récepteur 5-HT
Les récepteurs 5-HT, également connus sous le nom de récepteurs de la sérotonine, sont un groupe de récepteurs couplés aux protéines G (GPCR) qui médiatisent les effets de la sérotonine, un neurotransmetteur impliqué dans la régulation de l'humeur, l'anxiété, le sommeil, l'appétit et d'autres processus physiologiques. Ces récepteurs sont divisés en plusieurs sous-types, chacun ayant des fonctions et des propriétés pharmacologiques distinctes. Les modulateurs des récepteurs 5-HT sont largement étudiés pour leurs rôles dans le traitement de la dépression, des troubles anxieux et d'autres affections neuropsychiatriques. Chez CymitQuimica, nous offrons une gamme de modulateurs des récepteurs 5-HT de haute qualité pour soutenir vos recherches en neuropharmacologie, troubles de l'humeur et signalisation GPCR.
Produits appartenant à la catégorie "récepteur 5-HT"
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Azasetron hydrochloride
CAS :Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.Formule :C17H20ClN3O3·HClDegré de pureté :99.50%Couleur et forme :SolidMasse moléculaire :386.27Trimipramine maleate
CAS :Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.Formule :C24H30N2O4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :410.51Ritanserin
CAS :Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formule :C27H25F2N3OSDegré de pureté :99.45% - 99.89%Couleur et forme :SolidMasse moléculaire :477.57Flumexadol
CAS :Flumexadol is a selective 5-HT2C receptor agonist with an affinity (Ki) of 25 nM for the (+)-enantiomer and exhibits 40-fold selectivity over the 5-HT2A receptor. It is an orally active, non-narcotic analgesic.Formule :C11H12F3NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :231.21DREADD agonist 21
CAS :DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).Formule :C17H18N4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :278.35Ref: TM-T11095L
2mg34,00€5mg58,00€10mg85,00€25mg140,00€50mg221,00€100mg329,00€200mg472,00€1mL*10mM (DMSO)52,00€Mosapride Citrate
CAS :Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.Formule :C21H25ClFN3O3·C6H8O7Degré de pureté :99.70%Couleur et forme :White PowderMasse moléculaire :614.02Itasetron
CAS :Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.Formule :C16H20N4O2Degré de pureté :100% - 99.63%Couleur et forme :SolidMasse moléculaire :300.364-Chloro-L-phenylalanine
CAS :4-Chloro-L-phenalanine (L-PCPA) is an inhibitor of 5-HT biosynthesis and a non-specific antagonist of tryptophan hydroxylases (TPH1 and TPH2).Formule :C9H10ClNO2Degré de pureté :99.76% - 99.96%Couleur et forme :SolidMasse moléculaire :199.63Isocorynoxeine
CAS :Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Formule :C22H26N2O4Degré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :382.45Donitriptan
CAS :Donitriptan 是一种 5-HT 受体激动剂,对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。Formule :C23H25N5O2Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :403.485-MeO-pyr-T
CAS :5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.Formule :C15H20N2OCouleur et forme :SolidMasse moléculaire :244.33PRX-07034 hydrochloride
CAS :PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.Formule :C21H29Cl2N3O4SDegré de pureté :98.50%Couleur et forme :SolidMasse moléculaire :490.44Naftidrofuryl oxalate
CAS :Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.Formule :C26H35NO7Degré de pureté :97.12% - 98.38%Couleur et forme :SolidMasse moléculaire :473.567-Desmethyl-3-hydroxyagomelatine
CAS :7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.Formule :C14H15NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :245.27Etoperidone
CAS :Etoperidone is an antidepressant that acts as an orally active reuptake inhibitor for serotonin (serotonin) and noradrenaline (nor-adrenaline). It demonstrates specific binding affinities (Kd) for several receptors: 36 nM at the 5-HT2 receptor, 38 nM at the α1-adrenergic receptor (α1-adrenergic receptor), 85 nM at the 5-HT1A receptor, and 570 nM at the α2-adrenergic receptor (α2-adrenergic receptor).Formule :C19H28ClN5OCouleur et forme :SolidMasse moléculaire :377.91Org-12962
CAS :Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).Formule :C10H11ClF3N3Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :265.66Perphenazine
CAS :Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.Formule :C21H26ClN3OSDegré de pureté :99.3% - 99.72%Couleur et forme :SolidMasse moléculaire :403.97Eplivanserin
CAS :Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Formule :C19H21FN2O2Degré de pureté :97.04%Couleur et forme :SolidMasse moléculaire :328.38Zotepine
CAS :Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formule :C18H18ClNOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :331.86Jatrorrhizine
CAS :Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Formule :C20H20NO4Degré de pureté :97.18% - 99.06%Couleur et forme :SolidMasse moléculaire :338.38Pridefine
CAS :Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Formule :C19H21NDegré de pureté :99.05% - 99.23%Couleur et forme :SolidMasse moléculaire :263.38YM348
CAS :YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high affinity for the cloned human 5-HT2C receptor (Ki: 0.89 nM).Formule :C14H17N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :243.38-OH-Dpat
