Signalisation du cytosquelette
Les inhibiteurs de la signalisation du cytosquelette sont des composés qui perturbent les voies de signalisation régulant le cytosquelette, essentiel pour la forme, la motilité, la division des cellules et le transport intracellulaire. Ces inhibiteurs sont utilisés pour étudier la dynamique des protéines du cytosquelette, telles que l'actine et la tubuline, et leur rôle dans des processus comme la migration cellulaire, l'adhésion et la métastase du cancer. Les inhibiteurs de la signalisation du cytosquelette sont précieux dans la recherche en biologie cellulaire, en cancérologie et en neurobiologie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs de la signalisation du cytosquelette de haute qualité pour soutenir vos recherches dans ces domaines.
Produits appartenant à la catégorie "Signalisation du cytosquelette"
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Cenisertib
CAS :Cenisertib is A potent ATP-competitive multi-kinase inhibitor, showing inhibitory effects on the activity of Aurora-kinase-A/B, ABL1, AKT, STAT5, FLT3, as wellFormule :C24H30FN7OCouleur et forme :SolidMasse moléculaire :451.54XL228
CAS :XL228 is an inhibitor of multi-targeted tyrosine kinase (IC50s: 5, 3.1, 1.6, 6.1, 2 nM for Bcr-Abl, Aurora A, IGF-1R, Src, and Lyn, respectively).Formule :C22H31N9ODegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :437.54Ref: TM-T17267
1mg56,00€2mg78,00€5mg99,00€10mg149,00€25mg258,00€50mg393,00€100mg582,00€1mL*10mM (DMSO)110,00€Bisindolylmaleimide VIII acetate
CAS :Bisindolylmaleimide VIII acetate is a selective PKC inhibitor with an IC50 of 158 nM in rat brain and varying IC50s for different PKC isoforms.Formule :C26H26N4O4Degré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :458.51PKC-ε translocation inhibitor peptide
PKC-ε Translocation Inhibitor Peptide is a selective modulator that controls the FcγR-mediated internalization rate of opsonized beads without affecting FcαRDegré de pureté :98%Couleur et forme :Odour SolidArg-Gly-Asp TFA (99896-85-2(free base))
Arg-Gly-Asp TFA (RGD, 99896-85-2) is a tripeptide that promotes cell adhesion and integrin binding.Formule :C14H23F3N6O8Degré de pureté :99.2% - ≥98%Couleur et forme :SolidMasse moléculaire :460.36STX-100
PY314 is a CHO-expressed humanized monoclonal antibody targeting TREM2 with antitumor activity for the study of metastatic renal cell carcinoma.Degré de pureté :95% - 95%Couleur et forme :Odour LiquidEMD534085
CAS :EMD534085 is an effective and selective mitotic kinesin-5 inhibitor (IC50: 8 nM).Formule :C25H31F3N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :476.53Nilotinib monohydrochloride monohydrate
CAS :Nilotinib monohydrochloride monohydrate (Nilotinib (monohydrochloride monohydrate)) is significantly potent BCR-ABL against, is a second generation tyrosineFormule :C28H22F3N7O·HCl·H2ODegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :583.99Anti-Mouse IL-1a Antibody (ALF-161)
Anti-Mouse IL-1a Antibody is an IgG1 subtype inhibitor specific to mouse IL-1a, derived from the Armenian Hamster.Degré de pureté :98%Couleur et forme :Odour SolidDanicamtiv
CAS :Danicamtiv (MYK-491) is an inotropic agent and it also is a selective allosteric activator of cardiac myosin.Formule :C16H20F3N5O4SDegré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :435.42Ref: TM-T15050
1mg136,00€5mg274,00€10mg454,00€25mg750,00€50mg1.026,00€100mg1.406,00€1mL*10mM (DMSO)303,00€LY 379196
