Récepteur de la dopamine
Les récepteurs de la dopamine sont un groupe de récepteurs couplés aux protéines G (GPCR) qui répondent au neurotransmetteur dopamine, jouant un rôle clé dans la régulation du mouvement, de la motivation, de la récompense et de plusieurs fonctions cognitives. Ces récepteurs sont divisés en familles de type D1 et de type D2, chacune ayant des fonctions et des profils pharmacologiques distincts. Les modulateurs des récepteurs de la dopamine sont largement étudiés pour leurs applications dans le traitement de la maladie de Parkinson, de la schizophrénie, de la dépendance et d'autres troubles neuropsychiatriques. Chez CymitQuimica, nous offrons une large gamme de modulateurs de récepteurs de la dopamine de haute qualité pour soutenir vos recherches en neurosciences, santé mentale et signalisation GPCR.
Produits appartenant à la catégorie "Récepteur de la dopamine"
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NRA-0160
CAS :NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)Formule :C24H23F2N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.52Tiaspirone hydrochloride
CAS :Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity and influences the electrophysiological activity of dopaminergic neurons.Formule :C24H33ClN4O2SDegré de pureté :99.98%Couleur et forme :SoildMasse moléculaire :477.065-HT6/7 antagonist 1
CAS :5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.Formule :C22H20FN3O3Degré de pureté :98.55% - 98.78%Couleur et forme :SolidMasse moléculaire :393.41Benperidol
CAS :Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.Formule :C22H24FN3O2Degré de pureté :97.39%Couleur et forme :SolidMasse moléculaire :381.44Ref: TM-T26360
1mg116,00€5mg276,00€10mg410,00€25mg680,00€50mg938,00€100mg1.293,00€500mg2.593,00€1mL*10mM (DMSO)279,00€Liafensine
CAS :Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.Formule :C24H22N4Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :366.46Asenapine
CAS :Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophreniaFormule :C17H16ClNODegré de pureté :99.16%Couleur et forme :CoaMasse moléculaire :285.77SLV-310
CAS :SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.Formule :C25H24FN3O2Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :417.48D3R/MOR antagonist 1
Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nMFormule :C22H27Cl2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.38Metoclopramide hydrochloride
CAS :Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.Formule :C14H22ClN3O2·HClDegré de pureté :99.99%Couleur et forme :White To Off-White PowderMasse moléculaire :336.26NMI 8739
CAS :NMI 8739 (n-docosahexaenoyl dopamine) is an agonist of D2 autoreceptor.Formule :C30H41NO3Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :463.65Ref: TM-T11079
1mg40,00€5mg85,00€10mg120,00€25mg207,00€50mg303,00€100mg449,00€200mg652,00€1mL*10mM (DMSO)90,00€Itopride hydrochloride
CAS :Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.Formule :C20H27ClN2O4Degré de pureté :99.59%Couleur et forme :White Or Pale Brownish CrystalMasse moléculaire :394.9Oxolinic acid
CAS :Oxolinic acid (Nidantin) is a synthetic antimicrobial related to NALIDIXIC ACID and used in URINARY TRACT INFECTIONS.Formule :C13H11NO5Degré de pureté :98.39% - 99.72%Couleur et forme :Crystals From Dimethylformamide White Crystalline PowderMasse moléculaire :261.23Fluphenazine decanoate
CAS :Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.Formule :C32H44F3N3O2SDegré de pureté :100% - 98.14%Couleur et forme :SolidMasse moléculaire :591.77Benztropine mesylate
CAS :Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSONFormule :C21H25NO·CH4SO3Degré de pureté :98.41% - 99.96%Couleur et forme :White Crystalline Powder; Odourless Or Almost OdourlessMasse moléculaire :403.53Syrosingopine
CAS :Syrosingopine is a dual inhibitor of MCT1 and MCT4, 60 times more potent against MCT4, preventing lactate and H+ efflux.Cost-effective and quality-assured.Formule :C35H42N2O11Degré de pureté :99.25% - 99.78%Couleur et forme :SolidMasse moléculaire :666.71Ref: TM-TN2252
1mg66,00€5mg142,00€10mg212,00€25mg361,00€50mg543,00€100mg750,00€1mL*10mM (DMSO)202,00€GR 103691
CAS :GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).Formule :C30H35N3O3Degré de pureté :98.94% - 99.29%Couleur et forme :SolidMasse moléculaire :485.62Ref: TM-T11463
2mg46,00€5mg66,00€10mg99,00€25mg197,00€50mg311,00€100mg505,00€500mg1.121,00€1mL*10mM (DMSO)74,00€PF-00217830
CAS :PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.Formule :C26H30N4O2Degré de pureté :98.30%Couleur et forme :SolidMasse moléculaire :430.54Aniracetam
CAS :Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.Formule :C12H13NO3Degré de pureté :99.88% - 99.89%Couleur et forme :White Crystalline Or Crystalline PowdeMasse moléculaire :219.24Oxidopamine hydrobromide
CAS :Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.Formule :C8H12BrNO3Degré de pureté :98.1% - 99.88%Couleur et forme :Beige To Brown Fine Crystalline PowderMasse moléculaire :250.09Flunarizine dihydrochloride
CAS :Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.Formule :C26H28Cl2F2N2Degré de pureté :99.53% - 99.89%Couleur et forme :White Crystalline Powder Odorless And TastelessMasse moléculaire :477.42Pardoprunox
