Receptor de adenosina
Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.
Produtos da "Receptor de adenosina"
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KI-7
CAS:KI-7 is an adenosine A2B receptor positive allosteric modulator.Fórmula:C23H18N2O2Pureza:98.03%Cor e Forma:SolidPeso molecular:354.4Ref: TM-T9238
2mg38,00€5mg58,00€10mg90,00€25mg182,00€50mg279,00€100mg420,00€200mg592,00€1mL*10mM (DMSO)65,00€Acefylline
CAS:Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.Fórmula:C9H10N4O4Pureza:99.57%Cor e Forma:White Crystalline SolidPeso molecular:238.2YGZ-331
CAS:YGZ-331, a sedative hypnotic, acts by elevating GABA levels as a derivative of the adenosine nucleoside NGBA. It functions through activating A1R and A2aR, and inhibiting the phosphorylation of CaMKII (pCaMKII), thereby exerting its calming effects. Additionally, YGZ-331 reduces spontaneous motor activity in mice.Fórmula:C19H23N5O4Cor e Forma:SolidPeso molecular:385.42MRS1220
CAS:MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeuticFórmula:C21H14ClN5O2Pureza:96.59%Cor e Forma:SolidPeso molecular:403.82LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Fórmula:C18H14FN5OPureza:100% - 99.03%Cor e Forma:SolidPeso molecular:335.34Swertisin
CAS:Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.Fórmula:C22H22O10Pureza:99.74% - 99.79%Cor e Forma:SolidPeso molecular:446.4SCH 58261
CAS:SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Fórmula:C18H15N7OPureza:99.07% - 99.75%Cor e Forma:SolidPeso molecular:345.36Ref: TM-T6979
1mg40,00€2mg51,00€5mg85,00€10mg125,00€25mg225,00€50mg364,00€100mg582,00€1mL*10mM (DMSO)86,00€Diphylline
CAS:Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.Fórmula:C10H14N4O4Pureza:98.54%Cor e Forma:Crystals From Alcohol SolidPeso molecular:254.24MRS 1754
CAS:MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.Fórmula:C26H26N6O4Pureza:96.12% - 97.48%Cor e Forma:SolidPeso molecular:486.52A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effectiveFórmula:C28H34N6O6Pureza:98%Cor e Forma:SolidPeso molecular:550.61Taminadenant
CAS:Taminadenant is an adenosine receptor antagonist.Fórmula:C10H8BrN7Pureza:99.11%Cor e Forma:SolidPeso molecular:306.12Ref: TM-T16980
5mg51,00€10mg88,00€25mg127,00€50mg170,00€100mg250,00€200mg374,00€1mL*10mM (DMSO)57,00€BAY 60-6583
CAS:BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3Fórmula:C19H17N5O2SPureza:100% - 98.87%Cor e Forma:SolidPeso molecular:379.44Ref: TM-T14506
1mg44,00€5mg92,00€10mg123,00€25mg245,00€50mg418,00€100mg627,00€200mg877,00€1mL*10mM (DMSO)106,00€Rolofylline
CAS:Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Fórmula:C20H28N4O2Pureza:99.53%Cor e Forma:SolidPeso molecular:356.46VPC171
CAS:VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Fórmula:C18H12F3NOSPureza:99.52%Cor e Forma:SolidPeso molecular:347.35Ref: TM-T29112
1mg73,00€2mg96,00€5mg131,00€10mg182,00€25mg335,00€50mg467,00€100mg662,00€200mg892,00€1mL*10mM (DMSO)134,00€