LY 379196, a potent PKC-β inhibitor (IC 50: 50 nM for PKC βI and 30 nM for PKC βII), effectively suppresses the proliferation of bovine retinal microvascular endothelial cells (BREC) induced by VEGF, IGF-1, and bFGF. This compound serves as an antiproliferative agent for proliferative retinopathy.Formule :C30H34N4O5SCouleur et forme :SolidMasse moléculaire :562.68XL888
CAS :XL888 is an orally bioavailable Hsp90 inhibitor, blocking cell proliferation and inducing tumor regression with an IC50 of 24 nM.Formule :C29H37N5O3Degré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :503.64Loureirin A
CAS :Loureirin A inhibits platelet aggregation and PI3K/Akt signaling, promotes hair follicle repair, and has anti-fibrotic and anti-angiogenic properties.Formule :C17H18O4Degré de pureté :99.83% - 99.84%Couleur et forme :SolidMasse moléculaire :286.32Ref: TM-T5S0896
1mg74,00€5mg133,00€10mg188,00€25mg329,00€50mg490,00€100mg697,00€200mg938,00€1mL*10mM (DMSO)207,00€Mitoxantrone
CAS :Mitoxantrone: anthracenedione antibiotic, disrupts DNA/RNA replication, binds to topoisomerase II, less cardiotoxic than doxorubicin.Formule :C22H28N4O6Degré de pureté :97.97% - 98.74%Couleur et forme :Blue PowderMasse moléculaire :444.48CID-663143
CAS :CID-663143 inhibits cancer cell growth and shows microtubule-binding activity.Formule :C19H18N4O2SDegré de pureté :99.56% - 99.68%Couleur et forme :SolidMasse moléculaire :366.44Ref: TM-T23889
1mg77,00€5mg158,00€10mg225,00€25mg338,00€50mg475,00€100mg638,00€200mg845,00€1mL*10mM (DMSO)164,00€Soblidotin
CAS :Soblidotin (TZT-1027) (Auristatin PE) is an inhibitor of tubulin polymerization. It is also a novel synthetic Dolastatin 10 derivative.Formule :C39H67N5O6Degré de pureté :97.48%Couleur et forme :SolidMasse moléculaire :701.98DCPLA-ME
CAS :DCPLA-ME (2-[(2-Pentylcyclopropyl)methyl]cyclopropaneoctanoic acid methyl ester) is the methyl ester form of DCPLA and can be used to treat neurodegenerativeFormule :C21H38O2Degré de pureté :98.16%Couleur et forme :SolidMasse moléculaire :322.53Ref: TM-T10980
1mg65,00€5mg133,00€10mg180,00€25mg369,00€50mg605,00€100mg815,00€200mg1.111,00€1mL*10mM (DMSO)145,00€MT189
CAS :MT189 (Antiproliferative agent-14) inhibits tubulin polymerization (IC50 3.41 μM), arrests G2/M cell cycle, and is highly antiproliferative.Formule :C21H18FN3O2Degré de pureté :98.67%Couleur et forme :SoildMasse moléculaire :363.38G-5555 hydrochloride (1648863-90-4 free base)
G-5555 hydrochloride is a potent and selective p21-activated kinase 1 (PAK1) inhibitor with a Ki of 3.7 nM.Formule :C25H26Cl2N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :529.42TAS0612
CAS :TAS0612, a novel oral inhibitor of RSK, AKT, and S6K, exhibits broad-spectrum antitumor activity by impeding cell growth [1].Formule :C27H34F3N9O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :573.61Recilisib
CAS :Recilisib (ON 01210) is a radioprotectant,can activate AKT, PI3K activities in cells.Formule :C16H13ClO4SDegré de pureté :98.85% - 98.96%Couleur et forme :SolidMasse moléculaire :336.79Ref: TM-T13862
1mg46,00€2mg59,00€5mg87,00€10mg119,00€25mg187,00€50mg354,00€100mg528,00€500mg1.159,00€1mL*10mM (DMSO)105,00€LP-261
CAS :LP-261 is a novel tubulin targeting anticancer agent that binds at the colchicine site on tubulin, inducing G2/M arrest.Formule :C22H19N3O4SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :421.47Ref: TM-T9595
1mg38,00€2mg49,00€5mg79,00€10mg119,00€25mg187,00€50mg354,00€100mg528,00€1mL*10mM (DMSO)87,00€Sabizabulin