CAS :Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formule :C12H15N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :233.27Amisulpride
CAS :Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.Formule :C17H27N3O4SDegré de pureté :99.97%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :369.48Bendazol
CAS :Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.Formule :C14H12N2Degré de pureté :98.7% - 99.81%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :208.26Chlorprothixene hydrochloride
CAS :Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formule :C18H18ClNS·HClDegré de pureté :99.16%Couleur et forme :White PowderMasse moléculaire :352.32Aplindore Fumarate
CAS :Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Formule :C22H22N2O7Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :426.42SKF 38393 hydrochloride
CAS :SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.Formule :C16H17NO2·HClDegré de pureté :98.70% - 99.1%Couleur et forme :SolidMasse moléculaire :291.77Perphenazine
CAS :Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.Formule :C21H26ClN3OSDegré de pureté :99.3% - 99.72%Couleur et forme :SolidMasse moléculaire :403.97Zotepine
CAS :Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formule :C18H18ClNOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :331.86Glaucine
CAS :Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.Formule :C21H25NO4Degré de pureté :99.14% - 99.42%Couleur et forme :SolidMasse moléculaire :355.43Dexchlorpheniramine Maleate
CAS :Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.Formule :C20H23ClN2O4Degré de pureté :99.58%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :390.86Bromperidol
CAS :Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.Formule :C21H23BrFNO2Degré de pureté :99.89%Couleur et forme :Tan SolidMasse moléculaire :420.32Mesoridazine Besylate
CAS :Mesoridazine Besylate (Serentil), a piperidine antipsychotic and phenothiazine, treats schizophrenia; it's a thioridazine metabolite.Formule :C27H32N2O4S3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :544.75U 99194 maleate
CAS :U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.Formule :C21H31NO6Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :393.47Sertindole
CAS :Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).Formule :C24H26ClFN4ODegré de pureté :99.74%Couleur et forme :Off-White To Pale Yellow SolidMasse moléculaire :440.94PG 01037 dihydrochloride
CAS :PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.Formule :C26H28Cl4N4ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :554.34Ref: TM-T23143
1mg42,00€2mg52,00€5mg82,00€10mg105,00€25mg168,00€50mg249,00€100mg369,00€200mg522,00€1mL*10mM (DMSO)97,00€ABT 724 trihydrochloride
CAS :ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.Formule :C17H22Cl3N5Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :402.75Ref: TM-T22019
5mg40,00€10mg65,00€25mg126,00€50mg188,00€100mg283,00€200mg419,00€1mL*10mM (DMSO)44,00€7-Hydroxy-DPAT hydrobromide
CAS :7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.Formule :C16H26BrNODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :328.29Carmoxirole hydrochloride
CAS :Carmoxirole hydrochloride (EMD 45609 hydrochloride) is a selective dopamine D2 receptor agonist with antihypertensive activity in vivo.Formule :C24H27ClN2O2Degré de pureté :97.8% - 98.12%Couleur et forme :SolidMasse moléculaire :410.94Ref: TM-T10683
1mg58,00€5mg117,00€10mg178,00€25mg306,00€50mg452,00€100mg620,00€200mg835,00€1mL*10mM (DMSO)134,00€SKF-83566
CAS :SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.Formule :C17H18BrNODegré de pureté :95.00% - 99.82%Couleur et forme :SolidMasse moléculaire :332.23SKF83959
CAS :SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.Formule :C18H20ClNO2Degré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :317.81Ref: TM-T60835
1mg52,00€5mg103,00€10mg169,00€25mg359,00€50mg530,00€100mg758,00€1mL*10mM (DMSO)114,00€GSK163090
CAS :GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).Formule :C25H29N5ODegré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :415.53Ref: TM-TQ0311
1mg37,00€2mg52,00€5mg80,00€10mg125,00€25mgÀ demander50mgÀ demander1mL*10mM (DMSO)87,00€Tavapadon
CAS :Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Formule :C19H16F3N3O3Degré de pureté :99.33% - 99.8%Couleur et forme :SolidMasse moléculaire :391.34Ref: TM-T16999
1mg81,00€5mg170,00€10mg274,00€25mg502,00€50mg705,00€100mg938,00€1mL*10mM (DMSO)188,00€Mianserin hydrochloride
CAS :Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.Formule :C18H21ClN2Degré de pureté :99.63% - 99.82%Couleur et forme :White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedMasse moléculaire :300.83UNC9975
CAS :UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.Formule :C23H28Cl2N4O2Degré de pureté :99.02% - 99.02%Couleur et forme :SolidMasse moléculaire :463.4Risperidone
CAS :Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.Formule :C23H27FN4O2Degré de pureté :99.73%Couleur et forme :Crystalline SolidMasse moléculaire :410.48Pipamperone
CAS :Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.Formule :C21H30FN3O2Degré de pureté :99.94%Couleur et forme :White PowderMasse moléculaire :375.48Ref: TM-T12480
