récepteur 5-HT
Les récepteurs 5-HT, également connus sous le nom de récepteurs de la sérotonine, sont un groupe de récepteurs couplés aux protéines G (GPCR) qui médiatisent les effets de la sérotonine, un neurotransmetteur impliqué dans la régulation de l'humeur, l'anxiété, le sommeil, l'appétit et d'autres processus physiologiques. Ces récepteurs sont divisés en plusieurs sous-types, chacun ayant des fonctions et des propriétés pharmacologiques distinctes. Les modulateurs des récepteurs 5-HT sont largement étudiés pour leurs rôles dans le traitement de la dépression, des troubles anxieux et d'autres affections neuropsychiatriques. Chez CymitQuimica, nous offrons une gamme de modulateurs des récepteurs 5-HT de haute qualité pour soutenir vos recherches en neuropharmacologie, troubles de l'humeur et signalisation GPCR.
Produits appartenant à la catégorie "récepteur 5-HT"
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Azatadine dimaleate
CAS :Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).Formule :C28H30N2O8Degré de pureté :100% - 99.70%Couleur et forme :PowderMasse moléculaire :522.555-MeO-MET
CAS :5-MeO-MET (5-Methoxy-N-methyl-N-ethyltryptamine) is a compound belonging to the 5-methoxytryptamine class. It acts as an agonist for 5-HT1A and 5-HT2A receptors. In mice, 5-MeO-MET inhibits locomotion and has sedative effects.Formule :C14H20N2OCouleur et forme :SolidMasse moléculaire :232.32Terfenadine
CAS :Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Formule :C32H41NO2Degré de pureté :98.76% - 99.75%Couleur et forme :SolidMasse moléculaire :471.67GR 113808
CAS :GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.Formule :C19H27N3O4SDegré de pureté :98.16%Couleur et forme :SolidMasse moléculaire :393.5Pimavanserin
CAS :Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.Formule :C25H34FN3O2Degré de pureté :97.84% - 99.69%Couleur et forme :Pale Yellow To Pale Orange SolidMasse moléculaire :427.55Xaliproden hydrochloride
CAS :Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formule :C24H23ClF3NDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :417.89Ref: TM-T9272
1mg40,00€5mg85,00€10mg120,00€25mg235,00€50mg376,00€100mg540,00€200mg775,00€1mL*10mM (DMSO)96,00€PF-04995274
CAS :PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.Formule :C23H32N2O6Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :432.51Pellotine
CAS :Pellotine is an alkaloid isolated from Lophophora. It acts as an inverse agonist of the 5-HT7 receptor (5-HT7 receptor), with an EC50 of 291 nM. Pellotine shows strong affinity for the 5-HT1DR and 5-HT6R, with Ki values of 117 nM and 170 nM, respectively. Additionally, Pellotine reduces intracellular cAMP levels, thereby decreasing neuronal excitability and neurotransmitter release.Formule :C13H19NO3Couleur et forme :SolidMasse moléculaire :237.295Amperozide
CAS :Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Formule :C23H29F2N3ODegré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :401.49Ref: TM-T23733
1mg92,00€5mg188,00€10mg311,00€25mg525,00€50mg747,00€100mg1.017,00€500mg2.023,00€1mL*10mM (DMSO)339,00€Paroxetine hydrochloride hemihydrate
CAS :Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).Formule :C38H44Cl2F2N2O7Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :749.67BRL-15572 dihydrochloride
CAS :BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.Formule :C25H27ClN2O·2HClDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :479.874-Chloromethamphetamine hydrochloride
CAS :4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.Formule :C10H15Cl2NCouleur et forme :SolidMasse moléculaire :220.144F 4PP oxalate
CAS :4F 4PP oxalate is a 5-HT2A antagonist.Formule :C22H26FNO·C2H2O4Degré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :429.49Ref: TM-T22514
5mg46,00€10mg80,00€25mg131,00€50mg210,00€100mg313,00€200mg445,00€1mL*10mM (DMSO)49,00€Lintopride HCl
CAS :Lintopride HCl is a 5HT-4 antagonist.Formule :C14H20Cl2N4O2Degré de pureté :97.70% - 98.42%Couleur et forme :SoildMasse moléculaire :347.24Ramosetron hydrochloride
CAS :Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.Formule :C17H18ClN3ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :315.8RS 42358-197
CAS :RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Formule :C19H23ClN2ODegré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :330.85Ref: TM-T20739