CAS :8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.Formule :C16H25NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.38Ethylpropyltryptamine
CAS :Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.Formule :C15H22N2Couleur et forme :SolidMasse moléculaire :230.35Sarpogrelate hydrochloride
CAS :Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.Formule :C24H32ClNO6Degré de pureté :99.73%Couleur et forme :Colorless LiquidMasse moléculaire :465.97Dolasetron Mesylate
CAS :Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea followingFormule :C20H24N2O6SDegré de pureté :100%Couleur et forme :White PowderMasse moléculaire :420.48Deramciclane
CAS :Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Formule :C20H31NOCouleur et forme :SolidMasse moléculaire :301.47NPS ALX Compound 4a
CAS :NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formule :C25H25N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :431.55AAZ-A 154 benzoate
CAS :AAZ-A 154 benzoate is a selective, competitive, and non-hallucinogenic 5-HT2AR antagonist. This compound facilitates neuronal growth in rodents and produces lasting beneficial behavioral effects.Formule :C21H26N2O3Couleur et forme :SolidMasse moléculaire :354.44Nardosinonediol
CAS :Nardosinonediol is a natural compound derived from Nardostachys jatamansi that acts as a SERT inhibitor, regulating serotonin levels and antidepressant.Formule :C15H24O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :252.35Pimethixene
CAS :Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Formule :C19H19NSDegré de pureté :97.50%Couleur et forme :SolidMasse moléculaire :293.43Ref: TM-T12489
2mg34,00€5mg50,00€10mg65,00€25mg106,00€50mg158,00€100mg226,00€200mg339,00€1mL*10mM (DMSO)52,00€SB-269970 hydrochloride
CAS :SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivityFormule :C18H28N2O3S·HClDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :388.95Ogerin
CAS :Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).Formule :C17H17N5ODegré de pureté :99.50% - 99.75%Couleur et forme :SolidMasse moléculaire :307.35Ref: TM-T16378
1mg35,00€2mg52,00€5mg74,00€10mg115,00€25mg227,00€50mg380,00€100mg567,00€1mL*10mM (DMSO)86,00€Tandospirone citrate
CAS :Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Formule :C27H37N5O9Degré de pureté :97.84% - 99.83%Couleur et forme :SolidMasse moléculaire :575.61Quinupramine
CAS :Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formule :C21H24N2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :304.43PF-03382792
CAS :PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.Formule :C23H32FN3O4Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :433.52NPS ALX Compound 4a hydrochloride(1:1)
NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.Formule :C25H26ClN3O2SDegré de pureté :99.8%Couleur et forme :SoildMasse moléculaire :468.01Ref: TM-T12262L1
1mg52,00€5mg114,00€10mg172,00€25mg284,00€50mg411,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)138,00€Flesinoxan
CAS :Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor agonist (EC50: 24 nM).Formule :C22H26FN3O4Couleur et forme :SolidMasse moléculaire :415.46Serazapine
CAS :Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Formule :C22H23N3O2Degré de pureté :98.06% - 99%Couleur et forme :SolidMasse moléculaire :361.44VA012
CAS :VA012 (compound 11) acts as a positive allosteric modulator (PAM) of the serotonin 5-HT2C receptor. It has been shown to reduce food intake and prevent weight gain during subchronic administration without causing central nervous system-related discomfort. VA012 is applicable in obesity research.Formule :C21H19N3Couleur et forme :SolidMasse moléculaire :313.40Dapoxetine hydrochloride
CAS :Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature ejaculation.Formule :C21H23NO·HClDegré de pureté :99.5% - 99.70%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :341.87Amitriptyline hydrochloride
CAS :Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptiveFormule :C20H24ClNDegré de pureté :97% - 99.94%Couleur et forme :Crystals White To Off-White PowderMasse moléculaire :313.865-HT3-In-1
CAS :5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.Formule :C16H21ClN4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.82Piclozotan
CAS :Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)Formule :C23H24ClN3O2Degré de pureté :99%Couleur et forme :SolidMasse moléculaire :409.91NPS ALX Compound 4a dihydrochloride
CAS :NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formule :C25H27Cl2N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :504.47Facinicline hydrochloride
CAS :Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = 6 nM) and an antagonist of 5-HT3(Ki = 1.2 nM).Formule :C15H19ClN4ODegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :306.79BIMU 8
CAS :BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, and 540 nM for wild-type 5HT4 receptor, T3.36A, and W6.48A mutant 5-HT4.Formule :C19H27ClN4O2Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :378.9Ref: TM-T21946
1mg89,00€5mg172,00€10mg249,00€25mg416,00€50mg615,00€100mg873,00€500mg1.768,00€1mL*10mM (DMSO)185,00€Repinotan HCl