CAS :Sabizabulin (ABI-231) is a potent, orally bioavailable α- and β-tubulin inhibitor.Cost-effective and quality-assured.Formule :C21H19N3O4Degré de pureté :98.04% - 99.76%Couleur et forme :SolidMasse moléculaire :377.39Ref: TM-T17228
1mg145,00€2mg207,00€5mg354,00€10mg547,00€25mg880,00€50mg1.198,00€100mg1.596,00€500mg3.220,00€KOdiA-PC
CAS :KOdiA-PC is a truncated oxidized phospholipid and a CD36-targeting ligand found on oxLDL. It inhibits activation of TLR4 signaling components.Formule :C32H58NO11PCouleur et forme :SolidMasse moléculaire :663.78PKC β pseudosubstrate acetate
PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) is a selective cell-permeable inhibitor of PKC.Degré de pureté :95.01%Couleur et forme :SoildMps1-IN-2
CAS :Mps1-IN-2 is a potent, selective and ATP-competitive dual Mps1/Plk1 inhibitor.Formule :C26H36N6O3Degré de pureté :96.24% - 99.75%Couleur et forme :SolidMasse moléculaire :480.6Sotrastaurin
CAS :Sotrastaurin (AEB071) is a potent pan-PKC inhibitor (Kis: 0.95/0.64/2.1/3.2/1.8/0.22 nM for PKCα/βI/δ/ε/η/θ).Formule :C25H22N6O2Degré de pureté :98% - 99.70%Couleur et forme :SolidMasse moléculaire :438.48Ref: TM-T6278
1mg49,00€5mg96,00€10mg166,00€25mg313,00€50mg553,00€100mg790,00€500mg1.578,00€1mL*10mM (DMSO)115,00€K-80003
CAS :K-80003(TX-803) is a potent retinol-like X-receptor-alpha regulator that inhibits TRxrα-dependent Akt activation and tumor cell growth.Formule :C22H21FO2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :336.4Ref: TM-T11734
1mg49,00€5mg104,00€10mg166,00€25mg283,00€50mg430,00€100mg633,00€500mg1.349,00€1mL*10mM (DMSO)115,00€Bexotegrast
CAS :Bexotegrast (PLN-74809) is an αvβ6 and αvβ1 integrin inhibitor with antifibrotic properties for the study of idiopathic pulmonary fibrosis (IPF).Formule :C27H36N6O3Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :492.61Rotigaptide TFA(355151-12-1 free base)
Rotigaptide TFA is a Cx43 modulator & AAP that maintains gap junctions & cell communication under stress.Formule :C30H40F3N7O11Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :731.67PROTAC Hsp90α degrader 1
Compound X10g (PROTAC Hsp90α degrader 1) is a selective agent targeting Hsp90α for degradation and is utilized in breast cancer research.Formule :C43H50N6O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :762.89PF-562271 besylate
CAS :PF-562271 besylate: potent, ATP-competitive FAK inhibitor, IC50 1.5 nM, 10x less effective on Pyk2, highly selective vs other kinases.Formule :C21H20F3N7O3S·C6H6O3SDegré de pureté :97.65% - 99.01%Couleur et forme :SolidMasse moléculaire :665.66Ref: TM-T6177
1mg38,00€5mg79,00€10mg88,00€25mg145,00€50mg210,00€100mg313,00€200mg452,00€1mL*10mM (DMSO)95,00€Efalizumab
CAS :Efalizumab: humanized monoclonal antibody CD11a; modulates T cell activation/adhesion; for plaque psoriasis, psoriatic arthritis research.Degré de pureté :SDS-PAGE:95% SEC-HPLC:98.77%Couleur et forme :LiquidMasse moléculaire :146.14 kDaAntiangiogenic agent 4
Compound 3b, an antiangiogenic agent, inhibits Akt phosphorylation in both HFF and HUVEC cells and is utilized in cancer research [1].Formule :C21H24N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :380.44NAP1051
CAS :NAP1051, a biomimetic analog of Lipoxin A4, serves an anti-tumor role by targeting the inflammatory tumor microenvironment. It inhibits the chemotaxis of neutrophils to fMLP and stimulates macrophage efferocytosis by activating AKT. NAP1051 is utilized in research on colorectal cancer.Formule :C23H34O5Couleur et forme :SolidMasse moléculaire :390.51YM-53601