1mg166,00€5mg371,00€10mg557,00€25mg827,00€50mg1.111,00€100mg1.491,00€200mg2.015,00€1mL*10mM (DMSO)369,00€Lesopitron dihydrochloride
CAS :Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Formule :C15H23Cl3N6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :393.74RS 56812
CAS :RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive disorders.Formule :C18H21N3O2Degré de pureté :98.78%Couleur et forme :SoildMasse moléculaire :311.38Eptapirone
CAS :Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.Formule :C16H23N7O2Degré de pureté :99.39% - 99.65%Couleur et forme :SolidMasse moléculaire :345.4Talipexole dihydrochloride
CAS :Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical andFormule :C10H17Cl2N3SDegré de pureté :98.64%Couleur et forme :Light Yellow SolidMasse moléculaire :282.23Ref: TM-T14490
2mg38,00€5mg56,00€10mg89,00€25mg154,00€50mg264,00€100mg424,00€200mg613,00€500mg949,00€1mL*10mM (DMSO)63,00€RS102895 hydrochloride
CAS :RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).Formule :C21H22ClF3N2O2Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :426.86(-)-5-HT2C agonist-3
CAS :Compound (−)-19, also known as (-)-5-HT2C agonist-3, is a selective 5-HT2C agonist exhibiting a preference for Gq signaling. It demonstrates efficiency with EC50 values for 5-HT2 receptor subtypes as follows: 5-HT2C at 103 nM, 5-HT2B at 570 nM, and 5-HT2A at 72 nM. This compound is utilized in research on antipsychotics.Formule :C19H23ClFNO2Couleur et forme :SolidMasse moléculaire :351.84SCH-23390 maleate
CAS :SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formule :C21H22ClNO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :403.864i
CAS :4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.Formule :C16H12ClN3ODegré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :297.74Flibanserin
CAS :Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.Formule :C20H21F3N4ODegré de pureté :99.37% - 99.93%Couleur et forme :White PowderMasse moléculaire :390.4Flopropione
CAS :Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.Formule :C9H10O4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :182.17PRX-08066 Maleic acid
CAS :PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Formule :C23H21ClFN5O4SDegré de pureté :97.59%Couleur et forme :SolidMasse moléculaire :517.96Ref: TM-T6959
1mg90,00€5mg186,00€10mg252,00€25mg454,00€50mg660,00€100mg939,00€200mg1.276,00€1mL*10mM (DMSO)435,00€SCH-23390 hydrochloride
CAS :SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formule :C17H19Cl2NODegré de pureté :98% - 99.51%Couleur et forme :SolidMasse moléculaire :324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€F13714 fumarate
CAS :F13714 fumarate is a 5-HT1A receptor-biased agonist.Formule :C25H29ClF2N4O5Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :538.975-Carboxamidotryptamine maleate
CAS :5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.Formule :C15H17N3O5Degré de pureté :97.77%Couleur et forme :SolidMasse moléculaire :319.316-Fluoro-N,N-diethyltryptamine
CAS :6-Fluoro-N,N-diethyltryptamine (6-F-DET) exhibits affinity for the 5-HT2A receptor.Formule :C14H19FN2Couleur et forme :SolidMasse moléculaire :234.31SEP-363856 mesylate
CAS :SEP-363856 (SEP-856) mesylate is an orally active compound that acts as an agonist for both TAAR1 and 5-HT1A receptors. This compound exhibits antipsychotic activity in the central nervous system and has potential for the study of schizophrenia.Formule :C10H17NO4S2Couleur et forme :SolidMasse moléculaire :279.38AAZ-A 154 mesylate
CAS :AAZ-A 154 mesylate mesylate is a selective, competitive, and non-hallucinogenic antagonist of 5-HT2AR. It enhances neuronal growth in rodents and produces enduring beneficial behavioral effects.Formule :C15H24N2O4SCouleur et forme :SolidMasse moléculaire :328.43Ondansetron hydrochloride
CAS :Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiationFormule :C18H19N3O·HClDegré de pureté :99.78%Couleur et forme :White PowderMasse moléculaire :329.8225B-NBOH hydrochloride
CAS :25B-NBOH hydrochloride is a phenethylamine that exhibits high affinity for serotonin (5-HT) receptors 5-HT2A and 5-HT2C, with pKi values of 8.3 and 9.4, respectively.Formule :C17H21BrClNO3Couleur et forme :SolidMasse moléculaire :402.711SB-203186 hydrochloride
