Récepteur de la dopamine
Les récepteurs de la dopamine sont un groupe de récepteurs couplés aux protéines G (GPCR) qui répondent au neurotransmetteur dopamine, jouant un rôle clé dans la régulation du mouvement, de la motivation, de la récompense et de plusieurs fonctions cognitives. Ces récepteurs sont divisés en familles de type D1 et de type D2, chacune ayant des fonctions et des profils pharmacologiques distincts. Les modulateurs des récepteurs de la dopamine sont largement étudiés pour leurs applications dans le traitement de la maladie de Parkinson, de la schizophrénie, de la dépendance et d'autres troubles neuropsychiatriques. Chez CymitQuimica, nous offrons une large gamme de modulateurs de récepteurs de la dopamine de haute qualité pour soutenir vos recherches en neurosciences, santé mentale et signalisation GPCR.
Produits appartenant à la catégorie "Récepteur de la dopamine"
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NRA-0160
CAS :NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)Formule :C24H23F2N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.52Tiaspirone hydrochloride
CAS :Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity and influences the electrophysiological activity of dopaminergic neurons.Formule :C24H33ClN4O2SDegré de pureté :99.98%Couleur et forme :SoildMasse moléculaire :477.065-HT6/7 antagonist 1
CAS :5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.Formule :C22H20FN3O3Degré de pureté :98.55% - 98.78%Couleur et forme :SolidMasse moléculaire :393.41Benperidol
CAS :Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.Formule :C22H24FN3O2Degré de pureté :97.39%Couleur et forme :SolidMasse moléculaire :381.44Ref: TM-T26360
1mg116,00€5mg276,00€10mg410,00€25mg680,00€50mg938,00€100mg1.293,00€500mg2.593,00€1mL*10mM (DMSO)279,00€Liafensine
CAS :Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.Formule :C24H22N4Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :366.46Asenapine
CAS :Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophreniaFormule :C17H16ClNODegré de pureté :99.16%Couleur et forme :CoaMasse moléculaire :285.77SLV-310
CAS :SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.Formule :C25H24FN3O2Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :417.48D3R/MOR antagonist 1
Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nMFormule :C22H27Cl2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.38Metoclopramide hydrochloride
CAS :Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.Formule :C14H22ClN3O2·HClDegré de pureté :99.99%Couleur et forme :White To Off-White PowderMasse moléculaire :336.26NMI 8739
CAS :NMI 8739 (n-docosahexaenoyl dopamine) is an agonist of D2 autoreceptor.Formule :C30H41NO3Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :463.65Ref: TM-T11079
1mg40,00€5mg85,00€10mg120,00€25mg207,00€50mg303,00€100mg449,00€200mg652,00€1mL*10mM (DMSO)90,00€Itopride hydrochloride
CAS :Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.Formule :C20H27ClN2O4Degré de pureté :99.59%Couleur et forme :White Or Pale Brownish CrystalMasse moléculaire :394.9Oxolinic acid
CAS :Oxolinic acid (Nidantin) is a synthetic antimicrobial related to NALIDIXIC ACID and used in URINARY TRACT INFECTIONS.Formule :C13H11NO5Degré de pureté :98.39% - 99.72%Couleur et forme :Crystals From Dimethylformamide White Crystalline PowderMasse moléculaire :261.23Fluphenazine decanoate
CAS :Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.Formule :C32H44F3N3O2SDegré de pureté :100% - 98.14%Couleur et forme :SolidMasse moléculaire :591.77Benztropine mesylate
CAS :Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSONFormule :C21H25NO·CH4SO3Degré de pureté :98.41% - 99.96%Couleur et forme :White Crystalline Powder; Odourless Or Almost OdourlessMasse moléculaire :403.53Syrosingopine
CAS :Syrosingopine is a dual inhibitor of MCT1 and MCT4, 60 times more potent against MCT4, preventing lactate and H+ efflux.Cost-effective and quality-assured.Formule :C35H42N2O11Degré de pureté :99.25% - 99.78%Couleur et forme :SolidMasse moléculaire :666.71Ref: TM-TN2252
1mg66,00€5mg142,00€10mg212,00€25mg361,00€50mg543,00€100mg750,00€1mL*10mM (DMSO)202,00€GR 103691
CAS :GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).Formule :C30H35N3O3Degré de pureté :98.94% - 99.29%Couleur et forme :SolidMasse moléculaire :485.62Ref: TM-T11463
2mg46,00€5mg66,00€10mg99,00€25mg197,00€50mg311,00€100mg505,00€500mg1.121,00€1mL*10mM (DMSO)74,00€PF-00217830
CAS :PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.Formule :C26H30N4O2Degré de pureté :98.30%Couleur et forme :SolidMasse moléculaire :430.54Aniracetam
CAS :Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.Formule :C12H13NO3Degré de pureté :99.88% - 99.89%Couleur et forme :White Crystalline Or Crystalline PowdeMasse moléculaire :219.24Oxidopamine hydrobromide
CAS :Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.Formule :C8H12BrNO3Degré de pureté :98.1% - 99.88%Couleur et forme :Beige To Brown Fine Crystalline PowderMasse moléculaire :250.09Flunarizine dihydrochloride
CAS :Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.Formule :C26H28Cl2F2N2Degré de pureté :99.53% - 99.89%Couleur et forme :White Crystalline Powder Odorless And TastelessMasse moléculaire :477.42Pardoprunox
CAS :Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formule :C12H15N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :233.27Amisulpride
CAS :Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.Formule :C17H27N3O4SDegré de pureté :99.97%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :369.48Bendazol