CAS :Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.Formule :C21H25ClN2O4SDegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :436.95BF-1
CAS :BF-1 blocks 5-HT2B, may prevent migraines by hindering BW723C86/mCPP in guinea pigs.Formule :C22H25NO2SDegré de pureté :100% - 99.25%Couleur et forme :SolidMasse moléculaire :367.50Vortioxetine hydrobromide
CAS :Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Formule :C18H22N2S·HBrDegré de pureté :100% - 99.89%Couleur et forme :SolidMasse moléculaire :379.36BRL 54443
CAS :BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Formule :C14H18N2ODegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :230.31Melitracen hydrochloride
CAS :Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formule :C21H26ClNDegré de pureté :99.99%Couleur et forme :Crystalline SolidMasse moléculaire :327.9Ref: TM-T4274
10mg47,00€25mg67,00€50mg87,00€100mg116,00€200mg170,00€500mg279,00€1mL*10mM (DMSO)50,00€NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formule :C20H23Cl2F2N3O2Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :446.32Rotundine
CAS :Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formule :C21H25NO4Degré de pureté :100% - 99.8%Couleur et forme :Off-White SolidMasse moléculaire :355.43Iloperidone
CAS :Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Formule :C24H27FN2O4Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :426.48EMDT
CAS :EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Formule :C15H22N2ODegré de pureté :98.33% - 98.46%Couleur et forme :SolidMasse moléculaire :246.35Ref: TM-T11183
1mg92,00€2mg125,00€5mg170,00€10mg213,00€25mg474,00€50mg688,00€100mg938,00€500mg1.882,00€1mL*10mM (DMSO)170,00€Alniditan
CAS :Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.Formule :C17H26N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.41Ziprasidone hydrochloride monohydrate
CAS :Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFormule :C21H21ClN4OS·HCl·H2ODegré de pureté :98% - 99.83%Couleur et forme :Off-White PowderMasse moléculaire :467.12Lurasidone hydrochloride
CAS :Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Formule :C28H36N4O2S·HClDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :529.14(+)-OSU 6162
CAS :(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.Formule :C15H23NO2SDegré de pureté :99.81%Couleur et forme :SoildMasse moléculaire :281.41Ref: TM-T60027
1mg77,00€5mg155,00€10mg220,00€25mg338,00€50mg472,00€100mg632,00€200mg853,00€1mL*10mM (DMSO)163,00€Donitriptan hydrochloride
CAS :Donitriptan hydrochloride (Donitriptan monohydrochloride) is a potent, high efficacy agonist of 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectivelyFormule :C23H26ClN5O2Degré de pureté :99.8% - 99.8%Couleur et forme :SolidMasse moléculaire :439.94Ref: TM-T21666
2mg40,00€5mg49,00€10mg64,00€25mg135,00€50mg240,00€100mg339,00€200mg439,00€500mgÀ demanderSumatriptan succinate
CAS :Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.Formule :C18H27N3O6SDegré de pureté :97.53% - 99.51%Couleur et forme :White PowderMasse moléculaire :413.49Jatrorrhizine chloride
CAS :Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.Formule :C20H20ClNO4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :373.8rac Desmethyl Citalopram Hydrochloride
CAS :rac Desmethyl Citalopram Hydrochloride is a 5-hydroxy tryptamine uptake inhibitor with IC50 value of 0.013 μM.Formule :C19H20ClFN2ODegré de pureté :96.14%Couleur et forme :SolidMasse moléculaire :346.83Tegaserod
CAS :Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).Formule :C16H23N5ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :301.39Lurasidone
CAS :Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formule :C28H36N4O2SDegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :492.68PZ-1922
PZ-1922 (Compound 16), able to cross the blood-brain barrier, is a dual antagonist for 5-HT6R and 5-HT3R with K i values of 17 nM and 0.45 nM, respectively.Degré de pureté :98%Couleur et forme :Odour SolidAlprenolol
CAS :Alprenolol (Alpheprol) is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of the serotonin (5-HT) receptor subtypes 5-HT1AFormule :C15H23NO2Degré de pureté :99.73% - 99.78%Couleur et forme :SolidMasse moléculaire :249.35Mebhydrolin napadisylate
CAS :Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergicFormule :C19H20N2C10H8O6S2Degré de pureté :99.35% - 99.77%Couleur et forme :White Or Almost White CrystallineMasse moléculaire :420.52Zacopride hydrochloride
CAS :Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formule :C15H20ClN3O2·HClDegré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :346.26Ref: TM-T5336
1mg46,00€5mg87,00€10mg144,00€25mg283,00€50mg454,00€100mg655,00€200mg930,00€1mL*10mM (DMSO)97,00€Protriptyline hydrochloride
CAS :Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.Formule :C19H21N·HClDegré de pureté :98.54% - 99.98%Couleur et forme :SolidMasse moléculaire :299.84Sulamserod
CAS :Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular relatedFormule :C19H28ClN3O5SDegré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :445.965-HT2 antagonist 1
CAS :5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.Formule :C22H29FN4O2Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :400.49Ref: TM-T12597