CAS :YM-53601 is an SQS inhibitor that inhibits adipogenic biosynthesis and lipid secretion in rodents.YM-53601 is a cholesterol-lowering agent that inhibits FDFT1.Formule :C21H22ClFN2ODegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :372.86FAK-IN-10
CAS :FAK-IN-10 is an inhibitor of FAK (IC50:76.3 μM).FAK-IN-10 z MCF-7 and A431 cell lines showed antitumor activity with IC50 of 4.23 and 0.78 μM, respectively.Formule :C15H10BrN3O2SDegré de pureté :99.78%Couleur et forme :SoildMasse moléculaire :376.23FITC-Ahx-Gly-Arg-Gly-Asp-Ser-Pro
CAS :FITC-Ahx-Gly-Arg-Gly-Asp-Ser-Pro, also known as FITC-linked GRGDSP, is a fluorescent peptide with integrin inhibitory properties.Formule :C49H59N11O16SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1090.12Vodobatinib
CAS :Vodobatinib (K-0706) is a novel 3rd generation (3G) TKI effective against wild-type and mutated BCR-ABL1 with limited off-target activity.Formule :C27H20ClN3O2Degré de pureté :99.06% - 99.55%Couleur et forme :SolidMasse moléculaire :453.92Ref: TM-T8882
1mg37,00€5mg79,00€10mg116,00€25mg212,00€50mg340,00€100mg528,00€500mg1.275,00€1mL*10mM (DMSO)87,00€Obtustatin triacetate
Obtustatin triacetate, a 41-residue non-RGD disintegrin isolated from the venom of Vipera lebetina obtusa, serves as a potent and selective inhibitor of theFormule :C184H284N52O57S8·3C2H4O2Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :4573.21KW-2478
CAS :KW-2478 is a non-ansamycin HSP90 inhibitor with IC50 of 3.8 nM.Formule :C30H42N2O9Degré de pureté :98.68% - 99.52%Couleur et forme :SolidMasse moléculaire :574.66Ref: TM-T6558
1mg56,00€2mg81,00€5mg119,00€10mg187,00€25mg316,00€50mg472,00€100mg662,00€1mL*10mM (DMSO)205,00€Mavacamten
CAS :Mavacamten (MYK-461) is an orally bioavailable inhibitor of cardiac myosin ATPase,( IC50s of 490, 711 nM for bovine cardiac and human cardiac, respectively)Formule :C15H19N3O2Degré de pureté :99.53% - 99.98%Couleur et forme :SolidMasse moléculaire :273.33[Ala113]-MBP (104-118) acetate
[Ala113]MBP(104-118) acetate is an noncompetitive peptide inhibitors of protein kinase C (PKC), with IC50s ranging from 28-62 μM.Formule :C69H108N20O21Degré de pureté :97.72%Couleur et forme :SolidMasse moléculaire :1553.74Gypsogenin
CAS :Gypsogenin (639-14-5) is a naturally occurring biochemical that shows anti-ABL1 kinase and anti-chronic Myelogenous Leukemia activities.Formule :C30H46O4Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :470.68Ref: TM-T25476
1mg134,00€5mg315,00€10mg469,00€25mg748,00€50mg1.064,00€100mg1.415,00€1mL*10mM (DMSO)349,00€Tubulin inhibitor 7
CAS :Tubulin inhibitor 7 is an inhibitor of tubulin and a potent inhibitor of multiple cancer cell lines (tubulin polymerization (IC50: 0.52 μM), K562 cell growth (Formule :C21H14N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :358.35ICAM-1-IN-1
CAS :ICAM-1-IN-1 is a potent and selective E-selectin(IC50 = 7 nM) and ICAM-1(IC50 = 5 nM) inhibitor.Formule :C15H11BrN2O2SDegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :363.23Ref: TM-T13147
1mg185,00€5mg393,00€10mg587,00€25mg935,00€50mg1.264,00€100mg1.700,00€500mg3.410,00€1mL*10mM (DMSO)432,00€Benproperine phosphate
CAS :Benproperine phosphate (Pirexyl phosphate) is a cough suppressant.Formule :C21H30NO5PDegré de pureté :99.84%Couleur et forme :PowderMasse moléculaire :407.44Bimosiamose disodium
CAS :Bimosiamose disodium (TBC-1269Z), a pan-selectin inhibitor, has IC50s: E-selectin 88 μM, P-selectin 20 μM, L-selectin 86 μM; anti-inflammatory.Formule :C46H52Na2O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :906.88IPA-3