1mg62,00€2mg85,00€5mg119,00€10mg170,00€25mg283,00€50mg430,00€100mg622,00€1mL*10mM (DMSO)131,00€Promazine hydrochloride
CAS :Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Formule :C17H21ClN2SDegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :320.88Brexpiprazole
CAS :Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formule :C25H27N3O2SDegré de pureté :99.06% - 99.96%Couleur et forme :SolidMasse moléculaire :433.57lumateperone Tosylate
CAS :lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formule :C31H36FN3O4SDegré de pureté :95.83% - 98.57%Couleur et forme :SolidMasse moléculaire :565.7MLS1547
CAS :MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).Formule :C19H19ClN4ODegré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :354.83Sulpiride
CAS :Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.Formule :C15H23N3O4SDegré de pureté :99.94%Couleur et forme :White Crystalline PowderMasse moléculaire :341.43JNJ-37822681 dihydrochloride
CAS :JNJ-37822681 dihydrochloride 是特异性的、有中枢活性的,可快速解离的多巴胺 D2受体拮抗剂,与多巴胺 D2L 受体结合的亲和力适中 (Ki=158 nM)。JNJ-37822681 dihydrochloride 在精神分裂症和躁郁症领域有研究价值。Formule :C17H19Cl2F5N4Degré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :445.26Pramipexole dihydrochloride hydrate
CAS :Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.Formule :C10H17N3S·2HCl·H2ODegré de pureté :99.68%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :302.26Ref: TM-T6951
10mg47,00€25mg74,00€50mg119,00€100mg170,00€200mg255,00€500mg430,00€1mL*10mM (DMSO)47,00€Ziprasidone hydrochloride monohydrate
CAS :Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFormule :C21H21ClN4OS·HCl·H2ODegré de pureté :98% - 99.83%Couleur et forme :Off-White PowderMasse moléculaire :467.12D5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Couleur et forme :Odour SolidTrimethobenzamide hydrochloride
CAS :Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Formule :C21H29ClN2O5Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :424.92Fosopamine(HCl)
CAS :Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.Formule :C9H15ClNO5PDegré de pureté :100%Couleur et forme :SolidMasse moléculaire :283.65Alizapride hydrochloride
CAS :Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formule :C16H21N5O2·HClDegré de pureté :99.35% - 99.48%Couleur et forme :CoaMasse moléculaire :351.83Loxapine
CAS :Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.Formule :C18H18ClN3ODegré de pureté :99.88%Couleur et forme :Pale Yellowish Crystals From Petroleum Ether SolidMasse moléculaire :327.81Cabergoline
CAS :Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.Formule :C26H37N5O2Degré de pureté :99.86%Couleur et forme :White Crystalline SolidMasse moléculaire :451.6Ergocornine
CAS :Ergocornine is a naturally occurring ergot alkaloid and acts as a dopamine receptor (dopamine receptor) agonist.Formule :C31H39N5O5Couleur et forme :SolidMasse moléculaire :561.67Nomifensine
CAS :Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.Formule :C16H18N2Degré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :238.33Atomoxetine hydrochloride
CAS :Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.Formule :C17H22ClNODegré de pureté :99.86%Couleur et forme :White SolidMasse moléculaire :291.82Rotigotine Hydrochloride
CAS :Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.Formule :C19H26ClNOSDegré de pureté :99.53% - 99.56%Couleur et forme :Almost White To White Crystalline PowderMasse moléculaire :351.935-Benzyloxygramine
CAS :5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formule :C18H20N2ODegré de pureté :96.33%Couleur et forme :SolidMasse moléculaire :280.36Ropinirole hydrochloride
CAS :Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.Formule :C16H24N2O·HClDegré de pureté :99.87% - 99.98%Couleur et forme :Off-White SolidMasse moléculaire :296.84UCSF924
CAS :UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).Formule :C20H22N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :322.4Medifoxamine
CAS :Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.MedifoxamineFormule :C16H19NO2Degré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :257.33Ref: TM-T24444
1mg99,00€5mg235,00€10mg354,00€25mg635,00€50mg893,00€100mg1.159,00€1mL*10mM (DMSO)259,00€DOPEXAMINE
CAS :Dopexamine is a dopaminergic agonistFormule :C22H32N2O2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :356.5Ref: TM-T8653
1mg131,00€2mg188,00€5mg284,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€1mL*10mM (DMSO)306,00€Trimipramine maleate
CAS :Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.Formule :C24H30N2O4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :410.51Dopamine D2 receptor agonist-2
CAS :Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.Formule :C25H31Cl2N5OSDegré de pureté :98.93%Couleur et forme :SoildMasse moléculaire :520.52Ref: TM-T60075
1mg38,00€5mg71,00€10mg90,00€25mg148,00€50mg210,00€100mg314,00€200mg452,00€1mL*10mM (DMSO)90,00€Propionylpromazine hydrochloride
CAS :Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.Formule :C20H25ClN2OSDegré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :376.94Ritanserin