CAS :Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.Formule :C14H12N2Degré de pureté :98.7% - 99.81%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :208.26Chlorprothixene hydrochloride
CAS :Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formule :C18H18ClNS·HClDegré de pureté :99.16%Couleur et forme :White PowderMasse moléculaire :352.32Aplindore Fumarate
CAS :Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Formule :C22H22N2O7Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :426.42SKF 38393 hydrochloride
CAS :SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.Formule :C16H17NO2·HClDegré de pureté :98.70% - 99.1%Couleur et forme :SolidMasse moléculaire :291.77Perphenazine
CAS :Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.Formule :C21H26ClN3OSDegré de pureté :99.3% - 99.72%Couleur et forme :SolidMasse moléculaire :403.97Zotepine
CAS :Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formule :C18H18ClNOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :331.86Glaucine
CAS :Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.Formule :C21H25NO4Degré de pureté :99.14% - 99.42%Couleur et forme :SolidMasse moléculaire :355.43Dexchlorpheniramine Maleate
CAS :Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.Formule :C20H23ClN2O4Degré de pureté :99.58%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :390.86Bromperidol
CAS :Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.Formule :C21H23BrFNO2Degré de pureté :99.89%Couleur et forme :Tan SolidMasse moléculaire :420.32Mesoridazine Besylate
CAS :Mesoridazine Besylate (Serentil), a piperidine antipsychotic and phenothiazine, treats schizophrenia; it's a thioridazine metabolite.Formule :C27H32N2O4S3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :544.75U 99194 maleate
CAS :U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.Formule :C21H31NO6Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :393.47Sertindole
CAS :Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).Formule :C24H26ClFN4ODegré de pureté :99.74%Couleur et forme :Off-White To Pale Yellow SolidMasse moléculaire :440.94PG 01037 dihydrochloride
CAS :PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.Formule :C26H28Cl4N4ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :554.34Ref: TM-T23143
1mg42,00€2mg52,00€5mg82,00€10mg105,00€25mg168,00€50mg249,00€100mg369,00€200mg522,00€1mL*10mM (DMSO)97,00€ABT 724 trihydrochloride
CAS :ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.Formule :C17H22Cl3N5Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :402.75Ref: TM-T22019
5mg40,00€10mg65,00€25mg126,00€50mg188,00€100mg283,00€200mg419,00€1mL*10mM (DMSO)44,00€7-Hydroxy-DPAT hydrobromide
CAS :7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.Formule :C16H26BrNODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :328.29Carmoxirole hydrochloride
CAS :Carmoxirole hydrochloride (EMD 45609 hydrochloride) is a selective dopamine D2 receptor agonist with antihypertensive activity in vivo.Formule :C24H27ClN2O2Degré de pureté :97.8% - 98.12%Couleur et forme :SolidMasse moléculaire :410.94Ref: TM-T10683
1mg58,00€5mg117,00€10mg178,00€25mg306,00€50mg452,00€100mg620,00€200mg835,00€1mL*10mM (DMSO)134,00€SKF-83566
CAS :SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.Formule :C17H18BrNODegré de pureté :95.00% - 99.82%Couleur et forme :SolidMasse moléculaire :332.23SKF83959
CAS :SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.Formule :C18H20ClNO2Degré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :317.81Ref: TM-T60835
1mg52,00€5mg103,00€10mg169,00€25mg359,00€50mg530,00€100mg758,00€1mL*10mM (DMSO)114,00€GSK163090
CAS :GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).Formule :C25H29N5ODegré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :415.53Ref: TM-TQ0311
1mg37,00€2mg52,00€5mg80,00€10mg125,00€25mgÀ demander50mgÀ demander1mL*10mM (DMSO)87,00€Tavapadon
CAS :Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Formule :C19H16F3N3O3Degré de pureté :99.33% - 99.8%Couleur et forme :SolidMasse moléculaire :391.34Ref: TM-T16999
1mg81,00€5mg170,00€10mg274,00€25mg502,00€50mg705,00€100mg938,00€1mL*10mM (DMSO)188,00€Mianserin hydrochloride
CAS :Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.Formule :C18H21ClN2Degré de pureté :99.63% - 99.82%Couleur et forme :White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedMasse moléculaire :300.83UNC9975
CAS :UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.Formule :C23H28Cl2N4O2Degré de pureté :99.02% - 99.02%Couleur et forme :SolidMasse moléculaire :463.4Risperidone
CAS :Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.Formule :C23H27FN4O2Degré de pureté :99.73%Couleur et forme :Crystalline SolidMasse moléculaire :410.48Pipamperone
CAS :Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.Formule :C21H30FN3O2Degré de pureté :99.94%Couleur et forme :White PowderMasse moléculaire :375.48Ref: TM-T12480
1mg62,00€2mg85,00€5mg119,00€10mg170,00€25mg283,00€50mg430,00€100mg622,00€1mL*10mM (DMSO)131,00€Promazine hydrochloride
CAS :Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Formule :C17H21ClN2SDegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :320.88Brexpiprazole
CAS :Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formule :C25H27N3O2SDegré de pureté :99.06% - 99.96%Couleur et forme :SolidMasse moléculaire :433.57lumateperone Tosylate
CAS :lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formule :C31H36FN3O4SDegré de pureté :95.83% - 98.57%Couleur et forme :SolidMasse moléculaire :565.7MLS1547
CAS :MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).Formule :C19H19ClN4ODegré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :354.83
