récepteur 5-HT
Les récepteurs 5-HT, également connus sous le nom de récepteurs de la sérotonine, sont un groupe de récepteurs couplés aux protéines G (GPCR) qui médiatisent les effets de la sérotonine, un neurotransmetteur impliqué dans la régulation de l'humeur, l'anxiété, le sommeil, l'appétit et d'autres processus physiologiques. Ces récepteurs sont divisés en plusieurs sous-types, chacun ayant des fonctions et des propriétés pharmacologiques distinctes. Les modulateurs des récepteurs 5-HT sont largement étudiés pour leurs rôles dans le traitement de la dépression, des troubles anxieux et d'autres affections neuropsychiatriques. Chez CymitQuimica, nous offrons une gamme de modulateurs des récepteurs 5-HT de haute qualité pour soutenir vos recherches en neuropharmacologie, troubles de l'humeur et signalisation GPCR.
Produits appartenant à la catégorie "récepteur 5-HT"
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TIK-301
CAS :TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nMFormule :C14H17ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :280.75Alverine citrate
CAS :Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.Formule :C26H35NO7Degré de pureté :98.53% - 99.43%Couleur et forme :CoaMasse moléculaire :473.57Clomipramine
CAS :Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by hindering serotonin reuptake.Formule :C19H23ClN2Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :314.85Rizatriptan
CAS :Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.Formule :C15H19N5Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :269.35WAY-100635 Monomaleate
CAS :WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Formule :C25H34N4O2·C4H4O4Degré de pureté :99.26% - 99.68%Couleur et forme :SolidMasse moléculaire :538.64Ref: TM-T2631
2mg46,00€5mg66,00€10mg95,00€25mg180,00€50mg334,00€100mg495,00€200mg717,00€500mg1.111,00€1mL*10mM (DMSO)79,00€Sertraline hydrochloride
CAS :Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.Formule :C17H18Cl3NDegré de pureté :99.12% - 99.89%Couleur et forme :Solid PowderMasse moléculaire :342.691Ref: TM-T0482
5mg51,00€10mg63,00€25mg103,00€50mg180,00€100mg235,00€200mg304,00€500mg515,00€1mL*10mM (DMSO)57,00€4-Bromo-2,5-DMMA
CAS :4-Bromo-2,5-DMMA (Compound 2) demonstrates affinity for the 5-HT2 binding site and has an ED50 of 0.82 mg/kg in rat discrimination experiments.Formule :C12H18BrNO2Couleur et forme :SolidMasse moléculaire :288.18SB 699551 dihydrochloride
CAS :SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.Formule :C34H47Cl2N3ODegré de pureté :96.53%Couleur et forme :SolidMasse moléculaire :584.66Ref: TM-T23325
1mg52,00€5mg111,00€10mg180,00€25mg311,00€50mg449,00€100mg615,00€1mL*10mM (DMSO)150,00€Tianeptine sodium salt
CAS :Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。Formule :C21H24ClN2NaO4SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :458.93Vortioxetine
CAS :Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formule :C18H22N2SDegré de pureté :99.34% - 99.34%Couleur et forme :SolidMasse moléculaire :298.45Ref: TM-T2395
1g505,00€10mg50,00€25mg69,00€50mg95,00€100mg124,00€200mg215,00€500mg350,00€1mL*10mM (DMSO)48,00€Perospirone
CAS :Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formule :C23H30N4O2SDegré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :426.57Tropisetron hydrochloride
CAS :Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.Formule :C17H21ClN2O2Degré de pureté :99.72% - 99.83%Couleur et forme :SolidMasse moléculaire :320.82Cinanserin hydrochloride
CAS :Cinanserin hydrochloride (SQ 10643) is a 5-HT2 receptor blocker (Ki: 41 nM) and SARS-CoV 3C-like protease inhibitor.Formule :C20H25ClN2OSDegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :376.94Idalopirdine Hydrochloride
CAS :Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.Formule :C20H20ClF5N2ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :434.83Ref: TM-T22936
1mg64,00€2mg87,00€5mg116,00€10mg167,00€25mg283,00€50mg424,00€100mg598,00€200mg805,00€1mL*10mM (DMSO)125,00€3-AQC
CAS :3-AQC is a competitive antagonist of 5-HT3.Formule :C20H21N5O4Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :395.41Ref: TM-T8475
2mg35,00€5mg50,00€10mg66,00€25mg95,00€50mg140,00€100mg205,00€200mg304,00€1mL*10mM (DMSO)57,00€Rodatristat ethyl
CAS :Rodatristat ethyl is an oral TPH1 inhibitor reducing 5-HT levels & lowering PAH at low doses.Formule :C29H31ClF3N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :590.04LY 272015 hydrochloride