CAS :Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formule :C27H25F2N3OSDegré de pureté :99.45% - 99.89%Couleur et forme :SolidMasse moléculaire :477.57Fluphenazine dihydrochloride
CAS :Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.Formule :C22H28Cl2F3N3OSDegré de pureté :99.23%Couleur et forme :Off-White SolidMasse moléculaire :510.44Thiethylperazine dimaleate
CAS :Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor.Formule :C30H37N3O8S2Degré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :631.76carfenazine
CAS :carfenazine targets the Dopamine receptor and is used for schizophrenia research.Formule :C24H31N3O2SDegré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :425.59Trifluoperazine
CAS :Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.Formule :C21H24F3N3SDegré de pureté :98.3% - 99.46%Couleur et forme :White To Yellowish Crystalline PowderMasse moléculaire :407.5(-)-GSK598809 hydrochloride
CAS :(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.Formule :C22H24ClF4N5OSDegré de pureté :97.66%Couleur et forme :SoildMasse moléculaire :517.97Molindone
CAS :Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.Formule :C16H24N2O2Degré de pureté :98% - 99.37%Couleur et forme :Off-White SolidMasse moléculaire :276.37Foscarbidopa
CAS :Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.Formule :C10H15N2O7PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :306.21Dasotraline hydrochloride
CAS :Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formule :C16H16Cl3NDegré de pureté :98.92% - 99.6%Couleur et forme :SolidMasse moléculaire :328.66Nolomirole HCl
CAS :Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory effects on norepinephrine release, which can be used to studyFormule :C19H28ClNO4Degré de pureté :100% - 99.12%Couleur et forme :SolidMasse moléculaire :369.88Brexpiprazole S-oxide
CAS :Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).Formule :C25H27N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :449.57Tedatioxetine
CAS :Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Formule :C18H21NSDegré de pureté :100% - 98.58%Couleur et forme :SolidMasse moléculaire :283.43UNC10099984A
CAS :UNC10099984A (Compound 6) is a functionally selective ligand for the dopamine D2 receptor, exhibiting a Ki value of 4.6 nM and an EC50 of 6.2 nM for β-arrestin. This compound is useful for research into central nervous system diseases related to the D2 receptor.Formule :C24H29Cl2N3O2Couleur et forme :SolidMasse moléculaire :462.41Xaliproden hydrochloride
CAS :Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formule :C24H23ClF3NDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :417.89Ref: TM-T9272
1mg40,00€5mg85,00€10mg120,00€25mg235,00€50mg376,00€100mg540,00€200mg775,00€1mL*10mM (DMSO)96,00€Pimethixene
CAS :Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Formule :C19H19NSDegré de pureté :97.50%Couleur et forme :SolidMasse moléculaire :293.43Ref: TM-T12489
2mg34,00€5mg50,00€10mg65,00€25mg106,00€50mg158,00€100mg226,00€200mg339,00€1mL*10mM (DMSO)52,00€Methyldopa hydrate
CAS :Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.Formule :C10H13NO4H2ODegré de pureté :99.67%Couleur et forme :White SolidMasse moléculaire :238.24Tolnapersine TFA
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.Formule :C23H27F3N2O3Degré de pureté :98.10%Couleur et forme :SoildMasse moléculaire :436.47L-DOPA
CAS :L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is converted to dopamine by DOPA decarboxylase.Formule :C9H11NO4Degré de pureté :98.99% - 99.93%Couleur et forme :Colorless To White Crystals Or Crystalline Powder; Needles From Water SolidMasse moléculaire :197.19Abaperidone
CAS :Abaperidone is an atypical antipsychotic, antagonizes 5-HT2A (IC50=6.2 nM) and D2 receptors (IC50=17 nM), reduces hsp70 mRNA in rat brains.Formule :C25H25FN2O5Degré de pureté :94.35%Couleur et forme :SolidMasse moléculaire :452.47A-77636
CAS :A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50Formule :C20H27NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.43Diclofensine
CAS :Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.Formule :C17H17Cl2NODegré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :322.23Melitracen hydrochloride
CAS :Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formule :C21H26ClNDegré de pureté :99.99%Couleur et forme :Crystalline SolidMasse moléculaire :327.9Ref: TM-T4274
10mg47,00€25mg67,00€50mg87,00€100mg116,00€200mg170,00€500mg279,00€1mL*10mM (DMSO)50,00€BP 897
CAS :BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Formule :C26H31N3O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :417.54Ref: TM-T9100
1mg80,00€5mg162,00€10mg227,00€25mg379,00€50mg540,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)177,00€Rotundine
CAS :Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formule :C21H25NO4Degré de pureté :100% - 99.8%Couleur et forme :Off-White SolidMasse moléculaire :355.43Iloperidone
CAS :Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Formule :C24H27FN2O4Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :426.48D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.Formule :C27H37NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.59Methyldopa
