Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Productos de "Proteasa del VIH"
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HIV-1 protease-IN-12
CAS:HIV-1 protease-IN-12 (compound 35b) serves as a potent inhibitor of HIV-1 protease, exhibiting an IC50 value of 0.51 nM, and demonstrates efficacy against drug-Fórmula:C25H35N3O5SPureza:98%Forma y color:SolidPeso molecular:489.63Nandrolone decanoate
CAS:Nandrolone decanoate is an anabolic steroid similar to testosterone, stimulating muscle, bone growth, and red blood cell production.Fórmula:C28H44O3Pureza:98.43% - 99.03%Forma y color:SolidPeso molecular:428.65Vicriviroc maleate
CAS:Vicriviroc maleate (SCH-417690 (maleate))(Sch-417690) is a piperazine-based CCR5 receptor antagonist with activity against human immunodeficiency virus.Fórmula:C32H42F3N5O6Pureza:97.51% - 98.16%Forma y color:SolidPeso molecular:649.7Atazanavir
CAS:Atazanavir (BMS-232632)(BMS-232632) is an highly effective HIV-1 protease inhibitor.Fórmula:C38H52N6O7Pureza:98% - 99.95%Forma y color:Crystalline SolidPeso molecular:704.86Pirmitegravir
CAS:Pirmitegravir (STP0404) is a potent ALLINI, blocks LEDGF/p75 site, shows antiviral action against HIV.Fórmula:C27H31ClN4O3Pureza:100% - 99.79%Forma y color:SolidPeso molecular:495.01Bavtavirine
CAS:Bavtavirine is a non-nucleoside reverse HIV-1 transcriptase inhibitor (NNRTIs),inhibits HIV replication by preventing the transcription of viral RNA into DNA.Fórmula:C26H20N6Pureza:98.08%Forma y color:SolidPeso molecular:416.48Pentosan Polysulfate
CAS:Pentosan Polysulfate: anti-HIV, anti-inflammatory, supports cartilage, treats interstitial cystitis.Pureza:98%Forma y color:SolidPeso molecular:N/ARaltegravir
CAS:Raltegravir (MK-0518) is a pyrrolidinone derivative and HIV INTEGRASE INHIBITOR that is used in combination with other ANTI-HIV AGENTS for the treatment of HIVFórmula:C20H21FN6O5Pureza:100% - 99.86%Forma y color:SolidPeso molecular:444.42Escin IA
CAS:Escin IA (Escin IA;Aescin IA) is a triterpene saponin isolated from horse chestnut, which inhibits HIV-1 protease with IC50 values of 35 μM.Fórmula:C55H86O24Pureza:99.34% - 99.81%Forma y color:SolidPeso molecular:1131.26HIV-1 Nef-IN-1
CAS:HIV-1 Nef-IN-1 is an inhibitor of HIV-1 Nef protein. It efficiently competes for Nef-SH3Hck interactions(Kd : 6.7 μM).Fórmula:C18H16O2Pureza:99.90%Forma y color:SolidPeso molecular:264.32Ritonavir
CAS:Ritonavir (ABT 538) inhibits HIV-1/2 proteases; serum proteins limit it but it enhances other HIV drugs by hindering P450 degradation.Fórmula:C37H48N6O5S2Pureza:99.38% - 99.58%Forma y color:White PowderPeso molecular:720.94Ref: TM-T1525
1g502,00€5mg37,00€10mg49,00€25mg79,00€50mg101,00€100mg145,00€200mg202,00€500mg339,00€1mL*10mM (DMSO)49,00€MK-2048
CAS:MK-2048 is a potent inhibitor of integrase (IN) and INR263K with IC50 of 2.6 nM and 1.5 nM, respectively.Fórmula:C21H21ClFN5O4Pureza:98%Forma y color:SolidPeso molecular:461.87IMB-301
CAS:IMB-301 is a small molecular inhibitor via virtual screening according to the hA3G model.Fórmula:C19H17Cl2FN2OPureza:99.72%Forma y color:SolidPeso molecular:379.26Ref: TM-T9212
1mg48,00€5mg97,00€10mg156,00€25mg259,00€50mg369,00€100mg530,00€200mg720,00€1mL*10mM (DMSO)105,00€Probenecid
CAS:Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.Fórmula:C13H19NO4SPureza:98.47% - 99.95%Forma y color:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Peso molecular:285.36HIV-1 inhibitor-6
CAS:HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicingFórmula:C14H10N4O4SPureza:98.49%Forma y color:SolidPeso molecular:330.32TAK-779
CAS:TAK-779 (Takeda 779) is an antagonist of chemokine receptor 5 (CCR5), CCR2b, and CXC chemokine receptor 3 (CXCR3).Fórmula:C33H39ClN2O2Pureza:99.21%Forma y color:SolidPeso molecular:531.13RN-18
CAS:RN-18 is an inhibitor of HIV-1 viral infectivity factor (IC50: 6 μM in nonpermissive H9 cells).Fórmula:C20H16N2O4SPureza:97.21% - 98.39%Forma y color:SolidPeso molecular:380.42Aprepitant
CAS:Aprepitant (Aprepitant') is a Substance P/Neurokinin-1 Receptor Antagonist.Fórmula:C23H21F7N4O3Pureza:98% - 99.68%Forma y color:Off-White To Light Yellow Cyrstalline SolidPeso molecular:534.43Aplaviroc
CAS:Aplaviroc (AK 602), a SDP derivative, is a CCR5 antagonist. With IC50s of 0.1-0.4 nM for HIV-1Ba-L, HIV-1JRFL and HIV-1MOKW.Fórmula:C33H43N3O6Pureza:98.78% - 99.53%Forma y color:SolidPeso molecular:577.71HIV-1 inhibitor-81
HIV-1inhibitor-81 (Compound 14g) is an HIV-1 protease inhibitor with a Ki of 1.6 nM. This compound exhibits antiviral activity against HIV-1, with an EC50 value of 250 nM.Fórmula:C32H44N2O8SForma y color:SolidPeso molecular:616.77
