Récepteur d'adénosine
Les récepteurs de l'adénosine sont une classe de récepteurs GPCR qui répondent à la nucléoside endogène adénosine. Ces récepteurs sont impliqués dans la régulation de divers processus physiologiques, y compris la fonction cardiovasculaire, les cycles veille-sommeil et les réponses immunitaires. Les modulateurs des récepteurs de l'adénosine ont un potentiel thérapeutique pour traiter des affections telles que les arythmies cardiaques, l'inflammation et les maladies neurodégénératives. Chez CymitQuimica, nous offrons une sélection de modulateurs des récepteurs de l'adénosine de haute qualité pour soutenir vos recherches en biologie cardiovasculaire, neurosciences et immunologie.
Produits appartenant à la catégorie "Récepteur d'adénosine"
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MRS-3777 hemioxalate
CAS :MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.Formule :C17H19N5OC2H2O4Degré de pureté :97.10%Couleur et forme :SolidMasse moléculaire :354.39Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.Formule :C21H26NO10PDegré de pureté :95.50%Couleur et forme :SoildMasse moléculaire :483.41GS-6201
CAS :GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.Formule :C21H21F3N6O2Degré de pureté :98.32% - 99.74%Couleur et forme :SolidMasse moléculaire :446.43Ref: TM-T15418
1mg38,00€5mg79,00€10mg127,00€25mg261,00€50mg423,00€100mg635,00€200mg887,00€1mL*10mM (DMSO)87,00€A2B receptor antagonist 2
CAS :A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).Formule :C12H15N5Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :229.28Inosine
CAS :Inosine (NSC-20262) is a purine nucleoside that has hypoxanthine linked by the N9 nitrogen to the C1 carbon of ribose.Formule :C10H12N4O5Degré de pureté :99.51% - 99.78%Couleur et forme :SolidMasse moléculaire :268.23A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.Formule :C34H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.67PSB-603
CAS :PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.Formule :C24H25ClN6O4SDegré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :529.01Ref: TM-T23203
1mg37,00€5mg97,00€10mg160,00€25mg344,00€50mg562,00€100mg938,00€200mg1.264,00€1mL*10mM (DMSO)111,00€LUF6096
CAS :LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFormule :C22H21Cl2N3ODegré de pureté :100%Couleur et forme :SolidMasse moléculaire :414.33LAS38096
CAS :LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .Formule :C17H12N6ODegré de pureté :98.71% - 99.16%Couleur et forme :SolidMasse moléculaire :316.32A3AR antagonist 5
CAS :A3AR antagonist 5 (Compound 16) acts as a selective antagonist for the human adenosine A3 receptor (human adenosine A3 receptor), with an affinity expressed as a pC value of 4.542 μM.Formule :C18H16N2O2SCouleur et forme :SolidMasse moléculaire :324.40Selodenoson
CAS :Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.Formule :C17H24N6O4Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :376.41Adenosine antagonist-1
CAS :Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.Formule :C18H13N7SDegré de pureté :100% - 97%Couleur et forme :SolidMasse moléculaire :359.41A1/A3 AR antagonist 3
CAS :A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful inFormule :C22H19N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.42Theobromine
CAS :Theobromine (3,7-Dimethylxanthine), a xanthine alkaloid, is used as a bronchodilator and as a vasodilator.Formule :C7H8N4O2Degré de pureté :99.63% - 99.89%Couleur et forme :White To Yellow Crystalline PowderMasse moléculaire :180.16Theophylline
CAS :Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and centralFormule :C7H8N4O2Degré de pureté :99.47% - 99.97%Couleur et forme :White Solid PowderMasse moléculaire :180.16N 0861
CAS :N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.Formule :C13H17N5Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :243.31KFM19
CAS :KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.Formule :C16H22N4O3Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :318.37Zaladenant
CAS :Zaladenant is an adenosine receptor antagonist with antitumor properties.Formule :C19H15F3N6OCouleur et forme :SolidMasse moléculaire :400.357GR79236
CAS :GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Formule :C15H21N5O5Couleur et forme :SolidMasse moléculaire :351.36CPI-444
CAS :CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.Formule :C20H21N7O3Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :407.43ST3932
CAS :ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).Formule :C12H16N8ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :288.31A2AR-antagonist-1
CAS :Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.Formule :C27H25N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :451.52Binodenoson
CAS :Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.Formule :C17H25N7O4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :391.42Ref: TM-T9516
1mg103,00€5mg246,00€10mg369,00€25mg620,00€50mg825,00€100mg1.130,00€200mg1.549,00€1mL*10mM (DMSO)271,00€VUF 5574
CAS :VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.Formule :C21H17N5O2Degré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :371.39DPTN dihydrochloride