1mg678,00€5mg1.359,00€10mg1.833,00€25mg2.727,00€50mg3.676,00€100mg4.969,00€1mL*10mM (DMSO)1.605,00€Lumateperone
CAS :Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).Formule :C24H28FN3ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :393.5Rilapine
CAS :Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.Formule :C22H20ClN3Degré de pureté :99% - 99.66%Couleur et forme :SolidMasse moléculaire :361.87Masupirdine mesylate
CAS :Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's diseaseFormule :C23H32BrN3O9S3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :670.61Lerisetron
CAS :Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formule :C18H20N4Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :292.38SB-200646
CAS :SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormule :C15H14N4ODegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :266.3Ref: TM-T8357
1mg97,00€2mg150,00€5mg207,00€10mg311,00€25mg525,00€50mg757,00€100mg1.035,00€1mL*10mM (DMSO)216,00€AVN 322 free base
CAS :AVN 322 free base is an orally available, selective and potent 5-HT6R antagonist for the study of neuropathic system disorders such as Alzheimer's disease (AD) and schizophrenia.Formule :C17H19N5O2SDegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :357.435-HT2A&5-HT2C agonist-1
CAS :5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting the 5-HT2A and 5-HT2C receptors with respective IC50 values of 196 nM and 0.9 nM.Formule :C14H20N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :232.325-HT6R antagonist 6
5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.Formule :C24H26N4O2SMasse moléculaire :434.55Masupirdine free base
CAS :Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formule :C21H24BrN3O3SDegré de pureté :97.40% - 98.67%Couleur et forme :SolidMasse moléculaire :478.4Temanogrel
CAS :Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).Formule :C24H28N4O4Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :436.5Ref: TM-T17033
1mg69,00€5mg156,00€10mg225,00€25mg375,00€50mg533,00€100mg723,00€200mg938,00€1mL*10mM (DMSO)170,00€Lesopitron
CAS :Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.Formule :C15H21ClN6Degré de pureté :98.60% - 98.92%Couleur et forme :SolidMasse moléculaire :320.82Harmine
CAS :Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.Formule :C13H12N2ODegré de pureté :98.29% - 99.92%Couleur et forme :Off-White SolidMasse moléculaire :212.258-Hydroxy-DPAT hydrobromide
CAS :8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.Formule :C16H26BrNODegré de pureté :98.90% - 99.09%Couleur et forme :SolidMasse moléculaire :328.29Ketanserin
CAS :Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formule :C22H22FN3O3Degré de pureté :99.19% - 99.73%Couleur et forme :SolidMasse moléculaire :395.43CP94253 hydrochloride
CAS :CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).Formule :C15H20ClN3ODegré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :293.79Ref: TM-T22689
5mg70,00€10mg96,00€25mg216,00€50mg354,00€100mg567,00€200mg787,00€1mL*10mM (DMSO)70,00€Clozapine
CAS :Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.Formule :C18H19ClN4Degré de pureté :99.91% - 99.93%Couleur et forme :Yellow Crystals From Acetone-Petroleum Ether SolidMasse moléculaire :326.82Ref: TM-T0455
1g449,00€10mg35,00€25mg52,00€50mg70,00€100mg96,00€200mg170,00€500mg303,00€1mL*10mM (DMSO)47,00€L-694,247
CAS :L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.Formule :C20H21N5O3SDegré de pureté :98.36%Couleur et forme :White SolidMasse moléculaire :411.48Naftopidil dihydrochloride
CAS :Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.Formule :C24H28N2O3·2HClDegré de pureté :99.76%Couleur et forme :White SolidMasse moléculaire :465.41Phenylbiguanide
CAS :Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Formule :C8H11N5Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :177.21LP-533401 hydrochloride
CAS :LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formule :C27H23ClF4N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :562.94Brexpiprazole HCl
CAS :Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.Formule :C25H27N3O2S·xHClDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :433.6Ref: TM-T8690
1mg131,00€5mg286,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€500mg2.688,00€1mL*10mM (DMSO)338,00€S 16924
CAS :S 16924 is a 5-HT 1A agonist with potential anxiolytic effects and may be useful in the study of neurologic disorders.Formule :C22H24FNO4Degré de pureté :98.23% - 99.45%Couleur et forme :SolidMasse moléculaire :385.43Methamnetamine hydrochloride
CAS :Methamnetamine (PAL-1046) hydrochloride is a psychoactive substance derived from phenethylamine, known to cause excessive serotonin release.Formule :C14H18ClNCouleur et forme :SolidMasse moléculaire :235.75Palonosetron
CAS :Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).Formule :C19H24N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :296.41Syk Inhibitor II
CAS :Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formule :C14H15F3N6ODegré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :340.3SB-224289 hydrochloride
CAS :SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.Formule :C32H33ClN4O3Degré de pureté :97.82% - 98.09%Couleur et forme :SolidMasse moléculaire :557.085-HT2A receptor agonist-3
