Récepteur d'adénosine
Les récepteurs de l'adénosine sont une classe de récepteurs GPCR qui répondent à la nucléoside endogène adénosine. Ces récepteurs sont impliqués dans la régulation de divers processus physiologiques, y compris la fonction cardiovasculaire, les cycles veille-sommeil et les réponses immunitaires. Les modulateurs des récepteurs de l'adénosine ont un potentiel thérapeutique pour traiter des affections telles que les arythmies cardiaques, l'inflammation et les maladies neurodégénératives. Chez CymitQuimica, nous offrons une sélection de modulateurs des récepteurs de l'adénosine de haute qualité pour soutenir vos recherches en biologie cardiovasculaire, neurosciences et immunologie.
Produits appartenant à la catégorie "Récepteur d'adénosine"
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Nitrobenzylthioinosine
CAS :Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Formule :C17H17N5O6SDegré de pureté :98.83% - 99.69%Couleur et forme :Off-White SolidMasse moléculaire :419.41hA3AR agonist 2
hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.Formule :C11H14ClN5O2SCouleur et forme :SolidMasse moléculaire :315.78A2AR-agonist-1
CAS :A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).Formule :C20H22N6O4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :410.43Ref: TM-T10212
1mg96,00€2mg134,00€5mg188,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€500mg1.691,00€1mL*10mM (DMSO)217,00€CHEMBL241987
CAS :CHEMBL241987 targets the Adenosine receptor A3 (human)Formule :C16H11N3ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :261.28Ref: TM-T8598
2mg35,00€5mg50,00€10mg66,00€25mg108,00€50mg162,00€100mg235,00€200mg349,00€1mL*10mM (DMSO)50,00€ZM241385
CAS :ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.Formule :C16H15N7O2Degré de pureté :95.28% - 99.69%Couleur et forme :SolidMasse moléculaire :337.34Ref: TM-T7021
5mg57,00€10mg82,00€25mg133,00€50mg233,00€100mg432,00€200mg652,00€500mg1.026,00€1mL*10mM (DMSO)57,00€Tonapofylline
CAS :Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.Formule :C22H32N4O4Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :416.51Namodenoson
CAS :Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formule :C18H18ClIN6O4Degré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :544.73ATL444
CAS :ATL444 is an adenosine receptor antagonist with affinity (Ki values) for rA1AR, rA2AAR, rA2BAR, and rA3AR of 7.0, 2.5, 61.8, and >1000 nM, respectively.Formule :C17H19N5OCouleur et forme :SolidMasse moléculaire :309.37SCH442416
CAS :SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).Formule :C20H19N7O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :389.41Ref: TM-T23336
1mg48,00€2mg63,00€5mg93,00€10mg139,00€25mg281,00€50mg449,00€100mg658,00€1mL*10mM (DMSO)97,00€FSCPX
CAS :FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.Formule :C23H27FN4O6SDegré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :506.55Ref: TM-T39039
1mg111,00€5mg273,00€10mg409,00€25mg695,00€50mg929,00€100mg1.244,00€200mg1.681,00€1mL*10mM (DMSO)116,00€AZD4635
CAS :AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Formule :C15H11ClFN5Degré de pureté :99.15% - 99.90%Couleur et forme :SolidMasse moléculaire :315.73Ref: TM-T4265
1mg37,00€2mg52,00€5mg79,00€10mg116,00€25mg188,00€50mg296,00€100mg457,00€500mg1.008,00€1mL*10mM (DMSO)87,00€BAY-545
CAS :BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formule :C18H22F3N3O4SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :433.45Ref: TM-T8512
1mg88,00€5mg170,00€10mg248,00€25mg444,00€50mg638,00€100mg889,00€200mg1.198,00€1mL*10mM (DMSO)182,00€Kira8 Hydrochloride
CAS :Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.Formule :C31H30Cl2N6O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :637.58A2A receptor antagonist 1
CAS :A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.Formule :C16H12FN5ODegré de pureté :99.29% - 99.76%Couleur et forme :SolidMasse moléculaire :309.3Ref: TM-T37792
1mg37,00€5mg64,00€10mg92,00€25mg185,00€50mg284,00€100mg419,00€500mg883,00€1mL*10mM (DMSO)47,00€Norisoboldine
CAS :Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.Formule :C18H19NO4Degré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :313.35Adenosine amine congener
CAS :Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Formule :C28H32N8O6Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :576.6Theophylline monohydrate
CAS :Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calciumFormule :C7H8N4O2·H2ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :198.18Nelonicline
CAS :Nelonicline is a selective agonist of neuronal nicotinic receptors.Formule :C17H19N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.42Alloxazine
CAS :Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.Formule :C10H6N4O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :214.18N6-Cyclohexyladenosine
CAS :N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.Formule :C16H23N5O4Degré de pureté :99.84% - 99.98%Couleur et forme :SolidMasse moléculaire :349.38Xanthine amine congener trihydrochloride
CAS :Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Formule :C21H29ClN6O4Degré de pureté :97.85%Couleur et forme :SolidMasse moléculaire :464.95CCPA
CAS :CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptorFormule :C15H20ClN5O4Degré de pureté :99.10%Couleur et forme :Off-White To Light Yellow SolidMasse moléculaire :369.8PF-02575799
CAS :PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).Formule :C42H37FN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :680.77Piclidenoson
CAS :Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.Formule :C18H19IN6O4Degré de pureté :100% - ≥95%Couleur et forme :SolidMasse moléculaire :510.29Ref: TM-T7188