CAS :LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formule :C21H25ClN2O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :372.89Seganserin
CAS :Seganserin, a 5-HT2 antagonist, negates fluoxetine and quipazine's effects on hyperphagia, depression, and pain.Formule :C29H27F2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :471.54PRX-08066
CAS :PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.Formule :C19H17ClFN5SDegré de pureté :98.04% - 98.07%Couleur et forme :SolidMasse moléculaire :401.89Ref: TM-T16669
1mg60,00€5mg119,00€10mg170,00€25mg350,00€50mg522,00€100mg748,00€200mg1.026,00€1mL*10mM (DMSO)111,00€Vabicaserin hydrochloride
CAS :Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).Formule :C15H21ClN2Degré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :264.79Ref: TM-T13275
1mg84,00€5mg178,00€10mg264,00€25mg424,00€50mg562,00€100mg775,00€200mg1.026,00€1mL*10mM (DMSO)188,00€Alprenolol hydrochloride
CAS :Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.Formule :C15H24ClNO2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :285.81Tabernanthalog
CAS :TBG is a 5-HT2A agonist reducing alcohol/heroin cravings and promoting neuroplasticity with antidepressant effects in rodents.Formule :C14H18N2ODegré de pureté :98.57%Couleur et forme :SoildMasse moléculaire :230.31Ref: TM-T60221
1mg185,00€2mg279,00€5mg425,00€10mg625,00€25mg938,00€50mg1.311,00€100mg1.795,00€500mg3.591,00€1mL*10mM (DMSO)364,00€S 32212 hydrochloride
CAS :S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .Formule :C25H29ClN4O2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :452.98Osemozotan HCl
CAS :Osemozotan is a 5-HT1A receptor agonist potentially for the treatment of generalized anxiety disorder.Formule :C19H22ClNO5Degré de pureté :98.87% - 99.63%Couleur et forme :SolidMasse moléculaire :379.84Quetiapine
CAS :Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.Formule :C21H25N3O2SDegré de pureté :100% - 99.14%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :383.51SB-269970
CAS :SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).Formule :C18H28N2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.49SB 243213 dihydrochloride
CAS :SB 243213 dihydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8 forFormule :C22H21Cl2F3N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :501.33EMD 56551
CAS :EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.Formule :C24H31N3O2Degré de pureté :95.07% - 99.39%Couleur et forme :SolidMasse moléculaire :393.522Urapidil hydrochloride
CAS :Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.Formule :C20H29N5O3·HClDegré de pureté :99.58%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :423.94Serotonin hydrochloride
CAS :Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (Formule :C10H13ClN2ODegré de pureté :98.05% - 99.93%Couleur et forme :White To Cream PowderMasse moléculaire :212.6764-Hydroxy MET
CAS :4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.Formule :C13H18N2OCouleur et forme :SolidMasse moléculaire :218.3E6801
CAS :E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.Formule :C17H18ClN5O2S2Degré de pureté :100% - 96.66%Couleur et forme :SolidMasse moléculaire :423.94PNU-142633
CAS :PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; >18,000 nM for 5-HT1B.Formule :C24H30N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :422.52SB 216641
CAS :SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety disorders and depression.Formule :C28H30N4O4Degré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :486.56Fluvoxamine maleate
CAS :Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFormule :C19H25F3N2O6Degré de pureté :99.92% - 99.94%Couleur et forme :White Crystalline PowderMasse moléculaire :434.41Ref: TM-T1077
10mg51,00€25mg69,00€50mg85,00€100mg115,00€200mg170,00€500mg278,00€1mL*10mM (DMSO)52,00€Ramosetron
CAS :Ramosetron 是一种血清素 5-HT3 受体拮抗剂,用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。Formule :C17H17N3ODegré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :279.34Homoeriodictyol
CAS :Homoeriodictyol, a naturally occurring, bitter-masking flavanone, as a promising agent to increase appetite and food intake.Formule :C16H14O6Degré de pureté :99.34% - 99.96%Couleur et forme :SolidMasse moléculaire :302.282'-O-Methylisoliquiritigenin