CAS :SB 203186 hydrochloride is a potent 5-HT4 receptor antagonistFormule :C16H20N2O2·HClDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :308.81Loxapine succinate
CAS :Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.Formule :C22H24ClN3O5Degré de pureté :99.69%Couleur et forme :White To Of-White SolidMasse moléculaire :445.9Lecozotan HCl
CAS :Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.Formule :C28H30ClN5O3Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :520.02QF0301B
CAS :QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.Formule :C23H28N2O2Degré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :364.48Neocarzinostatin
CAS :Neocarzinostatin is an effective DNA-damaging, anti-tumor antibiotic.Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :N/ADapoxetine
CAS :Dapoxetine (Dapoxetina) is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation.Formule :C21H23NODegré de pureté :99.73%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :305.42Fananserin
CAS :Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Formule :C23H24FN3O2SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :425.52Ref: TM-T15270
2mg42,00€5mg56,00€10mg81,00€25mg116,00€50mg170,00€100mg250,00€200mg369,00€1mL*10mM (DMSO)62,00€Pimavanserin tartrate
CAS :Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.Formule :C50H68F2N6O4·C4H6O6Degré de pureté :100% - 99.98%Couleur et forme :SolidMasse moléculaire :1005.2Ziprasidone
CAS :Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.Formule :C21H21ClN4OSDegré de pureté :100% - 99.53%Couleur et forme :Tan SolidMasse moléculaire :412.94GM-60186
GM-60186, a potent inhibitor of the 5-HT receptor 2B (HTR2B) with an IC50 of 257 nM, effectively suppresses the proliferation and migration of colorectal cancer cells.Formule :C30H33FN2O4Couleur et forme :SolidMasse moléculaire :504.59Anpirtoline hydrochloride
CAS :Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.Formule :C10H14Cl2N2SDegré de pureté :100% - 100%Couleur et forme :SolidMasse moléculaire :265.20Quetiapine hemifumarate
CAS :Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formule :C46H54N6O8S2Degré de pureté :100% - 99.59%Couleur et forme :White Crystalline SolidMasse moléculaire :883.09Agomelatine
CAS :Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.Formule :C15H17NO2Degré de pureté :99.92%Couleur et forme :White SolidMasse moléculaire :243.3Rizatriptan benzoate
CAS :Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFormule :C22H25N5O2Degré de pureté :99% - 99.72%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :391.47Ref: TM-T1512
10mg47,00€25mg79,00€50mg126,00€100mg183,00€200mg273,00€500mg462,00€1mL*10mM (DMSO)50,00€Ansofaxine hydrochloride
CAS :Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formule :C24H32ClNO3Degré de pureté :99.57% - 99.77%Couleur et forme :SolidMasse moléculaire :417.97RS-127445 hydrochloride
CAS :RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).Formule :C17H17ClFN3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :317.795-HT6 agonist 1
Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting plateletFormule :C17H22Cl2N6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.37Paliperidone
CAS :Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.Formule :C23H27FN4O3Degré de pureté :95% - 99.08%Couleur et forme :Off White To Light Orange Coloured SolidMasse moléculaire :426.48Lintopride
CAS :Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Formule :C14H19ClN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.78(R)-Mirtazapine
CAS :(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formule :C17H19N3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :265.35Metergoline
CAS :Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formule :C25H29N3O2Degré de pureté :99.7% - 99.83%Couleur et forme :SolidMasse moléculaire :403.52F-15599
CAS :F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).Formule :C19H21ClF2N4ODegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :394.85Buclizine dihydrochloride
CAS :Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormule :C28H33ClN2·2HClDegré de pureté :98.05%Couleur et forme :Off-White PowderMasse moléculaire :505.95idalopirdine
CAS :Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Formule :C20H19F5N2ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :398.37Ref: TM-T7103
