Casein Kinase
Casein kinases are a family of serine/threonine protein kinases that regulate various cellular processes, including DNA repair, circadian rhythms, and signal transduction. These kinases are involved in the phosphorylation of numerous proteins and are implicated in diseases such as cancer, neurodegenerative disorders, and metabolic syndromes. At CymitQuimica, we offer a selection of casein kinase inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.
Products of "Casein Kinase"
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CK2-IN-4
CAS:CK2-IN-4 is a protein kinase (CK2) inhibitor with an IC50 value of 8.6 µM.Formula:C18H11N3O4SPurity:99.72%Color and Shape:SolidMolecular weight:365.36SR-3029
CAS:SR-3029 is a potent and highly specific CK1δ/CK1ε inhibitor.Formula:C23H19F3N8OPurity:99.64%Color and Shape:SolidMolecular weight:480.45CK1-IN-1
CAS:CK1-IN-1, a CK1 inhibitor with IC50: 15nM CK1δ, 16nM CK1ε, 73nM p38σ; patent WO2015119579A1.Formula:C24H15F2N3Purity:98.79%Color and Shape:SolidMolecular weight:383.39Ref: TM-T5393
1mg49.00€2mg65.00€5mg97.00€10mg160.00€25mg305.00€50mg472.00€100mg707.00€1mL*10mM (DMSO)106.00€Casein kinase 1δ-IN-30
CAS:Casein kinase1δ-IN-30 (Compound 581) is an inhibitor of casein kinase 1δ (CK1δ). It can be utilized in research related to neurodegenerative diseases.Formula:C18H15BrN6O2SColor and Shape:SolidMolecular weight:459.32CX-5011
CAS:CX-5011, a CK2 inhibitor, induces Rac1 activation and promotes apoptosis, effectively causing cancer cell death [1] [2].Formula:C20H12N4O2Purity:98%Color and Shape:SolidMolecular weight:340.33Casein kinase 1δ-IN-1
CAS:Casein kinase 1δ-IN-1 (WAY-643895) is an inhibitor of casein kinase 1δ (CK1δ), which inhibits CK1δ.Formula:C11H7N3OSPurity:99.46%Color and Shape:SolidMolecular weight:229.26Silmitasertib sodium salt
CAS:Silmitasertib sodium salt (CX-4945 sodium salt) is a potent and orally bioavailable, highly selective inhibitor of CK2(IC50 of 1 nM, CK2α).Formula:C19H11ClN3NaO2Purity:99.49% - 99.62%Color and Shape:SolidMolecular weight:371.75MGD-28
CAS:MGD-28 is a Cullin-CRBN-dependent IKZF family protein degrader for IKZF1 (Ikaros), IKZF2 (Helios), IKZF3 (Aiolos) ,and CK1α, antiproliferative.Formula:C33H34FN7O3Purity:99.39%Color and Shape:SolidMolecular weight:595.67SR-1277
CAS:SR-1277 is a potent, highly selective and ATP-competitive CK1δ/ε inhibitor, regulating Wee1 activity at the G2/M cell-cycle interface, and antiproliferative.Formula:C21H19N9O3SColor and Shape:SolidMolecular weight:477.5PI-828
CAS:PI-828 (LY 294002), a PI3K inhibitor, researches PI3K function and aids stem cell differentiation into mesoderm.Formula:C19H18N2O3Purity:99.39%Color and Shape:SolidMolecular weight:322.36Ref: TM-T16528
1mg35.00€5mg78.00€10mg117.00€25mg197.00€50mg283.00€100mg386.00€200mg550.00€1mL*10mM (DMSO)55.00€Orobol
CAS:Orobol (3’,4’,5,7-tetrahydroxy-isoflavon) is an inhibitor of tyrosine-specific protein kinase and phosphatidylinositol turnover.Formula:C15H10O6Purity:98% - 98%Color and Shape:SolidMolecular weight:286.24Casein kinase 1δ-IN-5
CAS:Casein kinase 1δ-IN-5 is a potent and selective CK-1δ inhibitor, exhibiting an IC50 of 47 nM, and demonstrates neuroprotective and anti-inflammatory effects inFormula:C16H11F3N2OSPurity:98%Color and Shape:SolidMolecular weight:336.33Casein kinase 1δ-IN-6
CAS:CK1δ-IN-6: potent, selective CK-1δ inhibitor, IC50 23 nM, neuroprotective, anti-inflammatory, for neurodegenerative research.Formula:C16H10ClF3N2OSPurity:99%Color and Shape:SoildMolecular weight:370.78Ref: TM-T77500
1mg127.00€2mg177.00€5mg283.00€10mg424.00€25mg740.00€50mg1,035.00€100mg1,454.00€500mg2,822.00€XL413 xHCl
CAS:BMS-863233 HCl is an ATP-competitive Cdc7 inhibitor (IC50: 3.4 nM) that is potent and selective.BMS-863233 HCl inhibited CK2 and PIM1 with IC50 values of 215Formula:C14H12ClN3O2·xHClPurity:99.42% - 99.67%Color and Shape:SolidMolecular weight:326.18dCK1α-2
dCK1α-2 is an orally effective CK1α molecular glue (Molecular Glue) degrader that targets p53 pathway-related targets. It demonstrates antitumor efficacy in mouse models by enhancing the expression of p53-related genes.Formula:C24H24ClN5O4Color and Shape:SolidMolecular weight:481.93LY-294002 hydrochloride
CAS:LY-294002 HCl (NSC 697286) is a stable PI3K inhibitor (IC50: 0.5-0.97 µM) and prevents autophagosome formation.Formula:C19H17NO3·HClPurity:99.95%Color and Shape:SolidMolecular weight:343.81SSTC3
CAS:SSTC3 is a casein kinase 1α (CK1α) activator with potential antitumor activity that inhibits WNT signaling.Formula:C23H17F3N4O3S2Purity:98.65%Color and Shape:SolidMolecular weight:518.53Casein kinase 1δ-IN-7
CAS:Casein kinase 1δ-IN-7 is a Casein kinase 1δ inhibitor for neurodegenerative diseases such as Alzheimer's disease.Formula:C17H14N4O2SPurity:98.6%Color and Shape:SolidMolecular weight:338.38Umbralisib
CAS:Umbralisib (TGR 1202) is a PI3Kδ inhibitor.Formula:C31H24F3N5O3Purity:99.56% - 99.56%Color and Shape:White SolidMolecular weight:571.55Ref: TM-T4976
1mg48.00€2mg65.00€5mg96.00€10mg170.00€25mg343.00€50mg449.00€100mg658.00€1mL*10mM (DMSO)120.00€Ellagic acid (hydrate)
CAS:Ellagic acid (hydrate) is a natural antioxidant and acts as a potent and ATP-competitive CK2 inhibitor (IC50:40 nM, Ki: 20 nM).Formula:C14H8O9Purity:98%Color and Shape:Green To Beige PowderMolecular weight:320.21