CAS :2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formule :C16H14O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :270.285-HT2A antagonist 1
CAS :5-HT2A antagonist 1, from US5728835A & JP 1007727, may treat gastrointestinal and circulatory issues.Formule :C26H28N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.53Vilazodone Hydrochloride
CAS :Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormule :C26H27N5O2·HClDegré de pureté :100% - 99.56%Couleur et forme :SolidMasse moléculaire :477.99SB 258585
CAS :SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.Formule :C18H22IN3O3SDegré de pureté :99.8%Couleur et forme :SoildMasse moléculaire :487.36Lamotrigine
CAS :Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.Formule :C9H7Cl2N5Degré de pureté :99.76% - 99.95%Couleur et forme :White To Pale Cream-Colored Powder Crystals From Isopropanol SolidMasse moléculaire :256.095-IAI hydrochloride
CAS :5-IAI hydrochloride is a psychoactive analog of para-iodoamphetamine. 5-IAI hydrochloride significantly reduces serotonin uptake sites and hippocampal serotonin levels in rats.Formule :C9H11ClINCouleur et forme :SolidMasse moléculaire :295.548HDAC6-IN-49
HDAC6-IN-49 (Compound 3) is an inhibitor of HDAC, with IC50 values of 0.012 and 0.735 µM against HDAC6 and HDAC1, respectively. Additionally, it inhibits MAO-B, cholinesterase (ChE), histamine receptor (H3R), and serotonin 6 receptor (5-HT6R). HDAC6-IN-49 exhibits neuroprotective effects in SH-SY5Y cells and enhances cognitive functions and motor abilities in fruit fly models of Parkinson's disease and C. elegans models of Alzheimer's disease.Couleur et forme :Odour Solid5-HT4 antagonist 1
CAS :5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).Formule :C23H36N4O5SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :480.62Sumatriptan
CAS :Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.Formule :C14H21N3O2SDegré de pureté :99.93%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :295.4(Iso)-Landipirdine
CAS :(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.Formule :C18H19FN2O3SDegré de pureté :97.27%Couleur et forme :SoildMasse moléculaire :362.42LY 344864 racemate
CAS :LY 344864 racemate is a 5-HT1F receptor agonist.Formule :C21H22FN3ODegré de pureté :99.47%Couleur et forme :SoildMasse moléculaire :351.42SB228357
CAS :SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.Formule :C22H17F4N3O2Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :431.38PU02
CAS :PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.Formule :C16H12N4SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :292.36Cericlamine
CAS :Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.Formule :C12H17Cl2NODegré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :262.18AVN-101
CAS :AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Formule :C21H25ClN2Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :340.89Ref: TM-T26690
1mg35,00€5mg80,00€10mg120,00€25mg216,00€50mg354,00€100mg588,00€200mg833,00€1mL*10mM (DMSO)97,00€SAX-187
CAS :SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formule :C15H13ClN4O2S2Degré de pureté :97.82% - 98%Couleur et forme :SolidMasse moléculaire :380.87Ref: TM-T3183
1mg84,00€5mg160,00€10mg259,00€25mg419,00€50mg562,00€100mg775,00€200mg1.026,00€1mL*10mM (DMSO)170,00€Granisetron
CAS :Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.Formule :C18H24N4OCouleur et forme :SolidMasse moléculaire :312.41Opiranserin hydrochloride
CAS :Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormule :C21H35ClN2O5Degré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :430.97Ref: TM-T9833
1mg96,00€5mg227,00€10mg359,00€25mg652,00€50mg929,00€100mg1.293,00€500mg2.593,00€1mL*10mM (DMSO)250,00€Zolmitriptan
CAS :Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Formule :C16H21N3O2Degré de pureté :99.69% - 99.91%Couleur et forme :White Or Kind Of White PowderMasse moléculaire :287.36ML 10302 hydrochloride
CAS :ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.Formule :C15H22Cl2N2O3Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :349.255-HT1A modulator 2 hydrochloride
CAS :5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.Formule :C11H16ClNODegré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :213.7LY310762