1mg88,00€2mg118,00€5mg188,00€10mg254,00€25mg429,00€50mg630,00€100mg898,00€1mL*10mM (DMSO)187,00€Org 13011
CAS :Org 13011 has CNS activity and induces conditioned taste aversion by mediating 5-HT 1A receptors.Formule :C18H25F3N4ODegré de pureté :98.98%Couleur et forme :SoildMasse moléculaire :370.41Ref: TM-T28258L
1mg185,00€5mg459,00€10mg657,00€25mg1.026,00€50mg1.415,00€100mg1.872,00€1mL*10mM (DMSO)469,00€Opiranserin
CAS :Opiranserin is a development as an injectable agent for the treatment of postoperative pain.Formule :C21H34N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.51Ampreloxetine
CAS :Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.Formule :C18H18F3NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.34Trazodone
CAS :Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.Formule :C19H22ClN5ODegré de pureté :99.79%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :371.86Arotinolol hydrochloride
CAS :Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.Formule :C15H22ClN3O2S3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :408Myristicin
CAS :Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.Formule :C11H12O3Degré de pureté :99.34%Couleur et forme :LiquidMasse moléculaire :192.21LY-2624803
CAS :LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Formule :C22H25N3O3Degré de pureté :100% - 99.87%Couleur et forme :SolidMasse moléculaire :379.45RS 67333 hydrochloride
CAS :RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Formule :C19H30Cl2N2O2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :389.36Naratriptan hydrochloride
CAS :Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.Formule :C17H25N3O2S·HClDegré de pureté :99.17% - 99.89%Couleur et forme :Beige SolidMasse moléculaire :371.93Ref: TM-T6602
10mg50,00€25mg88,00€50mg133,00€100mg188,00€200mg283,00€500mg467,00€1mL*10mM (DMSO)52,00€Prucalopride Succinate
CAS :Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formule :C18H26ClN3O3·C4H6O4Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :485.96Dehydroaripiprazole
CAS :Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.Formule :C23H25Cl2N3O2Degré de pureté :97.05%Couleur et forme :SolidMasse moléculaire :446.37THRX-194556
CAS :THRX-194556 is an agonist of the 5-HT4 receptor. It is applicable in the study of gastrointestinal functional disorders and Alzheimer's disease.Formule :C28H41N5O5SCouleur et forme :SolidMasse moléculaire :559.721Blonanserin
CAS :Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formule :C23H30FN3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :367.5Metoclopramide
CAS :Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formule :C14H22ClN3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :299.8Brilaroxazine
CAS :Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.Formule :C22H25Cl2N3O3Degré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :450.36Ref: TM-T14782
1mg105,00€5mg250,00€10mg406,00€25mg700,00€50mg1.008,00€100mg1.378,00€200mg1.833,00€1mL*10mM (DMSO)283,00€p-MPPI hydrochloride
CAS :p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.Formule :C25H28ClIN4O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :578.87Capeserod
CAS :Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive disorders and neurological disorders.Formule :C23H25ClN4O4Degré de pureté :98.82% - 99.37%Couleur et forme :SolidMasse moléculaire :456.92Azacyclonol
CAS :Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.Formule :C18H21NODegré de pureté :99.46%Couleur et forme :Solid PowderMasse moléculaire :267.37Cyproheptadine hydrochloride sesquihydrate
CAS :Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formule :C21H24ClNODegré de pureté :100% - 99.77%Couleur et forme :White To Slightly Yellowish Crystalline SolidMasse moléculaire :341.88Setiptiline maleate
CAS :Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.Formule :C23H23NO4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :377.43LE 300
CAS :LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.Formule :C20H22N2Degré de pureté :98.08% - 98.35%Couleur et forme :SolidMasse moléculaire :290.4Ro60-0175
CAS :Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.Formule :C11H12ClFN2Degré de pureté :97.09%Couleur et forme :SolidMasse moléculaire :226.68Ref: TM-T39161
