Receptor de adenosina
Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.
Produtos da "Receptor de adenosina"
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AZD4635
CAS:AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Fórmula:C15H11ClFN5Pureza:99.15% - 99.90%Cor e Forma:SolidPeso molecular:315.73Ref: TM-T4265
1mg37,00€2mg52,00€5mg79,00€10mg116,00€25mg188,00€50mg296,00€100mg457,00€500mg1.008,00€1mL*10mM (DMSO)87,00€BAY-545
CAS:BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Fórmula:C18H22F3N3O4SPureza:98.05%Cor e Forma:SolidPeso molecular:433.45Ref: TM-T8512
1mg88,00€5mg170,00€10mg248,00€25mg444,00€50mg638,00€100mg889,00€200mg1.198,00€1mL*10mM (DMSO)182,00€Kira8 Hydrochloride
CAS:Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.Fórmula:C31H30Cl2N6O3SPureza:98%Cor e Forma:SolidPeso molecular:637.58A2A receptor antagonist 1
CAS:A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.Fórmula:C16H12FN5OPureza:99.29% - 99.76%Cor e Forma:SolidPeso molecular:309.3Ref: TM-T37792
1mg37,00€5mg64,00€10mg92,00€25mg185,00€50mg284,00€100mg419,00€500mg883,00€1mL*10mM (DMSO)47,00€Norisoboldine
CAS:Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.Fórmula:C18H19NO4Pureza:98.12%Cor e Forma:SolidPeso molecular:313.35Adenosine amine congener
CAS:Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Fórmula:C28H32N8O6Pureza:97.86%Cor e Forma:SolidPeso molecular:576.6Theophylline monohydrate
CAS:Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calciumFórmula:C7H8N4O2·H2OPureza:99.78%Cor e Forma:SolidPeso molecular:198.18Nelonicline
CAS:Nelonicline is a selective agonist of neuronal nicotinic receptors.Fórmula:C17H19N3OSPureza:98%Cor e Forma:SolidPeso molecular:313.42Alloxazine
CAS:Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.Fórmula:C10H6N4O2Pureza:99.75%Cor e Forma:SolidPeso molecular:214.18N6-Cyclohexyladenosine
CAS:N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.Fórmula:C16H23N5O4Pureza:99.84% - 99.98%Cor e Forma:SolidPeso molecular:349.38Xanthine amine congener trihydrochloride
CAS:Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Fórmula:C21H29ClN6O4Pureza:97.85%Cor e Forma:SolidPeso molecular:464.95CCPA
CAS:CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptorFórmula:C15H20ClN5O4Pureza:99.10%Cor e Forma:Off-White To Light Yellow SolidPeso molecular:369.8PF-02575799
CAS:PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).Fórmula:C42H37FN4O4Pureza:98%Cor e Forma:SolidPeso molecular:680.77Piclidenoson
CAS:Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.Fórmula:C18H19IN6O4Pureza:100% - ≥95%Cor e Forma:SolidPeso molecular:510.29Ref: TM-T7188
2mg42,00€5mg62,00€10mg89,00€25mg183,00€50mg298,00€100mg464,00€200mg663,00€1mL*10mM (DMSO)70,00€ANR 94
CAS:ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.Fórmula:C9H13N5OPureza:98.21%Cor e Forma:SolidPeso molecular:207.23Ref: TM-T22031
2mg42,00€5mg64,00€10mg97,00€25mg188,00€50mg329,00€100mg465,00€200mg655,00€1mL*10mM (DMSO)63,00€CGS 15943
CAS:CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.Fórmula:C13H8ClN5OPureza:99.63%Cor e Forma:SolidPeso molecular:285.695-Iodotubercidin
CAS:5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.Fórmula:C11H13IN4O4Pureza:99.98%Cor e Forma:Tan SolidPeso molecular:392.15Ref: TM-T6745
1mg46,00€2mg57,00€5mg92,00€10mg155,00€25mg343,00€50mg509,00€100mg735,00€1mL*10mM (DMSO)97,00€Regadenoson
CAS:Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.Fórmula:C15H18N8O5Pureza:99.57% - 99.81%Cor e Forma:Off-White SolidPeso molecular:390.35Ref: TM-T2671
2mg47,00€5mg65,00€10mg92,00€25mg173,00€50mg273,00€100mg416,00€500mg935,00€1mL*10mM (DMSO)72,00€MIPS521
CAS:MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Fórmula:C19H10ClF6NOSPureza:99.76%Cor e Forma:SolidPeso molecular:449.8Ref: TM-T9330
1mg38,00€2mg49,00€5mg79,00€10mg111,00€25mg188,00€50mg329,00€100mg512,00€1mL*10mM (DMSO)87,00€PSB 1115
CAS:PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.Fórmula:C14H14N4O5SPureza:100% - 99.24%Cor e Forma:SolidPeso molecular:350.35
