Récepteur de la dopamine
Les récepteurs de la dopamine sont un groupe de récepteurs couplés aux protéines G (GPCR) qui répondent au neurotransmetteur dopamine, jouant un rôle clé dans la régulation du mouvement, de la motivation, de la récompense et de plusieurs fonctions cognitives. Ces récepteurs sont divisés en familles de type D1 et de type D2, chacune ayant des fonctions et des profils pharmacologiques distincts. Les modulateurs des récepteurs de la dopamine sont largement étudiés pour leurs applications dans le traitement de la maladie de Parkinson, de la schizophrénie, de la dépendance et d'autres troubles neuropsychiatriques. Chez CymitQuimica, nous offrons une large gamme de modulateurs de récepteurs de la dopamine de haute qualité pour soutenir vos recherches en neurosciences, santé mentale et signalisation GPCR.
Produits appartenant à la catégorie "Récepteur de la dopamine"
Trier par
Sulpiride
CAS :Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.Formule :C15H23N3O4SDegré de pureté :99.94%Couleur et forme :White Crystalline PowderMasse moléculaire :341.43JNJ-37822681 dihydrochloride
CAS :JNJ-37822681 dihydrochloride 是特异性的、有中枢活性的,可快速解离的多巴胺 D2受体拮抗剂,与多巴胺 D2L 受体结合的亲和力适中 (Ki=158 nM)。JNJ-37822681 dihydrochloride 在精神分裂症和躁郁症领域有研究价值。Formule :C17H19Cl2F5N4Degré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :445.26Pramipexole dihydrochloride hydrate
CAS :Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.Formule :C10H17N3S·2HCl·H2ODegré de pureté :99.68%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :302.26Ref: TM-T6951
10mg47,00€25mg74,00€50mg119,00€100mg170,00€200mg255,00€500mg430,00€1mL*10mM (DMSO)47,00€Ziprasidone hydrochloride monohydrate
CAS :Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFormule :C21H21ClN4OS·HCl·H2ODegré de pureté :98% - 99.83%Couleur et forme :Off-White PowderMasse moléculaire :467.12D5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Couleur et forme :Odour SolidTrimethobenzamide hydrochloride
CAS :Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Formule :C21H29ClN2O5Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :424.92Fosopamine(HCl)
CAS :Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.Formule :C9H15ClNO5PDegré de pureté :100%Couleur et forme :SolidMasse moléculaire :283.65Alizapride hydrochloride
CAS :Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formule :C16H21N5O2·HClDegré de pureté :99.35% - 99.48%Couleur et forme :CoaMasse moléculaire :351.83Loxapine
CAS :Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.Formule :C18H18ClN3ODegré de pureté :99.88%Couleur et forme :Pale Yellowish Crystals From Petroleum Ether SolidMasse moléculaire :327.81Cabergoline
CAS :Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.Formule :C26H37N5O2Degré de pureté :99.86%Couleur et forme :White Crystalline SolidMasse moléculaire :451.6Ergocornine
CAS :Ergocornine is a naturally occurring ergot alkaloid and acts as a dopamine receptor (dopamine receptor) agonist.Formule :C31H39N5O5Couleur et forme :SolidMasse moléculaire :561.67Nomifensine
CAS :Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.Formule :C16H18N2Degré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :238.33Atomoxetine hydrochloride
CAS :Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.Formule :C17H22ClNODegré de pureté :99.86%Couleur et forme :White SolidMasse moléculaire :291.82Rotigotine Hydrochloride
CAS :Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.Formule :C19H26ClNOSDegré de pureté :99.53% - 99.56%Couleur et forme :Almost White To White Crystalline PowderMasse moléculaire :351.935-Benzyloxygramine
CAS :5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formule :C18H20N2ODegré de pureté :96.33%Couleur et forme :SolidMasse moléculaire :280.36Ropinirole hydrochloride
CAS :Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.Formule :C16H24N2O·HClDegré de pureté :99.87% - 99.98%Couleur et forme :Off-White SolidMasse moléculaire :296.84UCSF924
CAS :UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).Formule :C20H22N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :322.4Medifoxamine
CAS :Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.MedifoxamineFormule :C16H19NO2Degré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :257.33Ref: TM-T24444
1mg99,00€5mg235,00€10mg354,00€25mg635,00€50mg893,00€100mg1.159,00€1mL*10mM (DMSO)259,00€DOPEXAMINE
CAS :Dopexamine is a dopaminergic agonistFormule :C22H32N2O2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :356.5Ref: TM-T8653
1mg131,00€2mg188,00€5mg284,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€1mL*10mM (DMSO)306,00€Trimipramine maleate
CAS :Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.Formule :C24H30N2O4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :410.51Dopamine D2 receptor agonist-2
CAS :Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.Formule :C25H31Cl2N5OSDegré de pureté :98.93%Couleur et forme :SoildMasse moléculaire :520.52Ref: TM-T60075
1mg38,00€5mg71,00€10mg90,00€25mg148,00€50mg210,00€100mg314,00€200mg452,00€1mL*10mM (DMSO)90,00€Propionylpromazine hydrochloride
CAS :Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.Formule :C20H25ClN2OSDegré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :376.94Ritanserin
CAS :Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formule :C27H25F2N3OSDegré de pureté :99.45% - 99.89%Couleur et forme :SolidMasse moléculaire :477.57Fluphenazine dihydrochloride