CAS :DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.Formule :C22H20Cl2N4OSDegré de pureté :100%Couleur et forme :SoildMasse moléculaire :459.39PD 117519
CAS :PD 117519 (CI947) is an agonist of adenosine receptorFormule :C19H21N5O4Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :383.4GW-493838
CAS :GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgiaFormule :C21H21ClFN7O4Degré de pureté :99.70% - 99.76%Couleur et forme :SolidMasse moléculaire :489.89Ref: TM-T27509
1mg152,00€5mg365,00€10mg520,00€25mg780,00€50mg1.054,00€100mg1.425,00€500mg2.793,00€1mL*10mM (DMSO)420,00€Ticlopidine hydrochloride
CAS :Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.Formule :C14H15Cl2NSDegré de pureté :99.82% - 99.98%Couleur et forme :White PowderMasse moléculaire :300.25ABT-702 dihydrochloride
CAS :ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.Formule :C22H21BrCl2N6ODegré de pureté :98.89% - 99%Couleur et forme :SolidMasse moléculaire :536.25Ref: TM-T4668
1mg62,00€2mg87,00€5mg119,00€10mg187,00€25mg350,00€50mg530,00€100mg748,00€500mg1.578,00€1mL*10mM (DMSO)140,00€YT 146
CAS :YT 146 is a biochemical.Formule :C18H25N5O4Degré de pureté :98.81% - 99.72%Couleur et forme :SolidMasse moléculaire :375.42PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM forFormule :C18H20N5O7S2·NH4·75H2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :532.09Aminophylline
CAS :Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.Formule :C7H8O2·C2H8N2Degré de pureté :99.31%Couleur et forme :White Or Slightly Yellowish Granules Or Powder SolidMasse moléculaire :420.43Istradefylline
CAS :Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.Formule :C20H24N4O4Degré de pureté :98.18% - 99.95%Couleur et forme :SolidMasse moléculaire :384.43N6-(2-Phenylethyl)adenosine
CAS :N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM forFormule :C18H21N5O4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :371.398-Cyclopentyl-1,3-dimethylxanthine
CAS :8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.Formule :C12H16N4O2Degré de pureté :100% - 98.58%Couleur et forme :SolidMasse moléculaire :248.28Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.Formule :C25H31F3N6O8Degré de pureté :98.40%Couleur et forme :SoildMasse moléculaire :600.55Evodenoson
CAS :Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.Formule :C23H29N7O6Degré de pureté :100% - 99.74%Couleur et forme :SolidMasse moléculaire :499.52Xanthine amine congener
CAS :Xanthine amine congener is an Adenosine receptor antagonist.Formule :C21H28N6O4Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :428.48CGS 21680 Hydrochloride
CAS :CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.Formule :C23H29N7O6·HClDegré de pureté :96.74% - 98.81%Couleur et forme :SolidMasse moléculaire :535.98Ref: TM-T6441
1mg40,00€2mg52,00€5mg86,00€10mg115,00€25mg226,00€50mg410,00€100mg607,00€1mL*10mM (DMSO)90,00€Trabodenoson
CAS :Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.Formule :C15H20N6O6Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :380.36Ref: TM-T34914
1mg131,00€2mg187,00€5mg311,00€10mg467,00€25mg747,00€50mg1.017,00€100mg1.359,00€1mL*10mM (DMSO)344,00€Tecadenoson
CAS :Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.Formule :C14H19N5O5Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :337.33Ref: TM-T17023
1mg50,00€5mg116,00€10mg178,00€25mg306,00€50mg434,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)128,00€N6-Cyclopentyladenosine
CAS :N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's ofFormule :C15H21N5O4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :335.36Vipadenant
CAS :Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formule :C16H15N7ODegré de pureté :97.25% - 97.36%Couleur et forme :SolidMasse moléculaire :321.34Ref: TM-T2373
1mg40,00€2mg52,00€5mg87,00€10mg119,00€25mg210,00€50mg350,00€100mg522,00€500mg1.130,00€1mL*10mM (DMSO)359,00€Tozadenant
CAS :Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Formule :C19H26N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.5Ref: TM-T7320
2mg38,00€5mg58,00€10mg96,00€25mg162,00€50mg273,00€100mg393,00€200mg563,00€1mL*10mM (DMSO)64,00€Doxofylline
CAS :Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.Formule :C11H14N4O4Degré de pureté :99.09% - 99.98%Couleur et forme :SolidMasse moléculaire :266.25Preladenant
CAS :Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosineFormule :C25H29N9O3Degré de pureté :97.32% - 98.18%Couleur et forme :SolidMasse moléculaire :503.56APNEA
CAS :APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Formule :C18H22N6O4Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :386.41Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.Formule :C24H29ClF3N5O5SDegré de pureté :96.67%Couleur et forme :SoildMasse moléculaire :592.03Derenofylline
CAS :Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)Formule :C18H20N4ODegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :308.38Capadenoson
CAS :Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Formule :C25H18ClN5O2S2Degré de pureté :98.85% - 99.62%Couleur et forme :SolidMasse moléculaire :520.03
