Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
Sort by
ML402
CAS:ML402 (ZINC3671497) is an activator of TREK-1 and TREK-2 with EC50s of 13.7 μM and 5.9 μM.Formula:C14H14ClNO2SPurity:98.93%Color and Shape:SolidMolecular weight:295.78Ref: TM-T16109
1mg37.00€2mg52.00€5mg79.00€10mg119.00€25mg235.00€50mg378.00€100mg560.00€500mg1,216.00€1mL*10mM (DMSO)87.00€Ersentilide
CAS:Ersentilide, a benzamide derivative, functions as both a β1-adrenergic receptor antagonist and an Ikr blocker. It has demonstrated efficacy in animal models of cardiac arrhythmias.Formula:C21H26N4O5SColor and Shape:SolidMolecular weight:446.52GSK369796 Dihydrochloride
CAS:GSK369796 Dihydrochloride (N-tert-butylisoquine),is an anti-malaria drug candidate.Formula:C20H24Cl3N3OPurity:100%Color and Shape:SolidMolecular weight:428.78Ref: TM-T7195
1mg79.00€2mg101.00€5mg149.00€10mg195.00€25mg373.00€50mg562.00€100mg802.00€1mL*10mM (DMSO)145.00€VU0134992 hydrochloride
CAS:VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).Formula:C20H32BrClN2O2Purity:100%Color and Shape:SolidMolecular weight:447.84Ref: TM-T13316
5mg39.00€10mg65.00€25mg108.00€50mg177.00€100mg304.00€200mg437.00€1mL*10mM (DMSO)44.00€BmP02
BmP02, a compound isolated from Chinese scorpion (Buthus martensi Karsch) venom, acts as a selective Kv1.3 channel blocker and a highly-selective Kv4.2Formula:C115H182N36O41S7Purity:98%Color and Shape:SolidMolecular weight:2949.35Sodium Channel inhibitor 4
CAS:Sodium Channel Inhibitor 4 is a compound that functions as a sodium channel inhibitor [1].Formula:C19H18ClN3O4S2Purity:98%Color and Shape:SolidMolecular weight:451.95SKA-111
CAS:SKA-111 activates KCa3.1 potassium channels, modulates membrane potential in endothelial cells, and dilates rat coronary arteries.Formula:C12H10N2SPurity:99.79%Color and Shape:SolidMolecular weight:214.29Ref: TM-T24799
1mg70.00€5mg153.00€10mg250.00€25mg504.00€50mg727.00€100mg1,017.00€500mg2,043.00€1mL*10mM (DMSO)167.00€Besipirdine
CAS:Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.Formula:C16H17N3Purity:97% - 98.59%Color and Shape:SolidMolecular weight:251.33GSK3395879
CAS:GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: 1 nM for hTRPV4).Formula:C20H15F4N3O5SPurity:98%Color and Shape:SolidMolecular weight:485.413′,4′,7-Trihydroxyflavone
CAS:7,3',4'-Trihydroxyflavone blocks osteoclast formation by inhibiting NFATc1 and RANKL-induced differentiation in BMMs.Formula:C15H10O5Purity:99.71% - 99.71%Color and Shape:SolidMolecular weight:270.24Ref: TM-TN3209
1mg106.00€5mg225.00€10mg334.00€25mg557.00€50mg793.00€100mg1,064.00€200mg1,415.00€1mL*10mM (DMSO)208.00€Olisutrigine bromide
CAS:Olisutrigine bromide is a sodium channel blocker used as an analgesic.Formula:C25H35BrN2Color and Shape:SolidMolecular weight:443.463Hypophyllanthin
CAS:Hypophyllanthin and phyllanthin have antitumour effects against Ehrlich Ascites Carcinoma in mice.Formula:C24H30O7Purity:98.39%Color and Shape:SolidMolecular weight:430.49Ciliobrevin D
CAS:Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.Formula:C17H8Cl3N3O2Purity:98.09%Color and Shape:SolidMolecular weight:392.62Ref: TM-T14965
1mg64.00€2mg92.00€5mg140.00€10mg215.00€25mg424.00€50mg625.00€100mg873.00€1mL*10mM (DMSO)157.00€LY2928057
LY2928057 is a humanized monoclonal antibody targeting the iron transporter SLC40A1, an iron-regulatory inhibitor used in cardiovascular disease research.Color and Shape:LiquidMolecular weight:145.5µ-Conotoxin BuIIIB
CAS:μ-Conotoxin BuIIIB (Mu-Conotoxin BuIIIB), a selective blocker of mammalian neuronal voltage-gated sodium channels (VGSC), is derived from Cone snail venom andFormula:C106H172N46O30S6Purity:98%Color and Shape:SolidMolecular weight:2763.18Xilmenolone
CAS:Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].Formula:C26H37N3O2Purity:98%Color and Shape:SolidMolecular weight:423.59NS-2710
CAS:NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.Formula:C22H20N4OPurity:98.10% - 99.82%Color and Shape:SolidMolecular weight:356.42Mebeverine hydrochloride
CAS:Mebeverine hydrochloride (Colofac Hydrochloride), a β-phenylethylamine derivative, is a potent α1 repector inhibitor, relaxing the muscles in and around the gutFormula:C25H35NO5Purity:99.81% - 99.81%Color and Shape:SolidMolecular weight:429.55(3S,6R)-NML
CAS:(3S,6R)-NML is an NMDA receptor antagonist with pIC50 values of 4.8 [GluN1-GluN2A], 4.6 [GluN1-GluN2B], 5.0 [GluN1-GluN2C], and 5.0 [GluN1-GluN2D]. It is applicable in the study of depression.Formula:C20H27NOColor and Shape:SolidMolecular weight:297.435LAU159
CAS:LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).Formula:C17H12ClN3O2Purity:98.70% - 99.38%Color and Shape:SolidMolecular weight:325.75Ref: TM-T11822
1mg116.00€2mg169.00€5mg230.00€10mg418.00€25mg690.00€50mg938.00€100mg1,311.00€500mg2,632.00€
