Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
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Products of "Membrane Transporter/Ion Channel"
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Vesnarinone HCl
Vesnarinone HCl is an oral PDE3 inhibitor improving heart contractility, affecting calcium and potassium flux. Used in heart failure research.Formula:C22H26ClN3O4Purity:99.17%Color and Shape:SoildMolecular weight:431.91Lanatoside C
CAS:Lanatoside C, a cardiac glycoside, treats heart failure and arrhythmia; taken orally or IV.Formula:C49H76O20Purity:100% - 99.8%Color and Shape:SolidMolecular weight:985.12Pramocaine hydrochloride
CAS:Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.Formula:C17H27NO3·HClPurity:99.15% - 99.61%Color and Shape:Crystals White Or Off White Crystalline PowderMolecular weight:329.86ML204
CAS:ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels.Formula:C15H18N2Purity:98.1% - 99.72%Color and Shape:SolidMolecular weight:226.32Ref: TM-T2298
2mg35.00€5mg50.00€10mg74.00€25mg111.00€50mg145.00€100mg220.00€200mg284.00€500mg467.00€1mL*10mM (DMSO)52.00€BMS-394136
CAS:BMS-394136 (BMS 394136) is a KV1.5 antagonist for the treatment of cardiovascular diseases such as arrhythmias and atrial fibrillation.Formula:C24H21Cl2FN4OPurity:98.25% - 98.67%Color and Shape:SolidMolecular weight:471.35Dc1a
Dc1a, a toxin isolated from the desert bush spider Diguetia canities [1], potently facilitates the opening of the German cockroach Na v channel (BgNa v 1).Formula:C276H414N76O84S8Purity:98%Color and Shape:SolidMolecular weight:6397.22Leptomycin A
CAS:Leptomycin A from Streptomyces inhibits CRM1, reducing HIV-1 replication, less potent than Leptomycin B, blocks protein nuclear export.Formula:C32H46O6Purity:98%Color and Shape:SolidMolecular weight:526.7PF 05089771 tosylate
CAS:PF-05089771 inhibits Nav1.7 channels (IC50: 11-33 nM), selective over Nav1.1-1.6/1.8, Ca+, K+ channels, TRPV1; 1000x affinity for half-inactivated state.Formula:C18H12Cl2FN5O3S2·C7H8O3SPurity:97.76%Color and Shape:SolidMolecular weight:672.56ASP7663
CAS:ASP7663 is a TRPA1 Receptor Agonist and exhibiting an abdominal analgesic effect in vivo.Formula:C14H14FNO3Purity:98.61%Color and Shape:SolidMolecular weight:263.26Ciclopirox
CAS:Ciclopirox is an antifungal that chelates Fe3+ and Al3+, inhibiting enzymes and has antibacterial and anti-inflammatory effects.Formula:C12H17NO2Purity:97.72% - 99.41%Color and Shape:SolidMolecular weight:207.27Clamikalant sodium
CAS:Clamikalant sodium (HMR 1098) is an ATP-dependent potassium channel (KATP) cardiac-selective blocker, used in the study of arrhythmias.Formula:C19H21ClN3NaO5S2Purity:99.95%Color and Shape:SolidMolecular weight:493.96Ref: TM-T63330
1mg52.00€5mg100.00€10mg191.00€25mg384.00€50mg595.00€100mg969.00€200mg1,296.00€1mL*10mM (DMSO)105.00€AVE-0118
CAS:AVE-0118 is a potassium channel blocker and suppresses persistent atrial fibrillation.Formula:C30H29N3O3Purity:98.89% - 99.52%Color and Shape:SolidMolecular weight:479.57Ref: TM-T26689
1mg73.00€5mg139.00€10mg183.00€25mg320.00€50mg474.00€100mg688.00€500mg1,444.00€1mL*10mM (DMSO)168.00€Pivagabine
CAS:Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.Formula:C9H17NO3Purity:99.87%Color and Shape:SolidMolecular weight:187.24Ref: TM-T12492
1mg35.00€2mg48.00€5mg70.00€10mg104.00€25mg167.00€50mg249.00€100mg369.00€500mg837.00€1mL*10mM (DMSO)50.00€Nisoxetine hydrochloride
CAS:Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitorFormula:C17H21NO2·HClPurity:98.52%Color and Shape:White SolidMolecular weight:307.82δ-Theraphotoxin-Hm1b
δ-Theraphotoxin-Hm1b, a 42-amino acid peptide derived from the Togo starburst tarantula (Heteroscodra maculata) venom, selectively inhibits the inactivation ofFormula:C169H241N45O50S6Purity:98%Color and Shape:SolidMolecular weight:3895.38Linoleoyl glycine
CAS:Linoleoyl glycine activates hKCNQ1/hKCNE1 channels, has analgesic properties, and is found in skin, spinal cord, and brain.Formula:C20H35NO3Purity:98.96%Color and Shape:SolidMolecular weight:337.5RY785
CAS:RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.Formula:C21H20N4O2SPurity:98.04%Color and Shape:SolidMolecular weight:392.47Ref: TM-T12786
1mg51.00€5mg144.00€10mg235.00€25mg399.00€50mg560.00€100mg787.00€200mg1,093.00€1mL*10mM (DMSO)131.00€Retusin
CAS:Retusin is derived from the leaves of Talinum triangulare. Retusin Retusin can be used in studies about acting as pre- and postemergent herbicides.Formula:C19H18O7Purity:99.00%Color and Shape:SolidMolecular weight:358.34VU590
CAS:VU590 is an inhibitor of extrarenal medullary potassium ROMK.VU590 inhibits Kir7.1 and modulates uterine myometrial contractility and melanocortin signalling.Formula:C24H32N4O7Purity:98.06%Color and Shape:SolidMolecular weight:488.53MZ82
MZ82, a derivative of Ko 143, is a potent inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2/BCRP), with an IC50 of approximately 23 nM. Compared to Ko 143, MZ82 exhibits significantly enhanced metabolic stability in liver microsomes and shows marked improvement in mice, along with the ability to penetrate the brain.Formula:C26H29N3O3Color and Shape:SolidMolecular weight:431.53