2mg42,00€5mg62,00€10mg89,00€25mg183,00€50mg298,00€100mg464,00€200mg663,00€1mL*10mM (DMSO)70,00€ANR 94
CAS :ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.Formule :C9H13N5ODegré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :207.23Ref: TM-T22031
2mg42,00€5mg64,00€10mg97,00€25mg188,00€50mg329,00€100mg465,00€200mg655,00€1mL*10mM (DMSO)63,00€CGS 15943
CAS :CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.Formule :C13H8ClN5ODegré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :285.695-Iodotubercidin
CAS :5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.Formule :C11H13IN4O4Degré de pureté :99.98%Couleur et forme :Tan SolidMasse moléculaire :392.15Ref: TM-T6745
1mg46,00€2mg57,00€5mg92,00€10mg155,00€25mg343,00€50mg509,00€100mg735,00€1mL*10mM (DMSO)97,00€Regadenoson
CAS :Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.Formule :C15H18N8O5Degré de pureté :99.57% - 99.81%Couleur et forme :Off-White SolidMasse moléculaire :390.35Ref: TM-T2671
2mg47,00€5mg65,00€10mg92,00€25mg173,00€50mg273,00€100mg416,00€500mg935,00€1mL*10mM (DMSO)72,00€MIPS521
CAS :MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Formule :C19H10ClF6NOSDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :449.8Ref: TM-T9330
1mg38,00€2mg49,00€5mg79,00€10mg111,00€25mg188,00€50mg329,00€100mg512,00€1mL*10mM (DMSO)87,00€PSB 1115
CAS :PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.Formule :C14H14N4O5SDegré de pureté :100% - 99.24%Couleur et forme :SolidMasse moléculaire :350.351-Ethyl-6-aminouracil
CAS :1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have highFormule :C6H9N3O2Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :155.15A2B receptor antagonist 1
CAS :A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.Formule :C21H24N6O2Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :392.45Ref: TM-T10058
1mg369,00€5mg735,00€10mg938,00€25mg1.473,00€50mg1.882,00€100mg2.670,00€1mL*10mM (DMSO)843,00€ISAM-140
CAS :ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.Formule :C19H19N3O3Degré de pureté :97.41%Couleur et forme :SolidMasse moléculaire :337.37N-[(4-Aminophenyl)methyl]adenosine
CAS :N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).Formule :C17H20N6O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :372.38Ref: TM-T16166
1mg92,00€5mg188,00€10mg283,00€25mg558,00€50mg885,00€100mg1.415,00€1mL*10mM (DMSO)240,00€FK-453
CAS :FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.Formule :C23H25N3O2Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :375.46Enprofylline
CAS :Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formule :C8H10N4O2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :194.19Ref: TM-T21389
2mg44,00€5mg65,00€10mg93,00€25mg149,00€50mg226,00€100mg335,00€200mg465,00€1mL*10mM (DMSO)63,00€5'-N-Ethylcarboxamidoadenosine
CAS :NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Formule :C12H16N6O4Degré de pureté :≥95%Couleur et forme :PowderMasse moléculaire :308.29Proxyphylline
CAS :Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.Formule :C10H14N4O3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :238.24GS-9667
CAS :GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia viaFormule :C21H24FN5O4SDegré de pureté :99.76% - 99.76%Couleur et forme :SolidMasse moléculaire :461.51Adenosine A1 receptor activator T62
CAS :Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and alsoFormule :C15H14ClNOSDegré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :291.8Ref: TM-T14127
1mg87,00€5mg183,00€10mg273,00€25mg439,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)280,00€Adenosine 5'-monophosphate monohydrate
CAS :Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.Formule :C10H14N5O7P·H2ODegré de pureté :97.68% - 98.49%Couleur et forme :White PowderMasse moléculaire :365.248-Chloro caffeine
CAS :8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.Formule :C8H9ClN4O2Couleur et forme :SolidMasse moléculaire :228.64ST-1535
CAS :ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.Formule :C12H16N8Degré de pureté :99.64% - 99.71%Couleur et forme :SolidMasse moléculaire :272.31SDZ WAG 994
CAS :SDZ WAG 994 is an A1 adenosine receptor agonist.Formule :C17H25N5O4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :363.41Ref: TM-T23347
1mg66,00€5mg120,00€10mg175,00€25mg316,00€50mg455,00€100mg620,00€200mg835,00€1mL*10mM (DMSO)127,00€2-Chloroadenosine
CAS :2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectivelyFormule :C10H12ClN5O4Degré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :301.69Adenosine receptor antagonist 4
CAS :Adenosine receptor antagonist 4 is an adenosine receptor antagonist.Formule :C10H13N3Degré de pureté :98.59% - 99.58%Couleur et forme :Off-White PowderMasse moléculaire :175.23Adenosine receptor agonist 1
Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.Formule :C12H14ClN5O2SeCouleur et forme :SolidMasse moléculaire :374.68AB928
CAS :AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].Formule :C23H22N8ODegré de pureté :100% - 98.55%Couleur et forme :SolidMasse moléculaire :426.47Ref: TM-T14078
1mg50,00€5mg124,00€10mg197,00€25mg389,00€50mg462,00€100mg663,00€1mL*10mM (DMSO)134,00€DPCPX
CAS :DPCPX (PD 116948) is an A1 adenosine receptor antagonistFormule :C16H24N4O2Degré de pureté :99.23% - 99.93%Couleur et forme :White SolidMasse moléculaire :304.39MRS-1706
CAS :MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.Formule :C27H29N5O5Degré de pureté :97.95%Couleur et forme :SolidMasse moléculaire :503.55Ref: TM-T16136
1mg37,00€2mg52,00€5mg79,00€10mg119,00€25mg240,00€50mg472,00€100mg687,00€1mL*10mM (DMSO)88,00€
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