Récepteur de la dopamine
Les récepteurs de la dopamine sont un groupe de récepteurs couplés aux protéines G (GPCR) qui répondent au neurotransmetteur dopamine, jouant un rôle clé dans la régulation du mouvement, de la motivation, de la récompense et de plusieurs fonctions cognitives. Ces récepteurs sont divisés en familles de type D1 et de type D2, chacune ayant des fonctions et des profils pharmacologiques distincts. Les modulateurs des récepteurs de la dopamine sont largement étudiés pour leurs applications dans le traitement de la maladie de Parkinson, de la schizophrénie, de la dépendance et d'autres troubles neuropsychiatriques. Chez CymitQuimica, nous offrons une large gamme de modulateurs de récepteurs de la dopamine de haute qualité pour soutenir vos recherches en neurosciences, santé mentale et signalisation GPCR.
Produits appartenant à la catégorie "Récepteur de la dopamine"
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Trazpiroben
CAS :Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Formule :C31H39N3O4Degré de pureté :98.85% - 99.41%Couleur et forme :SolidMasse moléculaire :517.66Fluoroclebopride
CAS :Fluoroclebopride is a dopamine (DA) D2 receptor ligand.Formule :C20H23ClFN3O2Degré de pureté :99.68% - 99.91%Couleur et forme :SolidMasse moléculaire :391.87Ref: TM-T3187
1mg35,00€5mg74,00€10mg96,00€25mg159,00€50mg235,00€100mg376,00€500mg867,00€1mL*10mM (DMSO)96,00€Duloxetine hydrochloride
CAS :Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.Formule :C18H20ClNOSDegré de pureté :100% - 99.93%Couleur et forme :White Or White Crystalline PowderMasse moléculaire :333.88Rotigotine-
CAS :Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formule :C19H25NOSDegré de pureté :98.08% - 99.59%Couleur et forme :SolidMasse moléculaire :315.47Ref: TM-T6647
5mg52,00€10mg78,00€25mg145,00€50mg255,00€100mg378,00€200mg552,00€500mg868,00€1mL*10mM (DMSO)55,00€D4R agonist-1
CAS :D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.Formule :C19H22N4SDegré de pureté :98.16%Couleur et forme :SolidMasse moléculaire :338.47Ref: TM-T78825
1mg333,00€5mg922,00€10mg1.140,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.664,00€PF-4363467
CAS :PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.Formule :C22H30N2O3SCouleur et forme :SolidMasse moléculaire :402.55Flupentixol dihydrochloride
CAS :Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.Formule :C23H27Cl2F3N2OSDegré de pureté :100% - 99.35%Couleur et forme :White Or Off-White SolidMasse moléculaire :507.43PD128907 HCl
CAS :PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.Formule :C14H20ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :285.77Zatebradine
CAS :Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).Formule :C26H36N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.57Remoxipride hydrochloride
CAS :Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-Formule :C16H24BrClN2O3Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :407.73BL-1020 Mesylate
CAS :BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.Formule :C28H45ClN4O11S4Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :777.39Dicarbine
CAS :Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.Formule :C13H18N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :202.3Ropinirole
CAS :Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.Formule :C16H24N2ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :260.38Tedatioxetine hydrobromide
CAS :Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.Formule :C18H22BrNSDegré de pureté :99.50%Couleur et forme :SolidMasse moléculaire :364.34Etilevodopa hydrochloride
CAS :Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.Formule :C11H16ClNO4Degré de pureté :95.00%Couleur et forme :SolidMasse moléculaire :261.7Losulazine
CAS :Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.Formule :C27H22F4N4O3SDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :558.55NGD 94-1
CAS :NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders such as cognitive impairment.Formule :C18H20N6Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :320.39Thioridazine hydrochloride
CAS :Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4Formule :C21H27ClN2S2Degré de pureté :99.55% - 99.55%Couleur et forme :White To Off-White SolidMasse moléculaire :407.04SB-277011
CAS :SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), <5.2 (5-HT1B).Formule :C28H30N4ODegré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :438.56Ref: TM-T12861
1mg47,00€5mg58,00€10mg93,00€25mg158,00€50mg254,00€100mgÀ demander1mL*10mM (DMSO)60,00€Tetrahydroberberine
CAS :Tetrahydroberberine (Canadine) is an isoquinoline alkaloid isolated from corydalis tuber, has a micromolar affinity for dopamine D(2) receptors.Formule :C20H21NO4Degré de pureté :96.65% - 99.89%Couleur et forme :SolidMasse moléculaire :339.39Neflumozide
CAS :Neflumozide (HRP 913) is an orally effective derivative of benzisoxazole, characterized by its potent dopamine antagonist properties and antipsychotic activity. It is utilized in research related to psychiatric disorders.Formule :C22H23FN4O2Couleur et forme :SolidMasse moléculaire :394.44FAUC-365
CAS :FAUC-365 is a D3 dopamine receptor agonist.Formule :C23H25Cl2N3OSDegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :462.44Ref: TM-T21667
1mg52,00€5mg111,00€10mg169,00€25mg323,00€50mg512,00€100mg740,00€500mg1.539,00€1mL*10mM (DMSO)123,00€Dexpramipexole dihydrochloride