CAS :IPA-3 is a selective non-ATP competitive Pak1 inhibitor with IC50 of 2.5 μM, no inhibition to group II PAKs (PAKs 4-6).Formule :C20H14O2S2Degré de pureté :96.7%Couleur et forme :SolidMasse moléculaire :350.45Peptide5 TFA
Peptide5 TFA, a connexin 43 mimetic peptide, mitigates swelling, astrogliosis, and neuronal cell death in animal models of spinal cord injury.Formule :C62H99F3N16O22SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1509.6α2β1 Integrin Ligand Peptide acetate
α2β1 Integrin Ligand Peptide acetate (α2β1 Integrin Ligand Peptide acetate (134580-64-6)) is a potential antagonist of α2β1 integrin receptor.Formule :C16H26N4O11Degré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :450.4Larixol
CAS :Larixol acts as both an fMLP inhibitor and a modulator of various signaling pathways by inhibiting Src kinase, ERK1/2, p38, and AKT phosphorylation critical forFormule :C20H34O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :306.48BGG463
CAS :BGG463 (K 0859) can inhibit c-ABL-T334I, BCR-ABL and BCR-ABL-T315I variants with an IC50 of 0.25 μM, 0.09 μM and 0.590 μM, respectively.Formule :C30H29F3N6O3Degré de pureté :100% - 95.05%Couleur et forme :SolidMasse moléculaire :578.58Ref: TM-T4618
1mg62,00€2mg87,00€5mg119,00€10mg188,00€25mg350,00€50mg505,00€100mg730,00€1mL*10mM (DMSO)154,00€Protein Kinase C (19-31) (TFA)(121545-65-1,free)
Protein Kinase C (19-31) TFA is a serine-modified PKCa-derived inhibitor for testing PKC activity.Formule :C69H119F3N26O18Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1657.842',4'-DIHYDROXYCHALCONE
CAS :2',4'-DIHYDROXYCHALCONE (2',4'-DHC) as a compound with Hsp90 inhibitory and antifungal effectsFormule :C15H12O3Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :240.25Ref: TM-T8829
2mg42,00€5mg62,00€10mg87,00€25mg154,00€50mg235,00€100mg354,00€200mg520,00€1mL*10mM (DMSO)65,00€Triclabendazole
CAS :Triclabendazole (CGA89317) has been used in trials studying Parasitic Disease.Formule :C14H9Cl3N2OSDegré de pureté :99.11%Couleur et forme :White To Brown Crystalline PowderMasse moléculaire :359.66Tubulin inhibitor 24
CAS :Tubulin inhibitor 24 is a potent inhibitor that can inhibit tubulin polymerization.Formule :C22H21N3O3Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :375.42Rocaglamide
CAS :Rocaglamide (Roc-A) from Aglaia treats coughs, injuries, asthma, skin issues, and inhibits NF-κB in T-cells.Formule :C29H31NO7Degré de pureté :95.32% - 98.46%Couleur et forme :SolidMasse moléculaire :505.56mP6
CAS :mP6 (Myr-FEEERA-OH), a myristoylated peptide, selectively inhibits Gα 13's interaction with integrin β 3 while preserving talin-dependent integrin function.Formule :C47H75N9O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :990.15HG-7-86-01
CAS :HG-7-86-01 is a selective type II tyrosine kinase inhibitor with antiproliferative activity against mutant T315I- Bcr-Abl for chronic myeloid leukemia (CML).Formule :C28H21F3N6O2SDegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :562.57Bisindolylmaleimide V
CAS :Bisindolylmaleimide V, a bisindolylmaleimide derivative, is an inactive of a kinase inhibitor.Formule :C21H15N3O2Degré de pureté :90%Couleur et forme :Red SolidMasse moléculaire :341.36Verubulin
CAS :Verubulin (MPC 6827) is a microtubule blocking agent with cytotoxic and potentially anticancer activity that disrupts newly formed blood vessels in xenografts.Formule :C17H17N3ODegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :279.34UMK57
