Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Productos de "Proteasa del VIH"
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HIV-1 protease-IN-9
CAS:HIV-1 protease-IN-9 (compound 5b), a potent HIV-1 protease inhibitor, exhibits strong antiviral efficacy with a dissociation constant (K_i) of 0.028 nM and aFórmula:C37H41N7O4SPureza:98%Forma y color:SolidPeso molecular:679.83CDK9-IN-30
CAS:CDK9-IN-30 is one of the Tat peptide derivatives and inhibits HIV-1 long terminal repeat-activated transcription.Fórmula:C16H20FNO3Pureza:99.76%Forma y color:SolidPeso molecular:293.33Ref: TM-T9632
1mg56,00€5mg119,00€10mg187,00€25mg316,00€50mg472,00€100mg658,00€500mg1.378,00€1mL*10mM (DMSO)114,00€Cenicriviroc
CAS:Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.Fórmula:C41H52N4O4SPureza:97.87%Forma y color:SolidPeso molecular:696.94Ref: TM-TQ0297
1mg69,00€5mg149,00€10mg235,00€25mg470,00€50mg610,00€100mg793,00€200mg1.064,00€1mL*10mM (DMSO)221,00€L-689502
CAS:L-689502 is a potent HIV-l protease inhibitor (IC50: 1 nM).Fórmula:C39H51N3O7Pureza:98%Forma y color:SolidPeso molecular:673.84Dimercaprol
CAS:Dimercaprol (Dicaptol) is an anti-gas warfare agent that is effective against Lewisite (dichloro(2-chlorovinyl)arsine) and formerly known as British Anti-Fórmula:C3H8OS2Pureza:98.91% - 99.64%Forma y color:Viscous Oily LiquidPeso molecular:124.22Tenofovir alafenamide hemifumarate
CAS:Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.Fórmula:C21H29N6O5PC4H4O4Pureza:99.33% - 99.96%Forma y color:SolidPeso molecular:534.51PTACH
CAS:PTACH (Cpd 51) (NCH-51) is a SAHA-based inhibitor of human HDAC. It can potently inhibit the growth of various human Y cells (EC50: 1 to 10 μM).Fórmula:C20H26N2O2S2Pureza:87.44% - 99.74%Forma y color:SolidPeso molecular:390.56Ref: TM-T3199
1mg50,00€5mg97,00€10mg154,00€25mg298,00€50mg447,00€100mg620,00€200mg843,00€1mL*10mM (DMSO)111,00€ST7612AA1
CAS:ST7612AA1: potent, oral HDAC inhibitor; reactivates HIV-1 latency; shows antitumor effects; may study malaria.Fórmula:C20H27N3O4SPureza:100%Forma y color:SolidPeso molecular:405.51Nelfinavir
CAS:Nelfinavir (AG1341), with Ki=2 nM, is an HIV treatment and broad-spectrum anticancer drug.Fórmula:C32H45N3O4SPureza:98.16% - 99.5%Forma y color:White To Off-White Crystalline PowderPeso molecular:567.78Ref: TM-T7779
1mg43,00€2mg56,00€5mg88,00€10mg111,00€25mg168,00€50mg216,00€100mg285,00€1mL*10mM (DMSO)97,00€Fosdevirine
CAS:Fosdevirine (GSK2248761), a non-nucleoside reverse transcriptase (NNRTI) inhibitor with anti-HIV activity, is used in the study of neurological related diseasesFórmula:C20H17ClN3O3PPureza:99.94%Forma y color:SolidPeso molecular:413.79Virstatin
CAS:Virstatin, an antiviral, inhibits replication of viruses like HSV, HIV, and influenza.Fórmula:C16H13NO4Pureza:99.94%Forma y color:SolidPeso molecular:283.2787Darunavir
CAS:Darunavir (TMC114) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Fórmula:C27H37N3O7SPureza:99.67% - 99.76%Forma y color:White Amorphous SolidPeso molecular:547.66I-XW-053
CAS:I-XW-053 is an inhibitor of capsid targeted HIV-1 replication using the hybrid structure based method to block the interface between CA N-terminal domains (NTD-Fórmula:C22H16N2O2Pureza:99.11%Forma y color:SolidPeso molecular:340.37TERT-IN-1
CAS:TERT-IN-1 has anti-HIV activity and can be used to study HIV infection.Fórmula:C16H20ClN3SPureza:99.31%Forma y color:SoildPeso molecular:321.87BMS-707035
CAS:BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM. Phase 2.Fórmula:C17H19FN4O5SPureza:99.78%Forma y color:SolidPeso molecular:410.42Ditiocarb sodium
CAS:Ditiocarb sodium (Sodium diethyldithiocarbamate) (sodium diethiocarbamate) is a copper reagent, which reacts with Cu2 + solution to form a complex and improvesFórmula:C5H10NNaS2Pureza:98%Forma y color:White Solid CrystallinePeso molecular:171.26GPI-1046
CAS:GPI-1046: immunophilin ligand, no antibiotic effect, reduces ethanol intake by boosting GLT1 in PFC and NAc-core.Fórmula:C20H28N2O4Pureza:99.69%Forma y color:SolidPeso molecular:360.45Ref: TM-T11451
1mg74,00€2mg94,00€5mg144,00€10mg235,00€25mg398,00€50mg567,00€100mg820,00€1mL*10mM (DMSO)131,00€Elsulfavirine
CAS:Elsulfavirine (VM-1500) is an HIV-1 infection reverse transcriptase inhibitor. It is a new anti-HIV drug.Fórmula:C24H17BrCl2FN3O5SPureza:99.66%Forma y color:SolidPeso molecular:629.28Ref: TM-T15210
1mg72,00€5mg156,00€10mg243,00€25mg487,00€50mg730,00€100mg1.026,00€1mL*10mM (DMSO)210,00€(2RS)-FPMPA
CAS:(2RS)-FPMPA(FPMPA) has antiviral activity with an IC50 value of 1.85 μM measured in human MT12 cells infected with SHIV (DH4R).Fórmula:C9H13FN5O4PPureza:100% - 99.90%Forma y color:SolidPeso molecular:305.2Azt-pmap
CAS:AZT-PMPA, an aryl phosphate derivative of AZT and a nucleoside analogue, demonstrates anti-HIV activity[1].Fórmula:C20H25N6O8PPureza:98%Forma y color:SolidPeso molecular:508.42