CAS :5-HT2A receptor agonist-3 represents the highest selectivity for the human 5-HT2A receptor currently identified, exhibiting a K i of 2.5 nM.Formule :C21H26BrNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.34Azatadine dimaleate
CAS :Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).Formule :C28H30N2O8Degré de pureté :100% - 99.70%Couleur et forme :PowderMasse moléculaire :522.555-MeO-MET
CAS :5-MeO-MET (5-Methoxy-N-methyl-N-ethyltryptamine) is a compound belonging to the 5-methoxytryptamine class. It acts as an agonist for 5-HT1A and 5-HT2A receptors. In mice, 5-MeO-MET inhibits locomotion and has sedative effects.Formule :C14H20N2OCouleur et forme :SolidMasse moléculaire :232.32Terfenadine
CAS :Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Formule :C32H41NO2Degré de pureté :98.76% - 99.75%Couleur et forme :SolidMasse moléculaire :471.67GR 113808
CAS :GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.Formule :C19H27N3O4SDegré de pureté :98.16%Couleur et forme :SolidMasse moléculaire :393.5Pimavanserin
CAS :Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.Formule :C25H34FN3O2Degré de pureté :97.84% - 99.69%Couleur et forme :Pale Yellow To Pale Orange SolidMasse moléculaire :427.55Xaliproden hydrochloride
CAS :Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formule :C24H23ClF3NDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :417.89Ref: TM-T9272
1mg40,00€5mg85,00€10mg120,00€25mg235,00€50mg376,00€100mg540,00€200mg775,00€1mL*10mM (DMSO)96,00€PF-04995274
CAS :PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.Formule :C23H32N2O6Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :432.51Pellotine
CAS :Pellotine is an alkaloid isolated from Lophophora. It acts as an inverse agonist of the 5-HT7 receptor (5-HT7 receptor), with an EC50 of 291 nM. Pellotine shows strong affinity for the 5-HT1DR and 5-HT6R, with Ki values of 117 nM and 170 nM, respectively. Additionally, Pellotine reduces intracellular cAMP levels, thereby decreasing neuronal excitability and neurotransmitter release.Formule :C13H19NO3Couleur et forme :SolidMasse moléculaire :237.295Amperozide
CAS :Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Formule :C23H29F2N3ODegré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :401.49Ref: TM-T23733
1mg92,00€5mg188,00€10mg311,00€25mg525,00€50mg747,00€100mg1.017,00€500mg2.023,00€1mL*10mM (DMSO)339,00€Paroxetine hydrochloride hemihydrate
CAS :Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).Formule :C38H44Cl2F2N2O7Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :749.67BRL-15572 dihydrochloride
CAS :BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.Formule :C25H27ClN2O·2HClDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :479.874-Chloromethamphetamine hydrochloride
CAS :4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.Formule :C10H15Cl2NCouleur et forme :SolidMasse moléculaire :220.144F 4PP oxalate
CAS :4F 4PP oxalate is a 5-HT2A antagonist.Formule :C22H26FNO·C2H2O4Degré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :429.49Ref: TM-T22514
5mg46,00€10mg80,00€25mg131,00€50mg210,00€100mg313,00€200mg445,00€1mL*10mM (DMSO)49,00€Lintopride HCl
CAS :Lintopride HCl is a 5HT-4 antagonist.Formule :C14H20Cl2N4O2Degré de pureté :97.70% - 98.42%Couleur et forme :SoildMasse moléculaire :347.24Ramosetron hydrochloride
CAS :Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.Formule :C17H18ClN3ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :315.8RS 42358-197
CAS :RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Formule :C19H23ClN2ODegré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :330.85Ref: TM-T20739
1mg166,00€5mg371,00€10mg557,00€25mg827,00€50mg1.111,00€100mg1.491,00€200mg2.015,00€1mL*10mM (DMSO)369,00€Lesopitron dihydrochloride
CAS :Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Formule :C15H23Cl3N6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :393.74RS 56812
CAS :RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive disorders.Formule :C18H21N3O2Degré de pureté :98.78%Couleur et forme :SoildMasse moléculaire :311.38Eptapirone
CAS :Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.Formule :C16H23N7O2Degré de pureté :99.39% - 99.65%Couleur et forme :SolidMasse moléculaire :345.4Talipexole dihydrochloride
CAS :Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical andFormule :C10H17Cl2N3SDegré de pureté :98.64%Couleur et forme :Light Yellow SolidMasse moléculaire :282.23Ref: TM-T14490
2mg38,00€5mg56,00€10mg89,00€25mg154,00€50mg264,00€100mg424,00€200mg613,00€500mg949,00€1mL*10mM (DMSO)63,00€RS102895 hydrochloride
CAS :RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).Formule :C21H22ClF3N2O2Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :426.86(-)-5-HT2C agonist-3
CAS :Compound (−)-19, also known as (-)-5-HT2C agonist-3, is a selective 5-HT2C agonist exhibiting a preference for Gq signaling. It demonstrates efficiency with EC50 values for 5-HT2 receptor subtypes as follows: 5-HT2C at 103 nM, 5-HT2B at 570 nM, and 5-HT2A at 72 nM. This compound is utilized in research on antipsychotics.Formule :C19H23ClFNO2Couleur et forme :SolidMasse moléculaire :351.84SCH-23390 maleate