CAS :UMK57 is a CENP-Ei and MCAK enhancer, selectively promoting k-MT attachment error correction to inhibit chromosome missegregation of small molecule compounds,Formule :C17H17N3SDegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :295.4Thiabendazole
CAS :Thiabendazole (2-(4-Thiazolyl)benzimidazole) is a benzimidazole derivative with anthelminthic property.Formule :C10H7N3SDegré de pureté :99.14%Couleur et forme :Light Yellow PowderMasse moléculaire :201.25PKCβII Peptide Inhibitor I
CAS :PKCβII Peptide Inhibitor I, a specific PKCβII inhibitor, exhibits cardioprotective properties in a rat cardiac ischemia/reperfusion injury model and mitigatesFormule :C61H94N12O19Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1299.47EL-102
CAS :EL-102 is a HIF1α inhibitor with anticancer activity that inhibits microtubule protein polymerization and can be used to study prostate cancer.Formule :C19H16N2O3S2Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :384.47Ref: TM-T15205
1mg87,00€5mg216,00€10mg349,00€25mg545,00€50mg740,00€100mg1.103,00€1mL*10mM (DMSO)183,00€AG957
CAS :Tyrphostin AG957, a tyrosine kinase inhibitor with anti-BCR/ABL tyrosine kinase activity restores beta1 integrin-mediated adhesion and inhibitory signaling inFormule :C15H15NO4Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :273.28Ref: TM-T21785
1mg89,00€5mg212,00€10mg315,00€25mg527,00€50mg750,00€100mg1.017,00€1mL*10mM (DMSO)265,00€Adaphostin
CAS :Adaphostin (NSC-680410) is a p210Bcr/Abl tyrosine kinase inhibitor with IC50 of 14 μM.Formule :C24H27NO4Degré de pureté :97.31%Couleur et forme :SolidMasse moléculaire :393.48Vaccarin
CAS :Vaccarin, a key flavonoid glycoside in Vaccariae semen, undergoes methylation, hydroxylation, glycosylation, and deglycosylation.Formule :C32H38O19Degré de pureté :99.16% - 99.97%Couleur et forme :SolidMasse moléculaire :726.63GSK-923295
CAS :GSK923295 is a selective allosteric inhibitor of CENP-E kinesin motor ATPase(Ki=3.2 nM).Formule :C32H38ClN5O4Degré de pureté :96.22% - 98.02%Couleur et forme :SolidMasse moléculaire :592.13Ref: TM-T2039
1mg49,00€2mg70,00€5mg97,00€10mg168,00€25mg331,00€50mg510,00€100mg737,00€1mL*10mM (DMSO)136,00€Mitoxantrone dihydrochloride
CAS :Mitoxantrone dihydrochloride (NSC-301739) is an anthracenedione antibiotic with antineoplastic activity. Mitoxantrone is a type II topoisomerase inhibitor.Formule :C22H30Cl2N4O6Degré de pureté :100% - 99.85%Couleur et forme :Blue-Black Solid From Water Ethanol SolidMasse moléculaire :517.4Feretoside
CAS :Feretoside is a natural product extracted from the barks of E. ulmoides. Feretoside shows inducible activity on the heat shock factor 1 (HSF1).Formule :C17H24O11Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :404.37Ref: TM-TQ0280
1mg85,00€5mg180,00€10mg274,00€25mg465,00€50mg663,00€100mg919,00€500mg1.833,00€1mL*10mM (DMSO)298,00€Ombrabulin
CAS :Ombrabulin is a derivative of CA-4 phosphate. It is known to show antivascular effects through selective disruption of the tubulin cytoskeleton of endothelial cells.Formule :C21H26N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :402.44GW406108X
CAS :GW406108X is a Kif15 and ULK1 inhibitor; IC50: 0.82 µM (ATPase), pIC50: 6.37; blocks autophagy.Formule :C20H11Cl2NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :400.2117-AEP-GA