CAS :Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.Formule :C22H28Cl2F3N3OSDegré de pureté :99.23%Couleur et forme :Off-White SolidMasse moléculaire :510.44Thiethylperazine dimaleate
CAS :Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor.Formule :C30H37N3O8S2Degré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :631.76carfenazine
CAS :carfenazine targets the Dopamine receptor and is used for schizophrenia research.Formule :C24H31N3O2SDegré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :425.59Trifluoperazine
CAS :Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.Formule :C21H24F3N3SDegré de pureté :98.3% - 99.46%Couleur et forme :White To Yellowish Crystalline PowderMasse moléculaire :407.5(-)-GSK598809 hydrochloride
CAS :(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.Formule :C22H24ClF4N5OSDegré de pureté :97.66%Couleur et forme :SoildMasse moléculaire :517.97Molindone
CAS :Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.Formule :C16H24N2O2Degré de pureté :98% - 99.37%Couleur et forme :Off-White SolidMasse moléculaire :276.37Foscarbidopa
CAS :Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.Formule :C10H15N2O7PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :306.21Dasotraline hydrochloride
CAS :Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formule :C16H16Cl3NDegré de pureté :98.92% - 99.6%Couleur et forme :SolidMasse moléculaire :328.66Nolomirole HCl
CAS :Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory effects on norepinephrine release, which can be used to studyFormule :C19H28ClNO4Degré de pureté :100% - 99.12%Couleur et forme :SolidMasse moléculaire :369.88Brexpiprazole S-oxide
CAS :Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).Formule :C25H27N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :449.57Tedatioxetine
CAS :Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Formule :C18H21NSDegré de pureté :100% - 98.58%Couleur et forme :SolidMasse moléculaire :283.43UNC10099984A
CAS :UNC10099984A (Compound 6) is a functionally selective ligand for the dopamine D2 receptor, exhibiting a Ki value of 4.6 nM and an EC50 of 6.2 nM for β-arrestin. This compound is useful for research into central nervous system diseases related to the D2 receptor.Formule :C24H29Cl2N3O2Couleur et forme :SolidMasse moléculaire :462.41Xaliproden hydrochloride
CAS :Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formule :C24H23ClF3NDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :417.89Ref: TM-T9272
1mg40,00€5mg85,00€10mg120,00€25mg235,00€50mg376,00€100mg540,00€200mg775,00€1mL*10mM (DMSO)96,00€Pimethixene
CAS :Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Formule :C19H19NSDegré de pureté :97.50%Couleur et forme :SolidMasse moléculaire :293.43Ref: TM-T12489
2mg34,00€5mg50,00€10mg65,00€25mg106,00€50mg158,00€100mg226,00€200mg339,00€1mL*10mM (DMSO)52,00€Methyldopa hydrate
CAS :Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.Formule :C10H13NO4H2ODegré de pureté :99.67%Couleur et forme :White SolidMasse moléculaire :238.24Tolnapersine TFA
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.Formule :C23H27F3N2O3Degré de pureté :98.10%Couleur et forme :SoildMasse moléculaire :436.47L-DOPA
CAS :L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is converted to dopamine by DOPA decarboxylase.Formule :C9H11NO4Degré de pureté :98.99% - 99.93%Couleur et forme :Colorless To White Crystals Or Crystalline Powder; Needles From Water SolidMasse moléculaire :197.19Abaperidone
CAS :Abaperidone is an atypical antipsychotic, antagonizes 5-HT2A (IC50=6.2 nM) and D2 receptors (IC50=17 nM), reduces hsp70 mRNA in rat brains.Formule :C25H25FN2O5Degré de pureté :94.35%Couleur et forme :SolidMasse moléculaire :452.47A-77636
CAS :A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50Formule :C20H27NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.43Diclofensine
CAS :Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.Formule :C17H17Cl2NODegré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :322.23Melitracen hydrochloride
CAS :Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formule :C21H26ClNDegré de pureté :99.99%Couleur et forme :Crystalline SolidMasse moléculaire :327.9Ref: TM-T4274
10mg47,00€25mg67,00€50mg87,00€100mg116,00€200mg170,00€500mg279,00€1mL*10mM (DMSO)50,00€BP 897
CAS :BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Formule :C26H31N3O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :417.54Ref: TM-T9100
1mg80,00€5mg162,00€10mg227,00€25mg379,00€50mg540,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)177,00€Rotundine
CAS :Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formule :C21H25NO4Degré de pureté :100% - 99.8%Couleur et forme :Off-White SolidMasse moléculaire :355.43Iloperidone
CAS :Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Formule :C24H27FN2O4Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :426.48D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.Formule :C27H37NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.59Methyldopa
CAS :Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFormule :C10H13NO4Degré de pureté :99.86% - 99.89%Couleur et forme :Less Or Almost Colorless Crystals Or White To Yellowish-White FineMasse moléculaire :211.21Lurasidone hydrochloride
CAS :Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Formule :C28H36N4O2S·HClDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :529.14