1mg87,00€5mg216,00€10mg354,00€25mg620,00€50mg847,00€100mg1.169,00€1mL*10mM (DMSO)197,00€5-HT3 antagonist 3
CAS :5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 receptors in rat brain cortical membranes (Ki: 0.25 nM).Formule :C20H21N3ODegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :319.4Ref: TM-T10162
1mg115,00€2mg172,00€5mg255,00€10mg375,00€25mg562,00€50mg792,00€100mg1.064,00€500mgÀ demanderElzasonan hydrochloride
CAS :Elzasonan hydrochloride is a serotonin 1B and serotonin 1D receptor antagonist. It is utilized in the study of depression.Formule :C22H24Cl3N3OSCouleur et forme :SolidMasse moléculaire :484.87ASP-2205
CAS :ASP-2205, a 5-HT2C receptor agonist (human 5-HT2C receptor, EC50=0.85 nM; rat 5-HT2C receptor, EC50=2.5 nM), enhances the urethral closure reflex mediated by the genital nerve, thereby preventing urinary incontinence.Formule :C19H28N2OCouleur et forme :SolidMasse moléculaire :300.44NAN-190 hydrobromide
CAS :NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.Formule :C23H28BrN3O3Degré de pureté :95.92%Couleur et forme :SolidMasse moléculaire :474.39BMY 7378 dihydrochloride
CAS :BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Formule :C22H33Cl2N3O3Degré de pureté :97.32% - 99.08%Couleur et forme :SolidMasse moléculaire :458.42R 59-022 hydrochloride
CAS :R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.Formule :C27H27ClFN3OSDegré de pureté :97.7%Couleur et forme :SolidMasse moléculaire :496.04Desvenlafaxine
CAS :Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.Formule :C16H25NO2Degré de pureté :99.46% - 99.81%Couleur et forme :White Crystalline PowderMasse moléculaire :263.38Pirenperone
CAS :Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Formule :C23H24FN3O2Degré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :393.4525E-NBOMe hydrochloride
CAS :25E-NBOMe hydrochloride is a derivative of 2C-E, featuring an N-(2-methoxybenzyl) addition to the amine group, and acts as a selective agonist of the 5-HT2A receptor.Formule :C20H28ClNO3Couleur et forme :SolidMasse moléculaire :365.89R-137696
CAS :R-137696 is an orally active 5-HT1A receptor agonist that facilitates the relaxation of the proximal stomach. It is utilized in research related to functional dyspepsia.Formule :C17H23N3O2Couleur et forme :SolidMasse moléculaire :301.38AAZ-A 154
CAS :AAZ-A 154 is a selective, competitive, and non-hallucinogenic antagonist of the 5-HT2AR. It promotes neuronal growth in rodents and results in lasting beneficial behavioral effects.Formule :C14H20N2OCouleur et forme :SolidMasse moléculaire :232.32AM9405
AM9405: peripheral CB1/5-HT3 agonist, suppresses gut motility, relieves GI disorder symptoms in mice.Formule :C24H33BrN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.44Roluperidone
CAS :Roluperidone (CYR-101) is a novel cyclic amide derivative.Formule :C22H23FN2O2Degré de pureté :96.46% - 97.77%Couleur et forme :SolidMasse moléculaire :366.43Cariprazine hydrochloride
CAS :Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formule :C21H33Cl3N4ODegré de pureté :100% - 98.52%Couleur et forme :SolidMasse moléculaire :463.87Fluoxetine hydrochloride
CAS :Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.Formule :C17H19ClF3NODegré de pureté :99.6% - 99.98%Couleur et forme :White To Off-White Crystalline Solid White To Off-White PowderMasse moléculaire :345.787Palonosetron hydrochloride
CAS :Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.Formule :C19H24N2O·HClDegré de pureté :99.84% - 99.92%Couleur et forme :White SolidMasse moléculaire :332.87Sevoflurane
CAS :Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.Formule :C4H3F7ODegré de pureté :99.78%Couleur et forme :Less Oil Colorless OilMasse moléculaire :200.05Ref: TM-T22425
2mg42,00€5mg57,00€10mg80,00€25mg116,00€50mg166,00€100mg240,00€200mg359,00€1mL*10mM (DMSO)59,00€Zalospirone
CAS :Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.Formule :C24H29N5O2Degré de pureté :100% - 99%Couleur et forme :SolidMasse moléculaire :419.52ALEPH hydrochloride
CAS :ALEPH (hydrochloride) acts as a partial agonist of h5-HT2A and h5-HT2B receptors, with EC50 values of 10.3 nM and 19.2 nM, respectively. It can induce head twitch responses in mice, with an ED50 of 0.80 mg/kg.Formule :C12H20ClNO2SCouleur et forme :SolidMasse moléculaire :277.81