CAS :17-AEP-GA is an HSP90 antagonist and a potent inhibitor of glioblastoma cell proliferation, survival, migration and invasion.Formule :C34H50N4O8Degré de pureté :97.77% - 99.56%Couleur et forme :SolidMasse moléculaire :642.78Tirofiban hydrochloride monohydrate
CAS :Tirofiban(MK383) hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.Formule :C22H39ClN2O6SDegré de pureté :95.83% - 99.94%Couleur et forme :White SolidMasse moléculaire :495.07Desmethylglycitein
CAS :Desmethylglycitein (6,7,4'-Trihydroxyisoflavone) , is a novel inhibitor of PKCα in suppressing solar UV-induced matrix metalloproteinase 1, which hasFormule :C15H10O5Degré de pureté :97.93%Couleur et forme :SolidMasse moléculaire :270.24Ref: TM-TN1299
1mg178,00€5mg540,00€10mg715,00€25mg1.103,00€50mg1.491,00€100mg2.005,00€500mg4.010,00€1mL*10mM (DMSO)442,00€PF-2771
CAS :PF-2771: potent CENP-E inhibitor, IC50 of 16.1 nM, used in cancer treatment.Formule :C29H36ClN5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :554.08PKCβ inhibitor 1
CAS :PKCβ inhibitor 1 (KUN79359)(KUN79359) is a potent, selective and ATP-competitive inhibitor of PKC isozymes(IC50s of 21 and 5 nM for human PKCβ1 and PKCβ2,Formule :C24H21N5O2Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :411.46Ref: TM-T8376
1mg154,00€5mg424,00€10mg605,00€25mg920,00€50mg1.216,00€100mg1.673,00€200mg2.252,00€500µg93,00€1mL*10mM (DMSO)401,00€Ingenol
CAS :Ingenol mebutate treats actinic keratosis, has anticancer properties, and may reactivate latent HIV.Formule :C20H28O5Degré de pureté :99.78% - 99.87%Couleur et forme :SolidMasse moléculaire :348.43Ref: TM-T5S2017
1mg52,00€5mg95,00€10mg127,00€25mg246,00€50mg467,00€100mg640,00€500mg1.359,00€1mL*10mM (DMSO)96,00€PF04929113
CAS :PF04929113 (SNX-5422), a synthetic small molecule Hsp90 inhibitor, offers potent efficacy orally for various cancers.Formule :C25H30F3N5O4Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :521.53Ref: TM-T6341
1mg39,00€2mg49,00€5mg84,00€10mg119,00€25mg187,00€50mg354,00€100mg527,00€1mL*10mM (DMSO)96,00€OXA-11
CAS :OXA-11 (FAK-IN-16) is a FAK inhibitor with anti-tumor activity, useful for cancer research.Formule :C37H49F3N7O5PDegré de pureté :98.70% - 99.20%Couleur et forme :SolidMasse moléculaire :759.8cSRC/BCR-ABL1-IN-1
cSRC/BCR-ABL1-IN-1 (compound 16a) is a dual-target inhibitor of the cSRC/BCR-ABL1 kinases.Formule :C24H27ClN6O4Couleur et forme :SolidMasse moléculaire :498.96HSP90-IN-19
CAS :HSP90-IN-19: potent Hsp90 inhibitor, IC50 = 0.27 μM, used in research on viral diseases, neurodegeneration, inflammation.Formule :C29H38O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :498.61ATM-3507
CAS :ATM-3507 is an inhibitor of tropomyosin. In human melanoma cell lines, the IC50s are from 3.83-6.84 μM.Formule :C37H46FN5O2Degré de pureté :96.36% - 99.10%Couleur et forme :SolidMasse moléculaire :611.79Asciminib
CAS :Asciminib (ABL001) (ABL001) is a potent and selective Bcr-Abl inhibitor (Kd: 0.5-0.8nM).Formule :C20H18ClF2N5O3Degré de pureté :97.93% - 99.45%Couleur et forme :SolidMasse moléculaire :449.84Ref: TM-T5177
1mg63,00€2mg92,00€5mg127,00€10mg187,00€25mg305,00€50mg427,00€100mg630,00€500mg1.320,00€1mL*10mM (DMSO)139,00€Natalizumab
CAS :Natalizumab used for the treatment of relapsing remitting multiple sclerosis and Crohn's disease.Degré de pureté :98.00%Couleur et forme :LiquidMasse moléculaire :N/AHSP90-IN-32
CAS :HSP90-IN-32, a carboxy-terminus inhibitor of Hsp90C, exhibits antiproliferative activity in various cell lines including SKMel173, SKMel103, SKMel19, and A375, with IC50 values of 1.01 μM, 0.782 μM, 0.607 μM, and 1.413 μM, respectively. This compound holds potential for research in anticancer agents.Formule :C33H40N2O4Couleur et forme :SolidMasse moléculaire :528.68CW-069
