€10mg170,00€25mg283,00€50mg432,00€100mg622,00€200mg873,00€1mL*10mM (DMSO)156,00€Emivirine
CAS:Emivirine (MKC-442) is a potent and selective nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1.Fórmula:C17H22N2O3Pureza:99.68%Forma y color:SolidPeso molecular:302.37BI 224436
CAS:BI 224436 is an inhibitor of HIV-1 noncatalytic site integrase. With EC50 values of less than 15 nM against different HIV-1 laboratory strains.Fórmula:C27H26N2O4Forma y color:SolidPeso molecular:442.51