CAS :SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formule :C21H22ClNO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :403.864i
CAS :4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.Formule :C16H12ClN3ODegré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :297.74Flibanserin
CAS :Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.Formule :C20H21F3N4ODegré de pureté :99.37% - 99.93%Couleur et forme :White PowderMasse moléculaire :390.4Flopropione
CAS :Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.Formule :C9H10O4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :182.17PRX-08066 Maleic acid
CAS :PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Formule :C23H21ClFN5O4SDegré de pureté :97.59%Couleur et forme :SolidMasse moléculaire :517.96Ref: TM-T6959
1mg90,00€5mg186,00€10mg252,00€25mg454,00€50mg660,00€100mg939,00€200mg1.276,00€1mL*10mM (DMSO)435,00€SCH-23390 hydrochloride
CAS :SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formule :C17H19Cl2NODegré de pureté :98% - 99.51%Couleur et forme :SolidMasse moléculaire :324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€F13714 fumarate
CAS :F13714 fumarate is a 5-HT1A receptor-biased agonist.Formule :C25H29ClF2N4O5Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :538.975-Carboxamidotryptamine maleate
CAS :5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.Formule :C15H17N3O5Degré de pureté :97.77%Couleur et forme :SolidMasse moléculaire :319.316-Fluoro-N,N-diethyltryptamine
CAS :6-Fluoro-N,N-diethyltryptamine (6-F-DET) exhibits affinity for the 5-HT2A receptor.Formule :C14H19FN2Couleur et forme :SolidMasse moléculaire :234.31SEP-363856 mesylate
CAS :SEP-363856 (SEP-856) mesylate is an orally active compound that acts as an agonist for both TAAR1 and 5-HT1A receptors. This compound exhibits antipsychotic activity in the central nervous system and has potential for the study of schizophrenia.Formule :C10H17NO4S2Couleur et forme :SolidMasse moléculaire :279.38AAZ-A 154 mesylate
CAS :AAZ-A 154 mesylate mesylate is a selective, competitive, and non-hallucinogenic antagonist of 5-HT2AR. It enhances neuronal growth in rodents and produces enduring beneficial behavioral effects.Formule :C15H24N2O4SCouleur et forme :SolidMasse moléculaire :328.43Ondansetron hydrochloride
CAS :Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiationFormule :C18H19N3O·HClDegré de pureté :99.78%Couleur et forme :White PowderMasse moléculaire :329.8225B-NBOH hydrochloride
CAS :25B-NBOH hydrochloride is a phenethylamine that exhibits high affinity for serotonin (5-HT) receptors 5-HT2A and 5-HT2C, with pKi values of 8.3 and 9.4, respectively.Formule :C17H21BrClNO3Couleur et forme :SolidMasse moléculaire :402.711SB-203186 hydrochloride
CAS :SB 203186 hydrochloride is a potent 5-HT4 receptor antagonistFormule :C16H20N2O2·HClDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :308.81Loxapine succinate
CAS :Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.Formule :C22H24ClN3O5Degré de pureté :99.69%Couleur et forme :White To Of-White SolidMasse moléculaire :445.9Lecozotan HCl
CAS :Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.Formule :C28H30ClN5O3Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :520.02QF0301B
CAS :QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.Formule :C23H28N2O2Degré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :364.48Neocarzinostatin
CAS :Neocarzinostatin is an effective DNA-damaging, anti-tumor antibiotic.Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :N/ADapoxetine
CAS :Dapoxetine (Dapoxetina) is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation.Formule :C21H23NODegré de pureté :99.73%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :305.42Fananserin
CAS :Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Formule :C23H24FN3O2SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :425.52Ref: TM-T15270
2mg42,00€5mg56,00€10mg81,00€25mg116,00€50mg170,00€100mg250,00€200mg369,00€1mL*10mM (DMSO)62,00€Pimavanserin tartrate
CAS :Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.Formule :C50H68F2N6O4·C4H6O6Degré de pureté :100% - 99.98%Couleur et forme :SolidMasse moléculaire :1005.2Ziprasidone
CAS :Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.Formule :C21H21ClN4OSDegré de pureté :100% - 99.53%Couleur et forme :Tan SolidMasse moléculaire :412.94GM-60186
GM-60186, a potent inhibitor of the 5-HT receptor 2B (HTR2B) with an IC50 of 257 nM, effectively suppresses the proliferation and migration of colorectal cancer cells.Formule :C30H33FN2O4Couleur et forme :SolidMasse moléculaire :504.59Anpirtoline hydrochloride
CAS :Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.Formule :C10H14Cl2N2SDegré de pureté :100% - 100%Couleur et forme :SolidMasse moléculaire :265.20Quetiapine hemifumarate
CAS :Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formule :C46H54N6O8S2Degré de pureté :100% - 99.59%Couleur et forme :White Crystalline SolidMasse moléculaire :883.09Agomelatine
CAS :Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.Formule :C15H17NO2Degré de pureté :99.92%Couleur et forme :White SolidMasse moléculaire :243.3Rizatriptan benzoate