CAS :Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFormule :C10H13NO4Degré de pureté :99.86% - 99.89%Couleur et forme :Less Or Almost Colorless Crystals Or White To Yellowish-White FineMasse moléculaire :211.21Lurasidone hydrochloride
CAS :Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Formule :C28H36N4O2S·HClDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :529.14Fallypride
CAS :Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.Formule :C20H29FN2O3Degré de pureté :100% - 99.17%Couleur et forme :SolidMasse moléculaire :364.45Ref: TM-T70302
1mg359,00€5mg842,00€10mg1.035,00€25mg1.663,00€50mg2.072,00€100mg2.660,00€1mL*10mM (DMSO)677,00€Loxapine succinate
CAS :Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.Formule :C22H24ClN3O5Degré de pureté :99.69%Couleur et forme :White To Of-White SolidMasse moléculaire :445.95-HT7R antagonist 3
CAS :Compound 6.4, also known as 5-HT7R antagonist 3, is a selective antagonist of the 5-HT7R with a Ki of 8 nM. It exhibits significantly less affinity towards D2R, 5-HT1AR, and 5-HT2AR with Ki values of 511 nM, 8930 nM, and 5786 nM, respectively. In mice, 5-HT7R antagonist 3 demonstrates anti-depressant and anti-anxiety activities.Formule :C30H33FN4O3Couleur et forme :SolidMasse moléculaire :516.61Pericyazine
CAS :Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.Formule :C21H23N3OSDegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :365.49Ref: TM-T16472
1mg46,00€2mg59,00€5mg93,00€10mg124,00€25mg235,00€50mg389,00€100mg567,00€500mg1.225,00€1mL*10mM (DMSO)77,00€Piribedil
CAS :Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.Formule :C16H18N4O2Degré de pureté :99.79% - 99.91%Couleur et forme :SolidMasse moléculaire :298.34Fananserin
CAS :Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Formule :C23H24FN3O2SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :425.52Ref: TM-T15270
2mg42,00€5mg56,00€10mg81,00€25mg116,00€50mg170,00€100mg250,00€200mg369,00€1mL*10mM (DMSO)62,00€Fipexide
CAS :Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983.Formule :C20H21ClN2O4Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :388.84Lurasidone
CAS :Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formule :C28H36N4O2SDegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :492.68(Rac)-Rotigotine hydrochloride
CAS :(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.Formule :C19H26ClNOSCouleur et forme :SolidMasse moléculaire :351.93Docosahexaenoic acid ethyl ester
CAS :Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.Formule :C24H36O2Couleur et forme :SolidMasse moléculaire :356.54Amantadine hydrochloride
CAS :Amantadine hydrochloride (CI-719) is an antiviral that is used in the prophylactic or symptomatic treatment of influenza A and Parkinson disease.Formule :C10H18ClNDegré de pureté :99.98%Couleur et forme :Solid CrystallineMasse moléculaire :187.71Sonepiprazole
CAS :Sonepiprazole (PNU-101387G) is a chemical compound known for its selective antagonistic properties toward D4 dopamine receptors, exhibiting dissociationFormule :C21H27N3O3SDegré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :401.52Ref: TM-T23380
2mg38,00€5mg58,00€10mg94,00€25mg180,00€50mg306,00€100mg442,00€200mg622,00€1mL*10mM (DMSO)71,00€UCM-1306
CAS :UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.Formule :C14H14FNO2SDegré de pureté :100%Couleur et forme :SoildMasse moléculaire :279.33Ansofaxine hydrochloride
CAS :Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formule :C24H32ClNO3Degré de pureté :99.57% - 99.77%Couleur et forme :SolidMasse moléculaire :417.97Paliperidone
CAS :Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.Formule :C23H27FN4O3Degré de pureté :95% - 99.08%Couleur et forme :Off White To Light Orange Coloured SolidMasse moléculaire :426.48Mesdopetam hemitartrate
CAS :Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.Formule :C28H42F2N2O12S2Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :700.77Lumateperone
CAS :Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).Formule :C24H28FN3ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :393.5Haloperidol
CAS :Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function.Formule :C21H23ClFNO2Degré de pureté :98.69% - 98.97%Couleur et forme :Crystals SolidMasse moléculaire :375.86Moperone
CAS :Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.Formule :C22H26FNO2Couleur et forme :SolidMasse moléculaire :355.45PD-168077 maleate
CAS :PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)Formule :C24H26N4O5Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :450.49Ref: TM-T5047
2mg35,00€5mg52,00€10mg80,00€25mg150,00€50mg245,00€100mg364,00€200mg517,00€1mL*10mM (DMSO)58,00€L-745870 hydrochloride
CAS :L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptorFormule :C18H20Cl2N4Degré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :363.28Ref: TM-T11799
5mg40,00€10mg65,00€25mg111,00€50mg178,00€100mg259,00€200mg374,00€1mL*10mM (DMSO)34,00€Levosulpiride
CAS :Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Formule :C15H23N3O4SDegré de pureté :98.20% - 99.88%Couleur et forme :White Crystalline PowderMasse moléculaire :341.43Diclofensine hydrochloride
CAS :Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Formule :C17H18Cl3NODegré de pureté :98.86% - 99.93%Couleur et forme :SolidMasse moléculaire :358.69FAUC 213