CAS :LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Formule :C24H27FN2O2·HClDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :430.94Metoclopramide hydrochloride hydrate
CAS :Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formule :C14H25Cl2N3O3Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :354.27Isobutyryl-L-carnitine
CAS :Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a product of the acyl-CoA dehydrogenases.Formule :C11H21NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :231.29Felcisetrag
CAS :Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.Formule :C25H37N5O3Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :455.59Ref: TM-T28934
1mg155,00€5mg378,00€10mg560,00€25mg898,00€50mg1.216,00€100mg1.644,00€500mg3.287,00€1mL*10mM (DMSO)415,00€Iferanserin
CAS :Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors.Formule :C23H28N2OCouleur et forme :SolidMasse moléculaire :348.483-Hydroxy agomelatine
CAS :3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.Formule :C15H17NO3Couleur et forme :SolidMasse moléculaire :259.3JNJ-18038683
CAS :JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.Formule :C26H28ClN3O7Degré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :529.97Ref: TM-T11720
2mg35,00€5mg50,00€10mg90,00€25mg170,00€50mg259,00€100mg383,00€200mg545,00€1mL*10mM (DMSO)55,00€7-Methyl DMT
CAS :7-Methyl DMT (7-TMT) acts as a 5-HT2 receptor agonist. Structurally, it is a tryptamine derivative and serves as an analytical reference for the psychoactive substance DOM. It is also applicable in research related to neurological disorders.Formule :C13H18N2Couleur et forme :SolidMasse moléculaire :202.32-Bromo-6-methoxynaphthalene
CAS :2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.Formule :C11H9BrODegré de pureté :98.51%Couleur et forme :White To Off-White PowderMasse moléculaire :237.09SB399885
CAS :SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.Formule :C18H21Cl2N3O4SDegré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :446.35Ref: TM-T19669
1mg87,00€5mg170,00€10mg253,00€25mg418,00€50mg562,00€100mg792,00€200mg1.064,00€1mL*10mM (DMSO)207,00€SB-215505
CAS :SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).Formule :C19H16ClN3ODegré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :337.8DOAM
CAS :DOAM is an antagonist of the 5-HT2 receptor.Formule :C16H27NO2Couleur et forme :SolidMasse moléculaire :265.39Azaphen
CAS :Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.Formule :C16H21Cl2N5ODegré de pureté :97.62%Couleur et forme :SolidMasse moléculaire :370.28Granisetron hydrochloride
CAS :Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapyFormule :C18H25ClN4ODegré de pureté :99.88% - 99.93%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :348.87Eltoprazine hydrochloride
CAS :Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formule :C12H17ClN2O2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :256.73Perospirone hydrochloride
CAS :Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formule :C23H31ClN4O2SDegré de pureté :99.37%Couleur et forme :White SolidMasse moléculaire :463RU 24969 free base
CAS :RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.Formule :C14H16N2ODegré de pureté :97.38%Couleur et forme :SolidMasse moléculaire :228.296-fluoro-DL-Tryptophan
CAS :6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.Formule :C11H11FN2O2Degré de pureté :99.25%Couleur et forme :Off-White PowderMasse moléculaire :222.22TG6-10-1
CAS :TG6-10-1 is an EP2 antagonist.Formule :C23H23F3N2O4Degré de pureté :100% - ≥95%Couleur et forme :SolidMasse moléculaire :448.43Epinastine hydrochloride
CAS :Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formule :C16H15N3·HClDegré de pureté :99.26% - 99.62%Couleur et forme :White SolidMasse moléculaire :285.77Binospirone
CAS :Binospirone (MDL 73005EF) is a 5-HT1A receptor agonist with anxiolytic activity used in the study of movement disorders associated with neurologic dysfunction.Formule :C20H26N2O4Degré de pureté :98.05% - 99.11%Couleur et forme :SoildMasse moléculaire :358.43AP521
CAS :AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).Formule :C20H19ClN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :402.89Hymenidin HCl
CAS :Hymenidin HCl is a natural alkaloid that acts as 5-HT receptor antagonist. Hymenidin HCl inhibits Kv and CDK5 and induces apoptosis in cancer cells.Formule :C11H13BrClN5ODegré de pureté :99.95%Couleur et forme :SoildMasse moléculaire :346.61E-3620