CAS :Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFormule :C22H25N5O2Degré de pureté :99% - 99.72%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :391.47Ref: TM-T1512
10mg47,00€25mg79,00€50mg126,00€100mg183,00€200mg273,00€500mg462,00€1mL*10mM (DMSO)50,00€Ansofaxine hydrochloride
CAS :Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formule :C24H32ClNO3Degré de pureté :99.57% - 99.77%Couleur et forme :SolidMasse moléculaire :417.97RS-127445 hydrochloride
CAS :RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).Formule :C17H17ClFN3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :317.795-HT6 agonist 1
Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting plateletFormule :C17H22Cl2N6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.37Paliperidone
CAS :Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.Formule :C23H27FN4O3Degré de pureté :95% - 99.08%Couleur et forme :Off White To Light Orange Coloured SolidMasse moléculaire :426.48Lintopride
CAS :Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Formule :C14H19ClN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.78(R)-Mirtazapine
CAS :(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formule :C17H19N3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :265.35Metergoline
CAS :Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formule :C25H29N3O2Degré de pureté :99.7% - 99.83%Couleur et forme :SolidMasse moléculaire :403.52F-15599
CAS :F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).Formule :C19H21ClF2N4ODegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :394.85Buclizine dihydrochloride
CAS :Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormule :C28H33ClN2·2HClDegré de pureté :98.05%Couleur et forme :Off-White PowderMasse moléculaire :505.95idalopirdine
CAS :Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Formule :C20H19F5N2ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :398.37Ref: TM-T7103
1mg88,00€2mg118,00€5mg188,00€10mg254,00€25mg429,00€50mg630,00€100mg898,00€1mL*10mM (DMSO)187,00€Org 13011
CAS :Org 13011 has CNS activity and induces conditioned taste aversion by mediating 5-HT 1A receptors.Formule :C18H25F3N4ODegré de pureté :98.98%Couleur et forme :SoildMasse moléculaire :370.41Ref: TM-T28258L
1mg185,00€5mg459,00€10mg657,00€25mg1.026,00€50mg1.415,00€100mg1.872,00€1mL*10mM (DMSO)469,00€Opiranserin
CAS :Opiranserin is a development as an injectable agent for the treatment of postoperative pain.Formule :C21H34N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.51Ampreloxetine
CAS :Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.Formule :C18H18F3NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.34Trazodone
CAS :Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.Formule :C19H22ClN5ODegré de pureté :99.79%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :371.86Arotinolol hydrochloride
CAS :Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.Formule :C15H22ClN3O2S3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :408Myristicin
CAS :Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.Formule :C11H12O3Degré de pureté :99.34%Couleur et forme :LiquidMasse moléculaire :192.21LY-2624803
CAS :LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Formule :C22H25N3O3Degré de pureté :100% - 99.87%Couleur et forme :SolidMasse moléculaire :379.45RS 67333 hydrochloride
CAS :RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Formule :C19H30Cl2N2O2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :389.36Naratriptan hydrochloride
CAS :Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.Formule :C17H25N3O2S·HClDegré de pureté :99.17% - 99.89%Couleur et forme :Beige SolidMasse moléculaire :371.93Ref: TM-T6602
10mg50,00€25mg88,00€50mg133,00€100mg188,00€200mg283,00€500mg467,00€1mL*10mM (DMSO)52,00€Prucalopride Succinate
CAS :Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formule :C18H26ClN3O3·C4H6O4Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :485.96Dehydroaripiprazole
CAS :Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.Formule :C23H25Cl2N3O2Degré de pureté :97.05%Couleur et forme :SolidMasse moléculaire :446.37THRX-194556
CAS :THRX-194556 is an agonist of the 5-HT4 receptor. It is applicable in the study of gastrointestinal functional disorders and Alzheimer's disease.Formule :C28H41N5O5SCouleur et forme :SolidMasse moléculaire :559.721Blonanserin
CAS :Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formule :C23H30FN3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :367.5Metoclopramide
CAS :Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formule :C14H22ClN3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :299.8Brilaroxazine
CAS :Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.Formule :C22H25Cl2N3O3Degré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :450.36Ref: TM-T14782
1mg105,00€5mg250,00€10mg406,00€25mg700,00€50mg1.008,00€100mg1.378,00€200mg1.833,00€1mL*10mM (DMSO)283,00€p-MPPI hydrochloride
CAS :p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.Formule :C25H28ClIN4O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :578.87Capeserod
CAS :Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive disorders and neurological disorders.Formule :C23H25ClN4O4Degré de pureté :98.82% - 99.37%Couleur et forme :SolidMasse moléculaire :456.92Azacyclonol