CAS :FAUC 213 is a selective full antagonist of the dopamine D4 receptor.Formule :C18H19ClN4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :326.82Nomifensine maleate
CAS :Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.Formule :C20H22N2O4Degré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :354.4Tolnapersine
CAS :Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.Formule :C21H26N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :322.44Clozapine
CAS :Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.Formule :C18H19ClN4Degré de pureté :99.91% - 99.93%Couleur et forme :Yellow Crystals From Acetone-Petroleum Ether SolidMasse moléculaire :326.82Ref: TM-T0455
1g449,00€10mg35,00€25mg52,00€50mg70,00€100mg96,00€200mg170,00€500mg303,00€1mL*10mM (DMSO)47,00€Brexpiprazole HCl
CAS :Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.Formule :C25H27N3O2S·xHClDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :433.6Ref: TM-T8690
1mg131,00€5mg286,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€500mg2.688,00€1mL*10mM (DMSO)338,00€A-381393
CAS :A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).Formule :C20H24N4Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :320.43Ref: TM-T5397
1mg40,00€5mg80,00€10mg117,00€25mg210,00€50mg304,00€100mg437,00€200mg615,00€1mL*10mM (DMSO)88,00€Hirsuteine
CAS :Hirsuteine: natural product; blocks nicotine effects on dopamine by hindering ion flow in receptor channels.Formule :C22H26N2O3Degré de pureté :99.36% - 99.63%Couleur et forme :SolidMasse moléculaire :366.45Pramipexole dihydrochloride
CAS :Pramipexole dihydrochloride could be used to treat Parkinson disease.Formule :C10H18ClN3SDegré de pureté :98%Couleur et forme :White Crystalline PowderMasse moléculaire :247.79D1R antagonist 1
CAS :Compound 12a (D1R antagonist 1) is a D1R antagonist that participates in both G-protein-coupled and β-arrestin-mediated signaling pathways [1].Formule :C22H26BrNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.35Tetrahydropalmatine hydrochloride
CAS :Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.Formule :C21H26ClNO4Degré de pureté :98% - 99.59%Couleur et forme :SolidMasse moléculaire :391.888PF2562
CAS :PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).Formule :C19H17N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.37AHN 1-055 hydrochloride
CAS :AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).Formule :C21H24ClF2NODegré de pureté :99.60%Couleur et forme :SolidMasse moléculaire :379.87Ref: TM-T39429
2mg35,00€5mg52,00€10mg80,00€25mg137,00€50mg202,00€100mg311,00€200mg467,00€1mL*10mM (DMSO)52,00€Talipexole dihydrochloride
CAS :Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical andFormule :C10H17Cl2N3SDegré de pureté :98.64%Couleur et forme :Light Yellow SolidMasse moléculaire :282.23Ref: TM-T14490
2mg38,00€5mg56,00€10mg89,00€25mg154,00€50mg264,00€100mg424,00€200mg613,00€500mg949,00€1mL*10mM (DMSO)63,00€PNU-96391
CAS :PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.Formule :C15H23NO2SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :281.41Ref: TM-T28435
1mg115,00€5mg249,00€10mg369,00€25mg562,00€50mg787,00€100mg1.054,00€200mg1.406,00€1mL*10mM (DMSO)235,00€Veralipride
CAS :Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.Formule :C17H25N3O5SDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :383.46N-0500 HCl
CAS :N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.Formule :C15H22ClNO2Degré de pureté :98.3% - 98.42%Couleur et forme :SolidMasse moléculaire :283.79SK609 HCl
CAS :SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.Formule :C10H15Cl2NDegré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :220.14SCH-23390 maleate
CAS :SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formule :C21H22ClNO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :403.86Flibanserin
CAS :Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.Formule :C20H21F3N4ODegré de pureté :99.37% - 99.93%Couleur et forme :White PowderMasse moléculaire :390.4Tetrahydropalmatine
CAS :Tetrahydropalmatine (DL-Tetrahydropalmatine) is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epilepticFormule :C21H25NO4Degré de pureté :99.91% - 99.95%Couleur et forme :SolidMasse moléculaire :355.43FGH31
FGH31 (Compound 24), a dopamine D4 agonist, exhibits potent and selective GRK2-dependency with a K i of 1.6 nM and partially activates β-arrestin [1].Formule :C33H36N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :520.66NGB 2904
CAS :NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Formule :C28H29Cl2N3ODegré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :494.46Ref: TM-T28167
2mg40,00€5mg58,00€10mg90,00€25mg163,00€50mg279,00€100mg394,00€500mgÀ demander1mL*10mM (DMSO)75,00€PD 168568 dihydrochloride
CAS :PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).Formule :C22H29Cl2N3ODegré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :422.39Ref: TM-T12383
5mg48,00€10mg58,00€25mg117,00€50mg170,00€100mg248,00€200mg348,00€1mL*10mM (DMSO)60,00€Pimethixene maleate
CAS :Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.Formule :C23H23NO4SDegré de pureté :100%Couleur et forme :SolidMasse moléculaire :409.5SCH-23390 hydrochloride