CAS :E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.Formule :C20H27Cl2N3O2Degré de pureté :98.88% - 98.88%Couleur et forme :SolidMasse moléculaire :412.35MK 212 hydrochloride
CAS :MK 212 hydrochloride is a 5-HT2C receptor agonistFormule :C8H11ClN4·HClDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :235.12CP-809101
CAS :CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formule :C15H17ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :304.77(4E)-SUN9221
CAS :(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity inFormule :C25H31FN4O3Degré de pureté :97.79%Couleur et forme :SolidMasse moléculaire :454.54Enciprazine
CAS :Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.Formule :C23H32N2O6Degré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :432.51Brompheniramine maleate
CAS :Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.Formule :C16H19BrN2·C4H4O4Degré de pureté :99.80%Couleur et forme :Crystal PowderMasse moléculaire :435.31Pancopride
CAS :Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-inducedFormule :C18H24ClN3O2Degré de pureté :93.64%Couleur et forme :SolidMasse moléculaire :349.86Norfluoxetine Hydrochloride
CAS :Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.Formule :C16H17ClF3NODegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :331.76Ref: TM-T21029
1mg48,00€5mg135,00€10mg205,00€25mg369,00€50mg502,00€100mg727,00€200mg1.017,00€1mL*10mM (DMSO)99,00€SB 258719
CAS :SB 258719 is a selective antagonist of 5-HT7 receptor with pKi of 7.5.Formule :C18H30N2O2SDegré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :338.51Ref: TM-T12855
2mg35,00€5mg55,00€10mg89,00€25mg163,00€50mg254,00€100mg375,00€200mg530,00€1mL*10mM (DMSO)62,00€Tandospirone
CAS :Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.Formule :C21H29N5O2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :383.49Ref: TM-TQ0315
2mg38,00€5mg57,00€10mg92,00€25mg148,00€50mg204,00€100mg325,00€200mg466,00€1mL*10mM (DMSO)63,00€ADR-851 free base
CAS :ADR-851 free base is an antagonist of the HT3 receptor.Formule :C14H18ClN3O2Degré de pureté :97.88% - 98.32%Couleur et forme :SolidMasse moléculaire :295.77Naluzotan
CAS :Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+Formule :C23H38N4O3SDegré de pureté :100%Couleur et forme :SolidMasse moléculaire :450.64Eplivanserin (mixture)
CAS :Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,Formule :C19H21FN2O2Couleur et forme :SolidMasse moléculaire :328.387Tegaserod maleate
CAS :Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March 30, 2007, due to heart risk concerns.Formule :C20H27N5O5Degré de pureté :98% - 99.06%Couleur et forme :White PowderMasse moléculaire :417.46Ref: TM-T1551
10mg47,00€25mg79,00€50mg119,00€100mg198,00€200mg301,00€500mg509,00€1mL*10mM (DMSO)50,00€Setiptiline
CAS :Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formule :C19H19NDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :261.36Sarizotan HCl
CAS :Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.Formule :C22H22ClFN2ODegré de pureté :96%Couleur et forme :SolidMasse moléculaire :384.87Spiperone
CAS :Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.Formule :C23H26FN3O2Degré de pureté :99.34% - 99.89%Couleur et forme :SolidMasse moléculaire :395.47Zatosetron maleate
CAS :Zatosetron maleate(LY 277359 maleate) is a potent and selective serotonin 5HT3 receptor antagonist for the study of acute migraine.Formule :C23H29ClN2O6Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :464.94Nuciferine
CAS :Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.Formule :C19H21NO2Degré de pureté :98.76% - 99.18%Couleur et forme :SolidMasse moléculaire :295.38Ricasetron
CAS :Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Formule :C19H27N3ODegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :313.44(±)-Fabesetron hydrochloride
CAS :FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist.Formule :C18H20ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.82PNU-282987 free base
CAS :PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.Formule :C14H17ClN2ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :264.75SB-616234-A
CAS :SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant activity.Formule :C32H36ClN5O3Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :574.11Ref: TM-T12847