CAS :Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.Formule :C18H21NODegré de pureté :99.46%Couleur et forme :Solid PowderMasse moléculaire :267.37Cyproheptadine hydrochloride sesquihydrate
CAS :Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formule :C21H24ClNODegré de pureté :100% - 99.77%Couleur et forme :White To Slightly Yellowish Crystalline SolidMasse moléculaire :341.88Setiptiline maleate
CAS :Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.Formule :C23H23NO4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :377.43LE 300
CAS :LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.Formule :C20H22N2Degré de pureté :98.08% - 98.35%Couleur et forme :SolidMasse moléculaire :290.4Ro60-0175
CAS :Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.Formule :C11H12ClFN2Degré de pureté :97.09%Couleur et forme :SolidMasse moléculaire :226.68Ref: TM-T39161
1mg87,00€5mg216,00€10mg354,00€25mg620,00€50mg847,00€100mg1.169,00€1mL*10mM (DMSO)197,00€5-HT3 antagonist 3
CAS :5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 receptors in rat brain cortical membranes (Ki: 0.25 nM).Formule :C20H21N3ODegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :319.4Ref: TM-T10162
1mg115,00€2mg172,00€5mg255,00€10mg375,00€25mg562,00€50mg792,00€100mg1.064,00€500mgÀ demanderElzasonan hydrochloride
CAS :Elzasonan hydrochloride is a serotonin 1B and serotonin 1D receptor antagonist. It is utilized in the study of depression.Formule :C22H24Cl3N3OSCouleur et forme :SolidMasse moléculaire :484.87ASP-2205
CAS :ASP-2205, a 5-HT2C receptor agonist (human 5-HT2C receptor, EC50=0.85 nM; rat 5-HT2C receptor, EC50=2.5 nM), enhances the urethral closure reflex mediated by the genital nerve, thereby preventing urinary incontinence.Formule :C19H28N2OCouleur et forme :SolidMasse moléculaire :300.44NAN-190 hydrobromide
CAS :NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.Formule :C23H28BrN3O3Degré de pureté :95.92%Couleur et forme :SolidMasse moléculaire :474.39BMY 7378 dihydrochloride
CAS :BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Formule :C22H33Cl2N3O3Degré de pureté :97.32% - 99.08%Couleur et forme :SolidMasse moléculaire :458.42R 59-022 hydrochloride
CAS :R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.Formule :C27H27ClFN3OSDegré de pureté :97.7%Couleur et forme :SolidMasse moléculaire :496.04Desvenlafaxine
CAS :Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.Formule :C16H25NO2Degré de pureté :99.46% - 99.81%Couleur et forme :White Crystalline PowderMasse moléculaire :263.38Pirenperone
CAS :Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Formule :C23H24FN3O2Degré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :393.4525E-NBOMe hydrochloride
CAS :25E-NBOMe hydrochloride is a derivative of 2C-E, featuring an N-(2-methoxybenzyl) addition to the amine group, and acts as a selective agonist of the 5-HT2A receptor.Formule :C20H28ClNO3Couleur et forme :SolidMasse moléculaire :365.89R-137696
CAS :R-137696 is an orally active 5-HT1A receptor agonist that facilitates the relaxation of the proximal stomach. It is utilized in research related to functional dyspepsia.Formule :C17H23N3O2Couleur et forme :SolidMasse moléculaire :301.38AAZ-A 154
CAS :AAZ-A 154 is a selective, competitive, and non-hallucinogenic antagonist of the 5-HT2AR. It promotes neuronal growth in rodents and results in lasting beneficial behavioral effects.Formule :C14H20N2OCouleur et forme :SolidMasse moléculaire :232.32AM9405
AM9405: peripheral CB1/5-HT3 agonist, suppresses gut motility, relieves GI disorder symptoms in mice.Formule :C24H33BrN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.44Roluperidone
CAS :Roluperidone (CYR-101) is a novel cyclic amide derivative.Formule :C22H23FN2O2Degré de pureté :96.46% - 97.77%Couleur et forme :SolidMasse moléculaire :366.43Cariprazine hydrochloride
CAS :Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formule :C21H33Cl3N4ODegré de pureté :100% - 98.52%Couleur et forme :SolidMasse moléculaire :463.87Fluoxetine hydrochloride
CAS :Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.Formule :C17H19ClF3NODegré de pureté :99.6% - 99.98%Couleur et forme :White To Off-White Crystalline Solid White To Off-White PowderMasse moléculaire :345.787Palonosetron hydrochloride
CAS :Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.Formule :C19H24N2O·HClDegré de pureté :99.84% - 99.92%Couleur et forme :White SolidMasse moléculaire :332.87Sevoflurane
CAS :Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.Formule :C4H3F7ODegré de pureté :99.78%Couleur et forme :Less Oil Colorless OilMasse moléculaire :200.05Ref: TM-T22425
2mg42,00€5mg57,00€10mg80,00€25mg116,00€50mg166,00€100mg240,00€200mg359,00€1mL*10mM (DMSO)59,00€Zalospirone
CAS :Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.Formule :C24H29N5O2Degré de pureté :100% - 99%Couleur et forme :SolidMasse moléculaire :419.52ALEPH hydrochloride
CAS :ALEPH (hydrochloride) acts as a partial agonist of h5-HT2A and h5-HT2B receptors, with EC50 values of 10.3 nM and 19.2 nM, respectively. It can induce head twitch responses in mice, with an ED50 of 0.80 mg/kg.Formule :C12H20ClNO2SCouleur et forme :SolidMasse moléculaire :277.81
