Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
Products of "Androgen Receptor"
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Cyproterone acetate
CAS:Cyproterone acetate (Cyproterone 17-O-acetate) binds the androgen receptor (AR), thereby preventing androgen-induced receptor activation in target tissues andFormula:C24H29ClO4Purity:98.43%Color and Shape:Crystals From Diisopropyl Ether OdourMolecular weight:416.943-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.Formula:C18H14N4OPurity:98.15%Color and Shape:SolidMolecular weight:302.33WCA-814
WCA-814, an androgen receptor (AR) antagonist-Hsp90 inhibitor conjugate, induces degradation of both full-length and AR-V7, exhibiting cytotoxic effects inFormula:C46H53ClN10O5Purity:98%Color and Shape:SolidMolecular weight:861.43Medroxyprogesterone Acetate
CAS:Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. Farlutin is a long-acting contraceptive.Formula:C24H34O4Purity:99.05% - 99.44%Color and Shape:White PowderMolecular weight:386.52BMS-986365
CAS:BMS-986365 (CC-94676) is an orally available, selective and highly potent AR degrader with potential anticancer activity that inhibits AR signaling and suppresses tumor growth for the study of prostate cancer.Formula:C41H45F3N8O5SPurity:98.77% - 99.96%Color and Shape:SoildMolecular weight:818.91Testosterone undecanoate
CAS:Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.Formula:C30H48O3Purity:99.45%Color and Shape:White Crystalline PowderMolecular weight:456.7LGD-2226
CAS:LGD-2226: selective oral androgen receptor modulator, EC50: 0.2nM, Ki: 1.5nM. Treats muscle loss, osteoporosis, sexual issues.Formula:C14H9F9N2OPurity:98%Color and Shape:SolidMolecular weight:392.22TLB 150 Benzoate
CAS:TLB 150 Benzoate (RAD150) is a modulator of the androgen receptor with an IC50 value of 0.13 μM.Formula:C27H20ClN5O3Color and Shape:SolidMolecular weight:497.93Topterone
CAS:Topterone (Win 17,665) is a potent topical antiandrogen that inhibits the stimulation of lumbar organ development by testosterone and dihydrotestosterone inFormula:C22H34O2Purity:100%Color and Shape:SolidMolecular weight:330.5Testosterone acetate
CAS:Testosterone acetate (NSC-523836) is a hormone with in vitro antitumor activity.Formula:C21H30O3Purity:99.60%Color and Shape:White To Off-White Crystalline PowderMolecular weight:330.46FL442
CAS:FL442 is an Androgen Receptor (AR) modulator. This compound exhibits potent inhibitory effects in AR-dependent prostate cancer cells, showing similar suppression efficiency to the traditional antiandrogen drugs Bicalutamide and Enzalutamide. It also maintains antiandrogen activity against the Enzalutamide-resistant AR mutant F876L. The pharmacokinetic properties of FL442 in mice reveal a longer half-life (8 hours), excellent targeting (prostate tissue), and metabolic stability. Additionally, it is effective at inhibiting LNCaP tumor growth at low plasma concentrations (30 ng/mL).Formula:C15H13F3N2OColor and Shape:SolidMolecular weight:294.27GSK-2881078
CAS:GSK-2881078 is a selective androgen receptor modulato (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting.Formula:C14H13F3N2O2SPurity:98.16% - 98.81%Color and Shape:SolidMolecular weight:330.33Lupeol
CAS:Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.Formula:C30H50OPurity:98% - 99.31%Color and Shape:Needles From Alcohol Acetone White PowderMolecular weight:426.72Bicalutamide
CAS:Bicalutamide (ICI-176334), a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting theFormula:C18H14F4N2O4SPurity:98% - 99.87%Color and Shape:Off-White Crystalline SolidMolecular weight:430.37Adrenosterone
CAS:Adrenosterone (11-ketoandrostenedione) is a steroid hormone isolated from the adrenal cortex.Formula:C19H24O3Purity:97.04% - 98.13%Color and Shape:SolidMolecular weight:300.39JNJ-63576253 free base
CAS:JNJ-63576253 free base (TRC253) is a potent and orally active full antagonist of androgen receptor (AR). JNJ-63576253 can be used for the research of CRPC.Formula:C23H21F3N6O2SPurity:98.32%Color and Shape:SolidMolecular weight:502.51Ref: TM-T8933
2mg40.00€5mg52.00€10mg89.00€25mg167.00€50mg258.00€100mg379.00€200mg540.00€1mL*10mM (DMSO)90.00€Apalutamide
CAS:Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.Formula:C21H15F4N5O2SPurity:99.03% - 99.91%Color and Shape:SolidMolecular weight:477.43MK-3984
CAS:MK-3984 is a selective androgen receptor modulator, used in the study of conditions caused by androgen deficiency.Formula:C17H12F7NO2Purity:100%Color and Shape:SolidMolecular weight:395.27DJ-V-159
CAS:DJ-V-159 is a GPRC6A agonist, targeting the G protein-coupled receptor family C group 6 member A (GPRC6A).Formula:C24H12F6N4O2Purity:99.85% - 99.96%Color and Shape:SolidMolecular weight:502.37Nandrolone phenylpropionate
CAS:Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosisFormula:C27H34O3Purity:99.2% - 99.46%Color and Shape:White Or Milky Crystalline PowderMolecular weight:406.56
![3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT9752.webp&w=3840&q=75)
