Receptor de adenosina
Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.
Produtos da "Receptor de adenosina"
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Tecadenoson
CAS:Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.Fórmula:C14H19N5O5Pureza:98.83%Cor e Forma:SolidPeso molecular:337.33Ref: TM-T17023
1mg50,00€5mg116,00€10mg178,00€25mg306,00€50mg434,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)128,00€N6-Cyclopentyladenosine
CAS:N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's ofFórmula:C15H21N5O4Pureza:99.84%Cor e Forma:SolidPeso molecular:335.36Vipadenant
CAS:Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Fórmula:C16H15N7OPureza:97.25% - 97.36%Cor e Forma:SolidPeso molecular:321.34Ref: TM-T2373
1mg40,00€2mg52,00€5mg87,00€10mg119,00€25mg210,00€50mg350,00€100mg522,00€500mg1.130,00€1mL*10mM (DMSO)359,00€Tozadenant
CAS:Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Fórmula:C19H26N4O4SPureza:98%Cor e Forma:SolidPeso molecular:406.5Ref: TM-T7320
2mg38,00€5mg58,00€10mg96,00€25mg162,00€50mg273,00€100mg393,00€200mg563,00€1mL*10mM (DMSO)64,00€Doxofylline
CAS:Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.Fórmula:C11H14N4O4Pureza:99.09% - 99.98%Cor e Forma:SolidPeso molecular:266.25Preladenant
CAS:Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosineFórmula:C25H29N9O3Pureza:97.32% - 98.18%Cor e Forma:SolidPeso molecular:503.56APNEA
CAS:APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Fórmula:C18H22N6O4Pureza:99.58%Cor e Forma:SolidPeso molecular:386.41Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.Fórmula:C24H29ClF3N5O5SPureza:96.67%Cor e Forma:SoildPeso molecular:592.03Derenofylline
CAS:Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)Fórmula:C18H20N4OPureza:98.09%Cor e Forma:SolidPeso molecular:308.38Capadenoson
CAS:Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Fórmula:C25H18ClN5O2S2Pureza:98.85% - 99.62%Cor e Forma:SolidPeso molecular:520.03Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Fórmula:C17H17N5O6SPureza:98.83% - 99.69%Cor e Forma:Off-White SolidPeso molecular:419.41hA3AR agonist 2
hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.Fórmula:C11H14ClN5O2SCor e Forma:SolidPeso molecular:315.78A2AR-agonist-1
CAS:A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).Fórmula:C20H22N6O4Pureza:99.82%Cor e Forma:SolidPeso molecular:410.43Ref: TM-T10212
1mg96,00€2mg134,00€5mg188,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€500mg1.691,00€1mL*10mM (DMSO)217,00€CHEMBL241987
CAS:CHEMBL241987 targets the Adenosine receptor A3 (human)Fórmula:C16H11N3OPureza:99.81%Cor e Forma:SolidPeso molecular:261.28Ref: TM-T8598
2mg35,00€5mg50,00€10mg66,00€25mg108,00€50mg162,00€100mg235,00€200mg349,00€1mL*10mM (DMSO)50,00€ZM241385
CAS:ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.Fórmula:C16H15N7O2Pureza:95.28% - 99.69%Cor e Forma:SolidPeso molecular:337.34Ref: TM-T7021
5mg57,00€10mg82,00€25mg133,00€50mg233,00€100mg432,00€200mg652,00€500mg1.026,00€1mL*10mM (DMSO)57,00€Tonapofylline
CAS:Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.Fórmula:C22H32N4O4Pureza:99.52%Cor e Forma:SolidPeso molecular:416.51Namodenoson
CAS:Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Fórmula:C18H18ClIN6O4Pureza:98.97%Cor e Forma:SolidPeso molecular:544.73ATL444
CAS:ATL444 is an adenosine receptor antagonist with affinity (Ki values) for rA1AR, rA2AAR, rA2BAR, and rA3AR of 7.0, 2.5, 61.8, and >1000 nM, respectively.Fórmula:C17H19N5OCor e Forma:SolidPeso molecular:309.37SCH442416
CAS:SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).Fórmula:C20H19N7O2Pureza:99.58%Cor e Forma:SolidPeso molecular:389.41Ref: TM-T23336
1mg48,00€2mg63,00€5mg93,00€10mg139,00€25mg281,00€50mg449,00€100mg658,00€1mL*10mM (DMSO)97,00€FSCPX
CAS:FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.Fórmula:C23H27FN4O6SPureza:98.00%Cor e Forma:SolidPeso molecular:506.55Ref: TM-T39039
1mg111,00€5mg273,00€10mg409,00€25mg695,00€50mg929,00€100mg1.244,00€200mg1.681,00€1mL*10mM (DMSO)116,00€