CAS :SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formule :C17H19Cl2NODegré de pureté :98% - 99.51%Couleur et forme :SolidMasse moléculaire :324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€Ordopidine
CAS :Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.Formule :C14H20FNO2SDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :285.38Spiroxatrine
CAS :Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.Formule :C22H25N3O3Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :379.45D-tetrahydropalmatine
CAS :D-Tetrahydropalmatine inhibits OCT1, reducing MCT uptake and hepatocyte damage in MDCK-hOCT1 cells and rat livers.Formule :C21H25NO4Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :355.43Ref: TM-T4S0779
2mg44,00€5mg64,00€10mg97,00€25mg182,00€50mg273,00€100mg393,00€200mg558,00€1mL*10mM (DMSO)65,00€Sultopride hydrochloride
CAS :Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.Formule :C17H27ClN2O4SDegré de pureté :≥95%Couleur et forme :White Or Yellowish PowderMasse moléculaire :390.93Droperidol
CAS :Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.Formule :C22H22FN3O2Degré de pureté :97.16% - 98%Couleur et forme :SolidMasse moléculaire :379.43Ro 10-5824 dihydrochloride
CAS :Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Formule :C17H22Cl2N4Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :353.29Ziprasidone
CAS :Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.Formule :C21H21ClN4OSDegré de pureté :100% - 99.53%Couleur et forme :Tan SolidMasse moléculaire :412.94Quetiapine hemifumarate
CAS :Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formule :C46H54N6O8S2Degré de pureté :100% - 99.59%Couleur et forme :White Crystalline SolidMasse moléculaire :883.09Seridopidine
CAS :Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.Formule :C14H20FNO2SDegré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :285.38Bromopride
CAS :Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.Formule :C14H22BrN3O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :344.25Ref: TM-T1175
2mg44,00€5mg65,00€10mg93,00€25mg178,00€50mg281,00€100mg454,00€200mg650,00€1mL*10mM (DMSO)71,00€CP-226269
CAS :CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.Formule :C18H19FN4Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :310.37Tetrabenazine
CAS :Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.Formule :C19H27NO3Degré de pureté :98% - 99.91%Couleur et forme :White To Off-White White To Off-White SolidMasse moléculaire :317.42Didesmethyl cariprazine
CAS :Didesmethyl cariprazine, Cariprazine's active metabolite, treats schizophrenia/bipolar with D3/D2 affinity; half-life 1-3 weeks.Formule :C19H28Cl2N4ODegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :399.36L-741626
CAS :L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3Formule :C20H21ClN2ODegré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :340.85Metergoline
CAS :Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formule :C25H29N3O2Degré de pureté :99.7% - 99.83%Couleur et forme :SolidMasse moléculaire :403.52Aripiprazole Lauroxil
CAS :Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.Formule :C36H51Cl2N3O4Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :660.71Ref: TM-T14319
10mg48,00€25mg72,00€50mg96,00€100mg130,00€200mg188,00€500mg318,00€1mL*10mM (DMSO)49,00€Dihydrexidine
CAS :Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity.Formule :C17H17NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :267.32Pentiapine
CAS :Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.Formule :C15H17N5SDegré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :299.39Ref: TM-T12405
1mg487,00€5mg753,00€10mg1.216,00€25mg1.691,00€50mg2.262,00€100mg3.068,00€1mL*10mM (DMSO)938,00€Domperidone
CAS :Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.Formule :C22H24ClN5O2Degré de pureté :98% - 99.82%Couleur et forme :SolidMasse moléculaire :425.91DOV-216,303 Free Base
CAS :DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.Formule :C11H11Cl2NDegré de pureté :96.7%Couleur et forme :SolidMasse moléculaire :228.12Acetophenazine dimaleate
CAS :Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.Formule :C31H37N3O10SDegré de pureté :99.39% - 99.48%Couleur et forme :SolidMasse moléculaire :643.71Eticlopride hydrochloride
CAS :Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).Formule :C17H25ClN2O3·HClDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.31Odapipam
CAS :Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).Formule :C19H20ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.82Tiospirone
CAS :Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.Formule :C24H32N4O2SDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :440.6Ref: TM-T24885
1mg130,00€5mg309,00€10mg567,00€25mg910,00€50mg1.225,00€100mg1.644,00€1mL*10mM (DMSO)374,00€Blonanserin
CAS :Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formule :C23H30FN3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :367.5Metoclopramide
CAS :Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formule :C14H22ClN3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :299.8Phenelzine