CAS :CW-069 (IC50=75 μM), an allosteric selective inhibitor of microtubule motor protein HSET, exhibits remarkable specificity over KSP.Formule :C23H21IN2O3Degré de pureté :97.52% - 98.59%Couleur et forme :SolidMasse moléculaire :500.33Ref: TM-T6209
1mg43,00€5mg90,00€10mg125,00€25mg216,00€50mg306,00€100mg432,00€500mg938,00€1mL*10mM (DMSO)89,00€DM4
CAS :DM4 (Ravtansine) can be used in the preparation of antibody drug conjugate and it is an antitubulin agent. It can inhibit cell division.Formule :C38H54ClN3O10SDegré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :780.37NQTrp
CAS :NQTrp is an inhibitor of the aggregation of the tau protein with generic anti-amyloidogenic effects.Formule :C21H16N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :360.36N-Phenylbenzylamine
CAS :A series of N-Phenylbenzylamine (Benzenemethanamine) as potential cytotoxic and antimitotic agents acting by inhibition of tubulin polymerizationFormule :C13H13NDegré de pureté :99.93%Couleur et forme :Colorless To Pale Yellow Crystalline PowderMasse moléculaire :183.25Curvulin
CAS :Curvulin is the active metabolite isolated from Paraphoma sp. VIZR 1.46. Curvularin inhibits iNOS expression and microtubule assembly.Formule :C12H14O5Degré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :238.24Ref: TM-T36850
1mg145,00€5mg319,00€10mg472,00€25mg753,00€50mg1.074,00€100mg1.444,00€1mL*10mM (DMSO)284,00€Hu7691 free base
CAS :Hu7691 free base is an Akt inhibitor that inhibits Akt1, Akt2 and Akt3 and induces differentiation of neuroblastoma cells.Formule :C22H21F3N4ODegré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :414.423H-Gly-Arg-Gly-Asp-Asn-Pro-OH
CAS :RGD peptide (GRGDNP) (RGD peptide GRGDNP(2TFA)) is a integrin-ligand interactions inhibitor.Formule :C23H38N10O10Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :614.61Phenamacril
CAS :Phenamacril (JS39919) is acyanoacrylate fungicide, has powerful inhibition against Fusarium species, especially to Fusarium graminearum.Formule :C12H12N2O2Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :216.24Ref: TM-T24214
1mg145,00€5mg319,00€10mg472,00€25mg753,00€50mg1.074,00€100mg1.444,00€500mg2.822,00€1mL*10mM (DMSO)274,00€α-Linolenic acid
CAS :α-Linolenic Acid (ALA) is an essential fatty acid. α-Linolenic acid improves memory, inhibits thrombosis, and lowers blood lipids. Cost-effective and quality-assured.Formule :C18H30O2Degré de pureté :98.19% - 99.81%Couleur et forme :Physical Description Clear Colorless Liquid (Ntp 1992)Masse moléculaire :278.43Cyclo(RGDfC) TFA
Zelminemab (AMG-301) is a humanized monoclonal antibody targeting ADCYAP1R1 for use in neurological disorders.Formule :C26H35F3N8O9SDegré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :692.67ɛPKC(85-92),Myristoylated
CAS :PKC(85-92),Myristoylated is a myristic acid-conjugated, cell-permeable peptide activator of PKC that has been shown to increase nitric oxide (NO) release inFormule :C53H80N10O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1097.26cRGDfK-thioacetyl ester
CAS :cRGDfK-thioacetyl ester, a bioactive polypeptide, exhibits selective affinity for integrins and can modify near-infrared (NIR) fluorescent probes for targetedFormule :C31H45N9O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :719.81
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