1mg105,00€5mg255,00€10mg368,00€25mg557,00€50mg752,00€100mg1.035,00€200mg1.396,00€1mL*10mM (DMSO)321,00€5-HT2A/5-HT2C inverse agonist 1
CAS :5-HT2A/5-HT2C inverse agonist 1 serves as a dual and potent inverse agonist for the 5-HT2A and 5-HT2C receptors, with hERG inhibition properties that mitigate cardiovascular risks. Demonstrating significant antipsychotic efficacy in the MK-801-induced mouse model, this compound holds potential for psychosis research.Formule :C24H35N5O2Couleur et forme :SolidMasse moléculaire :425.57Lofepramine
CAS :Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.Formule :C26H27ClN2ODegré de pureté :98.38%Couleur et forme :Crystals From Methanol Or Acetone SolidMasse moléculaire :418.96Escitalopram Oxalate
CAS :Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Formule :C22H23FN2O5Degré de pureté :97.39% - 99.73%Couleur et forme :White SolidMasse moléculaire :414.43Ref: TM-T6493
1g283,00€10mg39,00€25mg55,00€50mg66,00€100mg90,00€200mg125,00€500mg197,00€1mL*10mM (DMSO)44,00€SB-399885 hydrochloride
CAS :SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.Formule :C18H22Cl3N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.81CP-809101 hydrochloride
CAS :CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formule :C15H18Cl2N4ODegré de pureté :99.50%Couleur et forme :SolidMasse moléculaire :341.24Femoxetine hydrochloride
CAS :Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Formule :C20H26ClNO2Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :347.88Almotriptan
CAS :Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Formule :C17H25N3O2SDegré de pureté :99.85%Couleur et forme :Light Yellow Or White PowerMasse moléculaire :335.462-Methyl-5-HT hydrochloride
CAS :2-Methyl-5-HT hydrochloride (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.Formule :C11H15ClN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :226.7(S)-Mirtazapine
CAS :(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Formule :C17H19N3Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :265.35AS19
CAS :AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).Formule :C18H25N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :283.41CP 96021
CAS :"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."Formule :C29H21FN4OSDegré de pureté :97.81% - 99.11%Couleur et forme :SoildMasse moléculaire :492.57Nelotanserin
CAS :Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).Formule :C18H15BrF2N4O2Degré de pureté :98.01% - 98.42%Couleur et forme :SolidMasse moléculaire :437.24Ref: TM-T7350
1mg40,00€2mg52,00€5mg88,00€10mg119,00€25mg188,00€50mg350,00€100mg522,00€500mg1.130,00€1mL*10mM (DMSO)85,00€Piboserod
CAS :Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formule :C22H31N3O2Degré de pureté :97.21% - 99.49%Couleur et forme :SolidMasse moléculaire :369.5Ref: TM-T2278
1mg40,00€2mg52,00€5mg88,00€10mg125,00€25mg233,00€50mg424,00€100mg613,00€500mg1.264,00€1mL*10mM (DMSO)127,00€2,6-DMA hydrochloride
CAS :2,6-DMA hydrochloride is a phenethylamine and acts as an agonist of the serotonin 5-HT2 receptor, with a pA2 value of 5.09.Formule :C11H18ClNO2Couleur et forme :SolidMasse moléculaire :231.72Ketanserin tartrate
CAS :Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formule :C26H28FN3O9Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :545.51Paynantheine
CAS :Paynantheine is an alkaloid with antinociceptive properties, found in Mitragyna speciosa. It also acts as an agonist at 5-HT1AR and 5-HT2BR receptors, inducing lower lip contraction and providing antinociception in rats.Formule :C23H28N2O4Couleur et forme :SolidMasse moléculaire :396.48Maprotiline hydrochloride
CAS :Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.Formule :C20H24ClNDegré de pureté :99.68% - 99.84%Couleur et forme :White PowderMasse moléculaire :313.864Ticalopride
CAS :Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formule :C14H20ClN3O3Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :313.78cis-Urocanic acid
CAS :cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).Formule :C6H6N2O2Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :138.12Rotigotine-
CAS :Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formule :C19H25NOSDegré de pureté :98.08% - 99.59%Couleur et forme :SolidMasse moléculaire :315.47Ref: TM-T6647
5mg52,00€10mg78,00€25mg145,00€50mg255,00€100mg378,00€200mg552,00€500mg868,00€1mL*10mM (DMSO)55,00€
