Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Productos de "Proteasa del VIH"
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Darunavir Ethanolate
CAS:Darunavir Ethanolate (UIC 94017) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Fórmula:C29H43N3O8SPureza:99.84%Forma y color:SolidPeso molecular:593.74Ref: TM-T3335
5mg37,00€10mg52,00€25mg80,00€50mg111,00€100mg165,00€200mg236,00€500mg399,00€1mL*10mM (DMSO)48,00€Stercobilin hydrochloride (mixture of isomers)
CAS:Stercobilin hydrochloride (mixture of isomers) is a bile pigment metabolized by intestinal bacteria and also acts as an inhibitor of HIV protease (HIVProtease) with a Ki of 4 μM. This compound can induce pro-inflammatory activity in mouse macrophage RAW264 cells, including the production of TNF-α and IL-1β. Stercobilin hydrochloride (mixture of isomers) is utilized in research on inflammation and viral infections.Fórmula:C33H47ClN4O6Forma y color:SolidPeso molecular:631.20HIV-IN-6
CAS:HIV-IN-6, an anti-HIV agent, blocks replication by targeting SFKs like Hck involved with Nef protein.Fórmula:C20H16N4O3SPureza:97.12%Forma y color:SolidPeso molecular:392.43Oxindole
CAS:Oxindole (Indolin-2-one) is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure has been used in receptor tyrosine kinases (RTKs) inhibitors such as SU4984 and intedanib, the RTK family represents an important therapeutic target for anti-cancer drug development.Fórmula:C8H7NOPureza:99.34%Forma y color:Off-White Crystalline PowderPeso molecular:133.15Rolipram
CAS:Rolipram (SB 95952) is a phosphodiesterase 4 inhibitor with antidepressant properties.Fórmula:C16H21NO3Pureza:99.22% - 99.26%Forma y color:SolidPeso molecular:275.34Rosamultin
CAS:Rosamultin has antioxidant, antiinflammatory/antinociceptive properties,and has anti-human immunodeficiency virus (HIV) activity.Fórmula:C36H58O10Pureza:98% - 99.83%Forma y color:SolidPeso molecular:650.84Cabotegravir
CAS:Cabotegravir (S/GSK1265744) (GSK744, GSK1265744) is a long-acting HIV integrase inhibitor and inhibits the HIV-1 integrase catalyzed strand transfer reaction (Fórmula:C19H17F2N3O5Pureza:98.55% - 99.92%Forma y color:SolidPeso molecular:405.35Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2
CAS:Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2 is a fluorogenic substrate for the HIV-1 protease, facilitating the assessment of enzyme activity [1].Fórmula:C40H66N12O11Pureza:98%Forma y color:SolidPeso molecular:891.03L 756423
CAS:L756423 is a potent, selective HIV protease inhibitor (Ki=0.049 nM), effective against HIV spread in MT25 lymphocytes at 0.1-0.5 nM, useful for AIDS research.Fórmula:C39H48N4O5Pureza:100% - 100%Forma y color:SolidPeso molecular:652.82Mavorixafor trihydrochloride
CAS:Mavorixafor trihydrochloride blocks CXCR4 (IC50: 13 nM) and suppresses T-tropic HIV-1 replication (IC50: 1-9 nM). It's orally active.Fórmula:C21H30Cl3N5Pureza:98.00%Forma y color:SolidPeso molecular:458.86NBD-557
CAS:NBD-557 is a potentially HIV-1 inhibitor.Fórmula:C17H24BrN3O2Pureza:99.52%Forma y color:SolidPeso molecular:382.3Ref: TM-T7382
1mg48,00€5mg97,00€10mg156,00€25mg301,00€50mg437,00€100mg620,00€200mg843,00€1mL*10mM (DMSO)105,00€Bellidifolin
CAS:Bellidoferin: anti-oxidant, protects liver, fights inflammation/tumors, aids nerve injury, blocks MAO A, may improve type-2 diabetes, antifungal.Fórmula:C14H10O6Pureza:99.79% - 99.81%Forma y color:SolidPeso molecular:274.23Ref: TM-T3822
1mg96,00€5mg225,00€10mg323,00€25mg537,00€50mg752,00€100mg1.035,00€1mL*10mM (DMSO)202,00€Talviraline
CAS:Talviraline (Bay 10-8979) is an RNA-induced DNA polymerase inhibitor.Talviraline is a potent inhibitor of HIV-1-induced cell killing and HIV-1 replication in aFórmula:C15H20N2O3S2Pureza:99.82%Forma y color:SolidPeso molecular:340.46Lopinavir
CAS:Lopinavir (ABT-378) is a peptidomimetic HIV protease inhibitor that retains activity against HIV protease with the Val 82 mutation.Fórmula:C37H48N4O5Pureza:98% - 99.62%Forma y color:White Crystalline SolidPeso molecular:628.83-Deazaadenosine hydrochloride
CAS:3-Deazaadenosine HCl blocks SAH hydrolase (Ki: 3.9 μM), with anti-inflammatory, anti-proliferative, and anti-HIV effects.Fórmula:C11H15ClN4O4Pureza:98.48%Forma y color:SolidPeso molecular:302.71Ref: TM-T10111
1mg126,00€5mg216,00€10mg374,00€25mg620,00€50mg868,00€100mg1.169,00€1mL*10mM (DMSO)149,00€Maraviroc
CAS:Maraviroc: a CCR5 antagonist blocking HIV-1 entry; IC50s-MIP-1α: 3.3nM, MIP-1β: 7.2nM, RANTES: 5.2nM.Fórmula:C29H41F2N5OPureza:100% - 99.55%Forma y color:Brown SolidPeso molecular:513.67Ref: TM-T6016
5mg51,00€10mg95,00€25mg160,00€50mg273,00€100mg492,00€200mg633,00€500mg998,00€1mL*10mM (DMSO)59,00€HIV-1 inhibitor-53
CAS:HIV-1 Inhibitor-53 targets HIV-1 protease (IC50: 1.93 nM) and reverse transcriptase (IC50: 2.35 μM), aiding AIDS research.Fórmula:C30H34N2O8SPureza:98%Forma y color:SolidPeso molecular:582.66Raltegravir potassium
CAS:Raltegravir potassium (MK 0518 potassium salt) salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.Fórmula:C20H20FN6O5·KPureza:98% - 99.55%Forma y color:Off-White SolidPeso molecular:482.51Nevirapine
CAS:Nevirapine (NVP) is a benzodiazepine non-nucleoside reverse transcriptase inhibitor.Fórmula:C15H14N4OPureza:99.58% - 99.59%Forma y color:White Or Off-White Crystalline PowderPeso molecular:266.3Ro24-7429
CAS:Ro24-7429: oral HIV-1 Tat antagonist, RUNX1 inhibitor with anti-HIV, antifibrotic, and anti-inflammatory properties.Fórmula:C14H13ClN4Pureza:99.29% - 99.85%Forma y color:SolidPeso molecular:272.73Ref: TM-T28578
1mg92,00€5mg187,00€10mg298,00€25mg507,00€50mg730,00€100mg1.026,00€500mg2.877,00€1mL*10mM (DMSO)215,00€
