Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
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Products of "Membrane Transporter/Ion Channel"
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3α,21-Dihydroxy-5α-pregnan-20-one
CAS:3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.Formula:C21H34O3Purity:98.00%Color and Shape:SolidMolecular weight:334.49Rilmazolam
CAS:Rilmazolam is a triazolobenzodiazepine compound and serves as the active metabolite of Rilmazafone.Formula:C19H15Cl2N5OColor and Shape:SolidMolecular weight:400.26Pinacidil
CAS:Pinacidil (P 1134) is a guanidine that opens potassium channels and directly dilates peripheral blood vessels in small arteries, lowering blood pressure andFormula:C13H19N5Purity:99.92%Color and Shape:SolidMolecular weight:245.32TRAM 39
CAS:TRAM 39 (2-Chloro-α,α-diphenylbenzeneacetonitrile) is a selective blocker of intermediate-conductance Ca2+-activated K+channels.Formula:C20H14ClNPurity:99.51%Color and Shape:SolidMolecular weight:303.78Ref: TM-T23471
1mg35.00€2mg49.00€5mg74.00€10mg107.00€25mg210.00€50mg335.00€100mg530.00€500mg1,121.00€SLC13A5-IN-1
CAS:SLC13A5-IN-1 is a selective inhibitor of sodium-citrate co-transporter (SLC13A5),completely blocks the uptake of 14C-citrate(IC50 : 0.022 μM in HepG2 cells).Formula:C19H19Cl3N2O3SPurity:99.11%Color and Shape:SolidMolecular weight:461.79Ref: TM-T12931
1mg50.00€5mg97.00€10mg160.00€25mg283.00€50mg472.00€100mg658.00€200mg933.00€500mg1,378.00€1mL*10mM (DMSO)120.00€Meticrane
CAS:Meticrane (Arresten) is a sulphonamide-derivative with thiazide-like diuretic activity.Formula:C10H13NO4S2Purity:99.16%Color and Shape:SolidMolecular weight:275.34PF-06869206
CAS:PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).Formula:C15H14ClF3N4O2Purity:99.37% - 99.79%Color and Shape:SolidMolecular weight:374.75Talniflumate
CAS:Talniflumate (Somalgen) is a calcium-activated chloride channel (hCLCA1/mCLCA3) blocker that reduces mucin synthesis and releases in animal models and cellFormula:C21H13F3N2O4Purity:98% - 99.81%Color and Shape:White To Pale Yellow Crystalline PowderMolecular weight:414.33Ref: TM-T4503
1mg37.00€2mg52.00€5mg77.00€10mg97.00€25mg182.00€50mg300.00€100mg449.00€1mL*10mM (DMSO)85.00€AZD3965
CAS:AZD3965 (AZD-3965) is a selective inhibitor of monocarboxylate transporter 1 (MCT1).Formula:C21H24F3N5O5SPurity:98% - 99.87%Color and Shape:SolidMolecular weight:515.512'MeO6MF
CAS:2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFormula:C17H14O3Purity:99.28% - 99.63%Color and Shape:SolidMolecular weight:266.29Ref: TM-T8887
1mg51.00€5mg107.00€10mg160.00€25mg255.00€50mg359.00€100mg485.00€200mg662.00€1mL*10mM (DMSO)101.00€D-GsMTx4 TFA
D-GsMTx4 TFA, a selective spider venom peptide, is a TRPC1/6 and Piezo2 inhibitor that inhibits cation-permeable mechanosensitive channels (MSCs) belonging to the Piezo and TRP channel families, blocks cation-selective stretch-activated channels (SACs), and attenuates lysophosphatidylcholine (LPC)-induced astrocyte toxicity and microglia reactivity. toxicity and microglia reactivity.D-GsMTx4 TFA prevented myocardial infarction in a mouse model of ischemia/reperfusion and can be used to characterize the role of excitatory MSCs in normal physiology and pathology.Formula:C187H279F3N48O48S6Purity:99.29% - 99.65%Color and Shape:SoildMolecular weight:4216.93BPDBA
CAS:BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 andFormula:C19H20Cl2N2OPurity:99.24% - 99.86%Color and Shape:SolidMolecular weight:363.28Ref: TM-T26891
5mg40.00€10mg58.00€25mg109.00€50mg170.00€100mg273.00€200mg378.00€1mL*10mM (DMSO)78.00€Dipropofol
CAS:Dipropofol (4,4-Bis(2,6-di-isopropylphenol)) is a small molecule GABAA receptor agonist that can be used to study epilepsy.Formula:C24H34O2Purity:99.6%Color and Shape:SolidMolecular weight:354.53Mesendogen
CAS:Mesendogen is an inhibitor of transient receptor potential cation channel, subfamily M, member 6 (TRPM6) and 7 (TRPM7) and acts by inhibiting TRPM6/TRPM7Formula:C18H16ClF3N2OSPurity:98.90%Color and Shape:SolidMolecular weight:400.85Apcin A HCL
CAS:Apcin A HCL is an Apcin derivative. Apcin A HCL is an anaphase-promoting complex (APC) inhibitor. Apcin-A HCL interacts strongly with Cdc20, and inhibits the ubiquitination of Cdc20 substrates. Apcin-A HCL can be used to synthesize the PROTAC CP5V [1].Formula:C10H15Cl4N5O2Purity:99.30%Color and Shape:SolidMolecular weight:379.07Ref: TM-T001
1mgTo inquire2mg63.00€5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire200mgTo inquire500mg2,792.00€Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Formula:C20H25NO2S2Purity:99.24%Color and Shape:White To Off-White Crystalline SolidMolecular weight:375.55ASG-5ME
ASG-5ME is a drug-antibody coupling targeting SLC44A4 that shows anti-tumor activity in xenograft models and may be used to study pancreatic and gastric cancer.Color and Shape:LiquidMolecular weight:145.5 kDaVanilloid receptor antagonist 1
CAS:Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.Formula:C18H15N3O2Purity:98.14%Color and Shape:SolidMolecular weight:305.33Ref: TM-T9247
1mg99.00€5mg235.00€10mg354.00€25mg602.00€50mg847.00€100mg1,206.00€1mL*10mM (DMSO)47.00€Propanidid
CAS:Propanidid (Sombrevin) is a gamma-aminobutyric acid type A receptor (GABAA) agonist and an intravenous anesthetic that lowers arterial blood pressure.Formula:C18H27NO5Purity:99.39%Color and Shape:SolidMolecular weight:337.41Ref: TM-T34146
1mg43.00€5mg85.00€10mg106.00€25mg173.00€50mg255.00€100mg373.00€200mg550.00€500mg803.00€