CAS :Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.Formule :C8H12N2Degré de pureté :98%Couleur et forme :LiquidMasse moléculaire :136.19Ref: TM-T9540
5mgÀ demander10mgÀ demander25mgÀ demander50mgÀ demander100mgÀ demander200mgÀ demander500mgÀ demanderBrilaroxazine
CAS :Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.Formule :C22H25Cl2N3O3Degré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :450.36Ref: TM-T14782
1mg105,00€5mg250,00€10mg406,00€25mg700,00€50mg1.008,00€100mg1.378,00€200mg1.833,00€1mL*10mM (DMSO)283,00€A-437203
CAS :A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.Formule :C20H27F3N6OSDegré de pureté :98.62%Couleur et forme :SolidMasse moléculaire :456.53Ref: TM-T10213
1mg89,00€5mg198,00€10mg279,00€25mg434,00€50mg562,00€100mg780,00€200mg1.035,00€1mL*10mM (DMSO)227,00€Ecopipam
CAS :Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.Formule :C19H20ClNODegré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :313.82Dimethocaine
CAS :Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Formule :C16H26N2O2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :278.39LE 300
CAS :LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.Formule :C20H22N2Degré de pureté :98.08% - 98.35%Couleur et forme :SolidMasse moléculaire :290.4BMY 7378 dihydrochloride
CAS :BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Formule :C22H33Cl2N3O3Degré de pureté :97.32% - 99.08%Couleur et forme :SolidMasse moléculaire :458.42Raclopride
CAS :Raclopride is a selective antagonist of dopamine D2/D3 receptor.Formule :C15H20Cl2N2O3Degré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :347.24MPTP hydrochloride
CAS :MPTP hydrochloride is a precursor of MPP+, a dopamine neurotoxin with blood-brain barrier permeability.Formule :C12H16ClNDegré de pureté :100% - 99.73%Couleur et forme :SolidMasse moléculaire :209.72Ref: TM-T4081
1g758,00€5mg35,00€10mg52,00€25mg87,00€50mg145,00€100mg197,00€200mg313,00€500mg527,00€1mL*10mM (DMSO)55,00€MLS1082
CAS :MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.Formule :C24H23N3O2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :385.46L-745870 trihydrochloride
CAS :L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.Formule :C18H22Cl4N4Degré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :436.21Cariprazine hydrochloride
CAS :Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formule :C21H33Cl3N4ODegré de pureté :100% - 98.52%Couleur et forme :SolidMasse moléculaire :463.87Desipramine hydrochloride
CAS :Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.Formule :C18H23ClN2Degré de pureté :99.58% - 99.94%Couleur et forme :White To Off-White PowderMasse moléculaire :302.842BisfluoroModafinil
CAS :CRL-40940 is a selective dopaminergic reuptake inhibitorFormule :C15H13F2NO2SDegré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :309.33Ref: TM-T4262
1mg48,00€2mg64,00€5mg94,00€10mg139,00€25mg236,00€50mg359,00€100mg540,00€500mg1.130,00€1mL*10mM (DMSO)104,00€Zuclopenthixol
CAS :Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.Formule :C22H25ClN2OSDegré de pureté :98.90% - 99.82%Couleur et forme :SolidMasse moléculaire :400.96Halopemide
CAS :Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Formule :C21H22ClFN4O2Degré de pureté :96.29%Couleur et forme :SolidMasse moléculaire :416.88Dexpramipexole
CAS :Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.Formule :C10H17N3SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :211.33WAY-100635 Monomaleate
CAS :WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Formule :C25H34N4O2·C4H4O4Degré de pureté :99.26% - 99.68%Couleur et forme :SolidMasse moléculaire :538.64Ref: TM-T2631
2mg46,00€5mg66,00€10mg95,00€25mg180,00€50mg334,00€100mg495,00€200mg717,00€500mg1.111,00€1mL*10mM (DMSO)79,00€Bromocriptine mesylate
CAS :Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with highest affinity (Ki = 2.5 nM)Formule :C33H44BrN5O8SDegré de pureté :99.76% - 99.87%Couleur et forme :White SolidMasse moléculaire :750.7Perospirone
CAS :Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formule :C23H30N4O2SDegré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :426.57Timiperone
CAS :Timiperone exhibits a high affinity for cerebral dopamine D2 receptors, demonstrating antipsychotic activity as it mitigates stereotyped behavior.Formule :C22H24FN3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :397.51Roxindole
CAS :Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formule :C23H26N2ODegré de pureté :99.08% - 99.18%Couleur et forme :SolidMasse moléculaire :346.47Asenapine hydrochloride
CAS :Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.Formule :C17H17Cl2NOCouleur et forme :SolidMasse moléculaire :322.23SPD-473 citrate
CAS :SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.Formule :C23H31Cl2NO8SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :552.475,7-Dimethoxyluteolin
CAS :5,7-Dimethoxyluteolin is a natural product from Hovenia acerba. 5,7-Dimethoxyluteolin is a dopamine transporter (DAT) activator with an EC50 of 3.417 μM.Formule :C17H14O6Degré de pureté :99.56% - 99.56%Couleur et forme :SolidMasse moléculaire :314.29WAY-100635
CAS :WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .Formule :C25H34N4O2Couleur et forme :SolidMasse moléculaire :422.56