CAS :Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamineFormule :C10H19Cl2N3SDegré de pureté :99.75% - 99.88%Couleur et forme :SolidMasse moléculaire :284.25Ref: TM-T11011
5mg52,00€10mg79,00€25mg153,00€50mg250,00€100mg378,00€200mg552,00€1mL*10mM (DMSO)52,00€WAY-260022
CAS :WAY-260022 is the norepinephrine transporter inhibitor.Formule :C21H31F3N2O2Degré de pureté :98.65% - 99.06%Couleur et forme :SolidMasse moléculaire :400.48Azaperone
CAS :Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.Formule :C19H22FN3ODegré de pureté :98.73%Couleur et forme :White Or Off-White CrystallineMasse moléculaire :327.4SB-277011 hydrochloride
CAS :SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.Formule :C28H31ClN4ODegré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :475.03Olanzapine
CAS :Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Formule :C17H20N4SDegré de pureté :100% - ≥95%Couleur et forme :Yellowish Crystalline PowderMasse moléculaire :312.43Amitifadine hydrochloride
CAS :Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).Formule :C11H12Cl3NDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :264.58L-745870
CAS :L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.Formule :C18H19ClN4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :326.82cis-(Z)-Flupentixol dihydrochloride
CAS :cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.Formule :C23H27Cl2F3N2OSDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :507.44AMI-193
CAS :AMI-193 (Spiramide) is a selective 5-HT2 & D2 receptor antagonist with antipsychotic properties.Formule :C22H26FN3O2Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :383.46(+)-PD 128907 hydrochloride
CAS :(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .Formule :C14H20ClNO3Degré de pureté :97.76%Couleur et forme :SolidMasse moléculaire :285.77Ref: TM-T7553
2mg40,00€5mg58,00€10mg90,00€25mg164,00€50mg281,00€100mg409,00€200mg582,00€1mL*10mM (DMSO)88,00€Rotigotine
CAS :Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.Formule :C19H25NOSDegré de pureté :98.84% - 99.82%Couleur et forme :SolidMasse moléculaire :315.47GBR 12935 dihydrochloride
CAS :GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.Formule :C28H36Cl2N2ODegré de pureté :98.17% - ≥95%Couleur et forme :SolidMasse moléculaire :487.5JNJ-37822681
CAS :JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.Formule :C17H17F5N4Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :372.34Nefazodone
CAS :Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.Formule :C25H32ClN5O2Degré de pureté :99.85%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :470.01Ref: TM-T21451
2mg47,00€5mg69,00€10mg96,00€25mg199,00€50mg307,00€100mg471,00€200mg693,00€1mL*10mM (DMSO)100,00€SKF-83566 hydrochloride
CAS :SKF-83566 hydrochloride is a D1-like dopamine receptor antagonist, inhibiting dopamine transporters and mitigating GBP-induced CPP.Formule :C17H19BrClNODegré de pureté :99.27%Couleur et forme :SoildMasse moléculaire :368.69Octodrine
CAS :Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.Formule :C8H19NDegré de pureté :99.98%Couleur et forme :Clear Colorless To Light Yellow LiquidMasse moléculaire :129.24Methiothepin mesylate
CAS :Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.Formule :C21H28N2O3S3Degré de pureté :98% - 99.92%Couleur et forme :SolidMasse moléculaire :452.65Quinpirole Hydrochloride
CAS :Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and miceFormule :C13H22ClN3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :255.79ABT-670
CAS :ABT-670 is a selective agonist of dopamine D4 receptor. For human D4, ferret D4, and rat D4, the EC50 values are 89 nM, 160 nM, and 93 nM , respectively.Formule :C19H23N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :325.4Mirtazapine
CAS :Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.Formule :C17H19N3Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :265.35Clozapine N-Oxide
CAS :View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Formule :C18H19ClN4ODegré de pureté :98.43% - 99.94%Couleur et forme :SolidMasse moléculaire :342.82L-(R,S)-Tetrahydropalmatine
CAS :L-(R,S)-Tetrahydropalmatine (Rotundine) is extracted from Corydalis yanhusuo W. T. Wang.Formule :C21H25NO4Degré de pureté :99.63% - 99.76%Couleur et forme :SolidMasse moléculaire :355.43N-Methyl amisulpride
CAS :N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.Formule :C18H29N3O4SCouleur et forme :SolidMasse moléculaire :383.519-FLUORENOL
CAS :9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.Formule :C13H10ODegré de pureté :99.98%Couleur et forme :Off-White Crystalline PowderMasse moléculaire :182.22Talquetamab
CAS :Talquetamab (JNJ-64407564) is a T-cell retargeting GPRC5D bispecific antibody with antitumor activity for the treatment of multiple myeloma.Couleur et forme :LiquidMasse moléculaire :144.59 kDaZiprasidone hydrochloride
CAS :Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFormule :C21H22CL2N4OSDegré de pureté :97.97% - 99.82%Couleur et forme :SolidMasse moléculaire :449.4Dopamine hydrochloride
CAS :Dopamine hydrochloride (ASL279) is a naturally occurring catecholamine formed by decarboxylation of dihydroxyphenylalanine and a precursor of norepinephrine andFormule :C8H12ClNO2Degré de pureté :99.56% - 99.76%Couleur et forme :SolidMasse moléculaire :189.639A 77636 hydrochloride
CAS :A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).Formule :C20H28ClNO3Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :365.89
